Compile Data Set for Download or QSAR
maximum 50k data
Report error Found 105 Enz. Inhib. hit(s) with all data for entry = 50006019
TargetThromboxane-A synthase(Human)
Dr. Karl Thomae

Curated by ChEMBL
LigandPNGBDBM50043839((E)-6-[2-(4-Fluoro-benzenesulfonylamino)-indan-5-y...)
Affinity DataIC50:  1nMAssay Description:Inhibition test of thromboxane A2 synthetase in human gel-filtered platelets.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetThromboxane-A synthase(Human)
Dr. Karl Thomae

Curated by ChEMBL
LigandPNGBDBM50043826(6-{4-[2-(4-Chloro-benzenesulfonylamino)-ethyl]-phe...)
Affinity DataIC50:  2nMAssay Description:Inhibition test of thromboxane A2 synthetase in human gel-filtered platelets.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetThromboxane-A synthase(Human)
Dr. Karl Thomae

Curated by ChEMBL
LigandPNGBDBM50003795(5-[1-Pyridin-3-yl-1-(3-trifluoromethyl-phenyl)-met...)
Affinity DataIC50:  4nMAssay Description:Inhibition test of thromboxane A2 synthetase in human gel-filtered platelets.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMedDrugBank


TargetThromboxane-A synthase(Human)
Dr. Karl Thomae

Curated by ChEMBL
LigandPNGBDBM50003795(5-[1-Pyridin-3-yl-1-(3-trifluoromethyl-phenyl)-met...)
Affinity DataIC50:  4nMAssay Description:Inhibition test of thromboxane A2 synthetase in human gel-filtered platelets.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMedDrugBank


TargetThromboxane-A synthase(Human)
Dr. Karl Thomae

Curated by ChEMBL
LigandPNGBDBM50043827((E)-6-(4-{2-[(4-Chloro-benzenesulfonyl)-(2-morphol...)
Affinity DataIC50:  4nMAssay Description:Inhibition test of thromboxane A2 synthetase in human gel-filtered platelets.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetThromboxane-A synthase(Human)
Dr. Karl Thomae

Curated by ChEMBL
LigandPNGBDBM50043829((E)-6-{3-[2-(4-Chloro-benzenesulfonylamino)-ethyl]...)
Affinity DataIC50:  4nMAssay Description:Inhibition test of thromboxane A2 synthetase in human gel-filtered platelets.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetThromboxane-A synthase(Human)
Dr. Karl Thomae

Curated by ChEMBL
LigandPNGBDBM50043841((E)-6-{4-[2-(4-Chloro-benzenesulfonylamino)-ethyl]...)
Affinity DataIC50:  4nMAssay Description:Inhibition test of thromboxane A2 synthetase in human gel-filtered platelets.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetThromboxane-A synthase(Human)
Dr. Karl Thomae

Curated by ChEMBL
LigandPNGBDBM50043856((Z)-6-{5-[2-(4-Fluoro-benzenesulfonylamino)-ethyl]...)
Affinity DataIC50:  4nMAssay Description:Inhibition test of thromboxane A2 synthetase in human gel-filtered platelets.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetThromboxane-A synthase(Human)
Dr. Karl Thomae

Curated by ChEMBL
LigandPNGBDBM50043847(3-((E)-2-{4-[2-(4-Chloro-benzenesulfonylamino)-eth...)
Affinity DataIC50:  4nMAssay Description:Inhibition test of thromboxane A2 synthetase in human gel-filtered platelets.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetThromboxane-A synthase(Human)
Dr. Karl Thomae

Curated by ChEMBL
LigandPNGBDBM50043851((E)-6-(4-{2-[(4-Chloro-benzenesulfonyl)-ethyl-amin...)
Affinity DataIC50:  4nMAssay Description:Inhibition test of thromboxane A2 synthetase in human gel-filtered platelets.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetThromboxane-A synthase(Human)
Dr. Karl Thomae

Curated by ChEMBL
LigandPNGBDBM50043868((E)-6-{4-[2-(4-Fluoro-benzenesulfonylamino)-ethyl]...)
Affinity DataIC50:  4nMAssay Description:Inhibition test of thromboxane A2 synthetase in human gel-filtered platelets.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetThromboxane-A synthase(Human)
Dr. Karl Thomae

Curated by ChEMBL
LigandPNGBDBM50043855((E)-6-{4-[2-(3,4-Dimethoxy-benzenesulfonylamino)-e...)
Affinity DataIC50:  5nMAssay Description:Inhibition test of thromboxane A2 synthetase in human gel-filtered platelets.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetThromboxane-A synthase(Human)
Dr. Karl Thomae

Curated by ChEMBL
LigandPNGBDBM50043850((E)-6-{4-[2-(Butane-1-sulfonylamino)-ethyl]-phenyl...)
Affinity DataIC50:  5nMAssay Description:Inhibition test of thromboxane A2 synthetase in human gel-filtered platelets.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetThromboxane-A synthase(Human)
Dr. Karl Thomae

Curated by ChEMBL
LigandPNGBDBM50043833((E)-6-{4-[2-(4-Methoxy-benzenesulfonylamino)-ethyl...)
Affinity DataIC50:  5nMAssay Description:Inhibition test of thromboxane A2 synthetase in human gel-filtered platelets.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetThromboxane-A synthase(Human)
Dr. Karl Thomae

Curated by ChEMBL
LigandPNGBDBM50043843((E)-6-Pyridin-3-yl-6-{4-[2-(toluene-4-sulfonylamin...)
Affinity DataIC50:  5nMAssay Description:Inhibition test of thromboxane A2 synthetase in human gel-filtered platelets.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetThromboxane-A synthase(Human)
Dr. Karl Thomae

Curated by ChEMBL
LigandPNGBDBM50043844((E)-6-[4-(4-Chloro-benzenesulfonylamino)-phenyl]-6...)
Affinity DataIC50:  5nMAssay Description:Inhibition test of thromboxane A2 synthetase in human gel-filtered platelets.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetThromboxane-A synthase(Human)
Dr. Karl Thomae

Curated by ChEMBL
LigandPNGBDBM50043858((E)-6-[4-(2-Benzenesulfonylamino-ethyl)-phenyl]-6-...)
Affinity DataIC50:  5nMAssay Description:Inhibition test of thromboxane A2 synthetase in human gel-filtered platelets.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetThromboxane-A synthase(Human)
Dr. Karl Thomae

Curated by ChEMBL
LigandPNGBDBM50043838((E)-6-{3-[(4-Chloro-benzenesulfonylamino)-methyl]-...)
Affinity DataIC50:  5nMAssay Description:Inhibition test of thromboxane A2 synthetase in human gel-filtered platelets.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetThromboxane-A synthase(Human)
Dr. Karl Thomae

Curated by ChEMBL
LigandPNGBDBM50043845((E)-6-[4-(2-Phenylmethanesulfonylamino-ethyl)-phen...)
Affinity DataIC50:  5nMAssay Description:Inhibition test of thromboxane A2 synthetase in human gel-filtered platelets.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetThromboxane-A synthase(Human)
Dr. Karl Thomae

Curated by ChEMBL
LigandPNGBDBM50043852((E)-6-(4-{2-[Carbamoylmethyl-(4-chloro-benzenesulf...)
Affinity DataIC50:  5nMAssay Description:Inhibition test of thromboxane A2 synthetase in human gel-filtered platelets.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetThromboxane-A synthase(Human)
Dr. Karl Thomae

Curated by ChEMBL
LigandPNGBDBM50003776(8-(4-Chloro-benzenesulfonylamino)-4-(3-pyridin-3-y...)
Affinity DataIC50:  6nMAssay Description:Inhibition test of thromboxane A2 synthetase in human gel-filtered platelets.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetThromboxane A2 receptor(Human)
Dr. Karl Thomae

Curated by ChEMBL
LigandPNGBDBM50003776(8-(4-Chloro-benzenesulfonylamino)-4-(3-pyridin-3-y...)
Affinity DataIC50:  6nMAssay Description:Displacement of the high affinity radiolabeled ligand [3H]- SQ-29,548 from the PGH-2/TXA-2 receptor in human gel-filtered platelets.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetThromboxane-A synthase(Human)
Dr. Karl Thomae

Curated by ChEMBL
LigandPNGBDBM50043848((E)-6-Pyridin-3-yl-6-{4-[2-(4-trifluoromethyl-benz...)
Affinity DataIC50:  6nMAssay Description:Inhibition test of thromboxane A2 synthetase in human gel-filtered platelets.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetThromboxane-A synthase(Human)
Dr. Karl Thomae

Curated by ChEMBL
LigandPNGBDBM50003776(8-(4-Chloro-benzenesulfonylamino)-4-(3-pyridin-3-y...)
Affinity DataIC50:  6nMAssay Description:Inhibition test of thromboxane A2 synthetase in human gel-filtered platelets.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetThromboxane-A synthase(Human)
Dr. Karl Thomae

Curated by ChEMBL
LigandPNGBDBM50043828((E)-6-[3-(4-Chloro-benzenesulfonylamino)-phenyl]-6...)
Affinity DataIC50:  7nMAssay Description:Inhibition test of thromboxane A2 synthetase in human gel-filtered platelets.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetThromboxane-A synthase(Human)
Dr. Karl Thomae

Curated by ChEMBL
LigandPNGBDBM50043832((E)-6-{4-[(4-Chloro-benzenesulfonylamino)-methyl]-...)
Affinity DataIC50:  7nMAssay Description:Inhibition test of thromboxane A2 synthetase in human gel-filtered platelets.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetThromboxane-A synthase(Human)
Dr. Karl Thomae

Curated by ChEMBL
LigandPNGBDBM50043849((E)-6-[6-(4-Chloro-benzenesulfonylamino)-5,6,7,8-t...)
Affinity DataIC50:  8nMAssay Description:Inhibition test of thromboxane A2 synthetase in human gel-filtered platelets.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetThromboxane A2 receptor(Human)
Dr. Karl Thomae

Curated by ChEMBL
LigandPNGBDBM50043839((E)-6-[2-(4-Fluoro-benzenesulfonylamino)-indan-5-y...)
Affinity DataIC50:  9nMAssay Description:Displacement of the high affinity radiolabeled ligand [3H]- SQ-29,548 from the PGH-2/TXA-2 receptor in human gel-filtered platelets.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetThromboxane A2 receptor(Human)
Dr. Karl Thomae

Curated by ChEMBL
LigandPNGBDBM50043862((E)-4-{4-[2-(4-Chloro-benzenesulfonylamino)-ethyl]...)
Affinity DataIC50:  12nMAssay Description:Displacement of the high affinity radiolabeled ligand [3H]- SQ-29,548 from the PGH-2/TXA-2 receptor in human gel-filtered platelets.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetThromboxane A2 receptor(Human)
Dr. Karl Thomae

Curated by ChEMBL
LigandPNGBDBM50043824(4-Chloro-N-(2-{4-[(E)-1-pyridin-3-yl-5-(1H-tetrazo...)
Affinity DataIC50:  12nMAssay Description:Displacement of the high affinity radiolabeled ligand [3H]- SQ-29,548 from the PGH-2/TXA-2 receptor in human gel-filtered platelets.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetThromboxane A2 receptor(Human)
Dr. Karl Thomae

Curated by ChEMBL
LigandPNGBDBM50043829((E)-6-{3-[2-(4-Chloro-benzenesulfonylamino)-ethyl]...)
Affinity DataIC50:  12nMAssay Description:Displacement of the high affinity radiolabeled ligand [3H]- SQ-29,548 from the PGH-2/TXA-2 receptor in human gel-filtered platelets.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetThromboxane A2 receptor(Human)
Dr. Karl Thomae

Curated by ChEMBL
LigandPNGBDBM50043849((E)-6-[6-(4-Chloro-benzenesulfonylamino)-5,6,7,8-t...)
Affinity DataIC50:  13nMAssay Description:Displacement of the high affinity radiolabeled ligand [3H]- SQ-29,548 from the PGH-2/TXA-2 receptor in human gel-filtered platelets.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetThromboxane-A synthase(Human)
Dr. Karl Thomae

Curated by ChEMBL
LigandPNGBDBM50043823((E)-6-(4-{2-[(4-Chloro-benzenesulfonyl)-methyl-ami...)
Affinity DataIC50:  15nMAssay Description:Inhibition test of thromboxane A2 synthetase in human gel-filtered platelets.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetThromboxane A2 receptor(Human)
Dr. Karl Thomae

Curated by ChEMBL
LigandPNGBDBM50043841((E)-6-{4-[2-(4-Chloro-benzenesulfonylamino)-ethyl]...)
Affinity DataIC50:  19nMAssay Description:Displacement of the high affinity radiolabeled ligand [3H]- SQ-29,548 from the PGH-2/TXA-2 receptor in human gel-filtered platelets.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetThromboxane-A synthase(Human)
Dr. Karl Thomae

Curated by ChEMBL
LigandPNGBDBM50043861((E)-6-Pyridin-3-yl-6-{4-[2-(2,4,6-trimethyl-benzen...)
Affinity DataIC50:  19nMAssay Description:Inhibition test of thromboxane A2 synthetase in human gel-filtered platelets.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetThromboxane A2 receptor(Human)
Dr. Karl Thomae

Curated by ChEMBL
LigandPNGBDBM50043865((E)-7-{4-[2-(4-Chloro-benzenesulfonylamino)-ethyl]...)
Affinity DataIC50:  19nMAssay Description:Displacement of the high affinity radiolabeled ligand [3H]- SQ-29,548 from the PGH-2/TXA-2 receptor in human gel-filtered platelets.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetThromboxane-A synthase(Human)
Dr. Karl Thomae

Curated by ChEMBL
LigandPNGBDBM50043859((E)-5-{4-[2-(4-Chloro-benzenesulfonylamino)-ethyl]...)
Affinity DataIC50:  21nMAssay Description:Inhibition test of thromboxane A2 synthetase in human gel-filtered platelets.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetThromboxane-A synthase(Human)
Dr. Karl Thomae

Curated by ChEMBL
LigandPNGBDBM50043854((E)-6-[4-(2-Phenylacetylamino-ethyl)-phenyl]-6-pyr...)
Affinity DataIC50:  21nMAssay Description:Inhibition test of thromboxane A2 synthetase in human gel-filtered platelets.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetThromboxane A2 receptor(Human)
Dr. Karl Thomae

Curated by ChEMBL
LigandPNGBDBM50043838((E)-6-{3-[(4-Chloro-benzenesulfonylamino)-methyl]-...)
Affinity DataIC50:  21nMAssay Description:Displacement of the high affinity radiolabeled ligand [3H]- SQ-29,548 from the PGH-2/TXA-2 receptor in human gel-filtered platelets.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetThromboxane-A synthase(Human)
Dr. Karl Thomae

Curated by ChEMBL
LigandPNGBDBM50043824(4-Chloro-N-(2-{4-[(E)-1-pyridin-3-yl-5-(1H-tetrazo...)
Affinity DataIC50:  21nMAssay Description:Inhibition test of thromboxane A2 synthetase in human gel-filtered platelets.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetThromboxane-A synthase(Human)
Dr. Karl Thomae

Curated by ChEMBL
LigandPNGBDBM50043822((E)-9-(4-Chloro-benzenesulfonylamino)-6-pyridin-3-...)
Affinity DataIC50:  24nMAssay Description:Inhibition test of thromboxane A2 synthetase in human gel-filtered platelets.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetThromboxane-A synthase(Human)
Dr. Karl Thomae

Curated by ChEMBL
LigandPNGBDBM50043865((E)-7-{4-[2-(4-Chloro-benzenesulfonylamino)-ethyl]...)
Affinity DataIC50:  24nMAssay Description:Inhibition test of thromboxane A2 synthetase in human gel-filtered platelets.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetThromboxane-A synthase(Human)
Dr. Karl Thomae

Curated by ChEMBL
LigandPNGBDBM50043857((E)-6-(4-{2-[(4-Chloro-benzenesulfonyl)-isopropyl-...)
Affinity DataIC50:  25nMAssay Description:Inhibition test of thromboxane A2 synthetase in human gel-filtered platelets.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetThromboxane A2 receptor(Human)
Dr. Karl Thomae

Curated by ChEMBL
LigandPNGBDBM50043823((E)-6-(4-{2-[(4-Chloro-benzenesulfonyl)-methyl-ami...)
Affinity DataIC50:  25nMAssay Description:Displacement of the high affinity radiolabeled ligand [3H]- SQ-29,548 from the PGH-2/TXA-2 receptor in human gel-filtered platelets.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetThromboxane A2 receptor(Human)
Dr. Karl Thomae

Curated by ChEMBL
LigandPNGBDBM50043860(3-[1-{4-[2-(4-Chloro-benzenesulfonylamino)-ethyl]-...)
Affinity DataIC50:  26nMAssay Description:Displacement of the high affinity radiolabeled ligand [3H]- SQ-29,548 from the PGH-2/TXA-2 receptor in human gel-filtered platelets.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetThromboxane-A synthase(Human)
Dr. Karl Thomae

Curated by ChEMBL
LigandPNGBDBM50043867(4-((E)-2-{4-[2-(4-Chloro-benzenesulfonylamino)-eth...)
Affinity DataIC50:  27nMAssay Description:Inhibition test of thromboxane A2 synthetase in human gel-filtered platelets.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetThromboxane A2 receptor(Human)
Dr. Karl Thomae

Curated by ChEMBL
LigandPNGBDBM50043869(4-{[{2-[4-((E)-5-Carboxy-1-pyridin-3-yl-pent-1-eny...)
Affinity DataIC50:  28nMAssay Description:Displacement of the high affinity radiolabeled ligand [3H]- SQ-29,548 from the PGH-2/TXA-2 receptor in human gel-filtered platelets.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetThromboxane A2 receptor(Human)
Dr. Karl Thomae

Curated by ChEMBL
LigandPNGBDBM50043848((E)-6-Pyridin-3-yl-6-{4-[2-(4-trifluoromethyl-benz...)
Affinity DataIC50:  28nMAssay Description:Displacement of the high affinity radiolabeled ligand [3H]- SQ-29,548 from the PGH-2/TXA-2 receptor in human gel-filtered platelets.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetThromboxane-A synthase(Human)
Dr. Karl Thomae

Curated by ChEMBL
LigandPNGBDBM50043834(7-{4-[2-(4-Chloro-benzenesulfonylamino)-ethyl]-phe...)
Affinity DataIC50:  31nMAssay Description:Inhibition test of thromboxane A2 synthetase in human gel-filtered platelets.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetThromboxane A2 receptor(Human)
Dr. Karl Thomae

Curated by ChEMBL
LigandPNGBDBM50043851((E)-6-(4-{2-[(4-Chloro-benzenesulfonyl)-ethyl-amin...)
Affinity DataIC50:  33nMAssay Description:Displacement of the high affinity radiolabeled ligand [3H]- SQ-29,548 from the PGH-2/TXA-2 receptor in human gel-filtered platelets.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

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