Compile Data Set for Download or QSAR
Report error Found 30 Enz. Inhib. hit(s) with all data for entry = 50048911
TargetTransient receptor potential cation channel subfamily V member 1/2/4(Rat)
Sandoz Institute For Medical Research

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50231166BDBM50231166(CHEMBL58719)
Affinity DataEC50:  60nMAssay Description:Effective concentration for [Ca2+] uptake into dorsal root ganglia neurones in rat cultured spinal sensory neuronesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/5/2019
Entry Details Article
PubMed
TargetTransient receptor potential cation channel subfamily V member 1/2/4(Rat)
Sandoz Institute For Medical Research

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50231175BDBM50231175(CHEMBL76789)
Affinity DataEC50:  280nMAssay Description:Effective concentration for [Ca2+] uptake into dorsal root ganglia neurones in rat cultured spinal sensory neuronesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/5/2019
Entry Details Article
PubMed
TargetTransient receptor potential cation channel subfamily V member 1/2/4(Rat)
Sandoz Institute For Medical Research

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 20461BDBM20461(Zostrix | (E)-N-[(4-hydroxy-3-methoxyphenyl)methyl...)
Affinity DataEC50:  300nMAssay Description:Effective concentration for [Ca2+] uptake into dorsal root ganglia neurones in rat cultured spinal sensory neuronesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/5/2019
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetTransient receptor potential cation channel subfamily V member 1/2/4(Rat)
Sandoz Institute For Medical Research

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50044753BDBM50044753(2-(4-Hydroxy-3-methoxy-phenyl)-N-octyl-acetamide |...)
Affinity DataEC50:  300nMAssay Description:Effective concentration for [Ca2+] uptake into dorsal root ganglia neurones in rat cultured spinal sensory neuronesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/5/2019
Entry Details Article
PubMed
TargetTransient receptor potential cation channel subfamily V member 1/2/4(Rat)
Sandoz Institute For Medical Research

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50231155BDBM50231155(CHEMBL77186)
Affinity DataEC50:  360nMAssay Description:Effective concentration for [Ca2+] uptake into dorsal root ganglia neurones in rat cultured spinal sensory neuronesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/5/2019
Entry Details Article
PubMed
TargetTransient receptor potential cation channel subfamily V member 1/2/4(Rat)
Sandoz Institute For Medical Research

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50231161BDBM50231161(CHEMBL431379)
Affinity DataEC50:  530nMAssay Description:Effective concentration for [Ca2+] uptake into dorsal root ganglia neurones in rat cultured spinal sensory neuronesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/5/2019
Entry Details Article
PubMed
TargetTransient receptor potential cation channel subfamily V member 1/2/4(Rat)
Sandoz Institute For Medical Research

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50044767BDBM50044767(N-(4-hydroxy-3-methoxybenzyl)nonanamide | nonivami...)
Affinity DataEC50:  550nMAssay Description:Effective concentration for [Ca2+] uptake into dorsal root ganglia neurones in rat cultured spinal sensory neuronesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/5/2019
Entry Details Article
PubMed
TargetTransient receptor potential cation channel subfamily V member 1/2/4(Rat)
Sandoz Institute For Medical Research

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50231176BDBM50231176(CHEMBL76476)
Affinity DataEC50:  670nMAssay Description:Effective concentration for [Ca2+] uptake into dorsal root ganglia neurones in rat cultured spinal sensory neuronesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/5/2019
Entry Details Article
PubMed
TargetTransient receptor potential cation channel subfamily V member 1/2/4(Rat)
Sandoz Institute For Medical Research

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50231162BDBM50231162(CHEMBL431788)
Affinity DataEC50:  1.16E+3nMAssay Description:Effective concentration for [Ca2+] uptake into dorsal root ganglia neurones in rat cultured spinal sensory neuronesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/5/2019
Entry Details Article
PubMed
TargetTransient receptor potential cation channel subfamily V member 1/2/4(Rat)
Sandoz Institute For Medical Research

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50231153BDBM50231153(CHEMBL312611)
Affinity DataEC50:  1.17E+3nMAssay Description:Effective concentration for [Ca2+] uptake into dorsal root ganglia neurones in rat cultured spinal sensory neuronesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/5/2019
Entry Details Article
PubMed
TargetTransient receptor potential cation channel subfamily V member 1/2/4(Rat)
Sandoz Institute For Medical Research

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50231169BDBM50231169(CHEMBL76546)
Affinity DataEC50:  1.32E+3nMAssay Description:Effective concentration for [Ca2+] uptake into dorsal root ganglia neurones in rat cultured spinal sensory neuronesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/5/2019
Entry Details Article
PubMed
TargetTransient receptor potential cation channel subfamily V member 1/2/4(Rat)
Sandoz Institute For Medical Research

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50231174BDBM50231174(CHEMBL431200)
Affinity DataEC50:  2.13E+3nMAssay Description:Effective concentration for [Ca2+] uptake into dorsal root ganglia neurones in rat cultured spinal sensory neuronesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/5/2019
Entry Details Article
PubMed
TargetTransient receptor potential cation channel subfamily V member 1/2/4(Rat)
Sandoz Institute For Medical Research

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50231167BDBM50231167(CHEMBL80153)
Affinity DataEC50:  2.32E+3nMAssay Description:Effective concentration for [Ca2+] uptake into dorsal root ganglia neurones in rat cultured spinal sensory neuronesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/5/2019
Entry Details Article
PubMed
TargetTransient receptor potential cation channel subfamily V member 1/2/4(Rat)
Sandoz Institute For Medical Research

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50231151BDBM50231151(CHEMBL77349)
Affinity DataEC50:  2.57E+3nMAssay Description:Effective concentration for [Ca2+] uptake into dorsal root ganglia neurones in rat cultured spinal sensory neuronesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/5/2019
Entry Details Article
PubMed
TargetTransient receptor potential cation channel subfamily V member 1/2/4(Rat)
Sandoz Institute For Medical Research

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50231173BDBM50231173(CHEMBL80954)
Affinity DataEC50:  3.28E+3nMAssay Description:Effective concentration for [Ca2+] uptake into dorsal root ganglia neurones in rat cultured spinal sensory neuronesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/5/2019
Entry Details Article
PubMed
TargetTransient receptor potential cation channel subfamily V member 1/2/4(Rat)
Sandoz Institute For Medical Research

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50231157BDBM50231157(CHEMBL77304)
Affinity DataEC50:  3.78E+3nMAssay Description:Effective concentration for [Ca2+] uptake into dorsal root ganglia neurones in rat cultured spinal sensory neuronesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/5/2019
Entry Details Article
PubMed
TargetTransient receptor potential cation channel subfamily V member 1/2/4(Rat)
Sandoz Institute For Medical Research

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50231163BDBM50231163(CHEMBL76312)
Affinity DataEC50:  4.48E+3nMAssay Description:Effective concentration for [Ca2+] uptake into dorsal root ganglia neurones in rat cultured spinal sensory neuronesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/5/2019
Entry Details Article
PubMed
TargetTransient receptor potential cation channel subfamily V member 1/2/4(Rat)
Sandoz Institute For Medical Research

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50231159BDBM50231159(CHEMBL80539)
Affinity DataEC50:  6.29E+3nMAssay Description:Effective concentration for [Ca2+] uptake into dorsal root ganglia neurones in rat cultured spinal sensory neuronesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/5/2019
Entry Details Article
PubMed
TargetTransient receptor potential cation channel subfamily V member 1/2/4(Rat)
Sandoz Institute For Medical Research

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50231170BDBM50231170(CHEMBL80400)
Affinity DataEC50:  1.42E+4nMAssay Description:Effective concentration for [Ca2+] uptake into dorsal root ganglia neurones in rat cultured spinal sensory neuronesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/5/2019
Entry Details Article
PubMed
TargetTransient receptor potential cation channel subfamily V member 1/2/4(Rat)
Sandoz Institute For Medical Research

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50231165BDBM50231165(CHEMBL80559)
Affinity DataEC50:  1.79E+4nMAssay Description:Effective concentration for [Ca2+] uptake into dorsal root ganglia neurones in rat cultured spinal sensory neuronesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/5/2019
Entry Details Article
PubMed
TargetTransient receptor potential cation channel subfamily V member 1/2/4(Rat)
Sandoz Institute For Medical Research

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50231154BDBM50231154(CHEMBL76790)
Affinity DataEC50:  1.83E+4nMAssay Description:Effective concentration for [Ca2+] uptake into dorsal root ganglia neurones in rat cultured spinal sensory neuronesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/5/2019
Entry Details Article
PubMed
TargetTransient receptor potential cation channel subfamily V member 1/2/4(Rat)
Sandoz Institute For Medical Research

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50231152BDBM50231152(CHEMBL420027)
Affinity DataEC50: >1.00E+5nMAssay Description:Effective concentration for [Ca2+] uptake into dorsal root ganglia neurones in rat cultured spinal sensory neuronesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/5/2019
Entry Details Article
PubMed
TargetTransient receptor potential cation channel subfamily V member 1/2/4(Rat)
Sandoz Institute For Medical Research

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50231168BDBM50231168(CHEMBL80159)
Affinity DataEC50: >1.00E+5nMAssay Description:Effective concentration for [Ca2+] uptake into dorsal root ganglia neurones in rat cultured spinal sensory neuronesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/5/2019
Entry Details Article
PubMed
TargetTransient receptor potential cation channel subfamily V member 1/2/4(Rat)
Sandoz Institute For Medical Research

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50231177BDBM50231177(CHEMBL80387)
Affinity DataEC50: >1.00E+5nMAssay Description:Effective concentration for [Ca2+] uptake into dorsal root ganglia neurones in rat cultured spinal sensory neuronesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/5/2019
Entry Details Article
PubMed
TargetTransient receptor potential cation channel subfamily V member 1/2/4(Rat)
Sandoz Institute For Medical Research

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50231164BDBM50231164(CHEMBL309534)
Affinity DataEC50: >1.00E+5nMAssay Description:Effective concentration for [Ca2+] uptake into dorsal root ganglia neurones in rat cultured spinal sensory neuronesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/5/2019
Entry Details Article
PubMed
TargetTransient receptor potential cation channel subfamily V member 1/2/4(Rat)
Sandoz Institute For Medical Research

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50231160BDBM50231160(CHEMBL80956)
Affinity DataEC50: >1.00E+5nMAssay Description:Effective concentration for [Ca2+] uptake into dorsal root ganglia neurones in rat cultured spinal sensory neuronesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/5/2019
Entry Details Article
PubMed
TargetTransient receptor potential cation channel subfamily V member 1/2/4(Rat)
Sandoz Institute For Medical Research

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50231156BDBM50231156(CHEMBL77389)
Affinity DataEC50: >1.00E+5nMAssay Description:Effective concentration for [Ca2+] uptake into dorsal root ganglia neurones in rat cultured spinal sensory neuronesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/5/2019
Entry Details Article
PubMed
TargetTransient receptor potential cation channel subfamily V member 1/2/4(Rat)
Sandoz Institute For Medical Research

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50231171BDBM50231171(CHEMBL76777)
Affinity DataEC50: >1.00E+5nMAssay Description:Effective concentration for [Ca2+] uptake into dorsal root ganglia neurones in rat cultured spinal sensory neuronesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/5/2019
Entry Details Article
PubMed
TargetTransient receptor potential cation channel subfamily V member 1/2/4(Rat)
Sandoz Institute For Medical Research

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50231158BDBM50231158(CHEMBL312574)
Affinity DataEC50: >1.00E+5nMAssay Description:Effective concentration for [Ca2+] uptake into dorsal root ganglia neurones in rat cultured spinal sensory neuronesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/5/2019
Entry Details Article
PubMed
TargetTransient receptor potential cation channel subfamily V member 1/2/4(Rat)
Sandoz Institute For Medical Research

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50231172BDBM50231172(CHEMBL80813)
Affinity DataEC50: >1.00E+5nMAssay Description:Effective concentration for [Ca2+] uptake into dorsal root ganglia neurones in rat cultured spinal sensory neuronesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/5/2019
Entry Details Article
PubMed