Compile Data Set for Download or QSAR
Report error Found 25 Enz. Inhib. hit(s) with all data for entry = 50005623
TargetAmine oxidase [flavin-containing] A(Rat)
Burroughs Wellcome

Curated by ChEMBL
LigandPNGBDBM50038938(N-(6-Ethyl-9,10,10-trioxo-9,10-dihydro-10lambda*6*...)
Affinity DataIC50: 10nMAssay Description:Inhibitory activity against monoamine oxidase A (MAO A) from rat brain using a radiometric procedure with [3H]5-HTMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAmine oxidase [flavin-containing] A(Rat)
Burroughs Wellcome

Curated by ChEMBL
LigandPNGBDBM50038947(N-(10,10-Dioxo-10H-10lambda*6*-phenoxathiin-2-yl)-...)
Affinity DataIC50: 14nMAssay Description:Inhibitory activity against monoamine oxidase A (MAO A) from rat brain using a radiometric procedure with [3H]5-HTMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAmine oxidase [flavin-containing] A(Rat)
Burroughs Wellcome

Curated by ChEMBL
LigandPNGBDBM50038946(N-(9,10,10-Trioxo-6-propyl-9,10-dihydro-10lambda*6...)
Affinity DataIC50: 20nMAssay Description:Inhibitory activity against monoamine oxidase A (MAO A) from rat brain using a radiometric procedure with [3H]5-HTMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAmine oxidase [flavin-containing] A(Rat)
Burroughs Wellcome

Curated by ChEMBL
LigandPNGBDBM50038936(N-(9-Methyl-9H-carbazol-2-yl)-acetamide | CHEMBL63...)
Affinity DataIC50: 30nMAssay Description:Inhibitory activity against monoamine oxidase A (MAO A) from rat brain using a radiometric procedure with [3H]5-HTMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAmine oxidase [flavin-containing] A(Rat)
Burroughs Wellcome

Curated by ChEMBL
LigandPNGBDBM50038928(N-(6-Oxo-6H-benzo[c]chromen-3-yl)-acetamide | CHEM...)
Affinity DataIC50: 40nMAssay Description:Inhibitory activity against monoamine oxidase A (MAO A) from rat brain using a radiometric procedure with [3H]- serotonin.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAmine oxidase [flavin-containing] A(Rat)
Burroughs Wellcome

Curated by ChEMBL
LigandPNGBDBM50038930(N-(9-Oxo-9H-fluoren-2-yl)-acetamide | CHEMBL417970)
Affinity DataIC50: 40nMAssay Description:Inhibitory activity against monoamine oxidase A (MAO A) from rat brain using a radiometric procedure with [3H]5-HTMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAmine oxidase [flavin-containing] A(Rat)
Burroughs Wellcome

Curated by ChEMBL
LigandPNGBDBM50038944(N-(9H-Carbazol-2-yl)-acetamide | CHEMBL63669)
Affinity DataIC50: 43nMAssay Description:Inhibitory activity against monoamine oxidase A (MAO A) from rat brain using a radiometric procedure with [3H]- serotonin.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAmine oxidase [flavin-containing] A(Rat)
Burroughs Wellcome

Curated by ChEMBL
LigandPNGBDBM50038942(N-(9,10,10-Trioxo-9,10-dihydro-10lambda*6*-thioxan...)
Affinity DataIC50: 60nMAssay Description:Inhibitory activity against monoamine oxidase A (MAO A) from rat brain using a radiometric procedure with [3H]5-HTMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAmine oxidase [flavin-containing] A(Rat)
Burroughs Wellcome

Curated by ChEMBL
LigandPNGBDBM50038934(N-(9,10,10-Trioxo-9,10-dihydro-10lambda*6*-thioxan...)
Affinity DataIC50: 120nMAssay Description:Inhibitory activity against monoamine oxidase A (MAO A) from rat brain using a radiometric procedure with [3H]5-HTMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAmine oxidase [flavin-containing] A(Rat)
Burroughs Wellcome

Curated by ChEMBL
LigandPNGBDBM50038932(N-(9,10-Dioxo-9,10-dihydro-anthracen-2-yl)-acetami...)
Affinity DataIC50: 160nMAssay Description:Inhibitory activity against monoamine oxidase A (MAO A) from rat brain using a radiometric procedure with [3H]- serotonin.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAmine oxidase [flavin-containing] A(Rat)
Burroughs Wellcome

Curated by ChEMBL
LigandPNGBDBM50038937(N-(5,5-Dioxo-5H-5lambda*6*-dibenzothiophen-2-yl)-a...)
Affinity DataIC50: 260nMAssay Description:Inhibitory activity against monoamine oxidase A (MAO A) from rat brain using a radiometric procedure with [3H]5-HTMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAmine oxidase [flavin-containing] A(Rat)
Burroughs Wellcome

Curated by ChEMBL
LigandPNGBDBM50038929(N-(9-Hydroxy-9H-fluoren-2-yl)-acetamide | CHEMBL30...)
Affinity DataIC50: 300nMAssay Description:Inhibitory activity against monoamine oxidase A (MAO A) from rat brain using a radiometric procedure with [3H]5-HTMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAmine oxidase [flavin-containing] A(Rat)
Burroughs Wellcome

Curated by ChEMBL
LigandPNGBDBM50038935(N-Dibenzofuran-3-yl-acetamide | CHEMBL63423)
Affinity DataIC50: 300nMAssay Description:Inhibitory activity against monoamine oxidase A (MAO A) from rat brain using a radiometric procedure with [3H]5-HTMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAmine oxidase [flavin-containing] A(Rat)
Burroughs Wellcome

Curated by ChEMBL
LigandPNGBDBM50038941(N-(6-Methyl-9,10,10-trioxo-9,10-dihydro-10lambda*6...)
Affinity DataIC50: 700nMAssay Description:Inhibitory activity against monoamine oxidase A (MAO A) from rat brain using a radiometric procedure with [3H]5-HTMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAmine oxidase [flavin-containing] A(Rat)
Burroughs Wellcome

Curated by ChEMBL
LigandPNGBDBM50038933(5,5-Dioxo-5H-5lambda*6*-dibenzothiophen-2-ylamine ...)
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibitory activity against monoamine oxidase A (MAO A) from rat brain using a radiometric procedure with [3H]5-HTMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAmine oxidase [flavin-containing] A(Rat)
Burroughs Wellcome

Curated by ChEMBL
LigandPNGBDBM50038931(N-(5,5-Dioxo-5H-5lambda*6*-dibenzothiophen-2-yl)-f...)
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibitory activity against monoamine oxidase A (MAO A) from rat brain using a radiometric procedure with [3H]5-HTMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAmine oxidase [flavin-containing] A(Rat)
Burroughs Wellcome

Curated by ChEMBL
LigandPNGBDBM50038945(N-(9H-Carbazol-2-yl)-formamide | CHEMBL440488)
Affinity DataIC50: 1.10E+3nMAssay Description:Inhibitory activity against monoamine oxidase A (MAO A) from rat brain using a radiometric procedure with [3H]5-HTMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAmine oxidase [flavin-containing] A(Rat)
Burroughs Wellcome

Curated by ChEMBL
LigandPNGBDBM50038949(N-(5,5-Dioxo-5H-5lambda*6*-dibenzothiophen-2-yl)-p...)
Affinity DataIC50: 1.20E+3nMAssay Description:Inhibitory activity against monoamine oxidase A (MAO A) from rat brain using a radiometric procedure with [3H]5-HTMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAmine oxidase [flavin-containing] A(Rat)
Burroughs Wellcome

Curated by ChEMBL
LigandPNGBDBM50038940(N-(7-Nitro-9-oxo-9H-fluoren-2-yl)-acetamide | CHEM...)
Affinity DataIC50: 1.30E+3nMAssay Description:Inhibitory activity against monoamine oxidase A (MAO A) from rat brain using a radiometric procedure with [3H]5-HTMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAmine oxidase [flavin-containing] A(Rat)
Burroughs Wellcome

Curated by ChEMBL
LigandPNGBDBM50038943(N-(7-Acetylamino-10-methyl-5,5-dioxo-5,10-dihydro-...)
Affinity DataIC50: 2.00E+3nMAssay Description:Inhibitory activity against monoamine oxidase A (MAO A) from rat brain using a radiometric procedure with [3H]5-HT at 1 uMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAmine oxidase [flavin-containing] B(Rat)
Burroughs Wellcome

Curated by ChEMBL
LigandPNGBDBM50038932(N-(9,10-Dioxo-9,10-dihydro-anthracen-2-yl)-acetami...)
Affinity DataIC50: 3.50E+3nMAssay Description:Inhibitory activity against monoamine oxidase B (MAO B) from rat brain using a radiometric procedure with [14C]- phenethylamine.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAmine oxidase [flavin-containing] B(Rat)
Burroughs Wellcome

Curated by ChEMBL
LigandPNGBDBM50038943(N-(7-Acetylamino-10-methyl-5,5-dioxo-5,10-dihydro-...)
Affinity DataIC50: 7.00E+3nMAssay Description:Inhibitory activity against monoamine oxidase B (MAO B) from rat brain using a radiometric procedure with [14C]phenylethylamine at 1 uMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAmine oxidase [flavin-containing] B(Rat)
Burroughs Wellcome

Curated by ChEMBL
LigandPNGBDBM50038939(N-(5,5-Dioxo-5,10-dihydro-5lambda*6*-phenothiazin-...)
Affinity DataIC50: 2.20E+4nMAssay Description:Inhibitory activity against monoamine oxidase B (MAO B) from rat brain using a radiometric procedure with [14C]phenylethylamine at 10 uMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAmine oxidase [flavin-containing] B(Rat)
Burroughs Wellcome

Curated by ChEMBL
LigandPNGBDBM50038948(N-(2,3-Dimethyl-1H-indol-5-yl)-acetamide | CHEMBL2...)
Affinity DataIC50: 4.20E+4nMAssay Description:Inhibitory activity against monoamine oxidase B (MAO B) from rat brain using a radiometric procedure with [14C]phenylethylamine at 1 uMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAmine oxidase [flavin-containing] A(Rat)
Burroughs Wellcome

Curated by ChEMBL
LigandPNGBDBM50038939(N-(5,5-Dioxo-5,10-dihydro-5lambda*6*-phenothiazin-...)
Affinity DataIC50: 7.40E+4nMAssay Description:Inhibitory activity against monoamine oxidase A (MAO A) from rat brain using a radiometric procedure with [3H]5-HT at 10 uMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed