Compile Data Set for Download or QSAR
Report error Found 33 Enz. Inhib. hit(s) with all data for entry = 50004896
TargetEpidermal growth factor receptor(Human)
University of Paris

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50029741BDBM50029741(2'-Methoxymethoxy-[1,1';4',1'']terphenyl-4-carboxy...)
Affinity DataIC50: 1.00E+3nMAssay Description:In vitro inhibition of intrinsic tyrosine protein kinase activity of the Epidermal growth factor receptor using tripeptide RR-SrcMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetEpidermal growth factor receptor(Human)
University of Paris

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50029728BDBM50029728(2'-Hydroxy-[1,1';4',1'']terphenyl-4-carboxylic aci...)
Affinity DataIC50: 1.00E+3nMAssay Description:In vitro inhibition of intrinsic tyrosine protein kinase activity of the Epidermal growth factor receptor using tripeptide RR-SrcMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetEpidermal growth factor receptor(Human)
University of Paris

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50029741BDBM50029741(2'-Methoxymethoxy-[1,1';4',1'']terphenyl-4-carboxy...)
Affinity DataIC50: 1.10E+3nMAssay Description:In vitro inhibition of EGF-stimulated DNA synthesis of ER 22 cells by following the incorporation of methyl-[3H]thymidine.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetEpidermal growth factor receptor(Human)
University of Paris

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50029728BDBM50029728(2'-Hydroxy-[1,1';4',1'']terphenyl-4-carboxylic aci...)
Affinity DataIC50: 1.40E+3nMAssay Description:In vitro inhibition of EGF-stimulated DNA synthesis of ER 22 cells by following the incorporation of methyl-[3H]thymidine.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetEpidermal growth factor receptor(Human)
University of Paris

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50029740BDBM50029740(4'-tert-Butyl-2'-hydroxy-biphenyl-4-carboxylic aci...)
Affinity DataIC50: 5.00E+3nMAssay Description:In vitro inhibition of intrinsic tyrosine protein kinase activity of the Epidermal growth factor receptor using tripeptide RR-SrcMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetEpidermal growth factor receptor(Human)
University of Paris

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50029723BDBM50029723(2'-Hydroxy-[1,1';3',1'']terphenyl-4-carboxylic aci...)
Affinity DataIC50: 5.00E+3nMAssay Description:In vitro inhibition of EGF-stimulated DNA synthesis of ER 22 cells by following the incorporation of methyl-[3H]thymidine.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetEpidermal growth factor receptor(Human)
University of Paris

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50454012BDBM50454012(CHEMBL357040)
Affinity DataIC50: 5.00E+3nMAssay Description:In vitro inhibition of EGF-stimulated DNA synthesis of ER 22 cells by following the incorporation of methyl-[3H]thymidine.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetEpidermal growth factor receptor(Human)
University of Paris

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50029723BDBM50029723(2'-Hydroxy-[1,1';3',1'']terphenyl-4-carboxylic aci...)
Affinity DataIC50: 5.00E+3nMAssay Description:In vitro inhibition of intrinsic tyrosine protein kinase activity of the Epidermal growth factor receptor using tripeptide RR-SrcMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetEpidermal growth factor receptor(Human)
University of Paris

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50029722BDBM50029722(2'-Hydroxy-[1,1';3',1'']terphenyl-4-carboxylic aci...)
Affinity DataIC50: 5.00E+3nMAssay Description:In vitro inhibition of EGF-stimulated DNA synthesis of ER 22 cells by following the incorporation of methyl-[3H]thymidine.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetEpidermal growth factor receptor(Human)
University of Paris

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50454011BDBM50454011(CHEMBL359136)
Affinity DataIC50: 5.00E+3nMAssay Description:In vitro inhibition of EGF-stimulated DNA synthesis of ER 22 cells by following the incorporation of methyl-[3H]thymidine.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetEpidermal growth factor receptor(Human)
University of Paris

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50029729BDBM50029729(3'-tert-Butyl-5'-hydroxy-biphenyl-4-carboxylic aci...)
Affinity DataIC50: 5.00E+3nMAssay Description:In vitro inhibition of intrinsic tyrosine protein kinase activity of the Epidermal growth factor receptor using tripeptide RR-SrcMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetEpidermal growth factor receptor(Human)
University of Paris

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50454014BDBM50454014(CHEMBL141884)
Affinity DataIC50: 5.00E+3nMAssay Description:In vitro inhibition of EGF-stimulated DNA synthesis of ER 22 cells by following the incorporation of methyl-[3H]thymidine.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetEpidermal growth factor receptor(Human)
University of Paris

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50029727BDBM50029727(4'-tert-Butyl-2'-methoxymethoxy-biphenyl-4-carboxy...)
Affinity DataIC50: 5.00E+3nMAssay Description:In vitro inhibition of intrinsic tyrosine protein kinase activity of the Epidermal growth factor receptor using tripeptide RR-SrcMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetEpidermal growth factor receptor(Human)
University of Paris

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50454017BDBM50454017(CHEMBL142200)
Affinity DataIC50: 5.00E+3nMAssay Description:In vitro inhibition of EGF-stimulated DNA synthesis of ER 22 cells by following the incorporation of methyl-[3H]thymidine.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetEpidermal growth factor receptor(Human)
University of Paris

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50029729BDBM50029729(3'-tert-Butyl-5'-hydroxy-biphenyl-4-carboxylic aci...)
Affinity DataIC50: 5.40E+3nMAssay Description:In vitro inhibition of EGF-stimulated DNA synthesis of ER 22 cells by following the incorporation of methyl-[3H]thymidine.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetEpidermal growth factor receptor(Human)
University of Paris

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50454010BDBM50454010(CHEMBL142148)
Affinity DataIC50: 8.00E+3nMAssay Description:In vitro inhibition of EGF-stimulated DNA synthesis of ER 22 cells by following the incorporation of methyl-[3H]thymidine.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetEpidermal growth factor receptor(Human)
University of Paris

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50454013BDBM50454013(CHEMBL143899)
Affinity DataIC50: 1.00E+4nMAssay Description:In vitro inhibition of EGF-stimulated DNA synthesis of ER 22 cells by following the incorporation of methyl-[3H]thymidine.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetEpidermal growth factor receptor(Human)
University of Paris

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50029726BDBM50029726(3'-tert-Butyl-5'-hydroxy-biphenyl-4-carboxylic aci...)
Affinity DataIC50: 1.00E+4nMAssay Description:In vitro inhibition of intrinsic tyrosine protein kinase activity of the Epidermal growth factor receptor using tripeptide RR-SrcMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetEpidermal growth factor receptor(Human)
University of Paris

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50454018BDBM50454018(CHEMBL142745)
Affinity DataIC50: 1.00E+4nMAssay Description:In vitro inhibition of EGF-stimulated DNA synthesis of ER 22 cells by following the incorporation of methyl-[3H]thymidine.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetEpidermal growth factor receptor(Human)
University of Paris

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50029726BDBM50029726(3'-tert-Butyl-5'-hydroxy-biphenyl-4-carboxylic aci...)
Affinity DataIC50: 1.00E+4nMAssay Description:In vitro inhibition of EGF-stimulated DNA synthesis of ER 22 cells by following the incorporation of methyl-[3H]thymidine.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetEpidermal growth factor receptor(Human)
University of Paris

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50454015BDBM50454015(CHEMBL144921)
Affinity DataIC50: 1.00E+4nMAssay Description:In vitro inhibition of EGF-stimulated DNA synthesis of ER 22 cells by following the incorporation of methyl-[3H]thymidine.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetEpidermal growth factor receptor(Human)
University of Paris

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50029734BDBM50029734(4'-tert-Butyl-2'-methoxymethoxy-biphenyl-4-carboxy...)
Affinity DataIC50: 1.00E+4nMAssay Description:In vitro inhibition of EGF-stimulated DNA synthesis of ER 22 cells by following the incorporation of methyl-[3H]thymidine.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetEpidermal growth factor receptor(Human)
University of Paris

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50029736BDBM50029736(5-tert-Butyl-4'-hydroxymethyl-biphenyl-3-ol | CHEM...)
Affinity DataIC50: 1.00E+4nMAssay Description:In vitro inhibition of intrinsic tyrosine protein kinase activity of the Epidermal growth factor receptor using tripeptide RR-SrcMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetEpidermal growth factor receptor(Human)
University of Paris

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50029732BDBM50029732(4'-tert-Butyl-2'-hydroxy-biphenyl-4-carboxylic aci...)
Affinity DataIC50: 1.00E+4nMAssay Description:In vitro inhibition of EGF-stimulated DNA synthesis of ER 22 cells by following the incorporation of methyl-[3H]thymidine.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetEpidermal growth factor receptor(Human)
University of Paris

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50029734BDBM50029734(4'-tert-Butyl-2'-methoxymethoxy-biphenyl-4-carboxy...)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of Epidermal growth factor receptor activity against tripeptide RR-Src at 10 uMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetEpidermal growth factor receptor(Human)
University of Paris

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50454016BDBM50454016(CHEMBL142831)
Affinity DataIC50: 1.00E+4nMAssay Description:In vitro inhibition of EGF-stimulated DNA synthesis of ER 22 cells by following the incorporation of methyl-[3H]thymidine.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetEpidermal growth factor receptor(Human)
University of Paris

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50029732BDBM50029732(4'-tert-Butyl-2'-hydroxy-biphenyl-4-carboxylic aci...)
Affinity DataIC50: 1.00E+4nMAssay Description:In vitro inhibition of intrinsic tyrosine protein kinase activity of the Epidermal growth factor receptor using tripeptide RR-SrcMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetEpidermal growth factor receptor(Human)
University of Paris

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50029724BDBM50029724(2'-Hydroxy-[1,1';4',1'']terphenyl-4-carboxylic aci...)
Affinity DataIC50: 1.40E+4nMAssay Description:In vitro inhibition of intrinsic tyrosine protein kinase activity of the Epidermal growth factor receptor using tripeptide RR-SrcMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetEpidermal growth factor receptor(Human)
University of Paris

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50029737BDBM50029737(3'-tert-Butyl-5'-hydroxy-biphenyl-4-carboxylic aci...)
Affinity DataIC50: 2.00E+4nMAssay Description:In vitro inhibition of EGF-stimulated DNA synthesis of ER 22 cells by following the incorporation of methyl-[3H]thymidine.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetEpidermal growth factor receptor(Human)
University of Paris

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50029745BDBM50029745(2'-Methoxymethoxy-[1,1';4',1'']terphenyl-4-carboxy...)
Affinity DataIC50: 2.00E+4nMAssay Description:In vitro inhibition of intrinsic tyrosine protein kinase activity of the Epidermal growth factor receptor using tripeptide RR-SrcMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetEpidermal growth factor receptor(Human)
University of Paris

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50029722BDBM50029722(2'-Hydroxy-[1,1';3',1'']terphenyl-4-carboxylic aci...)
Affinity DataIC50: 2.00E+4nMAssay Description:In vitro inhibition of intrinsic tyrosine protein kinase activity of the Epidermal growth factor receptor using tripeptide RR-SrcMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetEpidermal growth factor receptor(Human)
University of Paris

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50029738BDBM50029738(4'-tert-Butyl-2'-methoxymethoxy-biphenyl-4-carboxy...)
Affinity DataIC50: 5.00E+4nMAssay Description:In vitro inhibition of intrinsic tyrosine protein kinase activity of the Epidermal growth factor receptor using tripeptide RR-SrcMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetEpidermal growth factor receptor(Human)
University of Paris

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50029737BDBM50029737(3'-tert-Butyl-5'-hydroxy-biphenyl-4-carboxylic aci...)
Affinity DataIC50: 5.00E+4nMAssay Description:In vitro inhibition of intrinsic tyrosine protein kinase activity of the Epidermal growth factor receptor using tripeptide RR-SrcMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed