Compile Data Set for Download or QSAR
Report error Found 47 Enz. Inhib. hit(s) with all data for entry = 50005414
TargetSigma non-opioid intracellular receptor 1(Human)
New York University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50036730BDBM50036730(3-[4-(4-Chloro-phenyl)-3,6-dihydro-2H-pyridin-1-yl...)
Affinity DataIC50: 0.5nMAssay Description:Binding affinity against sigma receptor in bovine cerebellum using 2.0 nM [3H]haloperidol in the presence of 25 nM unlabeled spiperoneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSigma non-opioid intracellular receptor 1(Human)
New York University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50007400BDBM50007400(CHEMBL1788131 | CHEMBL325238 | 4-Phenyl-1-(4-pheny...)
Affinity DataKi:  1nMAssay Description:Binding affinity against sigma receptor in bovine cerebellum using 2.0 nM [3H]haloperidol in the presence of 25 nM unlabeled spiperoneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSigma non-opioid intracellular receptor 1(Human)
New York University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50036722BDBM50036722(3-[4-(4-Fluoro-phenyl)-3,6-dihydro-2H-pyridin-1-yl...)
Affinity DataIC50: 4nMAssay Description:Binding affinity against sigma receptor in bovine cerebellum using 2.0 nM [3H]haloperidol in the presence of 25 nM unlabeled spiperoneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSigma non-opioid intracellular receptor 1(Human)
New York University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50036729BDBM50036729(1-Phenyl-3-(4-phenyl-piperidin-1-yl)-propan-1-one ...)
Affinity DataIC50: 7nMAssay Description:Binding affinity against sigma receptor in bovine cerebellum using 2.0 nM [3H]haloperidol in the presence of 25 nM unlabeled spiperoneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSigma non-opioid intracellular receptor 1(Human)
New York University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50036716BDBM50036716(1-Phenyl-3-(4-phenyl-3,6-dihydro-2H-pyridin-1-yl)-...)
Affinity DataIC50: 8nMAssay Description:Binding affinity against sigma receptor in bovine cerebellum using 2.0 nM [3H]haloperidol in the presence of 25 nM unlabeled spiperoneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSigma non-opioid intracellular receptor 1(Human)
New York University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50002245BDBM50002245(CHEMBL130356 | CHEMBL137776 | 4-[2-(1-Cyclopropylm...)
Affinity DataKi:  10nMAssay Description:Binding affinity against sigma receptor in bovine cerebellum using 2.0 nM [3H]- haloperidolMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSigma non-opioid intracellular receptor 1(Human)
New York University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50002218BDBM50002218(CHEMBL42228 | CHEMBL543412 | 2-(1-Cyclopropylmethy...)
Affinity DataKi:  10nMAssay Description:Binding affinity against sigma receptor in bovine cerebellum using 2.0 nM [3H]- haloperidolMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSigma non-opioid intracellular receptor 1(Human)
New York University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50036711BDBM50036711(1-(4-Fluoro-phenyl)-3-[4-(4-fluoro-phenyl)-3,6-dih...)
Affinity DataIC50: 23nMAssay Description:Binding affinity against sigma receptor in bovine cerebellum using 2.0 nM [3H]haloperidol in the presence of 25 nM unlabeled spiperoneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSigma non-opioid intracellular receptor 1(Human)
New York University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50036724BDBM50036724(1-(4-Chloro-phenyl)-3-[4-(4-fluoro-phenyl)-3,6-dih...)
Affinity DataIC50: 25nMAssay Description:Binding affinity against sigma receptor in bovine cerebellum using 2.0 nM [3H]haloperidol in the presence of 25 nM unlabeled spiperoneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSigma non-opioid intracellular receptor 1(Human)
New York University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50036712BDBM50036712(CHEMBL101664 | CHEMBL2011566 | 4-(4-Chloro-phenyl)...)
Affinity DataIC50: 50nMAssay Description:Binding affinity against sigma receptor in bovine cerebellum using 2.0 nM [3H]haloperidol in the presence of 25 nM unlabeled spiperoneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSigma non-opioid intracellular receptor 1(Human)
New York University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50036713BDBM50036713(1-(4-Bromo-phenyl)-3-[4-(4-fluoro-phenyl)-3,6-dihy...)
Affinity DataIC50: 66nMAssay Description:Binding affinity against sigma receptor in bovine cerebellum using 2.0 nM [3H]haloperidol in the presence of 25 nM unlabeled spiperoneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSigma non-opioid intracellular receptor 1(Human)
New York University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50036723BDBM50036723(1-(4-Bromo-phenyl)-3-[4-(4-chloro-phenyl)-3,6-dihy...)
Affinity DataIC50: 100nMAssay Description:Binding affinity against sigma receptor in bovine cerebellum using 2.0 nM [3H]haloperidol in the presence of 25 nM unlabeled spiperoneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSigma non-opioid intracellular receptor 1(Human)
New York University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50036728BDBM50036728(1-(2-Chloro-phenyl)-3-[4-(4-chloro-phenyl)-3,6-dih...)
Affinity DataIC50: 105nMAssay Description:Binding affinity against sigma receptor in bovine cerebellum using 2.0 nM [3H]haloperidol in the presence of 25 nM unlabeled spiperoneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSigma non-opioid intracellular receptor 1(Human)
New York University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50036717BDBM50036717(3-[4-(4-Chloro-phenyl)-3,6-dihydro-2H-pyridin-1-yl...)
Affinity DataIC50: 158nMAssay Description:Binding affinity against sigma receptor in bovine cerebellum using 2.0 nM [3H]haloperidol in the presence of 25 nM unlabeled spiperoneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSigma non-opioid intracellular receptor 1(Human)
New York University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50036719BDBM50036719(1-(4-Chloro-phenyl)-3-[4-(4-chloro-phenyl)-3,6-dih...)
Affinity DataIC50: 158nMAssay Description:Binding affinity against sigma receptor in bovine cerebellum using 2.0 nM [3H]haloperidol in the presence of 25 nM unlabeled spiperoneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSigma non-opioid intracellular receptor 1(Human)
New York University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50036721BDBM50036721(3-[4-(4-Chloro-phenyl)-3,6-dihydro-2H-pyridin-1-yl...)
Affinity DataIC50: 235nMAssay Description:Binding affinity against sigma receptor in bovine cerebellum using 2.0 nM [3H]haloperidol in the presence of 25 nM unlabeled spiperoneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSigma non-opioid intracellular receptor 1(Human)
New York University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50036720BDBM50036720(1-Benzo[1,3]dioxol-5-yl-3-[4-(4-chloro-phenyl)-3,6...)
Affinity DataIC50: 281nMAssay Description:Binding affinity against sigma receptor in bovine cerebellum using 2.0 nM [3H]haloperidol in the presence of 25 nM unlabeled spiperoneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Bovine)
New York University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50007400BDBM50007400(CHEMBL1788131 | CHEMBL325238 | 4-Phenyl-1-(4-pheny...)
Affinity DataIC50: 335nMAssay Description:Binding affinity against Dopamine receptor D2 in bovine striatal homogenate using 200 pM [3H]- spiperone and 250 nM unlabeled ketanserinMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSigma non-opioid intracellular receptor 1(Human)
New York University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50036710BDBM50036710(3-[4-(4-Chloro-phenyl)-3,6-dihydro-2H-pyridin-1-yl...)
Affinity DataIC50: 400nMAssay Description:Binding affinity against sigma receptor in bovine cerebellum using 2.0 nM [3H]haloperidol in the presence of 25 nM unlabeled spiperoneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSigma non-opioid intracellular receptor 1(Human)
New York University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50036726BDBM50036726(3-[4-(4-Chloro-phenyl)-3,6-dihydro-2H-pyridin-1-yl...)
Affinity DataIC50: 495nMAssay Description:Binding affinity against sigma receptor in bovine cerebellum using 2.0 nM [3H]haloperidol in the presence of 25 nM unlabeled spiperoneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSigma non-opioid intracellular receptor 1(Human)
New York University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50036714BDBM50036714(3-[4-(4-Chloro-phenyl)-3,6-dihydro-2H-pyridin-1-yl...)
Affinity DataIC50: 500nMAssay Description:Binding affinity against sigma receptor in bovine cerebellum using 2.0 nM [3H]haloperidol in the presence of 25 nM unlabeled spiperoneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSigma non-opioid intracellular receptor 1(Human)
New York University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50036718BDBM50036718(CHEMBL1901802 | 4-phenyl-1,2,3,6-tetrahydropyridin...)
Affinity DataIC50: 1.00E+3nMAssay Description:Binding affinity against sigma receptor in bovine cerebellum using 2.0 nM [3H]haloperidol in the presence of 25 nM unlabeled spiperoneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Bovine)
New York University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50002218BDBM50002218(CHEMBL42228 | CHEMBL543412 | 2-(1-Cyclopropylmethy...)
Affinity DataKi: >1.00E+3nMAssay Description:Binding affinity against Dopamine receptor D2 in bovine striatal homogenate using 200 pM [3H]- spiperone and 250 nM unlabeled ketanserinMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Bovine)
New York University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50002245BDBM50002245(CHEMBL130356 | CHEMBL137776 | 4-[2-(1-Cyclopropylm...)
Affinity DataKi: >1.00E+3nMAssay Description:Binding affinity against Dopamine receptor D2 in bovine striatal homogenate using 200 pM [3H]- spiperone and 250 nM unlabeled ketanserinMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSigma non-opioid intracellular receptor 1(Human)
New York University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50036727BDBM50036727(3-Dipropylamino-1-phenyl-propan-1-one | CHEMBL1267...)
Affinity DataIC50: 1.25E+3nMAssay Description:Binding affinity against sigma receptor in bovine cerebellum using 2.0 nM [3H]haloperidol in the presence of 25 nM unlabeled spiperoneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSigma non-opioid intracellular receptor 1(Human)
New York University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50036715BDBM50036715(3-Diethylamino-1-phenyl-propan-1-one | CHEMBL13052...)
Affinity DataIC50: 1.25E+3nMAssay Description:Binding affinity against sigma receptor in bovine cerebellum using 2.0 nM [3H]haloperidol in the presence of 25 nM unlabeled spiperoneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSigma non-opioid intracellular receptor 1(Human)
New York University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50036731BDBM50036731(3-Dimethylamino-1-phenyl-propan-1-one | CHEMBL5011...)
Affinity DataIC50: 5.00E+3nMAssay Description:Binding affinity against sigma receptor in bovine cerebellum using 2.0 nM [3H]haloperidol in the presence of 25 nM unlabeled spiperoneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Bovine)
New York University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50036712BDBM50036712(CHEMBL101664 | CHEMBL2011566 | 4-(4-Chloro-phenyl)...)
Affinity DataIC50: 5.00E+3nMAssay Description:Binding affinity against Dopamine receptor D2 in bovine striatal homogenate using 200 pM [3H]- spiperone and 250 nM unlabeled ketanserinMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Bovine)
New York University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50036718BDBM50036718(CHEMBL1901802 | 4-phenyl-1,2,3,6-tetrahydropyridin...)
Affinity DataIC50: 5.00E+3nMAssay Description:Binding affinity against Dopamine receptor D2 in bovine striatal homogenate using 200 pM [3H]- spiperone and 250 nM unlabeled ketanserinMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Bovine)
New York University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50036710BDBM50036710(3-[4-(4-Chloro-phenyl)-3,6-dihydro-2H-pyridin-1-yl...)
Affinity DataIC50: 5.00E+3nMAssay Description:Binding affinity against Dopamine receptor D2 in bovine striatal homogenate using 200 pM [3H]- spiperone and 250 nM unlabeled ketanserinMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Bovine)
New York University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50036720BDBM50036720(1-Benzo[1,3]dioxol-5-yl-3-[4-(4-chloro-phenyl)-3,6...)
Affinity DataIC50: 5.00E+3nMAssay Description:Binding affinity against Dopamine receptor D2 in bovine striatal homogenate using 200 pM [3H]- spiperone and 250 nM unlabeled ketanserinMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Bovine)
New York University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50036727BDBM50036727(3-Dipropylamino-1-phenyl-propan-1-one | CHEMBL1267...)
Affinity DataIC50: 5.00E+3nMAssay Description:Binding affinity against Dopamine receptor D2 in bovine striatal homogenate using 200 pM [3H]- spiperone and 250 nM unlabeled ketanserinMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Bovine)
New York University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50036719BDBM50036719(1-(4-Chloro-phenyl)-3-[4-(4-chloro-phenyl)-3,6-dih...)
Affinity DataIC50: 5.00E+3nMAssay Description:Binding affinity against Dopamine receptor D2 in bovine striatal homogenate using 200 pM [3H]- spiperone and 250 nM unlabeled ketanserinMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Bovine)
New York University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50036717BDBM50036717(3-[4-(4-Chloro-phenyl)-3,6-dihydro-2H-pyridin-1-yl...)
Affinity DataIC50: 5.00E+3nMAssay Description:Binding affinity against Dopamine receptor D2 in bovine striatal homogenate using 200 pM [3H]- spiperone and 250 nM unlabeled ketanserinMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Bovine)
New York University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50036729BDBM50036729(1-Phenyl-3-(4-phenyl-piperidin-1-yl)-propan-1-one ...)
Affinity DataIC50: 5.00E+3nMAssay Description:Binding affinity against Dopamine receptor D2 in bovine striatal homogenate using 200 pM [3H]- spiperone and 250 nM unlabeled ketanserinMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Bovine)
New York University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50036721BDBM50036721(3-[4-(4-Chloro-phenyl)-3,6-dihydro-2H-pyridin-1-yl...)
Affinity DataIC50: 5.00E+3nMAssay Description:Binding affinity against Dopamine receptor D2 in bovine striatal homogenate using 200 pM [3H]- spiperone and 250 nM unlabeled ketanserinMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Bovine)
New York University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50036714BDBM50036714(3-[4-(4-Chloro-phenyl)-3,6-dihydro-2H-pyridin-1-yl...)
Affinity DataIC50: 5.00E+3nMAssay Description:Binding affinity against Dopamine receptor D2 in bovine striatal homogenate using 200 pM [3H]- spiperone and 250 nM unlabeled ketanserinMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Bovine)
New York University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50036723BDBM50036723(1-(4-Bromo-phenyl)-3-[4-(4-chloro-phenyl)-3,6-dihy...)
Affinity DataIC50: 5.00E+3nMAssay Description:Binding affinity against Dopamine receptor D2 in bovine striatal homogenate using 200 pM [3H]- spiperone and 250 nM unlabeled ketanserinMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Bovine)
New York University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50036722BDBM50036722(3-[4-(4-Fluoro-phenyl)-3,6-dihydro-2H-pyridin-1-yl...)
Affinity DataIC50: 5.00E+3nMAssay Description:Binding affinity against Dopamine receptor D2 in bovine striatal homogenate using 200 pM [3H]- spiperone and 250 nM unlabeled ketanserinMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Bovine)
New York University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50036715BDBM50036715(3-Diethylamino-1-phenyl-propan-1-one | CHEMBL13052...)
Affinity DataIC50: 5.00E+3nMAssay Description:Binding affinity against Dopamine receptor D2 in bovine striatal homogenate using 200 pM [3H]- spiperone and 250 nM unlabeled ketanserinMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Bovine)
New York University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50036726BDBM50036726(3-[4-(4-Chloro-phenyl)-3,6-dihydro-2H-pyridin-1-yl...)
Affinity DataIC50: 5.00E+3nMAssay Description:Binding affinity against Dopamine receptor D2 in bovine striatal homogenate using 200 pM [3H]- spiperone and 250 nM unlabeled ketanserinMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Bovine)
New York University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50036716BDBM50036716(1-Phenyl-3-(4-phenyl-3,6-dihydro-2H-pyridin-1-yl)-...)
Affinity DataIC50: 5.00E+3nMAssay Description:Binding affinity against Dopamine receptor D2 in bovine striatal homogenate using 200 pM [3H]- spiperone and 250 nM unlabeled ketanserinMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Bovine)
New York University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50036731BDBM50036731(3-Dimethylamino-1-phenyl-propan-1-one | CHEMBL5011...)
Affinity DataIC50: 5.00E+3nMAssay Description:Binding affinity against Dopamine receptor D2 in bovine striatal homogenate using 200 pM [3H]- spiperone and 250 nM unlabeled ketanserinMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Bovine)
New York University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50036730BDBM50036730(3-[4-(4-Chloro-phenyl)-3,6-dihydro-2H-pyridin-1-yl...)
Affinity DataIC50: 5.00E+3nMAssay Description:Binding affinity against Dopamine receptor D2 in bovine striatal homogenate using 200 pM [3H]- spiperone and 250 nM unlabeled ketanserinMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Bovine)
New York University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50036711BDBM50036711(1-(4-Fluoro-phenyl)-3-[4-(4-fluoro-phenyl)-3,6-dih...)
Affinity DataIC50: 1.00E+4nMAssay Description:Binding affinity against Dopamine receptor D2 in bovine striatal homogenate using 200 pM [3H]- spiperone and 250 nM unlabeled ketanserinMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Bovine)
New York University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50036713BDBM50036713(1-(4-Bromo-phenyl)-3-[4-(4-fluoro-phenyl)-3,6-dihy...)
Affinity DataIC50: 1.30E+4nMAssay Description:Binding affinity against Dopamine receptor D2 in bovine striatal homogenate using 200 pM [3H]- spiperone and 250 nM unlabeled ketanserinMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Bovine)
New York University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50036724BDBM50036724(1-(4-Chloro-phenyl)-3-[4-(4-fluoro-phenyl)-3,6-dih...)
Affinity DataIC50: 1.50E+4nMAssay Description:Binding affinity against Dopamine receptor D2 in bovine striatal homogenate using 200 pM [3H]- spiperone and 250 nM unlabeled ketanserinMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed