Compile Data Set for Download or QSAR
maximum 50k data
Found 24 Enz. Inhib. hit(s) with all data for entry = 50034770
TargetNeuromedin-K receptor(GUINEA PIG)
TBA

Curated by ChEMBL
LigandPNGBDBM50050649(CHEMBL444832 | {(S)-1-[(R)-1-Methyl-2-phenyl-1-(7-...)
Affinity DataIC50:  9nMAssay Description:Binding affinity for NK3 receptor binding sites in guinea pig cortical membranes by using [125I][MePhe7]-NKB as radioligandMore data for this Ligand-Target Pair
In DepthDetails Article
TargetNeuromedin-K receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50079412((NKB)Asp-Met-His-Asp-Phe-Phe-Val-Gly-Leu-Met-NH2 |...)
Affinity DataIC50:  10nMAssay Description:Displacement of [125I][MePhe]-NKB from human NK3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails Article
TargetNeuromedin-K receptor(GUINEA PIG)
TBA

Curated by ChEMBL
LigandPNGBDBM50282774(CHEMBL295301 | {(S)-1-[(R)-1-(8-Carbamoyl-octylcar...)
Affinity DataIC50:  15nMAssay Description:Binding affinity for NK3 receptor binding sites in guinea pig cortical membranes by using [125I][MePhe7]-NKB as radioligandMore data for this Ligand-Target Pair
In DepthDetails Article
TargetNeuromedin-K receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50050649(CHEMBL444832 | {(S)-1-[(R)-1-Methyl-2-phenyl-1-(7-...)
Affinity DataIC50:  16nMAssay Description:Displacement of [125I][MePhe]-NKB from human NK3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails Article
TargetNeuromedin-K receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50052524((S)-N-((S)-1-{[(S)-1-({[(S)-1-((S)-1-Carbamoyl-3-m...)
Affinity DataIC50:  21nMAssay Description:Displacement of [125I][MePhe]-NKB from human NK3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails Article
TargetNeuromedin-K receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50282782(CHEMBL297327 | {(S)-1-[(R)-1-(8-Hydroxy-octylcarba...)
Affinity DataIC50:  22nMAssay Description:Binding affinity for NK3 receptor binding sites in guinea pig cortical membranes by using [125I][MePhe7]-NKB as radioligandMore data for this Ligand-Target Pair
In DepthDetails Article
TargetNeuromedin-K receptor(GUINEA PIG)
TBA

Curated by ChEMBL
LigandPNGBDBM50282782(CHEMBL297327 | {(S)-1-[(R)-1-(8-Hydroxy-octylcarba...)
Affinity DataIC50:  22nMAssay Description:Binding affinity for NK3 receptor binding sites in guinea pig cortical membranes by using [125I][MePhe7]-NKB as radioligandMore data for this Ligand-Target Pair
In DepthDetails Article
TargetNeuromedin-K receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50282775((S)-2-[2-((S)-2-{(S)-2-[2-(4-Hydroxy-phenyl)-acety...)
Affinity DataIC50:  28nMAssay Description:Displacement of [125I][MePhe]-NKB from human NK3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails Article
TargetNeuromedin-K receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50282774(CHEMBL295301 | {(S)-1-[(R)-1-(8-Carbamoyl-octylcar...)
Affinity DataIC50:  39nMAssay Description:Displacement of [125I][MePhe]-NKB from human NK3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails Article
TargetNeuromedin-K receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50282777(CHEMBL295982 | {(S)-1-[1-(8-Hydroxy-octylcarbamoyl...)
Affinity DataIC50:  92nMAssay Description:Displacement of [125I][MePhe]-NKB from human NK3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails Article
TargetNeuromedin-K receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50282783(CHEMBL47929 | {(S)-1-[1-(8-Methoxy-octylcarbamoyl)...)
Affinity DataIC50:  102nMAssay Description:Displacement of [125I][MePhe]-NKB from human NK3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails Article
TargetNeuromedin-K receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50282780(8-[2-((S)-2-tert-Butoxycarbonylamino-2-methyl-3-ph...)
Affinity DataIC50:  229nMAssay Description:Displacement of [125I][MePhe]-NKB from human NK3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails Article
TargetNeuromedin-K receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50282786(CHEMBL430952 | {(S)-1-[1-(4-Hydroxy-benzylcarbamoy...)
Affinity DataIC50:  425nMAssay Description:Displacement of [125I][MePhe]-NKB from human NK3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails Article
TargetNeuromedin-K receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50282784(CHEMBL46113 | [(S)-1-(1-Carbamoyl-2-phenyl-ethylca...)
Affinity DataIC50:  1.52E+3nMAssay Description:Displacement of [125I][MePhe]-NKB from human NK3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails Article
TargetNeuromedin-K receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50050675(CHEMBL33650 | [(S)-1-((S)-1-Carbamoyl-2-phenyl-eth...)
Affinity DataIC50:  1.55E+3nMAssay Description:Tested for binding affinity for human NK3 receptor expressed in CHO cells by using [125I][MePhe]-NKB as radioligand,More data for this Ligand-Target Pair
In DepthDetails Article
TargetNeuromedin-K receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50282779(CHEMBL298252 | {(S)-1-[(S)-1-(8-Hydroxy-octylcarba...)
Affinity DataIC50:  1.69E+3nMAssay Description:Displacement of [125I][MePhe]-NKB from human NK3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails Article
TargetSubstance-K receptor(HAMSTER)
TBA

Curated by ChEMBL
LigandPNGBDBM50282774(CHEMBL295301 | {(S)-1-[(R)-1-(8-Carbamoyl-octylcar...)
Affinity DataIC50:  5.02E+3nMAssay Description:Binding affinity for NK2 receptor binding sites in membranes prepared from hamster urinary bladder by using [125I]NKA as radioligandMore data for this Ligand-Target Pair
In DepthDetails Article
TargetNeuromedin-K receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50282781((S)-N-(1-Carbamoyl-2-phenyl-ethyl)-2-[2-(4-hydroxy...)
Affinity DataIC50:  5.89E+3nMAssay Description:Displacement of [125I][MePhe]-NKB from human NK3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails Article
TargetSubstance-K receptor(HAMSTER)
TBA

Curated by ChEMBL
LigandPNGBDBM50282782(CHEMBL297327 | {(S)-1-[(R)-1-(8-Hydroxy-octylcarba...)
Affinity DataIC50:  6.16E+3nMAssay Description:Binding affinity for NK2 receptor binding sites in membranes prepared from hamster urinary bladder by using [125I]NKA as radioligandMore data for this Ligand-Target Pair
In DepthDetails Article
TargetSubstance-K receptor(HAMSTER)
TBA

Curated by ChEMBL
LigandPNGBDBM50050649(CHEMBL444832 | {(S)-1-[(R)-1-Methyl-2-phenyl-1-(7-...)
Affinity DataIC50:  6.54E+3nMAssay Description:Binding affinity for NK2 receptor binding sites in membranes prepared from hamster urinary bladder by using [125I]NKA as radioligandMore data for this Ligand-Target Pair
In DepthDetails Article
TargetNeuromedin-K receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50282785(CHEMBL295041 | [(R)-1-(1-Carbamoyl-2-phenyl-ethylc...)
Affinity DataIC50:  1.00E+4nMAssay Description:Displacement of [125I][MePhe]-NKB from human NK3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails Article
TargetSubstance-P receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50282774(CHEMBL295301 | {(S)-1-[(R)-1-(8-Carbamoyl-octylcar...)
Affinity DataIC50:  1.00E+4nMAssay Description:Binding affinity for NK1 receptor binding sites in human lymphoma IM9 cells by using [125I]-Bolton-Hunter substance P as radioligandMore data for this Ligand-Target Pair
In DepthDetails Article
TargetSubstance-P receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50282782(CHEMBL297327 | {(S)-1-[(R)-1-(8-Hydroxy-octylcarba...)
Affinity DataIC50:  1.00E+4nMAssay Description:Binding affinity for NK1 receptor binding sites in human lymphoma IM9 cells by using [125I]-Bolton-Hunter substance P as radioligandMore data for this Ligand-Target Pair
In DepthDetails Article
TargetSubstance-P receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50050649(CHEMBL444832 | {(S)-1-[(R)-1-Methyl-2-phenyl-1-(7-...)
Affinity DataIC50:  1.00E+4nMAssay Description:Binding affinity for NK1 receptor binding sites in human lymphoma IM9 cells by using [125I]-Bolton-Hunter substance P as radioligandMore data for this Ligand-Target Pair
In DepthDetails Article