TargetSigma non-opioid intracellular receptor 1(Homo sapiens (Human))
George Washington University Medical Center
Curated by ChEMBL
George Washington University Medical Center
Curated by ChEMBL
Affinity DataKi: 1.64nMAssay Description:Binding affinity against sigma-1 receptor in guinea pig brain using [3H]-(+)-pentazocine as radioligand.More data for this Ligand-Target Pair
TargetSigma non-opioid intracellular receptor 1(Homo sapiens (Human))
George Washington University Medical Center
Curated by ChEMBL
George Washington University Medical Center
Curated by ChEMBL
Affinity DataKi: 1.70nMAssay Description:Binding affinity against sigma-1 receptor in guinea pig brain using [3H]-(+)-pentazocine as radioligand.More data for this Ligand-Target Pair
TargetSigma non-opioid intracellular receptor 1(Homo sapiens (Human))
George Washington University Medical Center
Curated by ChEMBL
George Washington University Medical Center
Curated by ChEMBL
Affinity DataKi: 3.02nMAssay Description:Binding affinity against sigma-1 receptor in guinea pig brain using [3H]-(+)-pentazocine as radioligandMore data for this Ligand-Target Pair
TargetSigma non-opioid intracellular receptor 1(Homo sapiens (Human))
George Washington University Medical Center
Curated by ChEMBL
George Washington University Medical Center
Curated by ChEMBL
Affinity DataKi: 4.60nMAssay Description:Binding affinity against sigma receptor of MCF cellsMore data for this Ligand-Target Pair
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
George Washington University Medical Center
Curated by ChEMBL
George Washington University Medical Center
Curated by ChEMBL
Affinity DataKi: 24.8nMAssay Description:Binding affinity against D-2 dopamine receptor in rat brain membranes using [3H]-(-)-sulpiride as radioligand.More data for this Ligand-Target Pair
TargetSigma non-opioid intracellular receptor 1(Homo sapiens (Human))
George Washington University Medical Center
Curated by ChEMBL
George Washington University Medical Center
Curated by ChEMBL
Affinity DataKi: 60nMAssay Description:Binding affinity against sigma receptor of MCF cellsMore data for this Ligand-Target Pair
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
George Washington University Medical Center
Curated by ChEMBL
George Washington University Medical Center
Curated by ChEMBL
Affinity DataKi: 63.4nMAssay Description:Binding affinity against D-2 dopamine receptor in rat brain membranes using [3H]-(-)-sulpiride as radioligand.More data for this Ligand-Target Pair
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
George Washington University Medical Center
Curated by ChEMBL
George Washington University Medical Center
Curated by ChEMBL
Affinity DataKi: 382nMAssay Description:Binding affinity against D-2 dopamine receptor in rat brain membranes using [3H]-(-)-sulpiride as radioligand.More data for this Ligand-Target Pair
TargetSigma non-opioid intracellular receptor 1(Homo sapiens (Human))
George Washington University Medical Center
Curated by ChEMBL
George Washington University Medical Center
Curated by ChEMBL
Affinity DataKd: 38.2nMAssay Description:Binding affinity against MCF cells in the membrane preparation using radioligand binding assay.More data for this Ligand-Target Pair