Compile Data Set for Download or QSAR
maximum 50k data
Found 10 Enz. Inhib. hit(s) with all data for entry = 50030210
TargetEndothelin-1 receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50292475(CHEMBL510130 | hypophyllanthin)
Affinity DataIC50:  4.00E+4nMAssay Description:Displacement of [125I]endothelin-1 from human recombinant ETA receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails Article
TargetEndothelin-1 receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50292476(CHEMBL453822 | nirtetralin)
Affinity DataIC50:  7.50E+4nMAssay Description:Displacement of [125I]endothelin-1 from human recombinant ETA receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails Article
TargetEndothelin-1 receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50292478((2S,4S)-5,8-dimethoxy-6-methyl-4-phenyl-1,2,3,4-te...)
Affinity DataIC50:  1.60E+5nMAssay Description:Displacement of [125I]endothelin-1 from human recombinant ETA receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails Article
TargetEndothelin-1 receptor(RAT)
TBA

Curated by ChEMBL
LigandPNGBDBM50292476(CHEMBL453822 | nirtetralin)
Affinity DataIC50:  4.00E+5nMAssay Description:Displacement of [125I]endothelin-1 from ETA receptor in rat A10 cells by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails Article
TargetEndothelin receptor type B(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50292477(CHEMBL453568 | phyllanthin)
Affinity DataIC50: >5.00E+5nMAssay Description:Displacement of [125I]endothelin-1 from human recombinant ETB receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails Article
TargetEndothelin receptor type B(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50292476(CHEMBL453822 | nirtetralin)
Affinity DataIC50: >5.00E+5nMAssay Description:Displacement of [125I]endothelin-1 from human recombinant ETB receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails Article
TargetEndothelin receptor type B(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50292475(CHEMBL510130 | hypophyllanthin)
Affinity DataIC50: >5.00E+5nMAssay Description:Displacement of [125I]endothelin-1 from human recombinant ETB receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails Article
TargetEndothelin-1 receptor(RAT)
TBA

Curated by ChEMBL
LigandPNGBDBM50292475(CHEMBL510130 | hypophyllanthin)
Affinity DataIC50:  5.80E+5nMAssay Description:Displacement of [125I]endothelin-1 from ETA receptor in rat A10 cells by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails Article
TargetEndothelin-1 receptor(RAT)
TBA

Curated by ChEMBL
LigandPNGBDBM50292477(CHEMBL453568 | phyllanthin)
Affinity DataIC50: >1.00E+6nMAssay Description:Displacement of [125I]endothelin-1 from ETA receptor in rat A10 cells by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails Article
TargetEndothelin-1 receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50292477(CHEMBL453568 | phyllanthin)
Affinity DataIC50: >1.00E+6nMAssay Description:Displacement of [125I]endothelin-1 from human recombinant ETA receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails Article