Compile Data Set for Download or QSAR
Report error Found 86 Enz. Inhib. hit(s) with all data for entry = 50048909
TargetType-1 angiotensin II receptor A/B(Rat)
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50230906(CHEMBL308261)
Affinity DataIC50: 0.410nMAssay Description:Inhibitory concentration against binding of [125I]angiotensin II to rat liver expressing Angiotensin II receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/2/2019
Entry Details Article
PubMed
TargetType-1 angiotensin II receptor A/B(Rat)
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50230919(CHEMBL307844 | CI-996)
Affinity DataIC50: 0.580nMAssay Description:Inhibitory concentration against binding of [125I]angiotensin II to rat liver expressing Angiotensin II receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/2/2019
Entry Details Article
PubMed
TargetType-1 angiotensin II receptor A/B(Rat)
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50230891(CHEMBL76166)
Affinity DataIC50: 0.800nMAssay Description:Inhibitory concentration against binding of [125I]angiotensin II to rat liver expressing Angiotensin II receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/2/2019
Entry Details Article
PubMed
TargetType-1 angiotensin II receptor A/B(Rat)
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50230883(CHEMBL309089)
Affinity DataIC50: 0.820nMAssay Description:Inhibitory concentration against binding of [125I]angiotensin II to rat liver expressing Angiotensin II receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/2/2019
Entry Details Article
PubMed
TargetType-1 angiotensin II receptor A/B(Rat)
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50230915(CHEMBL76169)
Affinity DataIC50: 0.900nMAssay Description:Inhibitory concentration against binding of [125I]angiotensin II to rat liver expressing Angiotensin II receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/2/2019
Entry Details Article
PubMed
TargetType-1 angiotensin II receptor A/B(Rat)
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50230887(CHEMBL306259)
Affinity DataIC50: 1nMAssay Description:Inhibitory concentration against binding of [125I]angiotensin II to rat liver expressing Angiotensin II receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/2/2019
Entry Details Article
PubMed
TargetType-1 angiotensin II receptor A/B(Rat)
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50230912(CHEMBL72922)
Affinity DataIC50: 1.20nMAssay Description:Inhibitory concentration against binding of [125I]angiotensin II to rat liver expressing Angiotensin II receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/2/2019
Entry Details Article
PubMed
TargetType-1 angiotensin II receptor A/B(Rat)
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50230886(CHEMBL307455)
Affinity DataIC50: 1.40nMAssay Description:Inhibitory concentration against binding of [125I]angiotensin II to rat liver expressing Angiotensin II receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/2/2019
Entry Details Article
PubMed
TargetType-1 angiotensin II receptor A/B(Rat)
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50230882(CARBOXYLIC ACID METABOLITE | CHEBI:74125 | E-3174)
Affinity DataIC50: 1.60nMAssay Description:Tested for inhibitory concentration against AT1 receptor binding affinity in rat liverMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/2/2019
Entry Details Article
PubMed
TargetType-1 angiotensin II receptor A/B(Rat)
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50230882(CARBOXYLIC ACID METABOLITE | CHEBI:74125 | E-3174)
Affinity DataIC50: 1.60nMAssay Description:Inhibitory concentration against binding of [125I]angiotensin II to rat liver expressing Angiotensin II receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/2/2019
Entry Details Article
PubMed
TargetType-1 angiotensin II receptor A/B(Rat)
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50230910(CHEMBL306066)
Affinity DataIC50: 1.60nMAssay Description:Inhibitory concentration against binding of [125I]angiotensin II to rat liver expressing Angiotensin II receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/2/2019
Entry Details Article
PubMed
TargetType-1/Type-2 angiotensin II receptor(Human)
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50230882(CARBOXYLIC ACID METABOLITE | CHEBI:74125 | E-3174)
Affinity DataIC50: 1.80nMAssay Description:Inhibitory concentration against [125I]angiotensin II(AII) induced contraction in rabbit aorta by 50%More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/2/2019
Entry Details Article
PubMed
TargetType-1/Type-2 angiotensin II receptor(Human)
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50230883(CHEMBL309089)
Affinity DataIC50: 2.40nMAssay Description:Inhibitory concentration against [125I]angiotensin II(AII) induced contraction in rabbit aorta by 50%More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/2/2019
Entry Details Article
PubMed
TargetType-1 angiotensin II receptor A/B(Rat)
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50230877(CHEMBL70371)
Affinity DataIC50: 2.40nMAssay Description:Inhibitory concentration against binding of [125I]angiotensin II to rat liver expressing Angiotensin II receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/2/2019
Entry Details Article
PubMed
TargetType-1 angiotensin II receptor A/B(Rat)
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50230900(CHEMBL73433)
Affinity DataIC50: 2.5nMAssay Description:Inhibitory concentration against binding of [125I]angiotensin II to rat liver expressing Angiotensin II receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/2/2019
Entry Details Article
PubMed
TargetType-1/Type-2 angiotensin II receptor(Human)
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50230891(CHEMBL76166)
Affinity DataIC50: 2.60nMAssay Description:Inhibitory concentration against [125I]angiotensin II(AII) induced contraction in rabbit aorta by 50%More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/2/2019
Entry Details Article
PubMed
TargetType-1 angiotensin II receptor A/B(Rat)
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50230893(CHEMBL308031)
Affinity DataIC50: 2.80nMAssay Description:Inhibitory concentration against binding of [125I]angiotensin II to rat liver expressing Angiotensin II receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/2/2019
Entry Details Article
PubMed
TargetType-1 angiotensin II receptor A/B(Rat)
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50230902(CHEMBL75518)
Affinity DataIC50: 2.80nMAssay Description:Inhibitory concentration against binding of [125I]angiotensin II to rat liver expressing Angiotensin II receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/2/2019
Entry Details Article
PubMed
TargetType-1/Type-2 angiotensin II receptor(Human)
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50230887(CHEMBL306259)
Affinity DataIC50: 2.90nMAssay Description:Inhibitory concentration against [125I]angiotensin II(AII) induced contraction in rabbit aorta by 50%More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/2/2019
Entry Details Article
PubMed
TargetType-1/Type-2 angiotensin II receptor(Human)
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50230906(CHEMBL308261)
Affinity DataIC50: 3.30nMAssay Description:Inhibitory concentration against [125I]angiotensin II(AII) induced contraction in rabbit aorta by 50%More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/2/2019
Entry Details Article
PubMed
TargetType-1 angiotensin II receptor A/B(Rat)
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50230881(CHEMBL308779)
Affinity DataIC50: 3.30nMAssay Description:Inhibitory concentration against binding of [125I]angiotensin II to rat liver expressing Angiotensin II receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/2/2019
Entry Details Article
PubMed
TargetType-1 angiotensin II receptor A/B(Rat)
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50230908(CHEMBL443269 | DuP-532)
Affinity DataIC50: 3.40nMAssay Description:Tested for inhibitory concentration against AT1 receptor binding affinity in rat liverMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/2/2019
Entry Details Article
PubMed
TargetType-1 angiotensin II receptor A/B(Rat)
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50230909(CHEMBL306852)
Affinity DataIC50: 3.60nMAssay Description:Inhibitory concentration against binding of [125I]angiotensin II to rat liver expressing Angiotensin II receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/2/2019
Entry Details Article
PubMed
TargetType-1 angiotensin II receptor A/B(Rat)
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50230897(CHEMBL275652)
Affinity DataIC50: 3.60nMAssay Description:Inhibitory concentration against binding of [125I]angiotensin II to rat liver expressing Angiotensin II receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/2/2019
Entry Details Article
PubMed
TargetType-1/Type-2 angiotensin II receptor(Human)
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50230919(CHEMBL307844 | CI-996)
Affinity DataIC50: 3.80nMAssay Description:Inhibitory concentration against [125I]angiotensin II(AII) induced contraction in rabbit aorta by 50%More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/2/2019
Entry Details Article
PubMed
TargetType-1 angiotensin II receptor A/B(Rat)
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50230914(CHEMBL431390)
Affinity DataIC50: 3.90nMAssay Description:Inhibitory concentration against binding of [125I]angiotensin II to rat liver expressing Angiotensin II receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/2/2019
Entry Details Article
PubMed
TargetType-1 angiotensin II receptor A/B(Rat)
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50230888(CHEMBL306612)
Affinity DataIC50: 4nMAssay Description:Inhibitory concentration against binding of [125I]angiotensin II to rat liver expressing Angiotensin II receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/2/2019
Entry Details Article
PubMed
TargetType-1/Type-2 angiotensin II receptor(Human)
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50230877(CHEMBL70371)
Affinity DataIC50: 4nMAssay Description:Inhibitory concentration against [125I]angiotensin II(AII) induced contraction in rabbit aorta by 50%More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/2/2019
Entry Details Article
PubMed
TargetType-1/Type-2 angiotensin II receptor(Human)
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50230915(CHEMBL76169)
Affinity DataIC50: 4.5nMAssay Description:Inhibitory concentration against [125I]angiotensin II(AII) induced contraction in rabbit aorta by 50%More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/2/2019
Entry Details Article
PubMed
TargetType-1/Type-2 angiotensin II receptor(Human)
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50230893(CHEMBL308031)
Affinity DataIC50: 4.80nMAssay Description:Inhibitory concentration against [125I]angiotensin II(AII) induced contraction in rabbit aorta by 50%More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/2/2019
Entry Details Article
PubMed
TargetType-1 angiotensin II receptor A/B(Rat)
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM82258(NSC_3961 | CAS_114798-26-4 | Losartan)
Affinity DataIC50: 5nMAssay Description:Tested for inhibitory concentration against AT1 receptor binding affinity in rat liverMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/2/2019
Entry Details Article
PubMed
TargetType-1 angiotensin II receptor A/B(Rat)
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM82258(NSC_3961 | CAS_114798-26-4 | Losartan)
Affinity DataIC50: 5nMAssay Description:Inhibitory concentration against binding of [125I]angiotensin II to rat liver expressing Angiotensin II receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/2/2019
Entry Details Article
PubMed
TargetType-1/Type-2 angiotensin II receptor(Human)
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50230912(CHEMBL72922)
Affinity DataIC50: 5.40nMAssay Description:Inhibitory concentration against [125I]angiotensin II(AII) induced contraction in rabbit aorta by 50%More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/2/2019
Entry Details Article
PubMed
TargetType-1 angiotensin II receptor A/B(Rat)
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50230899(CHEMBL75935)
Affinity DataIC50: 5.60nMAssay Description:Inhibitory concentration against binding of [125I]angiotensin II to rat liver expressing Angiotensin II receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/2/2019
Entry Details Article
PubMed
TargetType-1/Type-2 angiotensin II receptor(Human)
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50230910(CHEMBL306066)
Affinity DataIC50: 7nMAssay Description:Inhibitory concentration against [125I]angiotensin II(AII) induced contraction in rabbit aorta by 50%More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/2/2019
Entry Details Article
PubMed
TargetType-1 angiotensin II receptor A/B(Rat)
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50230885(CHEMBL72453)
Affinity DataIC50: 8.80nMAssay Description:Inhibitory concentration against binding of [125I]angiotensin II to rat liver expressing Angiotensin II receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/2/2019
Entry Details Article
PubMed
TargetType-1/Type-2 angiotensin II receptor(Human)
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50230918(CHEMBL73084)
Affinity DataIC50: 9nMAssay Description:Inhibitory concentration against [125I]angiotensin II(AII) induced contraction in rabbit aorta by 50%More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/2/2019
Entry Details Article
PubMed
TargetType-1 angiotensin II receptor A/B(Rat)
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50230911(CHEMBL306949)
Affinity DataIC50: 11nMAssay Description:Inhibitory concentration against binding of [125I]angiotensin II to rat liver expressing Angiotensin II receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/2/2019
Entry Details Article
PubMed
TargetType-1 angiotensin II receptor A/B(Rat)
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50230918(CHEMBL73084)
Affinity DataIC50: 11nMAssay Description:Inhibitory concentration against binding of [125I]angiotensin II to rat liver expressing Angiotensin II receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/2/2019
Entry Details Article
PubMed
TargetType-1 angiotensin II receptor A/B(Rat)
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50230890(CHEMBL73646)
Affinity DataIC50: 12nMAssay Description:Inhibitory concentration against binding of [125I]angiotensin II to rat liver expressing Angiotensin II receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/2/2019
Entry Details Article
PubMed
TargetType-1 angiotensin II receptor A/B(Rat)
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50230907(CHEMBL76393)
Affinity DataIC50: 14nMAssay Description:Inhibitory concentration against binding of [125I]angiotensin II to rat liver expressing Angiotensin II receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/2/2019
Entry Details Article
PubMed
TargetType-1 angiotensin II receptor A/B(Rat)
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50230879(CHEMBL309094)
Affinity DataIC50: 15nMAssay Description:Inhibitory concentration against binding of [125I]angiotensin II to rat liver expressing Angiotensin II receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/2/2019
Entry Details Article
PubMed
TargetType-1/Type-2 angiotensin II receptor(Human)
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50230900(CHEMBL73433)
Affinity DataIC50: 18nMAssay Description:Inhibitory concentration against [125I]angiotensin II(AII) induced contraction in rabbit aorta by 50%More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/2/2019
Entry Details Article
PubMed
TargetType-1/Type-2 angiotensin II receptor(Human)
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50230911(CHEMBL306949)
Affinity DataIC50: 19nMAssay Description:Inhibitory concentration against [125I]angiotensin II(AII) induced contraction in rabbit aorta by 50%More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/2/2019
Entry Details Article
PubMed
TargetType-1 angiotensin II receptor A/B(Rat)
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50230916(CHEMBL76330)
Affinity DataIC50: 19nMAssay Description:Inhibitory concentration against binding of [125I]angiotensin II to rat liver expressing Angiotensin II receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/2/2019
Entry Details Article
PubMed
TargetType-1/Type-2 angiotensin II receptor(Human)
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50230881(CHEMBL308779)
Affinity DataIC50: 21nMAssay Description:Inhibitory concentration against [125I]angiotensin II(AII) induced contraction in rabbit aorta by 50%More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/2/2019
Entry Details Article
PubMed
TargetType-1 angiotensin II receptor A/B(Rat)
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50230896(CHEMBL308961)
Affinity DataIC50: 21nMAssay Description:Inhibitory concentration against binding of [125I]angiotensin II to rat liver expressing Angiotensin II receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/2/2019
Entry Details Article
PubMed
TargetType-1 angiotensin II receptor A/B(Rat)
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50230892(CHEMBL73725)
Affinity DataIC50: 22nMAssay Description:Inhibitory concentration against binding of [125I]angiotensin II to rat liver expressing Angiotensin II receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/2/2019
Entry Details Article
PubMed
TargetType-1 angiotensin II receptor A/B(Rat)
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50230913(CHEMBL75092)
Affinity DataIC50: 22nMAssay Description:Inhibitory concentration against binding of [125I]angiotensin II to rat liver expressing Angiotensin II receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/2/2019
Entry Details Article
PubMed
TargetType-1 angiotensin II receptor A/B(Rat)
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50230920(CHEMBL307284)
Affinity DataIC50: 23nMAssay Description:Inhibitory concentration against binding of [125I]angiotensin II to rat liver expressing Angiotensin II receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/2/2019
Entry Details Article
PubMed
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