Compile Data Set for Download or QSAR
maximum 50k data
Found 5 Enz. Inhib. hit(s) with all data for entry = 50030062
TargetTyrosine-protein kinase ZAP-70(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50069336(CHEMBL439120 | NELNLGRREE | NQLPpYNELNLGRREEpYDVLD)
Affinity DataIC50:  30nMAssay Description:Antagonistic activity against SH2 domain of Zeta-chain (TCR) associated protein kinase, ZAP-70More data for this Ligand-Target Pair
In DepthDetails Article
TargetTyrosine-protein kinase ZAP-70(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50290773(CHEMBL443592 | Non-peptide bidentate ITAM analogue)
Affinity DataIC50:  250nMAssay Description:Antagonistic activity against SH2 domain of Zeta-chain (TCR) associated protein kinase, ZAP-70More data for this Ligand-Target Pair
In DepthDetails Article
TargetTyrosine-protein kinase ZAP-70(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50290771(CHEMBL386787 | Non-peptide bidentate ITAM analogue)
Affinity DataIC50:  320nMAssay Description:Antagonistic activity against SH2 domain of Zeta-chain (TCR) associated protein kinase, ZAP-70More data for this Ligand-Target Pair
In DepthDetails Article
TargetTyrosine-protein kinase ZAP-70(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50290774(CHEMBL99125 | [Difluoro-(4-{[hexanoyl-((8R,9S,13S,...)
Affinity DataIC50:  1.90E+3nMAssay Description:Antagonistic activity against SH2 domain of Zeta-chain (TCR) associated protein kinase, ZAP-70More data for this Ligand-Target Pair
In DepthDetails Article
TargetTyrosine-protein kinase ZAP-70(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50290772((4-{[Hexanoyl-((8R,9S,13S,14S,17S)-13-methyl-3-pro...)
Affinity DataIC50:  3.20E+3nMAssay Description:Antagonistic activity against SH2 domain of Zeta-chain (TCR) associated protein kinase, ZAP-70More data for this Ligand-Target Pair
In DepthDetails Article