Compile Data Set for Download or QSAR
Report error Found 16 Enz. Inhib. hit(s) with all data for entry = 50005213
TargetDelta-type opioid receptor(Human)
University of Minnesota

Curated by ChEMBL
LigandPNGBDBM50034407(1N-{3-[22-cyclopropylmethyl-2,16-dihydroxy-14-oxa-...)
Affinity DataKi:  0.0190nMAssay Description:Tested for binding affinity against delta1 opioid receptor using [3H]-DPDPE as a radioligand in the guinea pig brain membranes.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Human)
University of Minnesota

Curated by ChEMBL
LigandPNGBDBM50034407(1N-{3-[22-cyclopropylmethyl-2,16-dihydroxy-14-oxa-...)
Affinity DataKi:  0.0380nMAssay Description:Tested for binding affinity against delta2 opioid receptor using [3H]DSLET as a radioligand in the guinea pig brain membranes.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Human)
University of Minnesota

Curated by ChEMBL
LigandPNGBDBM50034405(22-cyclopropylmethyl-11-(2-isothiocyanatobenzyl)-1...)
Affinity DataKi:  2nMAssay Description:Tested for binding affinity against delta1 opioid receptor using [3H]-DPDPE as a radioligand in the guinea pig brain membranes.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Human)
University of Minnesota

Curated by ChEMBL
LigandPNGBDBM50034405(22-cyclopropylmethyl-11-(2-isothiocyanatobenzyl)-1...)
Affinity DataKi:  3.60nMAssay Description:Tested for binding affinity against delta2 opioid receptor using [3H]DSLET as a radioligand in the guinea pig brain membranes.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Human)
University of Minnesota

Curated by ChEMBL
LigandPNGBDBM50034408(22-cyclopropylmethyl-11-(3-isothiocyanatobenzyl)-1...)
Affinity DataKi:  4.20nMAssay Description:Tested for binding affinity against delta1 opioid receptor using [3H]-DPDPE as a radioligand in the guinea pig brain membranes.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Human)
University of Minnesota

Curated by ChEMBL
LigandPNGBDBM50034406(22-cyclopropylmethyl-11-(4-isothiocyanatobenzyl)-1...)
Affinity DataKi:  5nMAssay Description:Tested for binding affinity against delta2 opioid receptor using [3H]DSLET as a radioligand in the guinea pig brain membranes.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Human)
University of Minnesota

Curated by ChEMBL
LigandPNGBDBM50034406(22-cyclopropylmethyl-11-(4-isothiocyanatobenzyl)-1...)
Affinity DataKi:  5.30nMAssay Description:Tested for binding affinity against delta1 opioid receptor using [3H]-DPDPE as a radioligand in the guinea pig brain membranes.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Human)
University of Minnesota

Curated by ChEMBL
LigandPNGBDBM50034408(22-cyclopropylmethyl-11-(3-isothiocyanatobenzyl)-1...)
Affinity DataKi:  7nMAssay Description:Tested for binding affinity against delta2 opioid receptor using [3H]DSLET as a radioligand in the guinea pig brain membranes.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetKappa-type opioid receptor(Guinea pig)
University of Minnesota

Curated by ChEMBL
LigandPNGBDBM50034407(1N-{3-[22-cyclopropylmethyl-2,16-dihydroxy-14-oxa-...)
Affinity DataKi:  8.80nMAssay Description:Tested for binding affinity against Opioid receptor kappa 1 using [3H]U-69593 as a radioligand in the guinea pig brain membranes.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMu-type opioid receptor(Guinea pig)
University of Minnesota

Curated by ChEMBL
LigandPNGBDBM50034407(1N-{3-[22-cyclopropylmethyl-2,16-dihydroxy-14-oxa-...)
Affinity DataKi:  15nMAssay Description:Tested for binding affinity against mu opioid receptor using [3H]DAMGO as a radioligand in the guinea pig brain membranes.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMu-type opioid receptor(Guinea pig)
University of Minnesota

Curated by ChEMBL
LigandPNGBDBM50034408(22-cyclopropylmethyl-11-(3-isothiocyanatobenzyl)-1...)
Affinity DataKi:  66nMAssay Description:Tested for binding affinity against mu opioid receptor using [3H]DAMGO as a radioligand in the guinea pig brain membranes.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetKappa-type opioid receptor(Guinea pig)
University of Minnesota

Curated by ChEMBL
LigandPNGBDBM50034408(22-cyclopropylmethyl-11-(3-isothiocyanatobenzyl)-1...)
Affinity DataKi:  104nMAssay Description:Tested for binding affinity against Opioid receptor kappa 1 using [3H]U-69593 as a radioligand in the guinea pig brain membranes.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMu-type opioid receptor(Guinea pig)
University of Minnesota

Curated by ChEMBL
LigandPNGBDBM50034405(22-cyclopropylmethyl-11-(2-isothiocyanatobenzyl)-1...)
Affinity DataKi:  151nMAssay Description:Tested for binding affinity against mu opioid receptor using [3H]DAMGO as a radioligand in the guinea pig brain membranes.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetKappa-type opioid receptor(Guinea pig)
University of Minnesota

Curated by ChEMBL
LigandPNGBDBM50034406(22-cyclopropylmethyl-11-(4-isothiocyanatobenzyl)-1...)
Affinity DataKi:  245nMAssay Description:Tested for binding affinity against Opioid receptor kappa 1 using [3H]U-69593 as a radioligand in the guinea pig brain membranes.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMu-type opioid receptor(Guinea pig)
University of Minnesota

Curated by ChEMBL
LigandPNGBDBM50034406(22-cyclopropylmethyl-11-(4-isothiocyanatobenzyl)-1...)
Affinity DataKi:  289nMAssay Description:Tested for binding affinity against mu opioid receptor using [3H]DAMGO as a radioligand in the guinea pig brain membranes.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetKappa-type opioid receptor(Guinea pig)
University of Minnesota

Curated by ChEMBL
LigandPNGBDBM50034405(22-cyclopropylmethyl-11-(2-isothiocyanatobenzyl)-1...)
Affinity DataKi:  615nMAssay Description:Tested for binding affinity against Opioid receptor kappa 1 using [3H]U-69593 as a radioligand in the guinea pig brain membranes.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed