Compile Data Set for Download or QSAR
Report error Found 13 Enz. Inhib. hit(s) with all data for entry = 50036392
TargetNeurotensin receptor type 1(Rat)
Instituto De Qu£Mica M£Dica (Csic)

Curated by ChEMBL
LigandPNGBDBM50369070(CHEMBL1793839)
Affinity DataIC50: 5nMAssay Description:IC50 was measured as binding to rat cortex membranes using [3H]- NT(neurotensin) as tracerMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/31/2012
Entry Details Article
PubMed
TargetNeurotensin receptor type 1(Rat)
Instituto De Qu£Mica M£Dica (Csic)

Curated by ChEMBL
LigandPNGBDBM50033671((S)-2-{(R)-2-[2-({1-[2-(2-Amino-5-guanidino-pentan...)
Affinity DataIC50: 8nMAssay Description:IC50 was measured as binding to rat cortex membranes using [3H]- NT(neurotensin) as tracerMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/31/2012
Entry Details Article
PubMed
TargetNeurotensin receptor type 1(Rat)
Instituto De Qu£Mica M£Dica (Csic)

Curated by ChEMBL
LigandPNGBDBM50240845(2-{(S)-2-[2-({(S)-1-[(S)-2-((S)-2-Amino-5-guanidin...)
Affinity DataIC50: 10nMAssay Description:IC50 was measured as binding to rat cortex membranes using [3H]- NT(neurotensin) as tracerMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/31/2012
Entry Details Article
PubMed
TargetNeurotensin receptor type 1(Rat)
Instituto De Qu£Mica M£Dica (Csic)

Curated by ChEMBL
LigandPNGBDBM50033670((S)-2-[(R)-5-({1-[2-(2-Amino-5-guanidino-pentanoyl...)
Affinity DataIC50: 15nMAssay Description:IC50 was measured as binding to rat cortex membranes using [3H]- NT(neurotensin) as tracerMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/31/2012
Entry Details Article
PubMed
TargetNeurotensin receptor type 1(Rat)
Instituto De Qu£Mica M£Dica (Csic)

Curated by ChEMBL
LigandPNGBDBM50033677((S,R)5-[1-{1-[2-[1-amino-4-amino(imino)methylamino...)
Affinity DataIC50: 120nMAssay Description:IC50 was measured as binding to rat cortex membranes using [3H]- NT(neurotensin) as tracerMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/31/2012
Entry Details Article
PubMed
TargetNeurotensin receptor type 1(Rat)
Instituto De Qu£Mica M£Dica (Csic)

Curated by ChEMBL
LigandPNGBDBM50033667((S,S)2-{1-[2-{1-[2-[1-amino-4-amino(imino)methylam...)
Affinity DataIC50: 180nMAssay Description:IC50 was measured as binding to rat cortex membranes using [3H]- NT (neurotensin) as tracerMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/31/2012
Entry Details Article
PubMed
TargetNeurotensin receptor type 1(Rat)
Instituto De Qu£Mica M£Dica (Csic)

Curated by ChEMBL
LigandPNGBDBM50033668((R,S)5-[1-{1-[2-[1-amino-4-amino(imino)methylamino...)
Affinity DataIC50: 900nMAssay Description:IC50 was measured as binding to rat cortex membranes using [3H]- NT(neurotensin) as tracerMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/31/2012
Entry Details Article
PubMed
TargetNeurotensin receptor type 1(Rat)
Instituto De Qu£Mica M£Dica (Csic)

Curated by ChEMBL
LigandPNGBDBM50033678((S,S)5-[1-{1-[2-[1-amino-4-amino(imino)methylamino...)
Affinity DataIC50: 1.20E+3nMAssay Description:IC50 was measured as binding to rat cortex membranes using [3H]- NT(neurotensin) as tracerMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/31/2012
Entry Details Article
PubMed
TargetNeurotensin receptor type 1(Rat)
Instituto De Qu£Mica M£Dica (Csic)

Curated by ChEMBL
LigandPNGBDBM50033675((S)-2-[(S)-5-({1-[2-(2-Amino-5-guanidino-pentanoyl...)
Affinity DataIC50: 1.20E+3nMAssay Description:IC50 was measured as binding to rat cortex membranes using [3H]- NT(neurotensin) as tracerMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/31/2012
Entry Details Article
PubMed
TargetNeurotensin receptor type 1(Rat)
Instituto De Qu£Mica M£Dica (Csic)

Curated by ChEMBL
LigandPNGBDBM50033679((R,R)5-[1-{1-[2-[1-amino-4-amino(imino)methylamino...)
Affinity DataIC50: 1.50E+3nMAssay Description:IC50 was measured as binding to rat cortex membranes using [3H]- NT(neurotensin) as tracerMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/31/2012
Entry Details Article
PubMed
TargetNeurotensin receptor type 1(Rat)
Instituto De Qu£Mica M£Dica (Csic)

Curated by ChEMBL
LigandPNGBDBM50369071(CHEMBL1793838)
Affinity DataIC50: 6.31E+3nMAssay Description:IC50 was measured as binding to rat cortex membranes using [3H]- NT(neurotensin) as tracerMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/31/2012
Entry Details Article
PubMed
TargetNeurotensin receptor type 1(Rat)
Instituto De Qu£Mica M£Dica (Csic)

Curated by ChEMBL
LigandPNGBDBM50369072(CHEMBL1793837)
Affinity DataIC50: 8.00E+3nMAssay Description:IC50 was measured as binding to rat cortex membranes using [3H]- NT(neurotensin) as tracerMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/31/2012
Entry Details Article
PubMed
TargetNeurotensin receptor type 1(Rat)
Instituto De Qu£Mica M£Dica (Csic)

Curated by ChEMBL
LigandPNGBDBM50033674((S,S)2-{1-[2-{1-[2-[1-amino-4-amino(imino)methylam...)
Affinity DataIC50: 1.00E+4nMAssay Description:IC50 was measured as binding to rat cortex membranes using [3H]- NT (neurotensin) as tracerMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/31/2012
Entry Details Article
PubMed