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Report error Found 46 Enz. Inhib. hit(s) with all data for entry = 50036403
Target5-hydroxytryptamine receptor 1A(Mouse)
University of G£Teborg

Curated by ChEMBL
LigandPNGBDBM50016777(((R)-8-Hydroxy-1,2,3,4-tetrahydro-naphthalen-2-yl)...)
Affinity DataKi:  0.5nMAssay Description:In vitro binding affinity towards 5-hydroxytryptamine 1A receptor by using [3H]-8-OH-DPAT as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

Target5-hydroxytryptamine receptor 1A(Mouse)
University of G£Teborg

Curated by ChEMBL
LigandPNGBDBM50034366(CHEMBL28437 | Trifluoro-methanesulfonic acid 7-dip...)
Affinity DataKi:  0.800nMAssay Description:In vitro binding affinity towards 5-hydroxytryptamine 1A receptor by using [3H]-8-OH-DPAT as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

Target5-hydroxytryptamine receptor 1A(Mouse)
University of G£Teborg

Curated by ChEMBL
LigandPNGBDBM50407735(CHEMBL2021539)
Affinity DataKi:  1.30nMAssay Description:In vitro binding affinity towards 5-hydroxytryptamine 1A receptor by using [3H]-8-OH-DPAT as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

Target5-hydroxytryptamine receptor 1A(Mouse)
University of G£Teborg

Curated by ChEMBL
LigandPNGBDBM50034368(CHEMBL28313 | Trifluoro-methanesulfonic acid 7-pro...)
Affinity DataKi:  2.80nMAssay Description:In vitro binding affinity towards 5-hydroxytryptamine 1A receptor by using [3H]-8-OH-DPAT as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

Target5-hydroxytryptamine receptor 1D(Human)
University of G£Teborg

Curated by ChEMBL
LigandPNGBDBM50407735(CHEMBL2021539)
Affinity DataKi:  6.70nMAssay Description:In vitro binding affinity towards 5-hydroxytryptamine 1D receptor alpha by using [3H]5-HT as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetD(2) dopamine receptor(Human)
University of G£Teborg

Curated by ChEMBL
LigandPNGBDBM50407737(CHEMBL2021538)
Affinity DataKi:  8.70nMAssay Description:In vitro binding affinity towards Dopamine receptor D2 by using [3H]U-86170 as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

Target5-hydroxytryptamine receptor 1A(Mouse)
University of G£Teborg

Curated by ChEMBL
LigandPNGBDBM50407737(CHEMBL2021538)
Affinity DataKi:  10nMAssay Description:In vitro binding affinity towards 5-hydroxytryptamine 1A receptor by using [3H]-8-OH-DPAT as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

Target5-hydroxytryptamine receptor 1D(Human)
University of G£Teborg

Curated by ChEMBL
LigandPNGBDBM50034366(CHEMBL28437 | Trifluoro-methanesulfonic acid 7-dip...)
Affinity DataKi:  12nMAssay Description:In vitro binding affinity towards 5-hydroxytryptamine 1D receptor alpha by using [3H]5-HT as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

Target5-hydroxytryptamine receptor 1A(Mouse)
University of G£Teborg

Curated by ChEMBL
LigandPNGBDBM50407734(CHEMBL2021524)
Affinity DataKi:  13nMAssay Description:In vitro binding affinity towards 5-hydroxytryptamine 1A receptor by using [3H]-8-OH-DPAT as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetD(3) dopamine receptor(Human)
University of G£Teborg

Curated by ChEMBL
LigandPNGBDBM50407737(CHEMBL2021538)
Affinity DataKi:  15nMAssay Description:In vitro binding affinity towards Dopamine receptor D3 by using [3H]spiperone as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

Target5-hydroxytryptamine receptor 1D(Human)
University of G£Teborg

Curated by ChEMBL
LigandPNGBDBM50034368(CHEMBL28313 | Trifluoro-methanesulfonic acid 7-pro...)
Affinity DataKi:  15nMAssay Description:In vitro binding affinity towards 5-hydroxytryptamine 1D receptor alpha by using [3H]5-HT as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetD(2) dopamine receptor(Human)
University of G£Teborg

Curated by ChEMBL
LigandPNGBDBM50034365(CHEMBL554220 | Trifluoro-methanesulfonic acid (R)-...)
Affinity DataKi:  50nMAssay Description:In vitro binding affinity towards dopamine D2 receptor by using [3H]U-86170 as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetD(2) dopamine receptor(Human)
University of G£Teborg

Curated by ChEMBL
LigandPNGBDBM50034366(CHEMBL28437 | Trifluoro-methanesulfonic acid 7-dip...)
Affinity DataKi:  62nMAssay Description:In vitro binding affinity towards Dopamine receptor D2 by using [3H]U-86170 as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

Target5-hydroxytryptamine receptor 1D(Human)
University of G£Teborg

Curated by ChEMBL
LigandPNGBDBM50407737(CHEMBL2021538)
Affinity DataKi:  63nMAssay Description:In vitro binding affinity towards 5-hydroxytryptamine 1D receptor alpha by using [3H]5-HT as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetD(2) dopamine receptor(Human)
University of G£Teborg

Curated by ChEMBL
LigandPNGBDBM50407735(CHEMBL2021539)
Affinity DataKi:  69nMAssay Description:In vitro binding affinity towards Dopamine receptor D2 by using [3H]U-86170 as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetD(2) dopamine receptor(Human)
University of G£Teborg

Curated by ChEMBL
LigandPNGBDBM50016777(((R)-8-Hydroxy-1,2,3,4-tetrahydro-naphthalen-2-yl)...)
Affinity DataKi:  90nMAssay Description:In vitro binding affinity towards Dopamine receptor D2 by using [3H]U-86170 as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetD(2) dopamine receptor(Human)
University of G£Teborg

Curated by ChEMBL
LigandPNGBDBM50034368(CHEMBL28313 | Trifluoro-methanesulfonic acid 7-pro...)
Affinity DataKi:  108nMAssay Description:In vitro binding affinity towards Dopamine receptor D2 by using [3H]U-86170 as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetD(2) dopamine receptor(Human)
University of G£Teborg

Curated by ChEMBL
LigandPNGBDBM50407737(CHEMBL2021538)
Affinity DataKi:  115nMAssay Description:In vitro binding affinity towards Dopamine receptor D2 by using [3H]spiperone as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetD(3) dopamine receptor(Human)
University of G£Teborg

Curated by ChEMBL
LigandPNGBDBM50407736(CHEMBL2021525)
Affinity DataKi:  120nMAssay Description:In vitro binding affinity towards Dopamine receptor D3 by using [3H]spiperone as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

Target5-hydroxytryptamine receptor 1D(Human)
University of G£Teborg

Curated by ChEMBL
LigandPNGBDBM50034365(CHEMBL554220 | Trifluoro-methanesulfonic acid (R)-...)
Affinity DataKi:  125nMAssay Description:In vitro binding affinity towards 5-HT1D alpha receptor by using [3H]5-HT as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

Target5-hydroxytryptamine receptor 1D(Human)
University of G£Teborg

Curated by ChEMBL
LigandPNGBDBM50034366(CHEMBL28437 | Trifluoro-methanesulfonic acid 7-dip...)
Affinity DataKi:  127nMAssay Description:In vitro binding affinity towards 5-hydroxytryptamine 1D receptor alpha by using [3H]-5-HT as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

Target5-hydroxytryptamine receptor 1D(Human)
University of G£Teborg

Curated by ChEMBL
LigandPNGBDBM50407737(CHEMBL2021538)
Affinity DataKi:  130nMAssay Description:In vitro binding affinity towards 5-hydroxytryptamine 1D receptor beta by using [3H]5-HT as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

Target5-hydroxytryptamine receptor 1D(Human)
University of G£Teborg

Curated by ChEMBL
LigandPNGBDBM50407735(CHEMBL2021539)
Affinity DataKi:  138nMAssay Description:In vitro binding affinity towards 5-hydroxytryptamine 1D receptor beta by using [3H]5-HT as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

Target5-hydroxytryptamine receptor 1D(Human)
University of G£Teborg

Curated by ChEMBL
LigandPNGBDBM50407734(CHEMBL2021524)
Affinity DataKi:  157nMAssay Description:In vitro binding affinity towards 5-hydroxytryptamine 1D receptor alpha by using [3H]5-HT as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

Target5-hydroxytryptamine receptor 1D(Human)
University of G£Teborg

Curated by ChEMBL
LigandPNGBDBM50016777(((R)-8-Hydroxy-1,2,3,4-tetrahydro-naphthalen-2-yl)...)
Affinity DataKi:  164nMAssay Description:In vitro binding affinity towards 5-hydroxytryptamine 1D receptor alpha by using [3H]5-HT as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

Target5-hydroxytryptamine receptor 1D(Human)
University of G£Teborg

Curated by ChEMBL
LigandPNGBDBM50034368(CHEMBL28313 | Trifluoro-methanesulfonic acid 7-pro...)
Affinity DataKi:  169nMAssay Description:In vitro binding affinity towards 5-hydroxytryptamine 1D receptor beta by using [3H]5-HT as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetD(3) dopamine receptor(Human)
University of G£Teborg

Curated by ChEMBL
LigandPNGBDBM50016777(((R)-8-Hydroxy-1,2,3,4-tetrahydro-naphthalen-2-yl)...)
Affinity DataKi:  179nMAssay Description:In vitro binding affinity towards Dopamine receptor D3 by using [3H]spiperone as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

Target5-hydroxytryptamine receptor 1A(Mouse)
University of G£Teborg

Curated by ChEMBL
LigandPNGBDBM50034365(CHEMBL554220 | Trifluoro-methanesulfonic acid (R)-...)
Affinity DataKi:  222nMAssay Description:In vitro binding affinity towards 5-hydroxytryptamine 1A receptor by using [3H]-8-OH-DPAT as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetD(2) dopamine receptor(Human)
University of G£Teborg

Curated by ChEMBL
LigandPNGBDBM50407734(CHEMBL2021524)
Affinity DataKi:  225nMAssay Description:In vitro binding affinity towards Dopamine receptor D2 by using [3H]U-86170 as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetD(3) dopamine receptor(Human)
University of G£Teborg

Curated by ChEMBL
LigandPNGBDBM50034366(CHEMBL28437 | Trifluoro-methanesulfonic acid 7-dip...)
Affinity DataKi:  273nMAssay Description:In vitro binding affinity towards Dopamine receptor D3 by using [3H]spiperone as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetD(2) dopamine receptor(Human)
University of G£Teborg

Curated by ChEMBL
LigandPNGBDBM50407735(CHEMBL2021539)
Affinity DataKi:  311nMAssay Description:In vitro binding affinity towards Dopamine receptor D2 by using [3H]spiperone as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

Target5-hydroxytryptamine receptor 1D(Human)
University of G£Teborg

Curated by ChEMBL
LigandPNGBDBM50034365(CHEMBL554220 | Trifluoro-methanesulfonic acid (R)-...)
Affinity DataKi:  340nMAssay Description:In vitro binding affinity towards 5-hydroxytryptamine 1D receptor alpha by using [3H]-5-HT as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetD(3) dopamine receptor(Human)
University of G£Teborg

Curated by ChEMBL
LigandPNGBDBM50034365(CHEMBL554220 | Trifluoro-methanesulfonic acid (R)-...)
Affinity DataKi:  359nMAssay Description:In vitro binding affinity towards Dopamine receptor D3 by using [3H]spiperone as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetD(2) dopamine receptor(Human)
University of G£Teborg

Curated by ChEMBL
LigandPNGBDBM50034366(CHEMBL28437 | Trifluoro-methanesulfonic acid 7-dip...)
Affinity DataKi: >413nMAssay Description:In vitro binding affinity towards Dopamine receptor D2 by using [3H]spiperone as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetD(2) dopamine receptor(Human)
University of G£Teborg

Curated by ChEMBL
LigandPNGBDBM50407734(CHEMBL2021524)
Affinity DataKi: >413nMAssay Description:In vitro binding affinity towards Dopamine receptor D2 by using [3H]spiperone as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetD(2) dopamine receptor(Human)
University of G£Teborg

Curated by ChEMBL
LigandPNGBDBM50016777(((R)-8-Hydroxy-1,2,3,4-tetrahydro-naphthalen-2-yl)...)
Affinity DataKi: >413nMAssay Description:In vitro binding affinity towards Dopamine receptor D2 by using [3H]spiperone as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetD(2) dopamine receptor(Human)
University of G£Teborg

Curated by ChEMBL
LigandPNGBDBM50034368(CHEMBL28313 | Trifluoro-methanesulfonic acid 7-pro...)
Affinity DataKi: >413nMAssay Description:In vitro binding affinity towards Dopamine receptor D2 by using [3H]spiperone as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetD(3) dopamine receptor(Human)
University of G£Teborg

Curated by ChEMBL
LigandPNGBDBM50407735(CHEMBL2021539)
Affinity DataKi:  524nMAssay Description:In vitro binding affinity towards Dopamine receptor D3 by using [3H]spiperone as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

Target5-hydroxytryptamine receptor 1D(Human)
University of G£Teborg

Curated by ChEMBL
LigandPNGBDBM50016777(((R)-8-Hydroxy-1,2,3,4-tetrahydro-naphthalen-2-yl)...)
Affinity DataKi:  638nMAssay Description:In vitro binding affinity towards 5-hydroxytryptamine 1D receptor alpha by using [3H]-5-HT as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetD(3) dopamine receptor(Human)
University of G£Teborg

Curated by ChEMBL
LigandPNGBDBM50034368(CHEMBL28313 | Trifluoro-methanesulfonic acid 7-pro...)
Affinity DataKi:  691nMAssay Description:In vitro binding affinity towards Dopamine receptor D3 by using [3H]spiperone as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

Target5-hydroxytryptamine receptor 1A(Mouse)
University of G£Teborg

Curated by ChEMBL
LigandPNGBDBM50407736(CHEMBL2021525)
Affinity DataKi: >1.00E+3nMAssay Description:In vitro binding affinity towards 5-hydroxytryptamine 1A receptor by using [3H]-8-OH-DPAT as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

Target5-hydroxytryptamine receptor 1D(Human)
University of G£Teborg

Curated by ChEMBL
LigandPNGBDBM50407734(CHEMBL2021524)
Affinity DataKi:  1.26E+3nMAssay Description:In vitro binding affinity towards 5-hydroxytryptamine 1D receptor beta by using [3H]5-HT as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

Target5-hydroxytryptamine receptor 1D(Human)
University of G£Teborg

Curated by ChEMBL
LigandPNGBDBM50407736(CHEMBL2021525)
Affinity DataKi: >1.50E+3nMAssay Description:In vitro binding affinity towards 5-hydroxytryptamine 1D receptor alpha by using [3H]5-HT as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

Target5-hydroxytryptamine receptor 1D(Human)
University of G£Teborg

Curated by ChEMBL
LigandPNGBDBM50407736(CHEMBL2021525)
Affinity DataKi: >1.50E+3nMAssay Description:In vitro binding affinity towards 5-hydroxytryptamine 1D receptor alpha by using [3H]-5-HT as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetD(3) dopamine receptor(Human)
University of G£Teborg

Curated by ChEMBL
LigandPNGBDBM50407734(CHEMBL2021524)
Affinity DataKi:  1.57E+3nMAssay Description:In vitro binding affinity towards Dopamine receptor D3 by using [3H]spiperone as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetD(2) dopamine receptor(Human)
University of G£Teborg

Curated by ChEMBL
LigandPNGBDBM50407736(CHEMBL2021525)
Affinity DataKi: >3.80E+3nMAssay Description:In vitro binding affinity towards Dopamine receptor D2 by using [3H]U-86170 as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed