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Found 4 Enz. Inhib. hit(s) with all data for entry = 50034705
TargetTubulin alpha-1A chain(Sus scrofa (Pig))
TBA

Curated by ChEMBL
LigandPNGBDBM50280140(CHEMBL418565 | [6-(3,4,5-Trimethoxy-benzyloxy)-imi...)
Affinity DataKi:  750nMAssay Description:Compound was tested for competitive inhibition with radioligand [3H]colchicine at colchicine site of mammalian tubulinMore data for this Ligand-Target Pair
In DepthDetails Article
TargetTubulin alpha-1A chain(Sus scrofa (Pig))
TBA

Curated by ChEMBL
LigandPNGBDBM50139772(22-oxovincaleukoblastine | leurocristine | vincris...)
Affinity DataIC50:  220nMAssay Description:The compound was evaluated in vitro for the mammalian brain tubulin polymerization using standard assay.More data for this Ligand-Target Pair
In DepthDetails Article
TargetTubulin alpha-1A chain(Sus scrofa (Pig))
TBA

Curated by ChEMBL
LigandPNGBDBM50280140(CHEMBL418565 | [6-(3,4,5-Trimethoxy-benzyloxy)-imi...)
Affinity DataIC50:  310nMAssay Description:In vitro mammalian brain tubulin polymerization using standard assay.More data for this Ligand-Target Pair
In DepthDetails Article
TargetTubulin alpha-1A chain(Sus scrofa (Pig))
TBA

Curated by ChEMBL
LigandPNGBDBM50014846((S)-N-(5,6,7,9-tetrahydro-1,2,3,10-tetramethoxy-9-...)
Affinity DataIC50:  1.50E+3nMAssay Description:The compound was evaluated in vitro for the mammalian brain tubulin polymerization using standard assay.More data for this Ligand-Target Pair