Compile Data Set for Download or QSAR
Report error Found 10 Enz. Inhib. hit(s) with all data for entry = 50034704
LigandChemical structure of BindingDB Monomer ID 50280054BDBM50280054((S)-3-{(S)-2-[(S)-2-tert-Butoxycarbonylamino-3-(1H...)
Affinity DataIC50: 350nMAssay Description:Concentration of compound required to inhibit binding of [125I]J-BH-CCK-8 radioligand to CCKB in mouse fore brain membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/23/2012
Entry Details Article

TargetCholecystokinin receptor type A(Mouse)
TBA

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50280054BDBM50280054((S)-3-{(S)-2-[(S)-2-tert-Butoxycarbonylamino-3-(1H...)
Affinity DataIC50: 3.50E+3nMAssay Description:Concentration of compound required to inhibit binding of [125I]J-BH-CCK-8 radioligand to CCKA in mouse pancreatic membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/23/2012
Entry Details Article

TargetCholecystokinin receptor type A(Mouse)
TBA

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50280052BDBM50280052(7-Methyl-4,6,6a,7,8,9-hexahydro-indolo[4,3-fg]quin...)
Affinity DataIC50: 1.20E+4nMAssay Description:Concentration of compound required to inhibit binding of [125I]J-BH-CCK-8 radioligand to CCKA in mouse pancreatic membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/23/2012
Entry Details Article

LigandChemical structure of BindingDB Monomer ID 50027065BDBM50027065(12'-hydroxy-2'-methyl-5'alpha-(phenylmethyl)ergota...)
Affinity DataIC50: 1.70E+4nMAssay Description:Concentration of compound required to inhibit binding of [125I]J-BH-CCK-8 radioligand to CCKB in mouse fore brain membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/23/2012
Entry Details Article

LigandChemical structure of BindingDB Monomer ID 50295557BDBM50295557(CHEMBL1732 | 7-Methyl-4,6,6a,7,8,9-hexahydro-indol...)
Affinity DataIC50: 2.30E+4nMAssay Description:Concentration of compound required to inhibit binding of [125I]J-BH-CCK-8 radioligand to CCKB in mouse fore brain membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/23/2012
Entry Details Article

TargetCholecystokinin receptor type A(Mouse)
TBA

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50027065BDBM50027065(12'-hydroxy-2'-methyl-5'alpha-(phenylmethyl)ergota...)
Affinity DataIC50: 3.40E+4nMAssay Description:Concentration of compound required to inhibit binding of [125I]J-BH-CCK-8 radioligand to CCKA in mouse pancreatic membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/23/2012
Entry Details Article

LigandChemical structure of BindingDB Monomer ID 50390993BDBM50390993(CHEMBL1403281)
Affinity DataIC50: 8.00E+4nMAssay Description:Concentration of compound required to inhibit binding of [125I]J-BH-CCK-8 radioligand to CCKB in mouse fore brain membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/23/2012
Entry Details Article

TargetCholecystokinin receptor type A(Mouse)
TBA

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50295557BDBM50295557(CHEMBL1732 | 7-Methyl-4,6,6a,7,8,9-hexahydro-indol...)
Affinity DataIC50: 8.00E+4nMAssay Description:Concentration of compound required to inhibit binding of [125I]J-BH-CCK-8 radioligand to CCKA in mouse pancreatic membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/23/2012
Entry Details Article

TargetCholecystokinin receptor type A(Mouse)
TBA

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50390993BDBM50390993(CHEMBL1403281)
Affinity DataIC50: 8.00E+4nMAssay Description:Concentration of compound required to inhibit binding of [125I]J-BH-CCK-8 radioligand to CCKA in mouse pancreatic membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/23/2012
Entry Details Article

LigandChemical structure of BindingDB Monomer ID 50280052BDBM50280052(7-Methyl-4,6,6a,7,8,9-hexahydro-indolo[4,3-fg]quin...)
Affinity DataIC50: 8.00E+4nMAssay Description:Concentration of compound required to inhibit binding of [125I]J-BH-CCK-8 radioligand to CCKB in mouse fore brain membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/23/2012
Entry Details Article