Compile Data Set for Download or QSAR
Report error Found 11 Enz. Inhib. hit(s) with all data for entry = 5000
TargetAlpha-1A adrenergic receptor(Human)
National Children'S Medical Research Center

Curated by PDSP Ki Database
LigandPNGBDBM29568([3H]-Minipress | [3H]-Furazosin | PRAZOSIN HYDROCH...)
Affinity DataKi:  0.210nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/9/2012
Entry Details Article
PubMed
TargetAlpha-1A adrenergic receptor(Human)
National Children'S Medical Research Center

Curated by PDSP Ki Database
LigandPNGBDBM81444(NSC_185453 | CAS_185453 | WB 4101 | WB-4101)
Affinity DataKi:  0.230nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/9/2012
Entry Details Article
PubMed
TargetAlpha-1A adrenergic receptor(Human)
National Children'S Medical Research Center

Curated by PDSP Ki Database
LigandPNGBDBM31046(SMR000059054 | cid_91430 | 3-[4,5-dihydro-1H-imida...)
Affinity DataKi:  1.40nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/9/2012
Entry Details Article
PubMed
TargetAlpha-1A adrenergic receptor(Human)
National Children'S Medical Research Center

Curated by PDSP Ki Database
LigandPNGBDBM50033112(Urapidil-5-methyl | CHEMBL420060 | 6-{3-[4-(2-Meth...)
Affinity DataKi:  4.20nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/9/2012
Entry Details Article
PubMed
TargetAlpha-1A adrenergic receptor(Human)
National Children'S Medical Research Center

Curated by PDSP Ki Database
LigandPNGBDBM30712(SMR000059324 | Oxymetazoline | cid_66259 | 6-tert-...)
Affinity DataKi:  28nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/9/2012
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetAlpha-1A adrenergic receptor(Human)
National Children'S Medical Research Center

Curated by PDSP Ki Database
LigandPNGBDBM50013515(yohimbic acid methyl ester | 17alpha-hydroxyyohimb...)
Affinity DataKi:  770nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/9/2012
Entry Details Article
PubMed
TargetAlpha-1A adrenergic receptor(Human)
National Children'S Medical Research Center

Curated by PDSP Ki Database
LigandPNGBDBM84342(EPINEPHRINE | 4-[1-hydroxy-2-(methylamino)ethyl]be...)
Affinity DataKi:  2.50E+3nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/9/2012
Entry Details Article
PubMed
TargetAlpha-1A adrenergic receptor(Human)
National Children'S Medical Research Center

Curated by PDSP Ki Database
LigandPNGBDBM84342(EPINEPHRINE | 4-[1-hydroxy-2-(methylamino)ethyl]be...)
Affinity DataKi:  4.80E+3nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/9/2012
Entry Details Article
PubMed
TargetAlpha-1A adrenergic receptor(Human)
National Children'S Medical Research Center

Curated by PDSP Ki Database
LigandPNGBDBM35234(Noradrenaline,(+) | NOREPINEPHRINE | DL-[7-3H]nore...)
Affinity DataKi:  7.50E+3nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/9/2012
Entry Details Article
PubMed
TargetAlpha-1A adrenergic receptor(Human)
National Children'S Medical Research Center

Curated by PDSP Ki Database
LigandPNGBDBM25392(Isoproterenol,(+) | CHEMBL434 | 4-[1-hydroxy-2-(pr...)
Affinity DataKi: >1.00E+4nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/9/2012
Entry Details Article
PubMed
TargetAlpha-1A adrenergic receptor(Human)
National Children'S Medical Research Center

Curated by PDSP Ki Database
LigandPNGBDBM50026777(CHEMBL524 | Vasoxyl | 2-Amino-1-(2,5-dimethoxy-phe...)
Affinity DataKi: >1.00E+4nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/9/2012
Entry Details Article
PubMed