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Found 12 Enz. Inhib. hit(s) with all data for entry = 50034757
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
TBA

Curated by ChEMBL
LigandPNGBDBM50366327(CHEMBL192037)
Affinity DataIC50:  30nMAssay Description:Compound was evaluated for binding affinity to Dopamine receptor D2 labeled with [3H]-SND 919 (0.5 nM) in rat striatal membranesMore data for this Ligand-Target Pair
In DepthDetails Article
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
TBA

Curated by ChEMBL
LigandPNGBDBM50282001((4,5-Dihydro-3H-pyrazolo[4,5,1-ij]quinolin-4-yl)-d...)
Affinity DataIC50:  260nMAssay Description:Compound was evaluated for binding affinity to Dopamine receptor D2 labeled with [3H]-SND 919 (0.5 nM) in rat striatal membranesMore data for this Ligand-Target Pair
In DepthDetails Article
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
TBA

Curated by ChEMBL
LigandPNGBDBM50281999((4,5-Dihydro-3H-pyrazolo[4,5,1-ij]quinolin-4-yl)-p...)
Affinity DataIC50:  2.70E+3nMAssay Description:Compound was evaluated for binding affinity to Dopamine receptor D2 labeled with [3H]-SND 919 (0.5 nM) in rat striatal membranesMore data for this Ligand-Target Pair
In DepthDetails Article
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
TBA

Curated by ChEMBL
LigandPNGBDBM50282000(4,5-Dihydro-3H-pyrazolo[4,5,1-ij]quinolin-4-ylamin...)
Affinity DataIC50:  2.80E+3nMAssay Description:Compound was evaluated for binding affinity to Dopamine receptor D2 labeled with [3H]-SND 919 (0.5 nM) in rat striatal membranesMore data for this Ligand-Target Pair
In DepthDetails Article
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
TBA

Curated by ChEMBL
LigandPNGBDBM50366327(CHEMBL192037)
Affinity DataIC50:  7.10E+3nMAssay Description:Compound was evaluated for binding affinity to Dopamine receptor D2 labeled with [3H]spiroperidol (0.5 nM) in rat striatal membranesMore data for this Ligand-Target Pair
In DepthDetails Article
TargetD(1A) dopamine receptor(RAT)
TBA

Curated by ChEMBL
LigandPNGBDBM50366327(CHEMBL192037)
Affinity DataIC50:  1.45E+4nMAssay Description:Compound was evaluated for binding affinity to Dopamine receptor D1 labeled with [3H]-SCH- 23390 (0.3 nM) in rat striatal membranesMore data for this Ligand-Target Pair
In DepthDetails Article
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
TBA

Curated by ChEMBL
LigandPNGBDBM50282001((4,5-Dihydro-3H-pyrazolo[4,5,1-ij]quinolin-4-yl)-d...)
Affinity DataIC50:  5.04E+4nMAssay Description:Compound was evaluated for binding affinity to Dopamine receptor D2 labeled with [3H]spiroperidol (0.5 nM) in rat striatal membranesMore data for this Ligand-Target Pair
In DepthDetails Article
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
TBA

Curated by ChEMBL
LigandPNGBDBM50281999((4,5-Dihydro-3H-pyrazolo[4,5,1-ij]quinolin-4-yl)-p...)
Affinity DataIC50: >1.00E+5nMAssay Description:Compound was evaluated for binding affinity to Dopamine receptor D2 labeled with [3H]spiroperidol (0.5 nM) in rat striatal membranesMore data for this Ligand-Target Pair
In DepthDetails Article
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
TBA

Curated by ChEMBL
LigandPNGBDBM50282000(4,5-Dihydro-3H-pyrazolo[4,5,1-ij]quinolin-4-ylamin...)
Affinity DataIC50: >1.00E+5nMAssay Description:Compound was evaluated for binding affinity to Dopamine receptor D2 labeled with [3H]spiroperidol (0.5 nM) in rat striatal membranesMore data for this Ligand-Target Pair
In DepthDetails Article
TargetD(1A) dopamine receptor(RAT)
TBA

Curated by ChEMBL
LigandPNGBDBM50282000(4,5-Dihydro-3H-pyrazolo[4,5,1-ij]quinolin-4-ylamin...)
Affinity DataIC50: >1.00E+5nMAssay Description:Compound was evaluated for binding affinity to Dopamine receptor D1 labeled with [3H]-SCH- 23390 (0.3 nM) in rat striatal membranesMore data for this Ligand-Target Pair
In DepthDetails Article
TargetD(1A) dopamine receptor(RAT)
TBA

Curated by ChEMBL
LigandPNGBDBM50282001((4,5-Dihydro-3H-pyrazolo[4,5,1-ij]quinolin-4-yl)-d...)
Affinity DataIC50: >1.00E+5nMAssay Description:Compound was evaluated for binding affinity to Dopamine receptor D1 labeled with [3H]-SCH- 23390 (0.3 nM) in rat striatal membranesMore data for this Ligand-Target Pair
In DepthDetails Article
TargetD(1A) dopamine receptor(RAT)
TBA

Curated by ChEMBL
LigandPNGBDBM50281999((4,5-Dihydro-3H-pyrazolo[4,5,1-ij]quinolin-4-yl)-p...)
Affinity DataIC50: >1.00E+5nMAssay Description:Compound was evaluated for binding affinity to Dopamine receptor D1 labeled with [3H]-SCH- 23390 (0.3 nM) in rat striatal membranesMore data for this Ligand-Target Pair
In DepthDetails Article