Compile Data Set for Download or QSAR
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Found 12 Enz. Inhib. hit(s) with all data for entry = 50030073
TargetDelta-type opioid receptor(MOUSE)
TBA

Curated by ChEMBL
LigandPNGBDBM50060080(2-({2-[(R)-2-Amino-3-(4-hydroxy-2,6-dimethyl-pheny...)
Affinity DataKi:  191nMAssay Description:The compound was evaluated for the binding affinity towards delta-opioid receptor by displacement of [3H]p-CI-DPDPE radioligand from mouse vas defere...More data for this Ligand-Target Pair
In DepthDetails Article
TargetMu-type opioid receptor(GUINEA PIG)
TBA

Curated by ChEMBL
LigandPNGBDBM50060080(2-({2-[(R)-2-Amino-3-(4-hydroxy-2,6-dimethyl-pheny...)
Affinity DataKi:  2.84E+4nMAssay Description:The compound was evaluated for the binding affinity towards mu-opioid receptor by displacement of [3H]DAMGO radioligand from guinea pig ileumMore data for this Ligand-Target Pair
In DepthDetails Article
TargetDelta-type opioid receptor(MOUSE)
TBA

Curated by ChEMBL
LigandPNGBDBM50290894((S)-2-[(2S,3R)-2-Amino-3-(4-hydroxy-2,6-dimethyl-p...)
Affinity DataIC50:  9.30nMAssay Description:The compound was evaluated for the binding affinity towards delta-opioid receptor by displacement of [3H]-p-CI-DPDPE radioligand from mouse vas defer...More data for this Ligand-Target Pair
In DepthDetails Article
TargetDelta-type opioid receptor(MOUSE)
TBA

Curated by ChEMBL
LigandPNGBDBM50290890((S)-2-[2-tert-Butoxycarbonylamino-3-(4-hydroxy-2,6...)
Affinity DataIC50:  19nMAssay Description:The compound was evaluated for the binding affinity towards delta-opioid receptor by displacement of [3H]-p-CI-DPDPE radioligand from mouse vas defer...More data for this Ligand-Target Pair
In DepthDetails Article
TargetDelta-type opioid receptor(MOUSE)
TBA

Curated by ChEMBL
LigandPNGBDBM50290892((S)-2-[(2S,3S)-2-Amino-3-(4-hydroxy-2,6-dimethyl-p...)
Affinity DataIC50:  124nMAssay Description:The compound was evaluated for the binding affinity towards delta-opioid receptor by displacement of [3H]-p-CI-DPDPE radioligand from mouse vas defer...More data for this Ligand-Target Pair
In DepthDetails Article
TargetMu-type opioid receptor(GUINEA PIG)
TBA

Curated by ChEMBL
LigandPNGBDBM50290890((S)-2-[2-tert-Butoxycarbonylamino-3-(4-hydroxy-2,6...)
Affinity DataIC50:  8.40E+3nMAssay Description:The compound was evaluated for the binding affinity towards mu-opioid receptor by displacement of [3H]-DAMGO radioligand from guinea pig ileumMore data for this Ligand-Target Pair
In DepthDetails Article
TargetDelta-type opioid receptor(MOUSE)
TBA

Curated by ChEMBL
LigandPNGBDBM50290891((S)-2-[(2R,3R)-2-Amino-3-(4-hydroxy-2,6-dimethyl-p...)
Affinity DataIC50: >1.00E+4nMAssay Description:The compound was evaluated for the binding affinity towards delta-opioid receptor by displacement of [3H]-p-CI-DPDPE radioligand from mouse vas defer...More data for this Ligand-Target Pair
In DepthDetails Article
TargetDelta-type opioid receptor(MOUSE)
TBA

Curated by ChEMBL
LigandPNGBDBM50290889((S)-2-[(2R,3S)-2-Amino-3-(4-hydroxy-2,6-dimethyl-p...)
Affinity DataIC50: >1.00E+4nMAssay Description:The compound was evaluated for the binding affinity towards delta-opioid receptor by displacement of [3H]-p-CI-DPDPE radioligand from mouse vas defer...More data for this Ligand-Target Pair
In DepthDetails Article
TargetMu-type opioid receptor(GUINEA PIG)
TBA

Curated by ChEMBL
LigandPNGBDBM50290894((S)-2-[(2S,3R)-2-Amino-3-(4-hydroxy-2,6-dimethyl-p...)
Affinity DataIC50:  3.50E+4nMAssay Description:The compound was evaluated for the binding affinity towards mu-opioid receptor by displacement of [3H]-DAMGO radioligand from guinea pig ileumMore data for this Ligand-Target Pair
In DepthDetails Article
TargetMu-type opioid receptor(GUINEA PIG)
TBA

Curated by ChEMBL
LigandPNGBDBM50290892((S)-2-[(2S,3S)-2-Amino-3-(4-hydroxy-2,6-dimethyl-p...)
Affinity DataIC50: >8.00E+4nMAssay Description:The compound was evaluated for the binding affinity towards mu-opioid receptor by displacement of [3H]-DAMGO radioligand from guinea pig ileumMore data for this Ligand-Target Pair
In DepthDetails Article
TargetMu-type opioid receptor(GUINEA PIG)
TBA

Curated by ChEMBL
LigandPNGBDBM50290891((S)-2-[(2R,3R)-2-Amino-3-(4-hydroxy-2,6-dimethyl-p...)
Affinity DataIC50: >8.00E+4nMAssay Description:The compound was evaluated for the binding affinity towards mu-opioid receptor by displacement of [3H]-DAMGO radioligand from guinea pig ileumMore data for this Ligand-Target Pair
In DepthDetails Article
TargetMu-type opioid receptor(GUINEA PIG)
TBA

Curated by ChEMBL
LigandPNGBDBM50290889((S)-2-[(2R,3S)-2-Amino-3-(4-hydroxy-2,6-dimethyl-p...)
Affinity DataIC50: >8.00E+4nMAssay Description:The compound was evaluated for the binding affinity towards mu-opioid receptor by displacement of [3H]-DAMGO radioligand from guinea pig ileumMore data for this Ligand-Target Pair
In DepthDetails Article