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Found 42 Enz. Inhib. hit(s) with all data for entry = 50034857
TargetGastrin-releasing peptide receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM85484(Bombesin)
Affinity DataKi:  0.150nMAssay Description:Binding affinity against [125 I][4Tyr]-bombesin labeled cloned human GRP(gastrin releasing peptide) receptors stably expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails Article
TargetGastrin-releasing peptide receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50288252(Bombesin analogue | CHEMBL269432)
Affinity DataKi:  0.700nMAssay Description:Binding affinity against [125 I][4Tyr]-bombesin labeled cloned human GRP(gastrin releasing peptide) receptors stably expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails Article
TargetNeuromedin-B receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM85484(Bombesin)
Affinity DataKi:  2nMAssay Description:Binding affinity against [125 I][4Tyr]-bombesin labeled cloned human NMB receptor stably expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails Article
TargetNeuromedin-B receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50288252(Bombesin analogue | CHEMBL269432)
Affinity DataKi:  2.10nMAssay Description:Binding affinity against [125 I][4Tyr]-bombesin labeled cloned human NMB receptor stably expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails Article
TargetNeuromedin-B receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50071754((S)-2-[3-(2,6-Diisopropyl-phenyl)-ureido]-3-(1H-in...)
Affinity DataKi:  6.30nMAssay Description:Binding affinity against [125 I][4Tyr]-bombesin labeled cloned human NMB receptor stably expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails Article
TargetNeuromedin-B receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50071754((S)-2-[3-(2,6-Diisopropyl-phenyl)-ureido]-3-(1H-in...)
Affinity DataKi:  6.30nMAssay Description:Binding affinity against human NMB receptor was determinedMore data for this Ligand-Target Pair
In DepthDetails Article
TargetNeuromedin-B receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50288243(2-[3-(2,6-Diisopropyl-phenyl)-ureido]-3-(1H-indol-...)
Affinity DataKi:  7.80nMAssay Description:Binding affinity against [125 I][4Tyr]-bombesin labeled cloned human NMB receptor stably expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails Article
TargetNeuromedin-B receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50366467(CHEMBL1907865)
Affinity DataKi:  14nMAssay Description:Binding affinity against [125 I][4Tyr]-bombesin labeled cloned human NMB receptor stably expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails Article
TargetNeuromedin-B receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50288247((R) 2-[3-(2,6-Diisopropyl-phenyl)-ureido]-3-(1H-in...)
Affinity DataKi:  72nMAssay Description:Binding affinity against [125 I][4Tyr]-bombesin labeled cloned human NMB receptor stably expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails Article
TargetNeuromedin-B receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50366466(CHEMBL1907682)
Affinity DataKi:  76nMAssay Description:Binding affinity against [125 I][4Tyr]-bombesin labeled cloned human NMB receptor stably expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails Article
TargetNeuromedin-B receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50288238(2-[3-(2,6-Diisopropyl-phenyl)-ureido]-N-((S)-2,2-d...)
Affinity DataKi:  95nMAssay Description:Binding affinity against [125 I][4Tyr]-bombesin labeled cloned human NMB receptor stably expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails Article
TargetNeuromedin-B receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50288239(CHEMBL315660 | N-Cyclohexylmethyl-2-[3-(2,6-diisop...)
Affinity DataKi:  120nMAssay Description:Binding affinity against [125 I][4Tyr]-bombesin labeled cloned human NMB receptor stably expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails Article
TargetNeuromedin-B receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50288244(CHEMBL89153 | N-Cyclohexylmethyl-2-[3-(2,6-diisopr...)
Affinity DataKi:  125nMAssay Description:Binding affinity against [125 I][4Tyr]-bombesin labeled cloned human NMB receptor stably expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails Article
TargetNeuromedin-B receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50288237(CHEMBL88174 | N-Cyclohexylmethyl-2-[3-(2,6-diisopr...)
Affinity DataKi:  260nMAssay Description:Binding affinity against [125 I][4Tyr]-bombesin labeled cloned human NMB receptor stably expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails Article
TargetNeuromedin-B receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50288251(CHEMBL87090 | N-Cyclohexyl-2-[3-(2,6-diisopropyl-p...)
Affinity DataKi:  310nMAssay Description:Binding affinity against [125 I][4Tyr]-bombesin labeled cloned human NMB receptor stably expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails Article
TargetNeuromedin-B receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50288246(2-[3-(2,6-Diisopropyl-phenyl)-ureido]-3-(1H-indol-...)
Affinity DataKi:  310nMAssay Description:Binding affinity against [125 I][4Tyr]-bombesin labeled cloned human NMB receptor stably expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails Article
TargetNeuromedin-B receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50288250(2-[3-(2,6-Diisopropyl-phenyl)-ureido]-N-((R)-2,2-d...)
Affinity DataKi:  420nMAssay Description:Binding affinity against [125 I][4Tyr]-bombesin labeled cloned human NMB receptor stably expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails Article
TargetNeuromedin-B receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50288249(CHEMBL312851 | N-(1-Cyclohexyl-ethyl)-2-[3-(2,6-di...)
Affinity DataKi:  440nMAssay Description:Binding affinity against [125 I][4Tyr]-bombesin labeled cloned human NMB receptor stably expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails Article
TargetNeuromedin-B receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50288242(2-[3-(2,6-Diisopropyl-phenyl)-ureido]-3-(1H-indol-...)
Affinity DataKi:  450nMAssay Description:Binding affinity against [125 I][4Tyr]-bombesin labeled cloned human NMB receptor stably expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails Article
TargetNeuromedin-B receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50288241(CHEMBL328230 | N-Cyclohexylmethyl-2-[3-(2,6-diisop...)
Affinity DataKi:  490nMAssay Description:Binding affinity against [125 I][4Tyr]-bombesin labeled cloned human NMB receptor stably expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails Article
TargetNeuromedin-B receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50288236(2-[3-(2,6-Diisopropyl-phenyl)-ureido]-N-(2,2-dimet...)
Affinity DataKi:  630nMAssay Description:Binding affinity against [125 I][4Tyr]-bombesin labeled cloned human NMB receptor stably expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails Article
TargetNeuromedin-B receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50288253(CHEMBL328591 | N-Cyclohexylmethyl-2-[3-(2,6-diisop...)
Affinity DataKi:  760nMAssay Description:Binding affinity against [125 I][4Tyr]-bombesin labeled cloned human NMB receptor stably expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails Article
TargetGastrin-releasing peptide receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50288253(CHEMBL328591 | N-Cyclohexylmethyl-2-[3-(2,6-diisop...)
Affinity DataKi:  1.50E+3nMAssay Description:Binding affinity against [125 I][4Tyr]-bombesin labeled cloned human GRP(gastrin releasing peptide) receptors stably expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails Article
TargetNeuromedin-B receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50288245(2-[3-(2,6-Diisopropyl-phenyl)-ureido]-3-(1H-indol-...)
Affinity DataKi:  3.70E+3nMAssay Description:Binding affinity against [125 I][4Tyr]-bombesin labeled cloned human NMB receptor stably expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails Article
TargetGastrin-releasing peptide receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50288247((R) 2-[3-(2,6-Diisopropyl-phenyl)-ureido]-3-(1H-in...)
Affinity DataKi: >1.00E+4nMAssay Description:Binding affinity against [125 I][4Tyr]-bombesin labeled cloned human GRP(gastrin releasing peptide) receptors stably expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails Article
TargetGastrin-releasing peptide receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50288236(2-[3-(2,6-Diisopropyl-phenyl)-ureido]-N-(2,2-dimet...)
Affinity DataKi: >1.00E+4nMAssay Description:Binding affinity against [125 I][4Tyr]-bombesin labeled cloned human GRP(gastrin releasing peptide) receptors stably expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails Article
TargetGastrin-releasing peptide receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50288241(CHEMBL328230 | N-Cyclohexylmethyl-2-[3-(2,6-diisop...)
Affinity DataKi: >1.00E+4nMAssay Description:Binding affinity against [125 I][4Tyr]-bombesin labeled cloned human GRP(gastrin releasing peptide) receptors stably expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails Article
TargetGastrin-releasing peptide receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50288251(CHEMBL87090 | N-Cyclohexyl-2-[3-(2,6-diisopropyl-p...)
Affinity DataKi: >1.00E+4nMAssay Description:Binding affinity against [125 I][4Tyr]-bombesin labeled cloned human GRP(gastrin releasing peptide) receptors stably expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails Article
TargetGastrin-releasing peptide receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50288242(2-[3-(2,6-Diisopropyl-phenyl)-ureido]-3-(1H-indol-...)
Affinity DataKi: >1.00E+4nMAssay Description:Binding affinity against [125 I][4Tyr]-bombesin labeled cloned human GRP(gastrin releasing peptide) receptors stably expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails Article
TargetGastrin-releasing peptide receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50288250(2-[3-(2,6-Diisopropyl-phenyl)-ureido]-N-((R)-2,2-d...)
Affinity DataKi: >1.00E+4nMAssay Description:Binding affinity against [125 I][4Tyr]-bombesin labeled cloned human GRP(gastrin releasing peptide) receptors stably expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails Article
TargetGastrin-releasing peptide receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50288245(2-[3-(2,6-Diisopropyl-phenyl)-ureido]-3-(1H-indol-...)
Affinity DataKi: >1.00E+4nMAssay Description:Binding affinity against [125 I][4Tyr]-bombesin labeled cloned human GRP(gastrin releasing peptide) receptors stably expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails Article
TargetGastrin-releasing peptide receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50366467(CHEMBL1907865)
Affinity DataKi: >1.00E+4nMAssay Description:Binding affinity against [125 I][4Tyr]-bombesin labeled cloned human GRP(gastrin releasing peptide) receptors stably expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails Article
TargetGastrin-releasing peptide receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50288237(CHEMBL88174 | N-Cyclohexylmethyl-2-[3-(2,6-diisopr...)
Affinity DataKi: >1.00E+4nMAssay Description:Binding affinity against [125 I][4Tyr]-bombesin labeled cloned human GRP(gastrin releasing peptide) receptors stably expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails Article
TargetGastrin-releasing peptide receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50288246(2-[3-(2,6-Diisopropyl-phenyl)-ureido]-3-(1H-indol-...)
Affinity DataKi: >1.00E+4nMAssay Description:Binding affinity against [125 I][4Tyr]-bombesin labeled cloned human GRP(gastrin releasing peptide) receptors stably expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails Article
TargetGastrin-releasing peptide receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50288239(CHEMBL315660 | N-Cyclohexylmethyl-2-[3-(2,6-diisop...)
Affinity DataKi: >1.00E+4nMAssay Description:Binding affinity against [125 I][4Tyr]-bombesin labeled cloned human GRP(gastrin releasing peptide) receptors stably expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails Article
TargetGastrin-releasing peptide receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50288243(2-[3-(2,6-Diisopropyl-phenyl)-ureido]-3-(1H-indol-...)
Affinity DataKi: >1.00E+4nMAssay Description:Binding affinity against [125 I][4Tyr]-bombesin labeled cloned human GRP(gastrin releasing peptide) receptors stably expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails Article
TargetGastrin-releasing peptide receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50288249(CHEMBL312851 | N-(1-Cyclohexyl-ethyl)-2-[3-(2,6-di...)
Affinity DataKi: >1.00E+4nMAssay Description:Binding affinity against [125 I][4Tyr]-bombesin labeled cloned human GRP(gastrin releasing peptide) receptors stably expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails Article
TargetGastrin-releasing peptide receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50071754((S)-2-[3-(2,6-Diisopropyl-phenyl)-ureido]-3-(1H-in...)
Affinity DataKi: >1.00E+4nMAssay Description:Binding affinity against [125 I][4Tyr]-bombesin labeled cloned human GRP(gastrin releasing peptide) receptors stably expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails Article
TargetGastrin-releasing peptide receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50288238(2-[3-(2,6-Diisopropyl-phenyl)-ureido]-N-((S)-2,2-d...)
Affinity DataKi: >1.00E+4nMAssay Description:Binding affinity against [125 I][4Tyr]-bombesin labeled cloned human GRP(gastrin releasing peptide) receptors stably expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails Article
TargetGastrin-releasing peptide receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50288244(CHEMBL89153 | N-Cyclohexylmethyl-2-[3-(2,6-diisopr...)
Affinity DataKi: >1.00E+4nMAssay Description:Binding affinity against [125 I][4Tyr]-bombesin labeled cloned human GRP(gastrin releasing peptide) receptors stably expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails Article
TargetGastrin-releasing peptide receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50366466(CHEMBL1907682)
Affinity DataKi: >1.00E+4nMAssay Description:Binding affinity against [125 I][4Tyr]-bombesin labeled cloned human GRP(gastrin releasing peptide) receptors stably expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails Article
TargetNeuromedin-B receptor(RAT)
TBA

Curated by ChEMBL
LigandPNGBDBM50071754((S)-2-[3-(2,6-Diisopropyl-phenyl)-ureido]-3-(1H-in...)
Affinity DataIC50:  150nMAssay Description:Binding affinity against NMB receptor in rat olfactory bulb was determined using [125I]-[Tyr4] bombesin.More data for this Ligand-Target Pair
In DepthDetails Article