Compile Data Set for Download or QSAR
maximum 50k data
Found 5 Enz. Inhib. hit(s) with all data for entry = 50005205
TargetSubstance-P receptor(Homo sapiens (Human))
Merck Sharp And Dohme Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50034271(4-(3,5-Bis-trifluoromethyl-benzyloxymethyl)-4-phen...)
Affinity DataIC50:  0.950nMAssay Description:Antagonistic activity against human Tachykinin receptor 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(Homo sapiens (Human))
Merck Sharp And Dohme Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50034275(4-(3,5-Dichloro-benzyloxymethyl)-4-phenyl-piperidi...)
Affinity DataIC50:  4.60nMAssay Description:Antagonistic activity against human Tachykinin receptor 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(Homo sapiens (Human))
Merck Sharp And Dohme Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50034272(4-(3,5-Dimethyl-benzyloxymethyl)-4-phenyl-piperidi...)
Affinity DataIC50:  9nMAssay Description:Antagonistic activity against human Tachykinin receptor 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(Homo sapiens (Human))
Merck Sharp And Dohme Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50034273(4-Phenyl-4-(3-trifluoromethyl-benzyloxymethyl)-pip...)
Affinity DataIC50:  57nMAssay Description:Antagonistic activity against human Tachykinin receptor 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(Homo sapiens (Human))
Merck Sharp And Dohme Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50034274(4-Benzyloxymethyl-4-phenyl-piperidine | CHEMBL2268...)
Affinity DataIC50:  1.10E+3nMAssay Description:Antagonistic activity against human Tachykinin receptor 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed