Compile Data Set for Download or QSAR
Report error Found 84 Enz. Inhib. hit(s) with all data for entry = 50005177
Target5-hydroxytryptamine receptor 1A(Rat)
Università

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50033839BDBM50033839(1-(2-Methoxy-phenyl)-4-[3-(5-methoxy-1,2,3,4-tetra...)
Affinity DataIC50: 0.320nMAssay Description:In vitro binding affinity measured on serotonin 5-hydroxytryptamine 1A receptor using [3H]8-OH-DPAT as radioligand.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Rat)
Università

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50033843BDBM50033843(1-[3-(5-Methoxy-3,4-dihydro-2H-naphthalen-1-yliden...)
Affinity DataIC50: 0.350nMAssay Description:In vitro binding affinity measured on serotonin 5-hydroxytryptamine 1A receptor using [3H]8-OH-DPAT as radioligand.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Rat)
Università

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50033857BDBM50033857(1-[3-(5-Methoxy-1,2,3,4-tetrahydro-naphthalen-1-yl...)
Affinity DataIC50: 0.360nMAssay Description:In vitro binding affinity measured on serotonin 5-hydroxytryptamine 1A receptor using [3H]8-OH-DPAT as radioligand.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Rat)
Università

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50033851BDBM50033851(1-(2-Methoxy-phenyl)-4-[3-(1,2,3,4-tetrahydro-naph...)
Affinity DataIC50: 0.390nMAssay Description:In vitro binding affinity measured on serotonin 5-hydroxytryptamine 1A receptor using [3H]8-OH-DPAT as radioligand.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Rat)
Università

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50008735BDBM50008735(CHEMBL8514 | BUTACLAMOL,d- | (+)-3-(tert-butyl)-(3...)
Affinity DataIC50: 0.5nMAssay Description:In vitro binding affinity measured on dopamine receptor D2 using [3H]spiroperidol as radioligand.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Rat)
Università

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50033833BDBM50033833(1-{3-[5-Methoxy-3,4-dihydro-2H-naphthalen-(1E)-yli...)
Affinity DataIC50: 0.520nMAssay Description:In vitro binding affinity measured on serotonin 5-hydroxytryptamine 1A receptor using [3H]8-OH-DPAT as radioligand.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Rat)
Università

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50033852BDBM50033852(1-[3-(5-Methoxy-1,2,3,4-tetrahydro-naphthalen-1-yl...)
Affinity DataIC50: 0.580nMAssay Description:In vitro binding affinity measured on serotonin 5-hydroxytryptamine 1A receptor using [3H]8-OH-DPAT as radioligand.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Rat)
Università

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50033836BDBM50033836(1-(2-Methoxy-phenyl)-4-[2-(5-methoxy-1,2,3,4-tetra...)
Affinity DataIC50: 1.08nMAssay Description:In vitro binding affinity measured on serotonin 5-hydroxytryptamine 1A receptor using [3H]8-OH-DPAT as radioligand.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Rat)
Università

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 21393BDBM21393(cid_1220 | CHEMBL56 | 7-(dipropylamino)-5,6,7,8-te...)
Affinity DataIC50: 1.10nMAssay Description:In vitro binding affinity measured on serotonin 5-hydroxytryptamine 1A receptor using [3H]8-OH-DPAT as radioligand.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Rat)
Università

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50033859BDBM50033859(1-(2-Methoxy-phenyl)-4-[3-(4,5,6,7-tetrahydro-benz...)
Affinity DataIC50: 1.13nMAssay Description:In vitro binding affinity measured on serotonin 5-hydroxytryptamine 1A receptor using [3H]8-OH-DPAT as radioligand.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Rat)
Università

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50033853BDBM50033853(1-[3-(5-Methoxy-3,4-dihydro-naphthalen-1-yl)-propy...)
Affinity DataIC50: 1.40nMAssay Description:In vitro binding affinity measured on serotonin 5-hydroxytryptamine 1A receptor using [3H]8-OH-DPAT as radioligand.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Rat)
Università

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50033858BDBM50033858(1-(2-Methoxy-phenyl)-4-[3-(7-methoxy-1,2,3,4-tetra...)
Affinity DataIC50: 1.5nMAssay Description:In vitro binding affinity measured on serotonin 5-hydroxytryptamine 1A receptor using [3H]8-OH-DPAT as radioligand.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Rat)
Università

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50033831BDBM50033831(1-[4-(7-Methoxy-3,4-dihydro-naphthalen-1-yl)-butyl...)
Affinity DataIC50: 1.53nMAssay Description:In vitro binding affinity measured on serotonin 5-hydroxytryptamine 1A receptor using [3H]8-OH-DPAT as radioligand.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Rat)
Università

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50033835BDBM50033835(1-(2-Methoxy-phenyl)-4-[4-(5-methoxy-1,2,3,4-tetra...)
Affinity DataIC50: 1.73nMAssay Description:In vitro binding affinity measured on serotonin 5-hydroxytryptamine 1A receptor using [3H]8-OH-DPAT as radioligand.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Rat)
Università

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50033844BDBM50033844(1-{3-[3,4-Dihydro-2H-naphthalen-(1E)-ylidene]-prop...)
Affinity DataIC50: 1.84nMAssay Description:In vitro binding affinity measured on serotonin 5-hydroxytryptamine 1A receptor using [3H]8-OH-DPAT as radioligand.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Rat)
Università

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50033834BDBM50033834(1-[3-(7-Methoxy-3,4-dihydro-naphthalen-1-yl)-propy...)
Affinity DataIC50: 2nMAssay Description:In vitro binding affinity measured on serotonin 5-hydroxytryptamine 1A receptor using [3H]8-OH-DPAT as radioligand.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Rat)
Università

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50033841BDBM50033841(1-[3-(7-Methoxy-1,2,3,4-tetrahydro-naphthalen-1-yl...)
Affinity DataIC50: 3.38nMAssay Description:In vitro binding affinity measured on serotonin 5-hydroxytryptamine 1A receptor using [3H]8-OH-DPAT as radioligand.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSigma non-opioid intracellular receptor 1(Human)
Università

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 21398BDBM21398(4-[4-(4-Chloro-phenyl)-4-hydroxy-piperidin-1-yl]-1...)
Affinity DataIC50: 5.64nMAssay Description:In vitro binding affinity measured on sigma opioid receptor using [3H]DTG as radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMedPDB3D3D Structure (crystal)
Target5-hydroxytryptamine receptor 1A(Rat)
Università

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50033849BDBM50033849(1-(2-Methoxy-phenyl)-4-[2-(7-methoxy-1,2,3,4-tetra...)
Affinity DataIC50: 5.94nMAssay Description:In vitro binding affinity measured on serotonin 5-hydroxytryptamine 1A receptor using [3H]8-OH-DPAT as radioligand.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Rat)
Università

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50033847BDBM50033847({2-[4-(2-Methoxy-phenyl)-piperazin-1-yl]-ethyl}-(5...)
Affinity DataIC50: 7.01nMAssay Description:In vitro binding affinity measured on serotonin 5-hydroxytryptamine 1A receptor using [3H]8-OH-DPAT as radioligand.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Rat)
Università

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50033836BDBM50033836(1-(2-Methoxy-phenyl)-4-[2-(5-methoxy-1,2,3,4-tetra...)
Affinity DataIC50: 7.83nMAssay Description:In vitro binding affinity measured on dopamine receptor D2 using [3H]spiroperidol as radioligand.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Rat)
Università

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50033838BDBM50033838(1-[3-(5-Methoxy-3,4-dihydro-naphthalen-1-yl)-propy...)
Affinity DataIC50: 8.80nMAssay Description:In vitro binding affinity measured on serotonin 5-hydroxytryptamine 1A receptor using [3H]8-OH-DPAT as radioligand.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Rat)
Università

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50033842BDBM50033842(1-(2-Methoxy-phenyl)-4-[4-(7-methoxy-1,2,3,4-tetra...)
Affinity DataIC50: 8.83nMAssay Description:In vitro binding affinity measured on serotonin 5-hydroxytryptamine 1A receptor using [3H]8-OH-DPAT as radioligand.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Rat)
Università

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50033854BDBM50033854(1-[3-(7-Methoxy-1,2,3,4-tetrahydro-naphthalen-1-yl...)
Affinity DataIC50: 9.24nMAssay Description:In vitro binding affinity measured on serotonin 5-hydroxytryptamine 1A receptor using [3H]8-OH-DPAT as radioligand.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSigma non-opioid intracellular receptor 1(Human)
Università

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50033859BDBM50033859(1-(2-Methoxy-phenyl)-4-[3-(4,5,6,7-tetrahydro-benz...)
Affinity DataIC50: 9.70nMAssay Description:In vitro binding affinity measured on sigma opioid receptor using [3H]DTG as radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Rat)
Università

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50033831BDBM50033831(1-[4-(7-Methoxy-3,4-dihydro-naphthalen-1-yl)-butyl...)
Affinity DataIC50: 10.6nMAssay Description:In vitro binding affinity measured on dopamine receptor D2 using [3H]spiroperidol as radioligand.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Rat)
Università

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50033833BDBM50033833(1-{3-[5-Methoxy-3,4-dihydro-2H-naphthalen-(1E)-yli...)
Affinity DataIC50: 11.3nMAssay Description:In vitro binding affinity measured on dopamine receptor D2 using [3H]spiroperidol as radioligand.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Rat)
Università

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50033844BDBM50033844(1-{3-[3,4-Dihydro-2H-naphthalen-(1E)-ylidene]-prop...)
Affinity DataIC50: 12.7nMAssay Description:In vitro binding affinity measured on dopamine receptor D2 using [3H]spiroperidol as radioligand.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Rat)
Università

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50001859BDBM50001859(BUSPAR | CHEMBL49 | 8-[4-(4-Pyrimidin-2-yl-piperaz...)
Affinity DataIC50: 12.8nMAssay Description:In vitro binding affinity measured on serotonin 5-hydroxytryptamine 1A receptor using [3H]8-OH-DPAT as radioligand.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMedPDB3D3D Structure (crystal)
Target5-hydroxytryptamine receptor 1A(Rat)
Università

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50033848BDBM50033848(1-[4-(5-Methoxy-3,4-dihydro-naphthalen-1-yl)-butyl...)
Affinity DataIC50: 13nMAssay Description:In vitro binding affinity measured on serotonin 5-hydroxytryptamine 1A receptor using [3H]8-OH-DPAT as radioligand.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Rat)
Università

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50033835BDBM50033835(1-(2-Methoxy-phenyl)-4-[4-(5-methoxy-1,2,3,4-tetra...)
Affinity DataIC50: 15.4nMAssay Description:In vitro binding affinity measured on dopamine receptor D2 using [3H]spiroperidol as radioligand.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Rat)
Università

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50033838BDBM50033838(1-[3-(5-Methoxy-3,4-dihydro-naphthalen-1-yl)-propy...)
Affinity DataIC50: 17.4nMAssay Description:In vitro binding affinity measured on dopamine receptor D2 using [3H]spiroperidol as radioligand.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Rat)
Università

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50033850BDBM50033850(1-[3-(5-Methoxy-3,4-dihydro-naphthalen-1-yl)-propy...)
Affinity DataIC50: 18.3nMAssay Description:In vitro binding affinity measured on serotonin 5-hydroxytryptamine 1A receptor using [3H]8-OH-DPAT as radioligand.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Rat)
Università

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50033839BDBM50033839(1-(2-Methoxy-phenyl)-4-[3-(5-methoxy-1,2,3,4-tetra...)
Affinity DataIC50: 20nMAssay Description:In vitro binding affinity measured on dopamine receptor D2 using [3H]spiroperidol as radioligand.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Rat)
Università

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50033859BDBM50033859(1-(2-Methoxy-phenyl)-4-[3-(4,5,6,7-tetrahydro-benz...)
Affinity DataIC50: 24.1nMAssay Description:In vitro binding affinity measured on dopamine receptor D2 using [3H]spiroperidol as radioligand.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Rat)
Università

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50033851BDBM50033851(1-(2-Methoxy-phenyl)-4-[3-(1,2,3,4-tetrahydro-naph...)
Affinity DataIC50: 24.7nMAssay Description:In vitro binding affinity measured on dopamine receptor D2 using [3H]spiroperidol as radioligand.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Rat)
Università

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50033854BDBM50033854(1-[3-(7-Methoxy-1,2,3,4-tetrahydro-naphthalen-1-yl...)
Affinity DataIC50: 28nMAssay Description:In vitro binding affinity measured on dopamine receptor D2 using [3H]spiroperidol as radioligand.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSigma non-opioid intracellular receptor 1(Human)
Università

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50033838BDBM50033838(1-[3-(5-Methoxy-3,4-dihydro-naphthalen-1-yl)-propy...)
Affinity DataIC50: 33nMAssay Description:In vitro binding affinity measured on sigma opioid receptor using [3H]DTG as radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Rat)
Università

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50033846BDBM50033846({2-[4-(2-Methoxy-phenyl)-piperazin-1-yl]-ethyl}-(7...)
Affinity DataIC50: 40.3nMAssay Description:In vitro binding affinity measured on serotonin 5-hydroxytryptamine 1A receptor using [3H]8-OH-DPAT as radioligand.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Rat)
Università

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50033849BDBM50033849(1-(2-Methoxy-phenyl)-4-[2-(7-methoxy-1,2,3,4-tetra...)
Affinity DataIC50: 50.2nMAssay Description:In vitro binding affinity measured on dopamine receptor D2 using [3H]spiroperidol as radioligand.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Rat)
Università

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50033842BDBM50033842(1-(2-Methoxy-phenyl)-4-[4-(7-methoxy-1,2,3,4-tetra...)
Affinity DataIC50: 50.9nMAssay Description:In vitro binding affinity measured on dopamine receptor D2 using [3H]spiroperidol as radioligand.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Rat)
Università

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50033858BDBM50033858(1-(2-Methoxy-phenyl)-4-[3-(7-methoxy-1,2,3,4-tetra...)
Affinity DataIC50: 51.5nMAssay Description:In vitro binding affinity measured on dopamine receptor D2 using [3H]spiroperidol as radioligand.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSigma non-opioid intracellular receptor 1(Human)
Università

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50033853BDBM50033853(1-[3-(5-Methoxy-3,4-dihydro-naphthalen-1-yl)-propy...)
Affinity DataIC50: 52nMAssay Description:In vitro binding affinity measured on sigma opioid receptor using [3H]DTG as radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSigma non-opioid intracellular receptor 1(Human)
Università

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50033833BDBM50033833(1-{3-[5-Methoxy-3,4-dihydro-2H-naphthalen-(1E)-yli...)
Affinity DataIC50: 52.2nMAssay Description:In vitro binding affinity measured on sigma opioid receptor using [3H]DTG as radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSigma non-opioid intracellular receptor 1(Human)
Università

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50033831BDBM50033831(1-[4-(7-Methoxy-3,4-dihydro-naphthalen-1-yl)-butyl...)
Affinity DataIC50: 53.5nMAssay Description:In vitro binding affinity measured on sigma opioid receptor using [3H]DTG as radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSigma non-opioid intracellular receptor 1(Human)
Università

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50033850BDBM50033850(1-[3-(5-Methoxy-3,4-dihydro-naphthalen-1-yl)-propy...)
Affinity DataIC50: 54.4nMAssay Description:In vitro binding affinity measured on sigma opioid receptor using [3H]DTG as radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSigma non-opioid intracellular receptor 1(Human)
Università

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50033844BDBM50033844(1-{3-[3,4-Dihydro-2H-naphthalen-(1E)-ylidene]-prop...)
Affinity DataIC50: 55nMAssay Description:In vitro binding affinity measured on sigma opioid receptor using [3H]DTG as radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Rat)
Università

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50033837BDBM50033837(1-[3-(5-Methoxy-3,4-dihydro-naphthalen-1-yl)-propy...)
Affinity DataIC50: 55.9nMAssay Description:In vitro binding affinity measured on serotonin 5-hydroxytryptamine 1A receptor using [3H]8-OH-DPAT as radioligand.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSigma non-opioid intracellular receptor 1(Human)
Università

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50033839BDBM50033839(1-(2-Methoxy-phenyl)-4-[3-(5-methoxy-1,2,3,4-tetra...)
Affinity DataIC50: 59.9nMAssay Description:In vitro binding affinity measured on sigma opioid receptor using [3H]DTG as radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Rat)
Università

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50033856BDBM50033856(1-[3-(7-Methoxy-3,4-dihydro-naphthalen-1-yl)-propy...)
Affinity DataIC50: 63.6nMAssay Description:In vitro binding affinity measured on serotonin 5-hydroxytryptamine 1A receptor using [3H]8-OH-DPAT as radioligand.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
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