Compile Data Set for Download or QSAR
Report error Found 55 Enz. Inhib. hit(s) with all data for entry = 50005523
TargetGastrin/cholecystokinin type B receptor(Human)
Pfizer

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50037869BDBM50037869(N-tert-Butyl-2-{(3R,5R)-3-[3-(3-chloro-phenyl)-ure...)
Affinity DataIC50: 0.600nMAssay Description:In vitro affinity to the cholecystokinin type B receptor in guinea pig cortex assayed using [125I]BH-CCK-8 as radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGastrin/cholecystokinin type B receptor(Human)
Pfizer

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50037849BDBM50037849(N-tert-Butyl-2-{(3R,5R)-3-[3-(3-chloro-phenyl)-ure...)
Affinity DataIC50: 1nMAssay Description:In vitro affinity to the cholecystokinin type B receptor in guinea pig cortex assayed using [125I]BH-CCK-8 as radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGastrin/cholecystokinin type B receptor(Human)
Pfizer

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50037849BDBM50037849(N-tert-Butyl-2-{(3R,5R)-3-[3-(3-chloro-phenyl)-ure...)
Affinity DataIC50: 1nMAssay Description:In vitro affinity to the cholecystokinin type B receptor in guinea pig cortex assayed using [125I]BH-CCK-8 as radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGastrin/cholecystokinin type B receptor(Human)
Pfizer

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50037866BDBM50037866(N-tert-Butyl-2-{(3R,5R)-3-[3-(3-chloro-phenyl)-ure...)
Affinity DataIC50: 1.07nMAssay Description:In vitro affinity to the cholecystokinin type B receptor in guinea pig cortex assayed using [125I]BH-CCK-8 as radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGastrin/cholecystokinin type B receptor(Human)
Pfizer

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50037871BDBM50037871(2-{(3R,5S)-5-Benzyl-3-[3-(3-chloro-phenyl)-ureido]...)
Affinity DataIC50: 1.40nMAssay Description:In vitro affinity to the cholecystokinin type B receptor in guinea pig cortex assayed using [125I]BH-CCK-8 as radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGastrin/cholecystokinin type B receptor(Human)
Pfizer

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50037867BDBM50037867(N-tert-Butyl-2-{(3R,5R)-3-[3-(3-chloro-phenyl)-ure...)
Affinity DataIC50: 1.5nMAssay Description:In vitro affinity to the cholecystokinin type B receptor in guinea pig cortex assayed using [125I]BH-CCK-8 as radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGastrin/cholecystokinin type B receptor(Human)
Pfizer

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50037847BDBM50037847(N-tert-Butyl-2-{(3R,5R)-3-[3-(3-chloro-phenyl)-ure...)
Affinity DataIC50: 2nMAssay Description:In vitro affinity to the cholecystokinin type B receptor in guinea pig cortex assayed using [125I]BH-CCK-8 as radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGastrin/cholecystokinin type B receptor(Human)
Pfizer

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50037864BDBM50037864(N-tert-Butyl-2-{(3R,5R)-3-[3-(3-chloro-phenyl)-ure...)
Affinity DataIC50: 2.20nMAssay Description:In vitro affinity to the cholecystokinin type B receptor in guinea pig cortex assayed using [125I]BH-CCK-8 as radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGastrin/cholecystokinin type B receptor(Human)
Pfizer

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50037853BDBM50037853({(3R,5R)-3-[3-(3-Chloro-phenyl)-ureido]-8-methyl-2...)
Affinity DataIC50: 2.20nMAssay Description:In vitro affinity to the cholecystokinin type B receptor in guinea pig cortex assayed using [125I]BH-CCK-8 as radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGastrin/cholecystokinin type B receptor(Human)
Pfizer

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50037870BDBM50037870([(3R,5R)-2-Oxo-5-phenyl-3-(3-m-tolyl-ureido)-2,3,4...)
Affinity DataIC50: 2.5nMAssay Description:In vitro affinity to the cholecystokinin type B receptor in guinea pig cortex assayed using [125I]BH-CCK-8 as radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGastrin/cholecystokinin type B receptor(Human)
Pfizer

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50037856BDBM50037856(N-tert-Butyl-2-{(3R,5R)-3-[3-(3-chloro-phenyl)-ure...)
Affinity DataIC50: 3.40nMAssay Description:In vitro affinity to the cholecystokinin type B receptor in guinea pig cortex assayed using [125I]BH-CCK-8 as radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGastrin/cholecystokinin type B receptor(Human)
Pfizer

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50037863BDBM50037863(2-{(3R,5R)-3-[3-(3-Chloro-phenyl)-ureido]-2-oxo-5-...)
Affinity DataIC50: 3.80nMAssay Description:In vitro affinity to the cholecystokinin type B receptor in guinea pig cortex assayed using [125I]BH-CCK-8 as radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGastrin/cholecystokinin type B receptor(Human)
Pfizer

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50037854BDBM50037854(N-tert-Butyl-2-{(3R,5R)-5-(3-chloro-phenyl)-3-[3-(...)
Affinity DataIC50: 4nMAssay Description:In vitro affinity to the cholecystokinin type B receptor in guinea pig cortex assayed using [125I]BH-CCK-8 as radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCholecystokinin receptor type A(Guinea pig)
Pfizer

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50037867BDBM50037867(N-tert-Butyl-2-{(3R,5R)-3-[3-(3-chloro-phenyl)-ure...)
Affinity DataIC50: 4.20nMAssay Description:In vitro binding affinity for the cholecystokinin type A receptor in guinea pig pancreas assayed using [125I]BH-CCK-8 as radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGastrin/cholecystokinin type B receptor(Human)
Pfizer

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50037860BDBM50037860(N-tert-Butyl-2-{(3R,5R)-3-[3-(3-chloro-phenyl)-ure...)
Affinity DataIC50: 4.30nMAssay Description:In vitro affinity to the cholecystokinin type B receptor in guinea pig cortex assayed using [125I]BH-CCK-8 as radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGastrin/cholecystokinin type B receptor(Human)
Pfizer

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50037859BDBM50037859(N-tert-Butyl-2-{(3R,5R)-8-chloro-3-[3-(3-chloro-ph...)
Affinity DataIC50: 6.70nMAssay Description:In vitro affinity to the cholecystokinin type B receptor in guinea pig cortex assayed using [125I]BH-CCK-8 as radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGastrin/cholecystokinin type B receptor(Human)
Pfizer

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50037865BDBM50037865(2-{(3R,5R)-3-[3-(3-Chloro-phenyl)-ureido]-2-oxo-5-...)
Affinity DataIC50: 7.60nMAssay Description:In vitro affinity to the cholecystokinin type B receptor in guinea pig cortex assayed using [125I]BH-CCK-8 as radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGastrin/cholecystokinin type B receptor(Human)
Pfizer

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50037850BDBM50037850(N-tert-Butyl-2-{(3R,5R)-3-[3-(3-chloro-phenyl)-ure...)
Affinity DataIC50: 7.70nMAssay Description:In vitro affinity to the cholecystokinin type B receptor in guinea pig cortex assayed using [125I]BH-CCK-8 as radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGastrin/cholecystokinin type B receptor(Human)
Pfizer

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50006878BDBM50006878(1-(1-Methyl-2-oxo-5-phenyl-2,3-dihydro-1H-benzo[e]...)
Affinity DataIC50: 8.10nMAssay Description:In vitro affinity to the cholecystokinin type B receptor in guinea pig cortex assayed using [125I]BH-CCK-8 as radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGastrin/cholecystokinin type B receptor(Human)
Pfizer

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50037868BDBM50037868(N-tert-Butyl-2-[(3R,5R)-2-oxo-5-phenyl-3-(3-m-toly...)
Affinity DataIC50: 10.1nMAssay Description:In vitro affinity to the cholecystokinin type B receptor in guinea pig cortex assayed using [125I]BH-CCK-8 as radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGastrin/cholecystokinin type B receptor(Human)
Pfizer

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50037857BDBM50037857(2-{(3R,5R)-3-[3-(3-Chloro-phenyl)-ureido]-2-oxo-5-...)
Affinity DataIC50: 10.6nMAssay Description:In vitro affinity to the cholecystokinin type B receptor in guinea pig cortex assayed using [125I]BH-CCK-8 as radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGastrin/cholecystokinin type B receptor(Human)
Pfizer

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50037855BDBM50037855(N-tert-Butyl-2-{(3R,5R)-7-chloro-3-[3-(3-chloro-ph...)
Affinity DataIC50: 24nMAssay Description:In vitro affinity to the cholecystokinin type B receptor in guinea pig cortex assayed using [125I]BH-CCK-8 as radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGastrin/cholecystokinin type B receptor(Human)
Pfizer

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50037851BDBM50037851(N-tert-Butyl-2-{(3R,5R)-3-[3-(3-methoxy-phenyl)-ur...)
Affinity DataIC50: 30.4nMAssay Description:In vitro affinity to the cholecystokinin type B receptor in guinea pig cortex assayed using [125I]BH-CCK-8 as radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGastrin/cholecystokinin type B receptor(Human)
Pfizer

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50037846BDBM50037846(N-tert-Butyl-2-{(3R,5R)-3-[3-(3-chloro-phenyl)-ure...)
Affinity DataIC50: 32nMAssay Description:In vitro affinity to the cholecystokinin type B receptor in guinea pig cortex assayed using [125I]BH-CCK-8 as radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCholecystokinin receptor type A(Guinea pig)
Pfizer

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50037853BDBM50037853({(3R,5R)-3-[3-(3-Chloro-phenyl)-ureido]-8-methyl-2...)
Affinity DataIC50: 34nMAssay Description:In vitro binding affinity for the cholecystokinin type A receptor in guinea pig pancreas assayed using [125I]BH-CCK-8 as radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGastrin/cholecystokinin type B receptor(Human)
Pfizer

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50037852BDBM50037852(N-tert-Butyl-2-[(3R,5R)-2-oxo-5-phenyl-3-(3-p-toly...)
Affinity DataIC50: 35nMAssay Description:In vitro affinity to the cholecystokinin type B receptor in guinea pig cortex assayed using [125I]BH-CCK-8 as radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGastrin/cholecystokinin type B receptor(Human)
Pfizer

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50037861BDBM50037861(N-tert-Butyl-2-{(3S,5S)-3-[3-(3-chloro-phenyl)-ure...)
Affinity DataIC50: 35.7nMAssay Description:In vitro affinity to the cholecystokinin type B receptor in guinea pig cortex assayed using [125I]BH-CCK-8 as radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGastrin/cholecystokinin type B receptor(Human)
Pfizer

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50037858BDBM50037858(N-tert-Butyl-2-{(3R,5R)-3-[3-(4-chloro-phenyl)-ure...)
Affinity DataIC50: 43nMAssay Description:In vitro affinity to the cholecystokinin type B receptor in guinea pig cortex assayed using [125I]BH-CCK-8 as radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCholecystokinin receptor type A(Guinea pig)
Pfizer

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50037870BDBM50037870([(3R,5R)-2-Oxo-5-phenyl-3-(3-m-tolyl-ureido)-2,3,4...)
Affinity DataIC50: 50nMAssay Description:In vitro binding affinity for the cholecystokinin type A receptor in guinea pig pancreas assayed using [125I]BH-CCK-8 as radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGastrin/cholecystokinin type B receptor(Human)
Pfizer

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50037862BDBM50037862(N-tert-Butyl-2-[(3R,5R)-2-oxo-5-phenyl-3-(3-o-toly...)
Affinity DataIC50: 55nMAssay Description:In vitro affinity to the cholecystokinin type B receptor in guinea pig cortex assayed using [125I]BH-CCK-8 as radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCholecystokinin receptor type A(Guinea pig)
Pfizer

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50037854BDBM50037854(N-tert-Butyl-2-{(3R,5R)-5-(3-chloro-phenyl)-3-[3-(...)
Affinity DataIC50: 69nMAssay Description:In vitro binding affinity for the cholecystokinin type A receptor in guinea pig pancreas assayed using [125I]BH-CCK-8 as radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCholecystokinin receptor type A(Guinea pig)
Pfizer

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50037847BDBM50037847(N-tert-Butyl-2-{(3R,5R)-3-[3-(3-chloro-phenyl)-ure...)
Affinity DataIC50: 71nMAssay Description:In vitro binding affinity for the cholecystokinin type A receptor in guinea pig pancreas assayed using [125I]BH-CCK-8 as radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCholecystokinin receptor type A(Guinea pig)
Pfizer

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50037856BDBM50037856(N-tert-Butyl-2-{(3R,5R)-3-[3-(3-chloro-phenyl)-ure...)
Affinity DataIC50: 72nMAssay Description:In vitro binding affinity for the cholecystokinin type A receptor in guinea pig pancreas assayed using [125I]BH-CCK-8 as radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCholecystokinin receptor type A(Guinea pig)
Pfizer

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50037864BDBM50037864(N-tert-Butyl-2-{(3R,5R)-3-[3-(3-chloro-phenyl)-ure...)
Affinity DataIC50: 77nMAssay Description:In vitro binding affinity for the cholecystokinin type A receptor in guinea pig pancreas assayed using [125I]BH-CCK-8 as radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCholecystokinin receptor type A(Guinea pig)
Pfizer

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50006878BDBM50006878(1-(1-Methyl-2-oxo-5-phenyl-2,3-dihydro-1H-benzo[e]...)
Affinity DataIC50: 86nMAssay Description:In vitro binding affinity for the cholecystokinin type A receptor in guinea pig pancreas assayed using [125I]BH-CCK-8 as radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCholecystokinin receptor type A(Guinea pig)
Pfizer

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50037849BDBM50037849(N-tert-Butyl-2-{(3R,5R)-3-[3-(3-chloro-phenyl)-ure...)
Affinity DataIC50: 130nMAssay Description:In vitro binding affinity for the cholecystokinin type A receptor in guinea pig pancreas assayed using [125I]BH-CCK-8 as radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGastrin/cholecystokinin type B receptor(Human)
Pfizer

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50037848BDBM50037848(N-tert-Butyl-2-{(3S,5R)-3-[3-(3-chloro-phenyl)-ure...)
Affinity DataIC50: 130nMAssay Description:In vitro affinity to the cholecystokinin type B receptor in guinea pig cortex assayed using [125I]BH-CCK-8 as radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCholecystokinin receptor type A(Guinea pig)
Pfizer

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50037865BDBM50037865(2-{(3R,5R)-3-[3-(3-Chloro-phenyl)-ureido]-2-oxo-5-...)
Affinity DataIC50: 144nMAssay Description:In vitro binding affinity for the cholecystokinin type A receptor in guinea pig pancreas assayed using [125I]BH-CCK-8 as radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCholecystokinin receptor type A(Guinea pig)
Pfizer

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50037860BDBM50037860(N-tert-Butyl-2-{(3R,5R)-3-[3-(3-chloro-phenyl)-ure...)
Affinity DataIC50: 144nMAssay Description:In vitro binding affinity for the cholecystokinin type A receptor in guinea pig pancreas assayed using [125I]BH-CCK-8 as radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCholecystokinin receptor type A(Guinea pig)
Pfizer

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50037851BDBM50037851(N-tert-Butyl-2-{(3R,5R)-3-[3-(3-methoxy-phenyl)-ur...)
Affinity DataIC50: 166nMAssay Description:In vitro binding affinity for the cholecystokinin type A receptor in guinea pig pancreas assayed using [125I]BH-CCK-8 as radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCholecystokinin receptor type A(Guinea pig)
Pfizer

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50037866BDBM50037866(N-tert-Butyl-2-{(3R,5R)-3-[3-(3-chloro-phenyl)-ure...)
Affinity DataIC50: 171nMAssay Description:In vitro binding affinity for the cholecystokinin type A receptor in guinea pig pancreas assayed using [125I]BH-CCK-8 as radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCholecystokinin receptor type A(Guinea pig)
Pfizer

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50037855BDBM50037855(N-tert-Butyl-2-{(3R,5R)-7-chloro-3-[3-(3-chloro-ph...)
Affinity DataIC50: 287nMAssay Description:In vitro binding affinity for the cholecystokinin type A receptor in guinea pig pancreas assayed using [125I]BH-CCK-8 as radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCholecystokinin receptor type A(Guinea pig)
Pfizer

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50037868BDBM50037868(N-tert-Butyl-2-[(3R,5R)-2-oxo-5-phenyl-3-(3-m-toly...)
Affinity DataIC50: 288nMAssay Description:In vitro binding affinity for the cholecystokinin type A receptor in guinea pig pancreas assayed using [125I]BH-CCK-8 as radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCholecystokinin receptor type A(Guinea pig)
Pfizer

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50037846BDBM50037846(N-tert-Butyl-2-{(3R,5R)-3-[3-(3-chloro-phenyl)-ure...)
Affinity DataIC50: 317nMAssay Description:In vitro binding affinity for the cholecystokinin type A receptor in guinea pig pancreas assayed using [125I]BH-CCK-8 as radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCholecystokinin receptor type A(Guinea pig)
Pfizer

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50037859BDBM50037859(N-tert-Butyl-2-{(3R,5R)-8-chloro-3-[3-(3-chloro-ph...)
Affinity DataIC50: 320nMAssay Description:In vitro binding affinity for the cholecystokinin type A receptor in guinea pig pancreas assayed using [125I]BH-CCK-8 as radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCholecystokinin receptor type A(Guinea pig)
Pfizer

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50037861BDBM50037861(N-tert-Butyl-2-{(3S,5S)-3-[3-(3-chloro-phenyl)-ure...)
Affinity DataIC50: 363nMAssay Description:In vitro binding affinity for the cholecystokinin type A receptor in guinea pig pancreas assayed using [125I]BH-CCK-8 as radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCholecystokinin receptor type A(Guinea pig)
Pfizer

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50037858BDBM50037858(N-tert-Butyl-2-{(3R,5R)-3-[3-(4-chloro-phenyl)-ure...)
Affinity DataIC50: 399nMAssay Description:In vitro binding affinity for the cholecystokinin type A receptor in guinea pig pancreas assayed using [125I]BH-CCK-8 as radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCholecystokinin receptor type A(Guinea pig)
Pfizer

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50037850BDBM50037850(N-tert-Butyl-2-{(3R,5R)-3-[3-(3-chloro-phenyl)-ure...)
Affinity DataIC50: 417nMAssay Description:In vitro binding affinity for the cholecystokinin type A receptor in guinea pig pancreas assayed using [125I]BH-CCK-8 as radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCholecystokinin receptor type A(Guinea pig)
Pfizer

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50037857BDBM50037857(2-{(3R,5R)-3-[3-(3-Chloro-phenyl)-ureido]-2-oxo-5-...)
Affinity DataIC50: 460nMAssay Description:In vitro binding affinity for the cholecystokinin type A receptor in guinea pig pancreas assayed using [125I]BH-CCK-8 as radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCholecystokinin receptor type A(Guinea pig)
Pfizer

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50037863BDBM50037863(2-{(3R,5R)-3-[3-(3-Chloro-phenyl)-ureido]-2-oxo-5-...)
Affinity DataIC50: 467nMAssay Description:In vitro binding affinity for the cholecystokinin type A receptor in guinea pig pancreas assayed using [125I]BH-CCK-8 as radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
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