Compile Data Set for Download or QSAR
Report error Found 53 Enz. Inhib. hit(s) with all data for entry = 50003403
TargetType-1 angiotensin II receptor A/B(Rat)
Hoechst Roussel Pgu Cardiovascular Agents

Curated by ChEMBL
LigandPNGBDBM50470233(CHEMBL80177)
Affinity DataIC50: 0.0800nMAssay Description:Specific binding inhibition of [125I]AII to Angiotensin II receptor, type 1 in rat liver membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2020
Entry Details Article
PubMed
TargetType-1 angiotensin II receptor A/B(Rat)
Hoechst Roussel Pgu Cardiovascular Agents

Curated by ChEMBL
LigandPNGBDBM50470229(CHEMBL76870)
Affinity DataIC50: 0.0900nMAssay Description:Specific binding inhibition of [125I]AII to Angiotensin II receptor, type 1 in rat liver membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2020
Entry Details Article
PubMed
TargetType-1 angiotensin II receptor A/B(Rat)
Hoechst Roussel Pgu Cardiovascular Agents

Curated by ChEMBL
LigandPNGBDBM50470236(CHEMBL309313)
Affinity DataIC50: 0.100nMAssay Description:Specific binding inhibition of [125I]AII to Angiotensin II receptor, type 1 in rat liver membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2020
Entry Details Article
PubMed
TargetType-1 angiotensin II receptor A/B(Rat)
Hoechst Roussel Pgu Cardiovascular Agents

Curated by ChEMBL
LigandPNGBDBM50470239(CHEMBL311312)
Affinity DataIC50: 0.100nMAssay Description:Specific binding inhibition of [125I]AII to Angiotensin II receptor, type 1 in rat liver membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2020
Entry Details Article
PubMed
TargetType-1 angiotensin II receptor A/B(Rat)
Hoechst Roussel Pgu Cardiovascular Agents

Curated by ChEMBL
LigandPNGBDBM50470235(CHEMBL308135)
Affinity DataIC50: 0.200nMAssay Description:Specific binding inhibition of [125I]AII to Angiotensin II receptor, type 1 in rat liver membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2020
Entry Details Article
PubMed
TargetType-1 angiotensin II receptor A/B(Rat)
Hoechst Roussel Pgu Cardiovascular Agents

Curated by ChEMBL
LigandPNGBDBM50213557(CHEMBL309602)
Affinity DataIC50: 0.200nMAssay Description:Specific binding inhibition of [125I]AII to Angiotensin II receptor, type 1 in rat liver membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2020
Entry Details Article
PubMed
TargetType-1 angiotensin II receptor A/B(Rat)
Hoechst Roussel Pgu Cardiovascular Agents

Curated by ChEMBL
LigandPNGBDBM50470250(CHEMBL77308)
Affinity DataIC50: 0.200nMAssay Description:Specific binding inhibition of [125I]AII to Angiotensin II receptor, type 1 in rat liver membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2020
Entry Details Article
PubMed
TargetType-1 angiotensin II receptor A/B(Rat)
Hoechst Roussel Pgu Cardiovascular Agents

Curated by ChEMBL
LigandPNGBDBM50470206(CHEMBL445365)
Affinity DataIC50: 0.200nMAssay Description:Specific binding inhibition of [125I]AII to Angiotensin II receptor, type 1 in rat liver membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2020
Entry Details Article
PubMed
TargetType-1 angiotensin II receptor A/B(Rat)
Hoechst Roussel Pgu Cardiovascular Agents

Curated by ChEMBL
LigandPNGBDBM50031491(3-(2'-Propylaminocarbonylsulfamoyl-biphenyl-4-ylme...)
Affinity DataIC50: 0.200nMAssay Description:Specific binding inhibition of [125I]AII to Angiotensin II receptor, type 1 in rat liver membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2020
Entry Details Article
PubMed
TargetType-1 angiotensin II receptor A/B(Rat)
Hoechst Roussel Pgu Cardiovascular Agents

Curated by ChEMBL
LigandPNGBDBM50470225(CHEMBL80700)
Affinity DataIC50: 0.200nMAssay Description:Specific binding inhibition of [125I]AII to Angiotensin II receptor, type 1 in rat liver membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2020
Entry Details Article
PubMed
TargetType-1 angiotensin II receptor A/B(Rat)
Hoechst Roussel Pgu Cardiovascular Agents

Curated by ChEMBL
LigandPNGBDBM50470226(CHEMBL311827)
Affinity DataIC50: 0.200nMAssay Description:Specific binding inhibition of [125I]AII to Angiotensin II receptor, type 1 in rat liver membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2020
Entry Details Article
PubMed
TargetType-1 angiotensin II receptor A/B(Rat)
Hoechst Roussel Pgu Cardiovascular Agents

Curated by ChEMBL
LigandPNGBDBM50213569(CHEMBL78866)
Affinity DataIC50: 0.200nMAssay Description:Specific binding inhibition of [125I]AII to Angiotensin II receptor, type 1 in rat liver membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2020
Entry Details Article
PubMed
TargetType-1 angiotensin II receptor A/B(Rat)
Hoechst Roussel Pgu Cardiovascular Agents

Curated by ChEMBL
LigandPNGBDBM50470223(CHEMBL312386)
Affinity DataIC50: 0.300nMAssay Description:Specific binding inhibition of [125I]AII to Angiotensin II receptor, type 1 in rat liver membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2020
Entry Details Article
PubMed
TargetType-1 angiotensin II receptor A/B(Rat)
Hoechst Roussel Pgu Cardiovascular Agents

Curated by ChEMBL
LigandPNGBDBM50470249(CHEMBL309845)
Affinity DataIC50: 0.300nMAssay Description:Specific binding inhibition of [125I]AII to Angiotensin II receptor, type 1 in rat liver membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2020
Entry Details Article
PubMed
TargetType-1 angiotensin II receptor A/B(Rat)
Hoechst Roussel Pgu Cardiovascular Agents

Curated by ChEMBL
LigandPNGBDBM50031537(5-carboxyl imidazolyl biphenyl sulfonylurea deriva...)
Affinity DataIC50: 0.300nMAssay Description:Specific binding inhibition of [125I]AII to Angiotensin II receptor, type 1 in rat liver membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2020
Entry Details Article
PubMed
TargetType-1 angiotensin II receptor A/B(Rat)
Hoechst Roussel Pgu Cardiovascular Agents

Curated by ChEMBL
LigandPNGBDBM50470227(CHEMBL76538)
Affinity DataIC50: 0.300nMAssay Description:Specific binding inhibition of [125I]AII to Angiotensin II receptor, type 1 in rat liver membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2020
Entry Details Article
PubMed
TargetType-1 angiotensin II receptor A/B(Rat)
Hoechst Roussel Pgu Cardiovascular Agents

Curated by ChEMBL
LigandPNGBDBM50470241(CHEMBL305638)
Affinity DataIC50: 0.300nMAssay Description:Specific binding inhibition of [125I]AII to Angiotensin II receptor, type 1 in rat liver membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2020
Entry Details Article
PubMed
TargetType-1 angiotensin II receptor A/B(Rat)
Hoechst Roussel Pgu Cardiovascular Agents

Curated by ChEMBL
LigandPNGBDBM50470234(CHEMBL76948)
Affinity DataIC50: 0.400nMAssay Description:Specific binding inhibition of [125I]AII to Angiotensin II receptor, type 1 in rat liver membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2020
Entry Details Article
PubMed
TargetType-1 angiotensin II receptor A/B(Rat)
Hoechst Roussel Pgu Cardiovascular Agents

Curated by ChEMBL
LigandPNGBDBM50470228(CHEMBL80971)
Affinity DataIC50: 0.400nMAssay Description:Specific binding inhibition of [125I]AII to Angiotensin II receptor, type 1 in rat liver membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2020
Entry Details Article
PubMed
TargetType-1 angiotensin II receptor A/B(Rat)
Hoechst Roussel Pgu Cardiovascular Agents

Curated by ChEMBL
LigandPNGBDBM50031530(2-Butyl-4-(methylthio)-1-[[2'-[[[(propylamino)carb...)
Affinity DataIC50: 0.480nMAssay Description:Specific binding inhibition of [125I]AII to Angiotensin II receptor, type 1 in rat liver membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2020
Entry Details Article
PubMed
TargetType-1 angiotensin II receptor A/B(Rat)
Hoechst Roussel Pgu Cardiovascular Agents

Curated by ChEMBL
LigandPNGBDBM50470243(CHEMBL306157)
Affinity DataIC50: 0.5nMAssay Description:Specific binding inhibition of [125I]AII to Angiotensin II receptor, type 1 in rat liver membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2020
Entry Details Article
PubMed
TargetType-1 angiotensin II receptor A/B(Rat)
Hoechst Roussel Pgu Cardiovascular Agents

Curated by ChEMBL
LigandPNGBDBM50470219(CHEMBL305604)
Affinity DataIC50: 0.600nMAssay Description:Specific binding inhibition of [125I]AII to Angiotensin II receptor, type 1 in rat liver membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2020
Entry Details Article
PubMed
TargetType-1 angiotensin II receptor A/B(Rat)
Hoechst Roussel Pgu Cardiovascular Agents

Curated by ChEMBL
LigandPNGBDBM50470212(CHEMBL80622)
Affinity DataIC50: 0.600nMAssay Description:Specific binding inhibition of [125I]AII to Angiotensin II receptor, type 1 in rat liver membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2020
Entry Details Article
PubMed
TargetType-1 angiotensin II receptor A/B(Rat)
Hoechst Roussel Pgu Cardiovascular Agents

Curated by ChEMBL
LigandPNGBDBM50470214(CHEMBL77360)
Affinity DataIC50: 0.800nMAssay Description:Specific binding inhibition of [125I]AII to Angiotensin II receptor, type 1 in rat liver membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2020
Entry Details Article
PubMed
TargetType-1 angiotensin II receptor A/B(Rat)
Hoechst Roussel Pgu Cardiovascular Agents

Curated by ChEMBL
LigandPNGBDBM50470230(CHEMBL76799)
Affinity DataIC50: 0.800nMAssay Description:Specific binding inhibition of [125I]AII to Angiotensin II receptor, type 1 in rat liver membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2020
Entry Details Article
PubMed
TargetType-1 angiotensin II receptor A/B(Rat)
Hoechst Roussel Pgu Cardiovascular Agents

Curated by ChEMBL
LigandPNGBDBM50470217(CHEMBL77138)
Affinity DataIC50: 0.800nMAssay Description:Specific binding inhibition of [125I]AII to Angiotensin II receptor, type 1 in rat liver membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2020
Entry Details Article
PubMed
TargetType-1 angiotensin II receptor A/B(Rat)
Hoechst Roussel Pgu Cardiovascular Agents

Curated by ChEMBL
LigandPNGBDBM50470240(CHEMBL432158)
Affinity DataIC50: 0.800nMAssay Description:Specific binding inhibition of [125I]AII to Angiotensin II receptor, type 1 in rat liver membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2020
Entry Details Article
PubMed
TargetType-1 angiotensin II receptor A/B(Rat)
Hoechst Roussel Pgu Cardiovascular Agents

Curated by ChEMBL
LigandPNGBDBM50470208(CHEMBL80900)
Affinity DataIC50: 0.900nMAssay Description:Specific binding inhibition of [125I]AII to Angiotensin II receptor, type 1 in rat liver membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2020
Entry Details Article
PubMed
TargetType-1 angiotensin II receptor A/B(Rat)
Hoechst Roussel Pgu Cardiovascular Agents

Curated by ChEMBL
LigandPNGBDBM50470224(CHEMBL311189)
Affinity DataIC50: 0.900nMAssay Description:Specific binding inhibition of [125I]AII to Angiotensin II receptor, type 1 in rat liver membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2020
Entry Details Article
PubMed
TargetType-1 angiotensin II receptor A/B(Rat)
Hoechst Roussel Pgu Cardiovascular Agents

Curated by ChEMBL
LigandPNGBDBM50470248(CHEMBL311847)
Affinity DataIC50: 0.900nMAssay Description:Specific binding inhibition of [125I]AII to Angiotensin II receptor, type 1 in rat liver membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2020
Entry Details Article
PubMed
TargetType-1 angiotensin II receptor A/B(Rat)
Hoechst Roussel Pgu Cardiovascular Agents

Curated by ChEMBL
LigandPNGBDBM50470237(CHEMBL306778)
Affinity DataIC50: 1nMAssay Description:Specific binding inhibition of [125I]AII to Angiotensin II receptor, type 1 in rat liver membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2020
Entry Details Article
PubMed
TargetType-1 angiotensin II receptor A/B(Rat)
Hoechst Roussel Pgu Cardiovascular Agents

Curated by ChEMBL
LigandPNGBDBM50470231(CHEMBL76613)
Affinity DataIC50: 1nMAssay Description:Specific binding inhibition of [125I]AII to Angiotensin II receptor, type 1 in rat liver membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2020
Entry Details Article
PubMed
TargetType-1 angiotensin II receptor A/B(Rat)
Hoechst Roussel Pgu Cardiovascular Agents

Curated by ChEMBL
LigandPNGBDBM50470246(CHEMBL306085)
Affinity DataIC50: 1nMAssay Description:Specific binding inhibition of [125I]AII to Angiotensin II receptor, type 1 in rat liver membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2020
Entry Details Article
PubMed
TargetType-1 angiotensin II receptor A/B(Rat)
Hoechst Roussel Pgu Cardiovascular Agents

Curated by ChEMBL
LigandPNGBDBM50470222(CHEMBL443069)
Affinity DataIC50: 1.10nMAssay Description:Specific binding inhibition of [125I]AII to Angiotensin II receptor, type 1 in rat liver membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2020
Entry Details Article
PubMed
TargetType-1 angiotensin II receptor A/B(Rat)
Hoechst Roussel Pgu Cardiovascular Agents

Curated by ChEMBL
LigandPNGBDBM50470238(CHEMBL80908)
Affinity DataIC50: 1.10nMAssay Description:Specific binding inhibition of [125I]AII to Angiotensin II receptor, type 1 in rat liver membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2020
Entry Details Article
PubMed
TargetType-1 angiotensin II receptor A/B(Rat)
Hoechst Roussel Pgu Cardiovascular Agents

Curated by ChEMBL
LigandPNGBDBM50470216(CHEMBL310267)
Affinity DataIC50: 1.30nMAssay Description:Specific binding inhibition of [125I]AII to Angiotensin II receptor, type 1 in rat liver membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2020
Entry Details Article
PubMed
TargetType-1 angiotensin II receptor A/B(Rat)
Hoechst Roussel Pgu Cardiovascular Agents

Curated by ChEMBL
LigandPNGBDBM50470245(CHEMBL78169)
Affinity DataIC50: 1.5nMAssay Description:Specific binding inhibition of [125I]AII to Angiotensin II receptor, type 1 in rat liver membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2020
Entry Details Article
PubMed
TargetType-1 angiotensin II receptor A/B(Rat)
Hoechst Roussel Pgu Cardiovascular Agents

Curated by ChEMBL
LigandPNGBDBM50470207(CHEMBL413491)
Affinity DataIC50: 1.70nMAssay Description:Specific binding inhibition of [125I]AII to Angiotensin II receptor, type 1 in rat liver membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2020
Entry Details Article
PubMed
TargetType-1 angiotensin II receptor A/B(Rat)
Hoechst Roussel Pgu Cardiovascular Agents

Curated by ChEMBL
LigandPNGBDBM50470242(CHEMBL80181)
Affinity DataIC50: 1.80nMAssay Description:Specific binding inhibition of [125I]AII to Angiotensin II receptor, type 1 in rat liver membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2020
Entry Details Article
PubMed
TargetType-1 angiotensin II receptor A/B(Rat)
Hoechst Roussel Pgu Cardiovascular Agents

Curated by ChEMBL
LigandPNGBDBM50213556(CHEMBL310610)
Affinity DataIC50: 1.90nMAssay Description:Specific binding inhibition of [125I]AII to Angiotensin II receptor, type 1 in rat liver membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2020
Entry Details Article
PubMed
TargetType-1 angiotensin II receptor A/B(Rat)
Hoechst Roussel Pgu Cardiovascular Agents

Curated by ChEMBL
LigandPNGBDBM50470252(CHEMBL441990)
Affinity DataIC50: 2.10nMAssay Description:Specific binding inhibition of [125I]AII to Angiotensin II receptor, type 1 in rat liver membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2020
Entry Details Article
PubMed
TargetType-1 angiotensin II receptor A/B(Rat)
Hoechst Roussel Pgu Cardiovascular Agents

Curated by ChEMBL
LigandPNGBDBM50470221(CHEMBL78445)
Affinity DataIC50: 2.10nMAssay Description:Specific binding inhibition of [125I]AII to Angiotensin II receptor, type 1 in rat liver membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2020
Entry Details Article
PubMed
TargetType-1 angiotensin II receptor A/B(Rat)
Hoechst Roussel Pgu Cardiovascular Agents

Curated by ChEMBL
LigandPNGBDBM50470213(CHEMBL76760)
Affinity DataIC50: 2.60nMAssay Description:Specific binding inhibition of [125I]AII to Angiotensin II receptor, type 1 in rat liver membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2020
Entry Details Article
PubMed
TargetType-1 angiotensin II receptor A/B(Rat)
Hoechst Roussel Pgu Cardiovascular Agents

Curated by ChEMBL
LigandPNGBDBM50470247(CHEMBL306180)
Affinity DataIC50: 3.10nMAssay Description:Specific binding inhibition of [125I]AII to Angiotensin II receptor, type 1 in rat liver membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2020
Entry Details Article
PubMed
TargetType-1 angiotensin II receptor A/B(Rat)
Hoechst Roussel Pgu Cardiovascular Agents

Curated by ChEMBL
LigandPNGBDBM50470211(CHEMBL80212)
Affinity DataIC50: 3.20nMAssay Description:Specific binding inhibition of [125I]AII to Angiotensin II receptor, type 1 in rat liver membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2020
Entry Details Article
PubMed
TargetType-1 angiotensin II receptor A/B(Rat)
Hoechst Roussel Pgu Cardiovascular Agents

Curated by ChEMBL
LigandPNGBDBM50470215(CHEMBL79106)
Affinity DataIC50: 4.5nMAssay Description:Specific binding inhibition of [125I]AII to Angiotensin II receptor, type 1 in rat liver membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2020
Entry Details Article
PubMed
TargetType-1 angiotensin II receptor A/B(Rat)
Hoechst Roussel Pgu Cardiovascular Agents

Curated by ChEMBL
LigandPNGBDBM50470244(CHEMBL80901)
Affinity DataIC50: 4.70nMAssay Description:Specific binding inhibition of [125I]AII to Angiotensin II receptor, type 1 in rat liver membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2020
Entry Details Article
PubMed
TargetType-1 angiotensin II receptor A/B(Rat)
Hoechst Roussel Pgu Cardiovascular Agents

Curated by ChEMBL
LigandPNGBDBM50470209(CHEMBL75921)
Affinity DataIC50: 7.70nMAssay Description:Specific binding inhibition of [125I]AII to Angiotensin II receptor, type 1 in rat liver membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2020
Entry Details Article
PubMed
TargetType-1 angiotensin II receptor A/B(Rat)
Hoechst Roussel Pgu Cardiovascular Agents

Curated by ChEMBL
LigandPNGBDBM50470218(CHEMBL76675)
Affinity DataIC50: 15nMAssay Description:Specific binding inhibition of [125I]AII to Angiotensin II receptor, type 1 in rat liver membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2020
Entry Details Article
PubMed
TargetType-1 angiotensin II receptor A/B(Rat)
Hoechst Roussel Pgu Cardiovascular Agents

Curated by ChEMBL
LigandPNGBDBM50470210(CHEMBL79108)
Affinity DataIC50: 36nMAssay Description:Specific binding inhibition of [125I]AII to Angiotensin II receptor, type 1 in rat liver membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2020
Entry Details Article
PubMed
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