Compile Data Set for Download or QSAR
maximum 50k data
Found 40 Enz. Inhib. hit(s) with all data for entry = 50005343
TargetGastrin/cholecystokinin type B receptor(Homo sapiens (Human))
Washington University

Curated by ChEMBL
LigandPNGBDBM50035820(Ac-Trp-L-3-MPt(Pr)-Asp-Phe-NH2 | CHEMBL37830)
Affinity DataIC50:  0.450nMAssay Description:Binding affinity towards Cholecystokinin type B receptor by displacement of [125I]-BH-CCK-8 from human jurkat cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin/cholecystokinin type B receptor(Homo sapiens (Human))
Washington University

Curated by ChEMBL
LigandPNGBDBM50035832(Ac-Trp-L-3-MPt(Et)-Asp-Phe-NH2 | CHEMBL35471)
Affinity DataIC50:  1.80nMAssay Description:Binding affinity towards Cholecystokinin type B receptor by displacement of [125I]-BH-CCK-8 from human jurkat cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin/cholecystokinin type B receptor(Homo sapiens (Human))
Washington University

Curated by ChEMBL
LigandPNGBDBM50035825(Ac-Trp-L-3-MPt(Pr)-Asp-Phe-NH2 | CHEMBL34554)
Affinity DataIC50:  3.30nMAssay Description:Binding affinity towards Cholecystokinin type B receptor by displacement of [125I]-BH-CCK-8 from human jurkat cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin/cholecystokinin type B receptor(Homo sapiens (Human))
Washington University

Curated by ChEMBL
LigandPNGBDBM50035829(Ac-Trp-L-3-MPt(Et)-Asp-Phe-NH2 | CHEMBL34853)
Affinity DataIC50:  30nMAssay Description:Binding affinity towards Cholecystokinin type B receptor by displacement of [125I]-BH-CCK-8 from human jurkat cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin/cholecystokinin type B receptor(Homo sapiens (Human))
Washington University

Curated by ChEMBL
LigandPNGBDBM50035834(Ac-Trp-L-3-MPt(Me)-Asp-Phe-NH2 | CHEMBL287753)
Affinity DataIC50:  50nMAssay Description:Binding affinity towards Cholecystokinin type B receptor by displacement of [125I]-BH-CCK-8 from human jurkat cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin/cholecystokinin type B receptor(Homo sapiens (Human))
Washington University

Curated by ChEMBL
LigandPNGBDBM50035833(Ac-Trp-D-3-MPt(Pr)-Asp-Phe-NH2 | CHEMBL37984)
Affinity DataIC50:  70nMAssay Description:Binding affinity towards Cholecystokinin type B receptor by displacement of [125I]-BH-CCK-8 from human jurkat cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin/cholecystokinin type B receptor(Homo sapiens (Human))
Washington University

Curated by ChEMBL
LigandPNGBDBM50035822(Ac-Trp-L-3-MPc(Me)-Asp-Phe-NH2 | CHEMBL37983)
Affinity DataIC50:  300nMAssay Description:Binding affinity towards Cholecystokinin type B receptor by displacement of [125I]-BH-CCK-8 from human jurkat cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin/cholecystokinin type B receptor(Homo sapiens (Human))
Washington University

Curated by ChEMBL
LigandPNGBDBM50035823(Ac-Trp-D-Pro-Asp-Phe-NH2 | Ac-Trp-Pro-Asp-Phe-NH2 ...)
Affinity DataIC50:  600nMAssay Description:Binding affinity towards Cholecystokinin type B receptor by displacement of [125I]-BH-CCK-8 from human jurkat cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin/cholecystokinin type B receptor(Homo sapiens (Human))
Washington University

Curated by ChEMBL
LigandPNGBDBM50035828(Ac-Trp-D-3-MPt(Pr)-Asp-Phe-NH2 | CHEMBL37900)
Affinity DataIC50:  600nMAssay Description:Binding affinity towards Cholecystokinin type B receptor by displacement of [125I]-BH-CCK-8 from human jurkat cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin/cholecystokinin type B receptor(Homo sapiens (Human))
Washington University

Curated by ChEMBL
LigandPNGBDBM50035821(Ac-Trp-D-3-MPt(Et)-Asp-Phe-NH2 | CHEMBL34916)
Affinity DataIC50:  800nMAssay Description:Binding affinity towards Cholecystokinin type B receptor by displacement of [125I]-BH-CCK-8 from human jurkat cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholecystokinin receptor type A(RAT)
Washington University

Curated by ChEMBL
LigandPNGBDBM50035825(Ac-Trp-L-3-MPt(Pr)-Asp-Phe-NH2 | CHEMBL34554)
Affinity DataIC50: >1.00E+3nMAssay Description:Binding affinity towards Cholecystokinin type A receptor by displacement of [125I]-BH-CCK-8 from rat pancreatic aciniMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholecystokinin receptor type A(RAT)
Washington University

Curated by ChEMBL
LigandPNGBDBM50035828(Ac-Trp-D-3-MPt(Pr)-Asp-Phe-NH2 | CHEMBL37900)
Affinity DataIC50: >1.00E+3nMAssay Description:Compound was tested for binding affinity towards Cholecystokinin type A receptor by measuring its ability to displace [125I]-BH-CCK-8 from rat pancre...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholecystokinin receptor type A(RAT)
Washington University

Curated by ChEMBL
LigandPNGBDBM50035823(Ac-Trp-D-Pro-Asp-Phe-NH2 | Ac-Trp-Pro-Asp-Phe-NH2 ...)
Affinity DataIC50: >1.00E+3nMAssay Description:Binding affinity towards Cholecystokinin type A receptor by displacement of [125I]-BH-CCK-8 from rat pancreatic aciniMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholecystokinin receptor type A(RAT)
Washington University

Curated by ChEMBL
LigandPNGBDBM50035833(Ac-Trp-D-3-MPt(Pr)-Asp-Phe-NH2 | CHEMBL37984)
Affinity DataIC50: >1.00E+3nMAssay Description:Binding affinity towards Cholecystokinin type A receptor by displacement of [125I]-BH-CCK-8 from rat pancreatic aciniMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholecystokinin receptor type A(RAT)
Washington University

Curated by ChEMBL
LigandPNGBDBM50035820(Ac-Trp-L-3-MPt(Pr)-Asp-Phe-NH2 | CHEMBL37830)
Affinity DataIC50: >1.00E+3nMAssay Description:Binding affinity towards Cholecystokinin type A receptor by displacement of [125I]-BH-CCK-8 from rat pancreatic aciniMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin/cholecystokinin type B receptor(Homo sapiens (Human))
Washington University

Curated by ChEMBL
LigandPNGBDBM50035831(Ac-Trp-D-3-MPt(Et)-Asp-Phe-NH2 | CHEMBL290444)
Affinity DataIC50:  2.50E+3nMAssay Description:Binding affinity towards Cholecystokinin type B receptor by displacement of [125I]-BH-CCK-8 from human jurkat cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin/cholecystokinin type B receptor(Homo sapiens (Human))
Washington University

Curated by ChEMBL
LigandPNGBDBM50035836((S)-3-((S)-2-{[(S)-2-Acetylamino-3-(1H-indol-3-yl)...)
Affinity DataIC50:  4.00E+3nMAssay Description:Binding affinity towards Cholecystokinin type B receptor by displacement of [125I]-BH-CCK-8 from human jurkat cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin/cholecystokinin type B receptor(Homo sapiens (Human))
Washington University

Curated by ChEMBL
LigandPNGBDBM50035826((S)-3-((S)-2-{[(S)-2-Acetylamino-3-(1H-indol-3-yl)...)
Affinity DataIC50:  7.00E+3nMAssay Description:Binding affinity towards Cholecystokinin type B receptor by displacement of [125I]-BH-CCK-8 from human jurkat cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholecystokinin receptor type A(RAT)
Washington University

Curated by ChEMBL
LigandPNGBDBM50035829(Ac-Trp-L-3-MPt(Et)-Asp-Phe-NH2 | CHEMBL34853)
Affinity DataIC50:  9.00E+3nMAssay Description:Binding affinity towards Cholecystokinin type A receptor by displacement of [125I]-BH-CCK-8 from rat pancreatic aciniMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholecystokinin receptor type A(RAT)
Washington University

Curated by ChEMBL
LigandPNGBDBM50035831(Ac-Trp-D-3-MPt(Et)-Asp-Phe-NH2 | CHEMBL290444)
Affinity DataIC50: >1.00E+4nMAssay Description:Binding affinity towards Cholecystokinin type A receptor by displacement of [125I]-BH-CCK-8 from rat pancreatic aciniMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin/cholecystokinin type B receptor(Homo sapiens (Human))
Washington University

Curated by ChEMBL
LigandPNGBDBM50035835(CHEMBL285756 | Trp-D-4-MPt(Me)-Asp-Phe-NH2)
Affinity DataIC50: >1.00E+4nMAssay Description:Binding affinity towards Cholecystokinin type B receptor by displacement of [125I]-BH-CCK-8 from human jurkat cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholecystokinin receptor type A(RAT)
Washington University

Curated by ChEMBL
LigandPNGBDBM50035836((S)-3-((S)-2-{[(S)-2-Acetylamino-3-(1H-indol-3-yl)...)
Affinity DataIC50: >1.00E+4nMAssay Description:Binding affinity towards Cholecystokinin type A receptor by displacement of [125I]-BH-CCK-8 from rat pancreatic aciniMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholecystokinin receptor type A(RAT)
Washington University

Curated by ChEMBL
LigandPNGBDBM50035827(Ac-Trp-L-4-MPc(Me)-Asp-Phe-NH2 | Ac-Trp-L-4-MPt(Me...)
Affinity DataIC50: >1.00E+4nMAssay Description:Binding affinity towards Cholecystokinin type A receptor by displacement of [125I]-BH-CCK-8 from rat pancreatic aciniMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin/cholecystokinin type B receptor(Homo sapiens (Human))
Washington University

Curated by ChEMBL
LigandPNGBDBM50035827(Ac-Trp-L-4-MPc(Me)-Asp-Phe-NH2 | Ac-Trp-L-4-MPt(Me...)
Affinity DataIC50: >1.00E+4nMAssay Description:Binding affinity towards Cholecystokinin type B receptor by displacement of [125I]-BH-CCK-8 from human jurkat cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin/cholecystokinin type B receptor(Homo sapiens (Human))
Washington University

Curated by ChEMBL
LigandPNGBDBM50453646(CHEMBL2114402)
Affinity DataIC50: >1.00E+4nMAssay Description:Binding affinity towards Cholecystokinin type B receptor by displacement of [125I]-BH-CCK-8 from human jurkat cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholecystokinin receptor type A(RAT)
Washington University

Curated by ChEMBL
LigandPNGBDBM50035834(Ac-Trp-L-3-MPt(Me)-Asp-Phe-NH2 | CHEMBL287753)
Affinity DataIC50: >1.00E+4nMAssay Description:Binding affinity towards Cholecystokinin type A receptor by displacement of [125I]-BH-CCK-8 from rat pancreatic aciniMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholecystokinin receptor type A(RAT)
Washington University

Curated by ChEMBL
LigandPNGBDBM50035835(CHEMBL285756 | Trp-D-4-MPt(Me)-Asp-Phe-NH2)
Affinity DataIC50: >1.00E+4nMAssay Description:Binding affinity towards Cholecystokinin type A receptor by displacement of [125I]-BH-CCK-8 from rat pancreatic aciniMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin/cholecystokinin type B receptor(Homo sapiens (Human))
Washington University

Curated by ChEMBL
LigandPNGBDBM50035819(Ac-Trp-D-3-MPt(Me)-Asp-Phe-NH2 | CHEMBL37786)
Affinity DataIC50:  1.00E+4nMAssay Description:Binding affinity towards Cholecystokinin type B receptor by displacement of [125I]-BH-CCK-8 from human jurkat cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin/cholecystokinin type B receptor(Homo sapiens (Human))
Washington University

Curated by ChEMBL
LigandPNGBDBM50035830(Ac-Trp-D-Nle(Me)-Asp-Phe-NH2 | CHEMBL35394)
Affinity DataIC50: >1.00E+4nMAssay Description:Binding affinity towards Cholecystokinin type B receptor by displacement of [125I]-BH-CCK-8 from human jurkat cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin/cholecystokinin type B receptor(Homo sapiens (Human))
Washington University

Curated by ChEMBL
LigandPNGBDBM50035824(Ac-Trp-D-3-MPc(Me)-Asp-Phe-NH2 | CHEMBL285051)
Affinity DataIC50:  1.00E+4nMAssay Description:Binding affinity towards Cholecystokinin type B receptor by displacement of [125I]-BH-CCK-8 from human jurkat cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholecystokinin receptor type A(RAT)
Washington University

Curated by ChEMBL
LigandPNGBDBM50035822(Ac-Trp-L-3-MPc(Me)-Asp-Phe-NH2 | CHEMBL37983)
Affinity DataIC50:  1.00E+4nMAssay Description:Binding affinity towards Cholecystokinin type A receptor by displacement of [125I]-BH-CCK-8 from rat pancreatic aciniMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholecystokinin receptor type A(RAT)
Washington University

Curated by ChEMBL
LigandPNGBDBM50035830(Ac-Trp-D-Nle(Me)-Asp-Phe-NH2 | CHEMBL35394)
Affinity DataIC50: >1.00E+4nMAssay Description:Binding affinity towards Cholecystokinin type A receptor by displacement of [125I]-BH-CCK-8 from rat pancreatic aciniMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholecystokinin receptor type A(RAT)
Washington University

Curated by ChEMBL
LigandPNGBDBM50035832(Ac-Trp-L-3-MPt(Et)-Asp-Phe-NH2 | CHEMBL35471)
Affinity DataIC50: >1.00E+4nMAssay Description:Binding affinity towards Cholecystokinin type A receptor by displacement of [125I]-BH-CCK-8 from rat pancreatic aciniMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholecystokinin receptor type A(RAT)
Washington University

Curated by ChEMBL
LigandPNGBDBM50453646(CHEMBL2114402)
Affinity DataIC50: >1.00E+4nMAssay Description:Binding affinity towards Cholecystokinin type A receptor by displacement of [125I]-BH-CCK-8 from rat pancreatic aciniMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholecystokinin receptor type A(RAT)
Washington University

Curated by ChEMBL
LigandPNGBDBM50035826((S)-3-((S)-2-{[(S)-2-Acetylamino-3-(1H-indol-3-yl)...)
Affinity DataIC50: >1.00E+4nMAssay Description:Binding affinity towards Cholecystokinin type A receptor by displacement of [125I]-BH-CCK-8 from rat pancreatic aciniMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin/cholecystokinin type B receptor(Homo sapiens (Human))
Washington University

Curated by ChEMBL
LigandPNGBDBM50035827(Ac-Trp-L-4-MPc(Me)-Asp-Phe-NH2 | Ac-Trp-L-4-MPt(Me...)
Affinity DataIC50: >1.00E+4nMAssay Description:Binding affinity towards Cholecystokinin type B receptor by displacement of [125I]-BH-CCK-8 from human jurkat cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholecystokinin receptor type A(RAT)
Washington University

Curated by ChEMBL
LigandPNGBDBM50035824(Ac-Trp-D-3-MPc(Me)-Asp-Phe-NH2 | CHEMBL285051)
Affinity DataIC50: >1.00E+4nMAssay Description:Binding affinity towards Cholecystokinin type A receptor by displacement of [125I]-BH-CCK-8 from rat pancreatic aciniMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholecystokinin receptor type A(RAT)
Washington University

Curated by ChEMBL
LigandPNGBDBM50035819(Ac-Trp-D-3-MPt(Me)-Asp-Phe-NH2 | CHEMBL37786)
Affinity DataIC50: >1.00E+4nMAssay Description:Binding affinity towards Cholecystokinin type A receptor by displacement of [125I]-BH-CCK-8 from rat pancreatic aciniMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholecystokinin receptor type A(RAT)
Washington University

Curated by ChEMBL
LigandPNGBDBM50035827(Ac-Trp-L-4-MPc(Me)-Asp-Phe-NH2 | Ac-Trp-L-4-MPt(Me...)
Affinity DataIC50: >1.00E+4nMAssay Description:Binding affinity towards Cholecystokinin type A receptor by displacement of [125I]-BH-CCK-8 from rat pancreatic aciniMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholecystokinin receptor type A(RAT)
Washington University

Curated by ChEMBL
LigandPNGBDBM50035821(Ac-Trp-D-3-MPt(Et)-Asp-Phe-NH2 | CHEMBL34916)
Affinity DataIC50: >1.00E+4nMAssay Description:Binding affinity towards Cholecystokinin type A receptor by displacement of [125I]-BH-CCK-8 from rat pancreatic aciniMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed