Compile Data Set for Download or QSAR
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Report error Found 43 Enz. Inhib. hit(s) with all data for entry = 50036266
Target5-hydroxytryptamine receptor 1A(Rat)
Solvay Duphar Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50020178(CHEMBL294633 | CHEMBL555633 | N-[2-(4-Benzofuran-7...)
Affinity DataKi:  0.150nMAssay Description:Binding affinity to displace [3H]2-(di-N-propylamino)-8-hydroxy-tetralin from 5-hydroxytryptamine 1A (5-HT1A) receptor in rat frontal cortex homogena...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

Target5-hydroxytryptamine receptor 1A(Rat)
Solvay Duphar Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50039829(CHEMBL92242 | Cyclohexanecarboxylic acid [2-(4-ben...)
Affinity DataKi:  0.200nMAssay Description:Binding affinity to displace [3H]2-(di-N-propylamino)-8-hydroxy-tetralin from 5-hydroxytryptamine 1A (5-HT1A) receptor in rat frontal cortex homogena...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

Target5-hydroxytryptamine receptor 1A(Rat)
Solvay Duphar Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50039822(1-(2-Cyclohexyl-ethyl)-4-(2,3-dihydro-benzo[1,4]di...)
Affinity DataKi:  0.25nMAssay Description:Binding affinity to displace [3H]2-(di-N-propylamino)-8-hydroxy-tetralin from 5-hydroxytryptamine 1A (5-HT1A) receptor in rat frontal cortex homogena...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

Target5-hydroxytryptamine receptor 1A(Rat)
Solvay Duphar Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50039824(CHEMBL81728 | N-{2-[4-(2,3-Dihydro-benzo[1,4]dioxi...)
Affinity DataKi:  0.300nMAssay Description:Binding affinity to displace [3H]2-(di-N-propylamino)-8-hydroxy-tetralin from 5-hydroxytryptamine 1A (5-HT1A) receptor in rat frontal cortex homogena...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

Target5-hydroxytryptamine receptor 1A(Rat)
Solvay Duphar Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50039818(1-(2,3-Dihydro-benzo[1,4]dioxin-5-yl)-4-(4-phenyl-...)
Affinity DataKi:  0.320nMAssay Description:Binding affinity to displace [3H]2-(di-N-propylamino)-8-hydroxy-tetralin from 5-hydroxytryptamine 1A (5-HT1A) receptor in rat frontal cortex homogena...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

Target5-hydroxytryptamine receptor 1A(Rat)
Solvay Duphar Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50039798(1-Benzofuran-7-yl-4-phenethyl-piperazine; hydrochl...)
Affinity DataKi:  0.370nMAssay Description:Binding affinity to displace [3H]2-(di-N-propylamino)-8-hydroxy-tetralin from 5-hydroxytryptamine 1A (5-HT1A) receptor in rat frontal cortex homogena...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

Target5-hydroxytryptamine receptor 1A(Rat)
Solvay Duphar Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50039821(CHEMBL93421 | Cyclohexanecarboxylic acid {2-[4-(2,...)
Affinity DataKi:  0.440nMAssay Description:Binding affinity to displace [3H]2-(di-N-propylamino)-8-hydroxy-tetralin from 5-hydroxytryptamine 1A (5-HT1A) receptor in rat frontal cortex homogena...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

Target5-hydroxytryptamine receptor 1A(Rat)
Solvay Duphar Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50039810(1-Benzofuran-7-yl-4-(2-phenoxy-ethyl)-piperazine; ...)
Affinity DataKi:  0.460nMAssay Description:Binding affinity to displace [3H]2-(di-N-propylamino)-8-hydroxy-tetralin from 5-hydroxytryptamine 1A (5-HT1A) receptor in rat frontal cortex homogena...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

Target5-hydroxytryptamine receptor 1A(Rat)
Solvay Duphar Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50039800(1-(2,3-Dihydro-benzo[1,4]dioxin-5-yl)-4-phenethyl-...)
Affinity DataKi:  0.470nMAssay Description:Binding affinity to displace [3H]2-(di-N-propylamino)-8-hydroxy-tetralin from 5-hydroxytryptamine 1A (5-HT1A) receptor in rat frontal cortex homogena...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

Target5-hydroxytryptamine receptor 1A(Rat)
Solvay Duphar Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50039819(1-(2,3-Dihydro-benzo[1,4]dioxin-5-yl)-4-hexyl-pipe...)
Affinity DataKi:  0.5nMAssay Description:Binding affinity to displace [3H]2-(di-N-propylamino)-8-hydroxy-tetralin from 5-hydroxytryptamine 1A (5-HT1A) receptor in rat frontal cortex homogena...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

Target5-hydroxytryptamine receptor 1A(Rat)
Solvay Duphar Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50039805(1-Benzofuran-7-yl-4-hexyl-piperazine | CHEMBL27558)
Affinity DataKi:  0.540nMAssay Description:Binding affinity to displace [3H]2-(di-N-propylamino)-8-hydroxy-tetralin from 5-hydroxytryptamine 1A (5-HT1A) receptor in rat frontal cortex homogena...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

Target5-hydroxytryptamine receptor 1A(Rat)
Solvay Duphar Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50039796(1-(2,3-Dihydro-benzo[1,4]dioxin-5-yl)-4-octyl-pipe...)
Affinity DataKi:  0.610nMAssay Description:Binding affinity to displace [3H]2-(di-N-propylamino)-8-hydroxy-tetralin from 5-hydroxytryptamine 1A (5-HT1A) receptor in rat frontal cortex homogena...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

Target5-hydroxytryptamine receptor 1A(Rat)
Solvay Duphar Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50039814(4-[4-(2,3-Dihydro-benzo[1,4]dioxin-5-yl)-piperazin...)
Affinity DataKi:  0.670nMAssay Description:Binding affinity to displace [3H]2-(di-N-propylamino)-8-hydroxy-tetralin from 5-hydroxytryptamine 1A (5-HT1A) receptor in rat frontal cortex homogena...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

Target5-hydroxytryptamine receptor 1A(Rat)
Solvay Duphar Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50039807(1-(2,3-Dihydro-benzo[1,4]dioxin-5-yl)-4-(2-phenoxy...)
Affinity DataKi:  0.730nMAssay Description:Binding affinity to displace [3H]2-(di-N-propylamino)-8-hydroxy-tetralin from 5-hydroxytryptamine 1A (5-HT1A) receptor in rat frontal cortex homogena...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

Target5-hydroxytryptamine receptor 1A(Rat)
Solvay Duphar Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50039795(1-Benzofuran-7-yl-4-pentyl-piperazine | CHEMBL2683...)
Affinity DataKi:  0.810nMAssay Description:Binding affinity to displace [3H]2-(di-N-propylamino)-8-hydroxy-tetralin from 5-hydroxytryptamine 1A (5-HT1A) receptor in rat frontal cortex homogena...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

Target5-hydroxytryptamine receptor 1A(Rat)
Solvay Duphar Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50039802(1-Benzofuran-7-yl-4-(3-phenoxy-propyl)-piperazine;...)
Affinity DataKi:  0.850nMAssay Description:Binding affinity to displace [3H]2-(di-N-propylamino)-8-hydroxy-tetralin from 5-hydroxytryptamine 1A (5-HT1A) receptor in rat frontal cortex homogena...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

Target5-hydroxytryptamine receptor 1A(Rat)
Solvay Duphar Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50039827(1-(2,3-Dihydro-benzo[1,4]dioxin-5-yl)-4-(3-phenoxy...)
Affinity DataKi:  0.950nMAssay Description:Binding affinity to displace [3H]2-(di-N-propylamino)-8-hydroxy-tetralin from 5-hydroxytryptamine 1A (5-HT1A) receptor in rat frontal cortex homogena...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

Target5-hydroxytryptamine receptor 1A(Rat)
Solvay Duphar Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50039826(1-Decyl-4-(2,3-dihydro-benzo[1,4]dioxin-5-yl)-pipe...)
Affinity DataKi:  1nMAssay Description:Binding affinity to displace [3H]2-(di-N-propylamino)-8-hydroxy-tetralin from 5-hydroxytryptamine 1A (5-HT1A) receptor in rat frontal cortex homogena...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

Target5-hydroxytryptamine receptor 1A(Rat)
Solvay Duphar Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50020180(4-(4-Benzofuran-7-yl-piperazin-1-yl)-1-(4-fluoro-p...)
Affinity DataKi:  1nMAssay Description:Binding affinity to displace [3H]2-(di-N-propylamino)-8-hydroxy-tetralin from 5-hydroxytryptamine 1A (5-HT1A) receptor in rat frontal cortex homogena...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

Target5-hydroxytryptamine receptor 1A(Rat)
Solvay Duphar Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50039811(4-[4-(2,3-Dihydro-benzo[1,4]dioxin-5-yl)-piperazin...)
Affinity DataKi:  1.40nMAssay Description:Binding affinity to displace [3H]2-(di-N-propylamino)-8-hydroxy-tetralin from 5-hydroxytryptamine 1A (5-HT1A) receptor in rat frontal cortex homogena...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

Target5-hydroxytryptamine receptor 1A(Rat)
Solvay Duphar Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50039832(1-Benzofuran-7-yl-4-octyl-piperazine | CHEMBL26988)
Affinity DataKi:  1.70nMAssay Description:Binding affinity to displace [3H]2-(di-N-propylamino)-8-hydroxy-tetralin from 5-hydroxytryptamine 1A (5-HT1A) receptor in rat frontal cortex homogena...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

Target5-hydroxytryptamine receptor 1A(Rat)
Solvay Duphar Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50039806(1-(2,3-Dihydro-benzo[1,4]dioxin-5-yl)-4-pentyl-pip...)
Affinity DataKi:  2.20nMAssay Description:Binding affinity to displace [3H]2-(di-N-propylamino)-8-hydroxy-tetralin from 5-hydroxytryptamine 1A (5-HT1A) receptor in rat frontal cortex homogena...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

Target5-hydroxytryptamine receptor 1A(Rat)
Solvay Duphar Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50039792(1-(2,3-Dihydro-benzo[1,4]dioxin-5-yl)-4-(2,3-dihyd...)
Affinity DataKi:  4nMAssay Description:Binding affinity to displace [3H]2-(di-N-propylamino)-8-hydroxy-tetralin from 5-hydroxytryptamine 1A (5-HT1A) receptor in rat frontal cortex homogena...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

Target5-hydroxytryptamine receptor 1A(Rat)
Solvay Duphar Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50039799(1-Benzofuran-7-yl-4-(2,3-dihydro-benzo[1,4]dioxin-...)
Affinity DataKi:  5.80nMAssay Description:Binding affinity to displace [3H]2-(di-N-propylamino)-8-hydroxy-tetralin from 5-hydroxytryptamine 1A (5-HT1A) receptor in rat frontal cortex homogena...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

Target5-hydroxytryptamine receptor 1A(Rat)
Solvay Duphar Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50039809(1-Benzofuran-7-yl-4-butyl-piperazine | CHEMBL28082...)
Affinity DataKi:  5.90nMAssay Description:Binding affinity to displace [3H]2-(di-N-propylamino)-8-hydroxy-tetralin from 5-hydroxytryptamine 1A (5-HT1A) receptor in rat frontal cortex homogena...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

Target5-hydroxytryptamine receptor 1A(Rat)
Solvay Duphar Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50039816(1-Benzofuran-7-yl-4-cyclohexylmethyl-piperazine | ...)
Affinity DataKi:  7.70nMAssay Description:Binding affinity to displace [3H]2-(di-N-propylamino)-8-hydroxy-tetralin from 5-hydroxytryptamine 1A (5-HT1A) receptor in rat frontal cortex homogena...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

Target5-hydroxytryptamine receptor 1A(Rat)
Solvay Duphar Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50039804(1-Benzofuran-7-yl-4-decyl-piperazine | CHEMBL26355)
Affinity DataKi:  8nMAssay Description:Binding affinity to displace [3H]2-(di-N-propylamino)-8-hydroxy-tetralin from 5-hydroxytryptamine 1A (5-HT1A) receptor in rat frontal cortex homogena...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

Target5-hydroxytryptamine receptor 1A(Rat)
Solvay Duphar Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50039830(1-Benzofuran-7-yl-4-methyl-piperazine | CHEMBL2862...)
Affinity DataKi:  8.10nMAssay Description:Binding affinity to displace [3H]2-(di-N-propylamino)-8-hydroxy-tetralin from 5-hydroxytryptamine 1A (5-HT1A) receptor in rat frontal cortex homogena...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

Target5-hydroxytryptamine receptor 1A(Rat)
Solvay Duphar Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50039793(1-Cyclohexylmethyl-4-(2,3-dihydro-benzo[1,4]dioxin...)
Affinity DataKi:  11nMAssay Description:Binding affinity to displace [3H]2-(di-N-propylamino)-8-hydroxy-tetralin from 5-hydroxytryptamine 1A (5-HT1A) receptor in rat frontal cortex homogena...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

Target5-hydroxytryptamine receptor 1A(Rat)
Solvay Duphar Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50039803(1-Butyl-4-(2,3-dihydro-benzo[1,4]dioxin-5-yl)-pipe...)
Affinity DataKi:  12nMAssay Description:Binding affinity to displace [3H]2-(di-N-propylamino)-8-hydroxy-tetralin from 5-hydroxytryptamine 1A (5-HT1A) receptor in rat frontal cortex homogena...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

Target5-hydroxytryptamine receptor 1A(Rat)
Solvay Duphar Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50035042(1-Benzofuran-7-yl-piperazine | CHEMBL61032)
Affinity DataKi:  13nMAssay Description:Binding affinity to displace [3H]2-(di-N-propylamino)-8-hydroxy-tetralin from 5-hydroxytryptamine 1A (5-HT1A) receptor in rat frontal cortex homogena...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

Target5-hydroxytryptamine receptor 1A(Rat)
Solvay Duphar Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50039808(1-Benzofuran-7-yl-4-cyclopropylmethyl-piperazine |...)
Affinity DataKi:  20nMAssay Description:Binding affinity to displace [3H]2-(di-N-propylamino)-8-hydroxy-tetralin from 5-hydroxytryptamine 1A (5-HT1A) receptor in rat frontal cortex homogena...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

Target5-hydroxytryptamine receptor 1A(Rat)
Solvay Duphar Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50039794(1-Benzofuran-7-yl-4-benzyl-piperazine; hydrochlori...)
Affinity DataKi:  22nMAssay Description:Binding affinity to displace [3H]2-(di-N-propylamino)-8-hydroxy-tetralin from 5-hydroxytryptamine 1A (5-HT1A) receptor in rat frontal cortex homogena...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

Target5-hydroxytryptamine receptor 1A(Rat)
Solvay Duphar Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50039815(1-Benzofuran-7-yl-4-ethyl-piperazine | CHEMBL32924...)
Affinity DataKi:  23nMAssay Description:Binding affinity to displace [3H]2-(di-N-propylamino)-8-hydroxy-tetralin from 5-hydroxytryptamine 1A (5-HT1A) receptor in rat frontal cortex homogena...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

Target5-hydroxytryptamine receptor 1A(Rat)
Solvay Duphar Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50039813(1-(2,3-Dihydro-benzo[1,4]dioxin-5-yl)-4-methyl-pip...)
Affinity DataKi:  24nMAssay Description:Binding affinity to displace [3H]2-(di-N-propylamino)-8-hydroxy-tetralin from 5-hydroxytryptamine 1A (5-HT1A) receptor in rat frontal cortex homogena...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

Target5-hydroxytryptamine receptor 1A(Rat)
Solvay Duphar Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50039801(1-Benzyl-4-(2,3-dihydro-benzo[1,4]dioxin-5-yl)-pip...)
Affinity DataKi:  28nMAssay Description:Binding affinity to displace [3H]2-(di-N-propylamino)-8-hydroxy-tetralin from 5-hydroxytryptamine 1A (5-HT1A) receptor in rat frontal cortex homogena...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

Target5-hydroxytryptamine receptor 1A(Rat)
Solvay Duphar Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50039820(1-Benzofuran-7-yl-4-propyl-piperazine | CHEMBL2664...)
Affinity DataKi:  29nMAssay Description:Binding affinity to displace [3H]2-(di-N-propylamino)-8-hydroxy-tetralin from 5-hydroxytryptamine 1A (5-HT1A) receptor in rat frontal cortex homogena...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

Target5-hydroxytryptamine receptor 1A(Rat)
Solvay Duphar Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50035057((eltoprazine)1-(2,3-Dihydro-benzo[1,4]dioxin-5-yl)...)
Affinity DataKi:  40nMAssay Description:Binding affinity to displace [3H]2-(di-N-propylamino)-8-hydroxy-tetralin from 5-hydroxytryptamine 1A (5-HT1A) receptor in rat frontal cortex homogena...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

Target5-hydroxytryptamine receptor 1A(Rat)
Solvay Duphar Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50039828(1-Benzofuran-7-yl-4-isopropyl-piperazine | CHEMBL2...)
Affinity DataKi:  56nMAssay Description:Binding affinity to displace [3H]2-(di-N-propylamino)-8-hydroxy-tetralin from 5-hydroxytryptamine 1A (5-HT1A) receptor in rat frontal cortex homogena...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

Target5-hydroxytryptamine receptor 1A(Rat)
Solvay Duphar Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50039825(1-Benzofuran-7-yl-4-isobutyl-piperazine | CHEMBL96...)
Affinity DataKi:  64nMAssay Description:Binding affinity to displace [3H]2-(di-N-propylamino)-8-hydroxy-tetralin from 5-hydroxytryptamine 1A (5-HT1A) receptor in rat frontal cortex homogena...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

Target5-hydroxytryptamine receptor 1A(Rat)
Solvay Duphar Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50039823(1-Benzofuran-7-yl-4-cyclohexyl-piperazine | CHEMBL...)
Affinity DataKi:  64nMAssay Description:Binding affinity to displace [3H]2-(di-N-propylamino)-8-hydroxy-tetralin from 5-hydroxytryptamine 1A (5-HT1A) receptor in rat frontal cortex homogena...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

Target5-hydroxytryptamine receptor 1A(Rat)
Solvay Duphar Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50039831(1-(2,3-Dihydro-benzo[1,4]dioxin-5-yl)-4-ethyl-pipe...)
Affinity DataKi:  66nMAssay Description:Binding affinity to displace [3H]2-(di-N-propylamino)-8-hydroxy-tetralin from 5-hydroxytryptamine 1A (5-HT1A) receptor in rat frontal cortex homogena...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

Target5-hydroxytryptamine receptor 1A(Rat)
Solvay Duphar Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50039817(1-(2,3-Dihydro-benzo[1,4]dioxin-5-yl)-4-propyl-pip...)
Affinity DataKi:  80nMAssay Description:Binding affinity to displace [3H]2-(di-N-propylamino)-8-hydroxy-tetralin from 5-hydroxytryptamine 1A (5-HT1A) receptor in rat frontal cortex homogena...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed