Compile Data Set for Download or QSAR
Report error Found 32 Enz. Inhib. hit(s) with all data for entry = 50003423 Sort by
TargetMelatonin receptor type 1C(Chicken)
University College London

Curated by ChEMBL
LigandPNGBDBM50470712(CHEMBL417988)
Affinity DataKi:  0.0190nMAssay Description:Binding affinity in chicken brain membranes by using [2-125I]melatonin in a competition radioligand binding assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetMelatonin receptor type 1C(Chicken)
University College London

Curated by ChEMBL
LigandPNGBDBM50470694(CHEMBL14483)
Affinity DataKi:  0.0466nMAssay Description:Binding affinity in chicken brain membranes by using [2-125I]melatonin in a competition radioligand binding assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetMelatonin receptor type 1C(Chicken)
University College London

Curated by ChEMBL
LigandPNGBDBM50470711(CHEMBL14403)
Affinity DataKi:  0.0558nMAssay Description:Binding affinity in chicken brain membranes by using [2-125I]melatonin in a competition radioligand binding assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetMelatonin receptor type 1C(Chicken)
University College London

Curated by ChEMBL
LigandPNGBDBM50034110(Melatonin,2-Phenyl | CHEMBL15060 | N-[2-(5-Methoxy...)
Affinity DataKi:  0.0596nMAssay Description:Binding affinity in chicken brain membranes by using [2-125I]melatonin in a competition radioligand binding assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetMelatonin receptor type 1C(Chicken)
University College London

Curated by ChEMBL
LigandPNGBDBM50469784(CHEMBL14975)
Affinity DataKi:  0.305nMAssay Description:Binding affinity in chicken brain membranes by using [2-125I]melatonin in a competition radioligand binding assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetMelatonin receptor type 1C(Chicken)
University College London

Curated by ChEMBL
LigandPNGBDBM9019(CHEMBL45 | N-[2-(5-methoxy-1H-indol-3-yl)ethyl]ace...)
Affinity DataKi:  0.590nMAssay Description:Binding affinity in chicken brain membranes by using [2-125I]melatonin in a competition radioligand binding assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetMelatonin receptor type 1C(Chicken)
University College London

Curated by ChEMBL
LigandPNGBDBM50470708(CHEMBL14552)
Affinity DataKi:  2.70nMAssay Description:Binding affinity in chicken brain membranes by using [2-125I]melatonin in a competition radioligand binding assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetMelatonin receptor type 1C(Chicken)
University College London

Curated by ChEMBL
LigandPNGBDBM50470707(CHEMBL15048)
Affinity DataKi:  5.90nMAssay Description:Binding affinity in chicken brain membranes by using [2-125I]melatonin in a competition radioligand binding assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetMelatonin receptor type 1C(Chicken)
University College London

Curated by ChEMBL
LigandPNGBDBM50470704(CHEMBL14139)
Affinity DataKi:  33nMAssay Description:Binding affinity in chicken brain membranes by using [2-125I]melatonin in a competition radioligand binding assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetMelatonin receptor type 1C(Chicken)
University College London

Curated by ChEMBL
LigandPNGBDBM50212915(CHEMBL14559)
Affinity DataKi:  55nMAssay Description:Binding affinity in chicken brain membranes by using [2-125I]melatonin in a competition radioligand binding assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetMelatonin receptor type 1C(Chicken)
University College London

Curated by ChEMBL
LigandPNGBDBM50470695(CHEMBL14635)
Affinity DataKi:  63nMAssay Description:Binding affinity in chicken brain membranes by using [2-125I]melatonin in a competition radioligand binding assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetMelatonin receptor type 1C(Chicken)
University College London

Curated by ChEMBL
LigandPNGBDBM50212908(CHEMBL15013)
Affinity DataKi:  70nMAssay Description:Binding affinity in chicken brain membranes by using [2-125I]melatonin in a competition radioligand binding assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetMelatonin receptor type 1C(Chicken)
University College London

Curated by ChEMBL
LigandPNGBDBM50212913(CHEMBL15318)
Affinity DataKi:  100nMAssay Description:Binding affinity in chicken brain membranes by using [2-125I]melatonin in a competition radioligand binding assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetMelatonin receptor type 1C(Chicken)
University College London

Curated by ChEMBL
LigandPNGBDBM50212905(CHEMBL15147)
Affinity DataKi:  112nMAssay Description:Binding affinity in chicken brain membranes by using [2-125I]melatonin in a competition radioligand binding assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetMelatonin receptor type 1C(Chicken)
University College London

Curated by ChEMBL
LigandPNGBDBM50212921(CHEMBL278183)
Affinity DataKi:  148nMAssay Description:Binding affinity in chicken brain membranes by using [2-125I]melatonin in a competition radioligand binding assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetMelatonin receptor type 1C(Chicken)
University College London

Curated by ChEMBL
LigandPNGBDBM50470699(CHEMBL279864)
Affinity DataKi:  154nMAssay Description:Binding affinity in chicken brain membranes by using [2-125I]melatonin in a competition radioligand binding assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetMelatonin receptor type 1C(Chicken)
University College London

Curated by ChEMBL
LigandPNGBDBM50212907(CHEMBL274045)
Affinity DataKi:  213nMAssay Description:Binding affinity in chicken brain membranes by using [2-125I]melatonin in a competition radioligand binding assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetMelatonin receptor type 1C(Chicken)
University College London

Curated by ChEMBL
LigandPNGBDBM50470703(CHEMBL275616)
Affinity DataKi:  216nMAssay Description:Binding affinity in chicken brain membranes by using [2-125I]melatonin in a competition radioligand binding assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetMelatonin receptor type 1C(Chicken)
University College London

Curated by ChEMBL
LigandPNGBDBM50470698(CHEMBL278671)
Affinity DataKi:  222nMAssay Description:Binding affinity in chicken brain membranes by using [2-125I]melatonin in a competition radioligand binding assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetMelatonin receptor type 1C(Chicken)
University College London

Curated by ChEMBL
LigandPNGBDBM50470710(CHEMBL15271)
Affinity DataKi:  263nMAssay Description:Binding affinity in chicken brain membranes by using [2-125I]melatonin in a competition radioligand binding assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetMelatonin receptor type 1C(Chicken)
University College London

Curated by ChEMBL
LigandPNGBDBM50470702(CHEMBL279188)
Affinity DataKi:  350nMAssay Description:Binding affinity in chicken brain membranes by using [2-125I]melatonin in a competition radioligand binding assay.More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetMelatonin receptor type 1C(Chicken)
University College London

Curated by ChEMBL
LigandPNGBDBM50470705(CHEMBL280493)
Affinity DataKi:  410nMAssay Description:Binding affinity in chicken brain membranes by using [2-125I]melatonin in a competition radioligand binding assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetMelatonin receptor type 1C(Chicken)
University College London

Curated by ChEMBL
LigandPNGBDBM50034101(N-CBCPT | Compound 6 | CHEMBL14701 | Cyclobutaneca...)
Affinity DataKi:  565nMAssay Description:Binding affinity in chicken brain membranes by using [2-125I]melatonin in a competition radioligand binding assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetMelatonin receptor type 1C(Chicken)
University College London

Curated by ChEMBL
LigandPNGBDBM50470706(CHEMBL276511)
Affinity DataKi:  633nMAssay Description:Binding affinity in chicken brain membranes by using [2-125I]melatonin in a competition radioligand binding assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetMelatonin receptor type 1C(Chicken)
University College London

Curated by ChEMBL
LigandPNGBDBM50470692(CHEMBL14372)
Affinity DataKi:  659nMAssay Description:Binding affinity in chicken brain membranes by using [2-125I]melatonin in a competition radioligand binding assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetMelatonin receptor type 1C(Chicken)
University College London

Curated by ChEMBL
LigandPNGBDBM50470700(CHEMBL14793)
Affinity DataKi:  726nMAssay Description:Binding affinity in chicken brain membranes by using [2-125I]melatonin in a competition radioligand binding assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetMelatonin receptor type 1C(Chicken)
University College London

Curated by ChEMBL
LigandPNGBDBM50470701(CHEMBL14800)
Affinity DataKi:  1.10E+3nMAssay Description:Binding affinity in chicken brain membranes by using [2-125I]melatonin in a competition radioligand binding assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetMelatonin receptor type 1C(Chicken)
University College London

Curated by ChEMBL
LigandPNGBDBM50470697(CHEMBL14846)
Affinity DataKi:  1.10E+3nMAssay Description:Binding affinity in chicken brain membranes by using [2-125I]melatonin in a competition radioligand binding assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetMelatonin receptor type 1C(Chicken)
University College London

Curated by ChEMBL
LigandPNGBDBM50470691(CHEMBL278658)
Affinity DataKi:  1.55E+3nMAssay Description:Binding affinity in chicken brain membranes by using [2-125I]melatonin in a competition radioligand binding assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetMelatonin receptor type 1C(Chicken)
University College London

Curated by ChEMBL
LigandPNGBDBM50470693(CHEMBL276581)
Affinity DataKi:  1.90E+3nMAssay Description:Binding affinity in chicken brain membranes by using [2-125I]melatonin in a competition radioligand binding assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetMelatonin receptor type 1C(Chicken)
University College London

Curated by ChEMBL
LigandPNGBDBM50470709(CHEMBL15188)
Affinity DataKi:  6.50E+3nMAssay Description:Binding affinity in chicken brain membranes by using [2-125I]melatonin in a competition radioligand binding assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetMelatonin receptor type 1C(Chicken)
University College London

Curated by ChEMBL
LigandPNGBDBM50470696(CHEMBL14607)
Affinity DataKi:  7.00E+3nMAssay Description:Binding affinity in chicken brain membranes by using [2-125I]melatonin in a competition radioligand binding assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed