Compile Data Set for Download or QSAR
Report error Found 29 Enz. Inhib. hit(s) with all data for entry = 50048910
TargetType-1 angiotensin II receptor A/B(Rat)
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50231010BDBM50231010(CHEMBL312066)
Affinity DataKi:  0.400nMAssay Description:Binding affinity of compound in presence of bovine serum albumin (BSA) at 0% against rat adrenal Angiotensin II receptor, type 1More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/3/2019
Entry Details Article
PubMed
TargetType-1 angiotensin II receptor A/B(Rat)
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50231010BDBM50231010(CHEMBL312066)
Affinity DataKi:  1.30nMAssay Description:Binding affinity of compound in presence of bovine serum albumin (BSA) at 0.01% against rat adrenal Angiotensin II receptor, type 1More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/3/2019
Entry Details Article
PubMed
TargetType-1 angiotensin II receptor A/B(Rat)
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50231010BDBM50231010(CHEMBL312066)
Affinity DataKi:  1.30nMAssay Description:Binding affinity for Angiotensin II receptor, type 1 in rat adrenal cortical membranes using [125I]Sar1, Ile8-angiotensin IIMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/3/2019
Entry Details Article
PubMed
TargetType-1 angiotensin II receptor A/B(Rat)
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50231140BDBM50231140(CHEMBL77029)
Affinity DataKi:  4.5nMAssay Description:Binding affinity for Angiotensin II receptor, type 1 in rat adrenal cortical membranes using [125I]Sar1, Ile8-angiotensin IIMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/3/2019
Entry Details Article
PubMed
TargetType-1 angiotensin II receptor A/B(Rat)
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50231145BDBM50231145(CHEMBL76785)
Affinity DataKi:  5.5nMAssay Description:Binding affinity of compound in presence of bovine serum albumin (BSA) at 0% against rat Angiotensin II receptor, type 1More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/3/2019
Entry Details Article
PubMed
TargetType-1 angiotensin II receptor A/B(Rat)
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50231150BDBM50231150(CHEMBL77935)
Affinity DataKi:  7.40nMAssay Description:Binding affinity for Angiotensin II receptor, type 1 in rat adrenal cortical membranes using [125I]Sar1, Ile8-angiotensin IIMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/3/2019
Entry Details Article
PubMed
TargetType-1 angiotensin II receptor A/B(Rat)
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50231139BDBM50231139(CHEMBL77827)
Affinity DataKi:  9nMAssay Description:Binding affinity for Angiotensin II receptor, type 1 in rat adrenal cortical membranes using [125I]Sar1, Ile8-angiotensin IIMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/3/2019
Entry Details Article
PubMed
TargetType-1 angiotensin II receptor A/B(Rat)
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50231149BDBM50231149(CHEMBL306278)
Affinity DataKi:  15nMAssay Description:Binding affinity for Angiotensin II receptor, type 1 in rat adrenal cortical membranes using [125I]Sar1, Ile8-angiotensin IIMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/3/2019
Entry Details Article
PubMed
TargetType-1 angiotensin II receptor A/B(Rat)
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50231143BDBM50231143(CHEMBL75053)
Affinity DataKi:  17nMAssay Description:Binding affinity for Angiotensin II receptor, type 1 in rat adrenal cortical membranes using [125I]Sar1, Ile8-angiotensin IIMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/3/2019
Entry Details Article
PubMed
TargetType-1 angiotensin II receptor A/B(Rat)
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50231007BDBM50231007(CHEMBL74445)
Affinity DataKi:  21nMAssay Description:Binding affinity for Angiotensin II receptor, type 1 in rat adrenal cortical membranes using [125I]Sar1, Ile8-angiotensin IIMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/3/2019
Entry Details Article
PubMed
TargetType-1 angiotensin II receptor A/B(Rat)
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50231142BDBM50231142(CHEMBL312068)
Affinity DataKi:  22nMAssay Description:Binding affinity for Angiotensin II receptor, type 1 in rat adrenal cortical membranes using [125I]Sar1, Ile8-angiotensin IIMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/3/2019
Entry Details Article
PubMed
TargetType-1 angiotensin II receptor A/B(Rat)
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50231148BDBM50231148(CHEMBL77376)
Affinity DataKi:  28nMAssay Description:Binding affinity for Angiotensin II receptor, type 1 in rat adrenal cortical membranes using [125I]Sar1, Ile8-angiotensin IIMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/3/2019
Entry Details Article
PubMed
TargetType-1 angiotensin II receptor A/B(Rat)
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50231011BDBM50231011(CHEMBL309489)
Affinity DataKi:  44nMAssay Description:Binding affinity for Angiotensin II receptor, type 1 in rat adrenal cortical membranes using [125I]Sar1, Ile8-angiotensin IIMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/3/2019
Entry Details Article
PubMed
TargetType-1 angiotensin II receptor A/B(Rat)
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50231145BDBM50231145(CHEMBL76785)
Affinity DataKi:  46nMAssay Description:Binding affinity of compound in presence of bovine serum albumin (BSA) at 0.01% against rat Angiotensin II receptor, type 1More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/3/2019
Entry Details Article
PubMed
TargetType-1 angiotensin II receptor A/B(Rat)
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50231145BDBM50231145(CHEMBL76785)
Affinity DataKi:  46nMAssay Description:Binding affinity for Angiotensin II receptor, type 1 in rat adrenal cortical membranes using [125I]Sar1, Ile8-angiotensin IIMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/3/2019
Entry Details Article
PubMed
TargetType-1 angiotensin II receptor A/B(Rat)
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50231009BDBM50231009(CHEMBL76765)
Affinity DataKi:  50nMAssay Description:Binding affinity for Angiotensin II receptor, type 1 in rat adrenal cortical membranes using [125I]Sar1, Ile8-angiotensin IIMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/3/2019
Entry Details Article
PubMed
TargetType-1 angiotensin II receptor A/B(Rat)
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50231147BDBM50231147(CHEMBL433310)
Affinity DataKi:  68nMAssay Description:Binding affinity for Angiotensin II receptor, type 1 in rat adrenal cortical membranes using [125I]Sar1, Ile8-angiotensin IIMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/3/2019
Entry Details Article
PubMed
TargetType-1 angiotensin II receptor A/B(Rat)
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50231008BDBM50231008(CHEMBL75101)
Affinity DataKi:  71nMAssay Description:Binding affinity for Angiotensin II receptor, type 1 in rat adrenal cortical membranes using [125I]Sar1, Ile8-angiotensin IIMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/3/2019
Entry Details Article
PubMed
TargetType-1 angiotensin II receptor A/B(Rat)
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50231008BDBM50231008(CHEMBL75101)
Affinity DataKi:  71nMAssay Description:Binding affinity of compound in presence of bovine serum albumin (BSA) at 0.01% against rat adrenal Angiotensin II receptor, type 1More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/3/2019
Entry Details Article
PubMed
TargetType-1 angiotensin II receptor A/B(Rat)
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50231144BDBM50231144(CHEMBL76943)
Affinity DataKi:  137nMAssay Description:Binding affinity for Angiotensin II receptor, type 1 in rat adrenal cortical membranes using [125I]Sar1, Ile8-angiotensin IIMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/3/2019
Entry Details Article
PubMed
TargetType-1 angiotensin II receptor A/B(Rat)
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50231141BDBM50231141(CHEMBL77266)
Affinity DataKi:  190nMAssay Description:Binding affinity for Angiotensin II receptor, type 1 in rat adrenal cortical membranes using [125I]Sar1, Ile8-angiotensin IIMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/3/2019
Entry Details Article
PubMed
TargetType-1 angiotensin II receptor A/B(Rat)
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50231146BDBM50231146(CHEMBL77185)
Affinity DataKi:  550nMAssay Description:Binding affinity of compound in presence of bovine serum albumin (BSA) at 0.01% against rat adrenal Angiotensin II receptor, type 1More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/3/2019
Entry Details Article
PubMed
TargetType-1 angiotensin II receptor A/B(Rat)
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50231146BDBM50231146(CHEMBL77185)
Affinity DataKi:  550nMAssay Description:Binding affinity for Angiotensin II receptor, type 1 in rat adrenal cortical membranes using [125I]Sar1, Ile8-angiotensin IIMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/3/2019
Entry Details Article
PubMed
TargetType-1 angiotensin II receptor A/B(Rat)
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50231008BDBM50231008(CHEMBL75101)
Affinity DataKi:  580nMAssay Description:Binding affinity of compound in presence of bovine serum albumin (BSA) at 0.22% against rat adrenal Angiotensin II receptor, type 1More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/3/2019
Entry Details Article
PubMed
TargetType-1 angiotensin II receptor A/B(Rat)
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50231144BDBM50231144(CHEMBL76943)
Affinity DataKi:  2.20E+3nMAssay Description:Binding affinity of compound in presence of bovine serum albumin (BSA) at 0.22% against rat adrenal Angiotensin II receptor, type 1More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/3/2019
Entry Details Article
PubMed
TargetType-1 angiotensin II receptor A/B(Rat)
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50231006BDBM50231006(CHEMBL307946)
Affinity DataKi:  3.45E+3nMAssay Description:Binding affinity of compound in presence of bovine serum albumin (BSA) at 0.01% against rat Angiotensin II receptor, type 1More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/3/2019
Entry Details Article
PubMed
TargetType-1 angiotensin II receptor A/B(Rat)
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50231006BDBM50231006(CHEMBL307946)
Affinity DataKi:  3.45E+3nMAssay Description:Binding affinity for Angiotensin II receptor, type 1 in rat adrenal cortical membranes using [125I]Sar1, Ile8-angiotensin IIMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/3/2019
Entry Details Article
PubMed
TargetType-1 angiotensin II receptor A/B(Rat)
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50231146BDBM50231146(CHEMBL77185)
Affinity DataKi:  2.44E+4nMAssay Description:Binding affinity of compound in presence of bovine serum albumin (BSA) at 0.22% against rat adrenal Angiotensin II receptor, type 1More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/3/2019
Entry Details Article
PubMed
TargetType-1 angiotensin II receptor A/B(Rat)
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50231006BDBM50231006(CHEMBL307946)
Affinity DataKi:  4.00E+4nMAssay Description:Binding affinity of compound in presence of bovine serum albumin (BSA) at 0.22% against rat Angiotensin II receptor, type 1More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/3/2019
Entry Details Article
PubMed