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Report error Found 43 Enz. Inhib. hit(s) with all data for entry = 50044023
Target5-hydroxytryptamine receptor 3A/3B(Rat)
Syntex Research

Curated by ChEMBL
LigandPNGBDBM50417287(Aloxi | Aurothioglucose | PALONOSETRON | PALONOSET...)
Affinity DataKi:  0.0400nMAssay Description:Binding affinity against 5-hydroxytryptamine 3 (5-HT3) receptor in rat brain cortical membranes using radioligand [3H]quipazineChecked by AuthorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMedPDB3D3D Structure (crystal)

Target5-hydroxytryptamine receptor 3A/3B(Rat)
Syntex Research

Curated by ChEMBL
LigandPNGBDBM50000523(CHEMBL544784)
Affinity DataKi:  0.160nMAssay Description:Binding affinity against 5-hydroxytryptamine 3 (5-HT3) receptor in rat brain cortical membranes using radioligand [3H]quipazineChecked by AuthorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

Target5-hydroxytryptamine receptor 3A/3B(Rat)
Syntex Research

Curated by ChEMBL
LigandPNGBDBM50000453(CHEMBL540055)
Affinity DataKi:  0.160nMAssay Description:Binding affinity against 5-hydroxytryptamine 3 (5-HT3) receptor in rat brain cortical membranes using radioligand [3H]quipazineChecked by AuthorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

Target5-hydroxytryptamine receptor 3A/3B(Rat)
Syntex Research

Curated by ChEMBL
LigandPNGBDBM50000471(CHEMBL542900)
Affinity DataKi:  0.200nMAssay Description:Binding affinity against 5-hydroxytryptamine 3 (5-HT3) receptor in rat brain cortical membranes using radioligand [3H]quipazineChecked by AuthorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

Target5-hydroxytryptamine receptor 3A/3B(Rat)
Syntex Research

Curated by ChEMBL
LigandPNGBDBM50000457(CHEMBL542904)
Affinity DataKi:  0.200nMAssay Description:Binding affinity against 5-hydroxytryptamine 3 (5-HT3) receptor in rat brain cortical membranes using radioligand [3H]quipazineChecked by AuthorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

Target5-hydroxytryptamine receptor 3A/3B(Rat)
Syntex Research

Curated by ChEMBL
LigandPNGBDBM50000450(CHEMBL542669)
Affinity DataKi:  0.200nMAssay Description:Binding affinity against 5-hydroxytryptamine 3 (5-HT3) receptor in rat brain cortical membranes using radioligand [3H]quipazineChecked by AuthorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

Target5-hydroxytryptamine receptor 3A/3B(Rat)
Syntex Research

Curated by ChEMBL
LigandPNGBDBM50056419(4-Amino-N-(1-aza-bicyclo[2.2.2]oct-3-yl)-5-chloro-...)
Affinity DataKi:  0.25nMAssay Description:Binding affinity against 5-hydroxytryptamine 3 (5-HT3) receptor in rat brain cortical membranes using radioligand [3H]quipazineChecked by AuthorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

Target5-hydroxytryptamine receptor 3A/3B(Rat)
Syntex Research

Curated by ChEMBL
LigandPNGBDBM50000460(CHEMBL540057)
Affinity DataKi:  0.320nMAssay Description:Binding affinity against 5-hydroxytryptamine 3 (5-HT3) receptor in rat brain cortical membranes using radioligand [3H]quipazineChecked by AuthorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

Target5-hydroxytryptamine receptor 3A/3B(Rat)
Syntex Research

Curated by ChEMBL
LigandPNGBDBM50000475(CHEMBL555068)
Affinity DataKi:  0.320nMAssay Description:Binding affinity against 5-hydroxytryptamine 3 (5-HT3) receptor in rat brain cortical membranes using radioligand [3H]quipazineChecked by AuthorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

Target5-hydroxytryptamine receptor 3A/3B(Rat)
Syntex Research

Curated by ChEMBL
LigandPNGBDBM50000469(CHEMBL542903)
Affinity DataKi:  0.400nMAssay Description:Binding affinity against 5-hydroxytryptamine 3 (5-HT3) receptor in rat brain cortical membranes using radioligand [3H]quipazineChecked by AuthorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

Target5-hydroxytryptamine receptor 3A/3B(Rat)
Syntex Research

Curated by ChEMBL
LigandPNGBDBM50000455(CHEMBL2093898)
Affinity DataKi:  0.400nMAssay Description:Binding affinity against 5-hydroxytryptamine 3 (5-HT3) receptor in rat brain cortical membranes using radioligand [3H]quipazineChecked by AuthorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

Target5-hydroxytryptamine receptor 3A/3B(Rat)
Syntex Research

Curated by ChEMBL
LigandPNGBDBM50000445(CHEMBL555038)
Affinity DataKi:  0.630nMAssay Description:Binding affinity against 5-hydroxytryptamine 3 (5-HT3) receptor in rat brain cortical membranes using radioligand [3H]quipazineChecked by AuthorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

Target5-hydroxytryptamine receptor 3A/3B(Rat)
Syntex Research

Curated by ChEMBL
LigandPNGBDBM50000462(CHEMBL545719)
Affinity DataKi:  0.630nMAssay Description:Binding affinity against 5-hydroxytryptamine 3 (5-HT3) receptor in rat brain cortical membranes using radioligand [3H]quipazineChecked by AuthorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

Target5-hydroxytryptamine receptor 3A/3B(Rat)
Syntex Research

Curated by ChEMBL
LigandPNGBDBM50449636(BRL-43694 | GRANISETRON | Kytril | LY-278584 | San...)
Affinity DataKi:  0.790nMAssay Description:Binding affinity against 5-hydroxytryptamine 3 (5-HT3) receptor in rat brain cortical membranes using radioligand [3H]quipazineChecked by AuthorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

Target5-hydroxytryptamine receptor 3A/3B(Rat)
Syntex Research

Curated by ChEMBL
LigandPNGBDBM50000446(CHEMBL88565)
Affinity DataKi:  0.790nMAssay Description:Binding affinity against 5-hydroxytryptamine 3 (5-HT3) receptor in rat brain cortical membranes using radioligand [3H]quipazineChecked by AuthorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

Target5-hydroxytryptamine receptor 3A/3B(Rat)
Syntex Research

Curated by ChEMBL
LigandPNGBDBM50000468(CHEMBL539020)
Affinity DataKi:  1nMAssay Description:Binding affinity against 5-hydroxytryptamine 3 (5-HT3) receptor in rat brain cortical membranes using radioligand [3H]quipazineChecked by AuthorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

Target5-hydroxytryptamine receptor 3A/3B(Rat)
Syntex Research

Curated by ChEMBL
LigandPNGBDBM50000472(CHEMBL555199)
Affinity DataKi:  2nMAssay Description:Binding affinity against 5-hydroxytryptamine 3 (5-HT3) receptor in rat brain cortical membranes using radioligand [3H]quipazineChecked by AuthorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

Target5-hydroxytryptamine receptor 3A/3B(Rat)
Syntex Research

Curated by ChEMBL
LigandPNGBDBM50108392((3-ENDO)-8-METHYL-8-AZABICYCLO[3.2.1]OCT-3-YL 1H-I...)
Affinity DataKi:  2nMAssay Description:Binding affinity against 5-hydroxytryptamine 3 (5-HT3) receptor in rat brain cortical membranes using radioligand [3H]quipazineChecked by AuthorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMedPDB3D3D Structure (crystal)

Target5-hydroxytryptamine receptor 3A/3B(Rat)
Syntex Research

Curated by ChEMBL
LigandPNGBDBM50000466(CHEMBL540040)
Affinity DataKi:  2.5nMAssay Description:Binding affinity against 5-hydroxytryptamine 3 (5-HT3) receptor in rat brain cortical membranes using radioligand [3H]quipazineChecked by AuthorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

Target5-hydroxytryptamine receptor 3A/3B(Rat)
Syntex Research

Curated by ChEMBL
LigandPNGBDBM50000467(CHEMBL544785)
Affinity DataKi:  2.5nMAssay Description:Binding affinity against 5-hydroxytryptamine 3 (5-HT3) receptor in rat brain cortical membranes using radioligand [3H]quipazineChecked by AuthorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

Target5-hydroxytryptamine receptor 3A/3B(Rat)
Syntex Research

Curated by ChEMBL
LigandPNGBDBM50000449(CHEMBL545717)
Affinity DataKi:  2.5nMAssay Description:Binding affinity against 5-hydroxytryptamine 3 (5-HT3) receptor in rat brain cortical membranes using radioligand [3H]quipazineChecked by AuthorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

Target5-hydroxytryptamine receptor 3A/3B(Rat)
Syntex Research

Curated by ChEMBL
LigandPNGBDBM50000454(CHEMBL540568)
Affinity DataKi:  2.5nMAssay Description:Binding affinity against 5-hydroxytryptamine 3 (5-HT3) receptor in rat brain cortical membranes using radioligand [3H]quipazineChecked by AuthorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

Target5-hydroxytryptamine receptor 3A/3B(Rat)
Syntex Research

Curated by ChEMBL
LigandPNGBDBM50000459(CHEMBL553733)
Affinity DataKi:  2.5nMAssay Description:Binding affinity against 5-hydroxytryptamine 3 (5-HT3) receptor in rat brain cortical membranes using radioligand [3H]quipazineChecked by AuthorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

Target5-hydroxytryptamine receptor 3A/3B(Rat)
Syntex Research

Curated by ChEMBL
LigandPNGBDBM50031475(4-Amino-N-(1-aza-bicyclo[2.2.2]oct-3-yl)-5-chloro-...)
Affinity DataKi:  3.20nMAssay Description:Binding affinity against 5-hydroxytryptamine 3 (5-HT3) receptor in rat brain cortical membranes using radioligand [3H]quipazineChecked by AuthorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

Target5-hydroxytryptamine receptor 3A/3B(Rat)
Syntex Research

Curated by ChEMBL
LigandPNGBDBM85330(CAS_68647 | NSC_68647 | ONDANSETRON | Ondansetron ...)
Affinity DataKi:  3.20nMAssay Description:Binding affinity against 5-hydroxytryptamine 3 (5-HT3) receptor in rat brain cortical membranes using radioligand [3H]quipazineChecked by AuthorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMedPDB3D3D Structure (crystal)

Target5-hydroxytryptamine receptor 3A/3B(Rat)
Syntex Research

Curated by ChEMBL
LigandPNGBDBM50000464(CHEMBL540820)
Affinity DataKi:  4nMAssay Description:Binding affinity against 5-hydroxytryptamine 3 (5-HT3) receptor in rat brain cortical membranes using radioligand [3H]quipazineChecked by AuthorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

Target5-hydroxytryptamine receptor 3A/3B(Rat)
Syntex Research

Curated by ChEMBL
LigandPNGBDBM50000476(CHEMBL543136)
Affinity DataKi:  4nMAssay Description:Binding affinity against 5-hydroxytryptamine 3 (5-HT3) receptor in rat brain cortical membranes using radioligand [3H]quipazineChecked by AuthorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

Target5-hydroxytryptamine receptor 3A/3B(Rat)
Syntex Research

Curated by ChEMBL
LigandPNGBDBM50000448(CHEMBL315518)
Affinity DataKi:  5nMAssay Description:Binding affinity against 5-hydroxytryptamine 3 (5-HT3) receptor in rat brain cortical membranes using radioligand [3H]quipazineChecked by AuthorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

Target5-hydroxytryptamine receptor 3A/3B(Rat)
Syntex Research

Curated by ChEMBL
LigandPNGBDBM50000456(CHEMBL555582)
Affinity DataKi:  5nMAssay Description:Binding affinity against 5-hydroxytryptamine 3 (5-HT3) receptor in rat brain cortical membranes using radioligand [3H]quipazineChecked by AuthorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

Target5-hydroxytryptamine receptor 3A/3B(Rat)
Syntex Research

Curated by ChEMBL
LigandPNGBDBM50000530(CHEMBL540547)
Affinity DataKi:  7.90nMAssay Description:Binding affinity against 5-hydroxytryptamine 3 (5-HT3) receptor in rat brain cortical membranes using radioligand [3H]quipazineChecked by AuthorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

Target5-hydroxytryptamine receptor 3A/3B(Rat)
Syntex Research

Curated by ChEMBL
LigandPNGBDBM50000500(CHEMBL539275)
Affinity DataKi:  10nMAssay Description:Binding affinity against 5-hydroxytryptamine 3 (5-HT3) receptor in rat brain cortical membranes using radioligand [3H]quipazineChecked by AuthorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

Target5-hydroxytryptamine receptor 3A/3B(Rat)
Syntex Research

Curated by ChEMBL
LigandPNGBDBM50000461(CHEMBL539785)
Affinity DataKi:  10nMAssay Description:Binding affinity against 5-hydroxytryptamine 3 (5-HT3) receptor in rat brain cortical membranes using radioligand [3H]quipazineChecked by AuthorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

Target5-hydroxytryptamine receptor 3A/3B(Rat)
Syntex Research

Curated by ChEMBL
LigandPNGBDBM50000452(CHEMBL554341)
Affinity DataKi:  10nMAssay Description:Binding affinity against 5-hydroxytryptamine 3 (5-HT3) receptor in rat brain cortical membranes using radioligand [3H]quipazineChecked by AuthorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

Target5-hydroxytryptamine receptor 3A/3B(Rat)
Syntex Research

Curated by ChEMBL
LigandPNGBDBM50000458(CHEMBL554259)
Affinity DataKi:  13nMAssay Description:Binding affinity against 5-hydroxytryptamine 3 (5-HT3) receptor in rat brain cortical membranes using radioligand [3H]quipazineChecked by AuthorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

Target5-hydroxytryptamine receptor 3A/3B(Rat)
Syntex Research

Curated by ChEMBL
LigandPNGBDBM50000529(CHEMBL540823)
Affinity DataKi:  13nMAssay Description:Binding affinity against 5-hydroxytryptamine 3 (5-HT3) receptor in rat brain cortical membranes using radioligand [3H]quipazineChecked by AuthorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

Target5-hydroxytryptamine receptor 3A/3B(Rat)
Syntex Research

Curated by ChEMBL
LigandPNGBDBM50000463(CHEMBL541844)
Affinity DataKi:  25nMAssay Description:Binding affinity against 5-hydroxytryptamine 3 (5-HT3) receptor in rat brain cortical membranes using radioligand [3H]quipazineChecked by AuthorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

Target5-hydroxytryptamine receptor 3A/3B(Rat)
Syntex Research

Curated by ChEMBL
LigandPNGBDBM50000447(CHEMBL538027)
Affinity DataKi:  40nMAssay Description:Binding affinity against 5-hydroxytryptamine 3 (5-HT3) receptor in rat brain cortical membranes using radioligand [3H]quipazineChecked by AuthorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

Target5-hydroxytryptamine receptor 3A/3B(Rat)
Syntex Research

Curated by ChEMBL
LigandPNGBDBM50000470(CHEMBL555523)
Affinity DataKi:  158nMAssay Description:Binding affinity against 5-hydroxytryptamine 3 (5-HT3) receptor in rat brain cortical membranes using radioligand [3H]quipazineChecked by AuthorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

Target5-hydroxytryptamine receptor 3A/3B(Rat)
Syntex Research

Curated by ChEMBL
LigandPNGBDBM50000451(CHEMBL542668)
Affinity DataKi:  158nMAssay Description:Binding affinity against 5-hydroxytryptamine 3 (5-HT3) receptor in rat brain cortical membranes using radioligand [3H]quipazineChecked by AuthorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

Target5-hydroxytryptamine receptor 3A/3B(Rat)
Syntex Research

Curated by ChEMBL
LigandPNGBDBM50000465(CHEMBL555402)
Affinity DataKi:  200nMAssay Description:Binding affinity against 5-hydroxytryptamine 3 (5-HT3) receptor in rat brain cortical membranes using radioligand [3H]quipazineChecked by AuthorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

Target5-hydroxytryptamine receptor 3A/3B(Rat)
Syntex Research

Curated by ChEMBL
LigandPNGBDBM50000474(CHEMBL541843)
Affinity DataKi:  398nMAssay Description:Binding affinity against 5-hydroxytryptamine 3 (5-HT3) receptor in rat brain cortical membranes using radioligand [3H]quipazineChecked by AuthorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

Target5-hydroxytryptamine receptor 3A/3B(Rat)
Syntex Research

Curated by ChEMBL
LigandPNGBDBM50000477(CHEMBL538775)
Affinity DataKi:  501nMAssay Description:Binding affinity against 5-hydroxytryptamine 3 (5-HT3) receptor in rat brain cortical membranes using radioligand [3H]quipazineChecked by AuthorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

Target5-hydroxytryptamine receptor 3A/3B(Rat)
Syntex Research

Curated by ChEMBL
LigandPNGBDBM50000473(CHEMBL555080)
Affinity DataKi:  631nMAssay Description:Binding affinity against 5-hydroxytryptamine 3 (5-HT3) receptor in rat brain cortical membranes using radioligand [3H]quipazineChecked by AuthorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed