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maximum 50k data
Found 18 Enz. Inhib. hit(s) with all data for entry = 50005798
TargetPurine nucleoside phosphorylase(Homo sapiens (Human))
Ciba-Geigy

Curated by ChEMBL
LigandPNGBDBM50039559(CHEMBL267803 | [5-(2-Amino-6-oxo-1,6-dihydro-purin...)
Affinity DataKi:  170nMAssay Description:Inhibition of human erythrocytic PNP (purine nucleoside phosphorylase) in 1 mM phosphateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPurine nucleoside phosphorylase(Homo sapiens (Human))
Ciba-Geigy

Curated by ChEMBL
LigandPNGBDBM50039552(CHEMBL267312 | [3,3-Dimethyl-5-(6-oxo-1,6-dihydro-...)
Affinity DataKi:  210nMAssay Description:Inhibition of human erythrocytic PNP (purine nucleoside phosphorylase) in 1 mM phosphateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPurine nucleoside phosphorylase(Homo sapiens (Human))
Ciba-Geigy

Curated by ChEMBL
LigandPNGBDBM50039555(CHEMBL13130 | [5-(6-Oxo-1,6-dihydro-purin-9-yl)-pe...)
Affinity DataKi:  1.10E+3nMAssay Description:Inhibition of human erythrocytic PNP (purine nucleoside phosphorylase) in 1 mM phosphateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPurine nucleoside phosphorylase(Homo sapiens (Human))
Ciba-Geigy

Curated by ChEMBL
LigandPNGBDBM50041099(9-(3,3-Dimethyl-pentyl)-1,9-dihydro-purin-6-one | ...)
Affinity DataKi:  1.10E+5nMAssay Description:Inhibition of human erythrocytic PNP (purine nucleoside phosphorylase) in 1 mM phosphateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPurine nucleoside phosphorylase(Rattus norvegicus)
Ciba-Geigy

Curated by ChEMBL
LigandPNGBDBM50039551(CHEMBL13448 | [5-(2-Amino-6-oxo-1,6-dihydro-purin-...)
Affinity DataIC50:  44nMAssay Description:Inhibition of calf spleen PNP (purine nucleoside phosphorylase) in 1 mM phosphateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPurine nucleoside phosphorylase(Rattus norvegicus)
Ciba-Geigy

Curated by ChEMBL
LigandPNGBDBM50041095(5-(2-Amino-6-oxo-1,6-dihydro-purin-9-yl)-3,3-dimet...)
Affinity DataIC50:  180nMAssay Description:Inhibition of calf spleen PNP (purine nucleoside phosphorylase) in 1 mM phosphateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPurine nucleoside phosphorylase(Rattus norvegicus)
Ciba-Geigy

Curated by ChEMBL
LigandPNGBDBM50039551(CHEMBL13448 | [5-(2-Amino-6-oxo-1,6-dihydro-purin-...)
Affinity DataIC50:  2.00E+3nMAssay Description:Inhibition of calf spleen PNP (purine nucleoside phosphorylase) in 50 mM phosphateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPurine nucleoside phosphorylase(Rattus norvegicus)
Ciba-Geigy

Curated by ChEMBL
LigandPNGBDBM50041097(6-(2-Amino-6-oxo-1,6-dihydro-purin-9-yl)-4,4-dimet...)
Affinity DataIC50:  8.00E+3nMAssay Description:Inhibition of calf spleen PNP (purine nucleoside phosphorylase) in 1 mM phosphateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPurine nucleoside phosphorylase(Rattus norvegicus)
Ciba-Geigy

Curated by ChEMBL
LigandPNGBDBM50041095(5-(2-Amino-6-oxo-1,6-dihydro-purin-9-yl)-3,3-dimet...)
Affinity DataIC50:  9.00E+3nMAssay Description:Inhibition of calf spleen PNP (purine nucleoside phosphorylase) in 50 mM phosphateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPurine nucleoside phosphorylase(Rattus norvegicus)
Ciba-Geigy

Curated by ChEMBL
LigandPNGBDBM50041096(2-Amino-9-(5-mercapto-3,3-dimethyl-pentyl)-1,9-dih...)
Affinity DataIC50:  5.00E+4nMAssay Description:Inhibition of calf spleen PNP (purine nucleoside phosphorylase) in 1 mM phosphateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPurine nucleoside phosphorylase(Rattus norvegicus)
Ciba-Geigy

Curated by ChEMBL
LigandPNGBDBM50041096(2-Amino-9-(5-mercapto-3,3-dimethyl-pentyl)-1,9-dih...)
Affinity DataIC50:  9.50E+4nMAssay Description:Inhibition of calf spleen PNP (purine nucleoside phosphorylase) in 50 mM phosphateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPurine nucleoside phosphorylase(Rattus norvegicus)
Ciba-Geigy

Curated by ChEMBL
LigandPNGBDBM50041093(5-(2-Amino-6-oxo-1,6-dihydro-purin-9-yl)-3,3-dimet...)
Affinity DataIC50:  1.00E+5nMAssay Description:Inhibition of calf spleen PNP (purine nucleoside phosphorylase) in 1 mM phosphateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPurine nucleoside phosphorylase(Rattus norvegicus)
Ciba-Geigy

Curated by ChEMBL
LigandPNGBDBM50041098(6-(2-Amino-6-oxo-1,6-dihydro-purin-9-yl)-4,4-dimet...)
Affinity DataIC50:  2.00E+5nMAssay Description:Inhibition of calf spleen PNP (purine nucleoside phosphorylase) in 1 mM phosphateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPurine nucleoside phosphorylase(Rattus norvegicus)
Ciba-Geigy

Curated by ChEMBL
LigandPNGBDBM50041094(6-(2-Amino-6-oxo-1,6-dihydro-purin-9-yl)-4,4-dimet...)
Affinity DataIC50:  2.60E+5nMAssay Description:Inhibition of calf spleen PNP (purine nucleoside phosphorylase) in 1 mM phosphateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPurine nucleoside phosphorylase(Rattus norvegicus)
Ciba-Geigy

Curated by ChEMBL
LigandPNGBDBM50041097(6-(2-Amino-6-oxo-1,6-dihydro-purin-9-yl)-4,4-dimet...)
Affinity DataIC50:  2.90E+5nMAssay Description:Inhibition of calf spleen PNP (purine nucleoside phosphorylase) in 50 mM phosphateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPurine nucleoside phosphorylase(Rattus norvegicus)
Ciba-Geigy

Curated by ChEMBL
LigandPNGBDBM50041094(6-(2-Amino-6-oxo-1,6-dihydro-purin-9-yl)-4,4-dimet...)
Affinity DataIC50: >3.00E+5nMAssay Description:Inhibition of calf spleen PNP (purine nucleoside phosphorylase) in 50 mM phosphateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPurine nucleoside phosphorylase(Rattus norvegicus)
Ciba-Geigy

Curated by ChEMBL
LigandPNGBDBM50041093(5-(2-Amino-6-oxo-1,6-dihydro-purin-9-yl)-3,3-dimet...)
Affinity DataIC50: >3.00E+5nMAssay Description:Inhibition of calf spleen PNP (purine nucleoside phosphorylase) in 50 mM phosphateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPurine nucleoside phosphorylase(Rattus norvegicus)
Ciba-Geigy

Curated by ChEMBL
LigandPNGBDBM50041098(6-(2-Amino-6-oxo-1,6-dihydro-purin-9-yl)-4,4-dimet...)
Affinity DataIC50: >3.00E+5nMAssay Description:Inhibition of calf spleen PNP (purine nucleoside phosphorylase) in 50 mM phosphateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed