Compile Data Set for Download or QSAR
Report error Found 58 Enz. Inhib. hit(s) with all data for entry = 50006173
Target5-hydroxytryptamine receptor 1A(Rat)
Solvay Duphar Research Laboratories

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50039822BDBM50039822(CHEMBL543851 | CHEMBL28143 | 1-(2-Cyclohexyl-ethyl...)
Affinity DataKi:  0.25nMAssay Description:Displacement of radioligand [3H]2-(di-N-propylamino)-8-hydroxytetralin from 5-hydroxytryptamine 1A receptor in rat frontal cortex homogenateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Rat)
Solvay Duphar Research Laboratories

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50039819BDBM50039819(1-(2,3-Dihydro-benzo[1,4]dioxin-5-yl)-4-hexyl-pipe...)
Affinity DataKi:  0.5nMAssay Description:Displacement of radioligand [3H]2-(di-N-propylamino)-8-hydroxytetralin from 5-hydroxytryptamine 1A receptor in rat frontal cortex homogenateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Rat)
Solvay Duphar Research Laboratories

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50039805BDBM50039805(1-Benzofuran-7-yl-4-hexyl-piperazine | CHEMBL27558)
Affinity DataKi:  0.540nMAssay Description:Displacement of radioligand [3H]2-(di-N-propylamino)-8-hydroxytetralin from 5-hydroxytryptamine 1A receptor in rat frontal cortex homogenateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Rat)
Solvay Duphar Research Laboratories

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50039796BDBM50039796(1-(2,3-Dihydro-benzo[1,4]dioxin-5-yl)-4-octyl-pipe...)
Affinity DataKi:  0.610nMAssay Description:Displacement of radioligand [3H]2-(di-N-propylamino)-8-hydroxytetralin from 5-hydroxytryptamine 1A receptor in rat frontal cortex homogenateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Rat)
Solvay Duphar Research Laboratories

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50039795BDBM50039795(1-Benzofuran-7-yl-4-pentyl-piperazine | CHEMBL2683...)
Affinity DataKi:  0.810nMAssay Description:Displacement of radioligand [3H]2-(di-N-propylamino)-8-hydroxytetralin from 5-hydroxytryptamine 1A receptor in rat frontal cortex homogenateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Rat)
Solvay Duphar Research Laboratories

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50039826BDBM50039826(1-Decyl-4-(2,3-dihydro-benzo[1,4]dioxin-5-yl)-pipe...)
Affinity DataKi:  1nMAssay Description:Displacement of radioligand [3H]2-(di-N-propylamino)-8-hydroxytetralin from 5-hydroxytryptamine 1A receptor in rat frontal cortex homogenateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Rat)
Solvay Duphar Research Laboratories

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50039832BDBM50039832(1-Benzofuran-7-yl-4-octyl-piperazine | CHEMBL26988)
Affinity DataKi:  1.70nMAssay Description:Displacement of radioligand [3H]2-(di-N-propylamino)-8-hydroxytetralin from 5-hydroxytryptamine 1A receptor in rat frontal cortex homogenateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Rat)
Solvay Duphar Research Laboratories

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50039806BDBM50039806(1-(2,3-Dihydro-benzo[1,4]dioxin-5-yl)-4-pentyl-pip...)
Affinity DataKi:  2.20nMAssay Description:Displacement of radioligand [3H]2-(di-N-propylamino)-8-hydroxytetralin from 5-hydroxytryptamine 1A receptor in rat frontal cortex homogenateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Rat)
Solvay Duphar Research Laboratories

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50005135BDBM50005135(CHEMBL279906 | 1-(3-Chloro-phenyl)-4-hexyl-piperaz...)
Affinity DataKi:  2.70nMAssay Description:Displacement of radioligand [3H]2-(di-N-propylamino)-8-hydroxytetralin from 5-hydroxytryptamine 1A receptor in rat frontal cortex homogenateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Rat)
Solvay Duphar Research Laboratories

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 21393BDBM21393(cid_1220 | CHEMBL56 | 7-(dipropylamino)-5,6,7,8-te...)
Affinity DataKi:  2.80nMAssay Description:Displacement of radioligand [3H]2-(di-N-propylamino)-8-hydroxytetralin from 5-hydroxytryptamine 1A receptor in rat frontal cortex homogenateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Rat)
Solvay Duphar Research Laboratories

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50005127BDBM50005127(1,1-Dioxo-2-[4-(4-pyrimidin-2-yl-piperazin-1-yl)-b...)
Affinity DataKi:  5.5nMAssay Description:Displacement of radioligand [3H]2-(di-N-propylamino)-8-hydroxytetralin from 5-hydroxytryptamine 1A receptor in rat frontal cortex homogenateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Rat)
Solvay Duphar Research Laboratories

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50005140BDBM50005140(CHEMBL27378 | 1-(3-Chloro-phenyl)-4-pentyl-piperaz...)
Affinity DataKi:  5.5nMAssay Description:Displacement of radioligand [3H]2-(di-N-propylamino)-8-hydroxytetralin from 5-hydroxytryptamine 1A receptor in rat frontal cortex homogenate (experim...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Rat)
Solvay Duphar Research Laboratories

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50039809BDBM50039809(1-Benzofuran-7-yl-4-butyl-piperazine | CHEMBL28082...)
Affinity DataKi:  5.90nMAssay Description:Displacement of radioligand [3H]2-(di-N-propylamino)-8-hydroxytetralin from 5-hydroxytryptamine 1A receptor in rat frontal cortex homogenateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Rat)
Solvay Duphar Research Laboratories

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50039816BDBM50039816(1-Benzofuran-7-yl-4-cyclohexylmethyl-piperazine | ...)
Affinity DataKi:  7.70nMAssay Description:Displacement of radioligand [3H]2-(di-N-propylamino)-8-hydroxytetralin from 5-hydroxytryptamine 1A receptor in rat frontal cortex homogenateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Rat)
Solvay Duphar Research Laboratories

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50005140BDBM50005140(CHEMBL27378 | 1-(3-Chloro-phenyl)-4-pentyl-piperaz...)
Affinity DataKi:  7.80nMAssay Description:Displacement of radioligand [3H]2-(di-N-propylamino)-8-hydroxytetralin from 5-hydroxytryptamine 1A receptor in rat frontal cortex homogenate (experim...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Rat)
Solvay Duphar Research Laboratories

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50039804BDBM50039804(1-Benzofuran-7-yl-4-decyl-piperazine | CHEMBL26355)
Affinity DataKi:  8nMAssay Description:Displacement of radioligand [3H]2-(di-N-propylamino)-8-hydroxytetralin from 5-hydroxytryptamine 1A receptor in rat frontal cortex homogenateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Rat)
Solvay Duphar Research Laboratories

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50039830BDBM50039830(1-Benzofuran-7-yl-4-methyl-piperazine | CHEMBL2862...)
Affinity DataKi:  8.10nMAssay Description:Displacement of radioligand [3H]2-(di-N-propylamino)-8-hydroxytetralin from 5-hydroxytryptamine 1A receptor in rat frontal cortex homogenateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Rat)
Solvay Duphar Research Laboratories

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50039793BDBM50039793(CHEMBL554093 | CHEMBL282205 | 1-Cyclohexylmethyl-4...)
Affinity DataKi:  11nMAssay Description:Displacement of radioligand [3H]2-(di-N-propylamino)-8-hydroxytetralin from 5-hydroxytryptamine 1A receptor in rat frontal cortex homogenateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Rat)
Solvay Duphar Research Laboratories

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50005129BDBM50005129(CHEMBL80574 | 1-(3-Chloro-phenyl)-4-octyl-piperazi...)
Affinity DataKi:  11nMAssay Description:Displacement of radioligand [3H]2-(di-N-propylamino)-8-hydroxytetralin from 5-hydroxytryptamine 1A receptor in rat frontal cortex homogenateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Rat)
Solvay Duphar Research Laboratories

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50039803BDBM50039803(1-Butyl-4-(2,3-dihydro-benzo[1,4]dioxin-5-yl)-pipe...)
Affinity DataKi:  12nMAssay Description:Displacement of radioligand [3H]2-(di-N-propylamino)-8-hydroxytetralin from 5-hydroxytryptamine 1A receptor in rat frontal cortex homogenateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Rat)
Solvay Duphar Research Laboratories

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50035042BDBM50035042(1-Benzofuran-7-yl-piperazine | CHEMBL61032)
Affinity DataKi:  13nMAssay Description:Displacement of radioligand [3H]2-(di-N-propylamino)-8-hydroxytetralin from 5-hydroxytryptamine 1A receptor in rat frontal cortex homogenateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Rat)
Solvay Duphar Research Laboratories

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50005134BDBM50005134(CHEMBL26650 | 1-Butyl-4-(3-chloro-phenyl)-piperazi...)
Affinity DataKi:  18nMAssay Description:Displacement of radioligand [3H]2-(di-N-propylamino)-8-hydroxytetralin from 5-hydroxytryptamine 1A receptor in rat frontal cortex homogenateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Rat)
Solvay Duphar Research Laboratories

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50039808BDBM50039808(1-Benzofuran-7-yl-4-cyclopropylmethyl-piperazine |...)
Affinity DataKi:  20nMAssay Description:Displacement of radioligand [3H]2-(di-N-propylamino)-8-hydroxytetralin from 5-hydroxytryptamine 1A receptor in rat frontal cortex homogenateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Rat)
Solvay Duphar Research Laboratories

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50039815BDBM50039815(1-Benzofuran-7-yl-4-ethyl-piperazine | CHEMBL32924...)
Affinity DataKi:  23nMAssay Description:Displacement of radioligand [3H]2-(di-N-propylamino)-8-hydroxytetralin from 5-hydroxytryptamine 1A receptor in rat frontal cortex homogenateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Rat)
Solvay Duphar Research Laboratories

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50039813BDBM50039813(1-(2,3-Dihydro-benzo[1,4]dioxin-5-yl)-4-methyl-pip...)
Affinity DataKi:  24nMAssay Description:Displacement of radioligand [3H]2-(di-N-propylamino)-8-hydroxytetralin from 5-hydroxytryptamine 1A receptor in rat frontal cortex homogenateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Rat)
Solvay Duphar Research Laboratories

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50039820BDBM50039820(1-Benzofuran-7-yl-4-propyl-piperazine | CHEMBL2664...)
Affinity DataKi:  29nMAssay Description:Displacement of radioligand [3H]2-(di-N-propylamino)-8-hydroxytetralin from 5-hydroxytryptamine 1A receptor in rat frontal cortex homogenateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50231235BDBM50231235(CHEMBL441636)
Affinity DataIC50: 30nMAssay Description:Tested for displacement of radioligand [3H]-Naloxone from opiate receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Rat)
Solvay Duphar Research Laboratories

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50035057BDBM50035057(1-(2,3-Dihydro-benzo[1,4]dioxin-5-yl)-piperazine |...)
Affinity DataKi:  40nMAssay Description:Displacement of radioligand [3H]2-(di-N-propylamino)-8-hydroxytetralin from 5-hydroxytryptamine 1A receptor in rat frontal cortex homogenateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50231227BDBM50231227(CHEMBL328583)
Affinity DataIC50: 55nMAssay Description:Tested for displacement of radioligand [3H]-Naloxone from opiate receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Rat)
Solvay Duphar Research Laboratories

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50039828BDBM50039828(1-Benzofuran-7-yl-4-isopropyl-piperazine | CHEMBL2...)
Affinity DataKi:  56nMAssay Description:Displacement of radioligand [3H]2-(di-N-propylamino)-8-hydroxytetralin from 5-hydroxytryptamine 1A receptor in rat frontal cortex homogenateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Rat)
Solvay Duphar Research Laboratories

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50039823BDBM50039823(1-Benzofuran-7-yl-4-cyclohexyl-piperazine | CHEMBL...)
Affinity DataKi:  64nMAssay Description:Displacement of radioligand [3H]2-(di-N-propylamino)-8-hydroxytetralin from 5-hydroxytryptamine 1A receptor in rat frontal cortex homogenateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Rat)
Solvay Duphar Research Laboratories

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50039825BDBM50039825(1-Benzofuran-7-yl-4-isobutyl-piperazine | CHEMBL96...)
Affinity DataKi:  64nMAssay Description:Displacement of radioligand [3H]2-(di-N-propylamino)-8-hydroxytetralin from 5-hydroxytryptamine 1A receptor in rat frontal cortex homogenateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Rat)
Solvay Duphar Research Laboratories

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50039831BDBM50039831(1-(2,3-Dihydro-benzo[1,4]dioxin-5-yl)-4-ethyl-pipe...)
Affinity DataKi:  66nMAssay Description:Displacement of radioligand [3H]2-(di-N-propylamino)-8-hydroxytetralin from 5-hydroxytryptamine 1A receptor in rat frontal cortex homogenateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Rat)
Solvay Duphar Research Laboratories

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50039817BDBM50039817(1-(2,3-Dihydro-benzo[1,4]dioxin-5-yl)-4-propyl-pip...)
Affinity DataKi:  80nMAssay Description:Displacement of radioligand [3H]2-(di-N-propylamino)-8-hydroxytetralin from 5-hydroxytryptamine 1A receptor in rat frontal cortex homogenateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Rat)
Solvay Duphar Research Laboratories

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50005123BDBM50005123(CHEMBL27192 | 1-(3-Chlorophenyl)-4-propylpiperazin...)
Affinity DataKi:  122nMAssay Description:Displacement of radioligand [3H]2-(di-N-propylamino)-8-hydroxytetralin from 5-hydroxytryptamine 1A receptor in rat frontal cortex homogenateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Rat)
Solvay Duphar Research Laboratories

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50001915BDBM50001915(mCPP | 1-(3-chlorophenyl)piperazine | CHEMBL478 | ...)
Affinity DataKi:  143nMAssay Description:Displacement of radioligand [3H]2-(di-N-propylamino)-8-hydroxytetralin from 5-hydroxytryptamine 1A receptor in rat frontal cortex homogenate (experim...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50231230BDBM50231230(CHEMBL328019)
Affinity DataIC50: 150nMAssay Description:Tested for displacement of radioligand [3H]-Naloxone from opiate receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Rat)
Solvay Duphar Research Laboratories

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50005124BDBM50005124(CHEMBL26737 | 1-(3-Chloro-phenyl)-4-methyl-piperaz...)
Affinity DataKi:  152nMAssay Description:Displacement of radioligand [3H]2-(di-N-propylamino)-8-hydroxytetralin from 5-hydroxytryptamine 1A receptor in rat frontal cortex homogenateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Rat)
Solvay Duphar Research Laboratories

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50005142BDBM50005142(CHEMBL307204 | 1-(3-Chloro-phenyl)-4-isopropyl-pip...)
Affinity DataKi:  159nMAssay Description:Displacement of radioligand [3H]2-(di-N-propylamino)-8-hydroxytetralin from 5-hydroxytryptamine 1A receptor in rat frontal cortex homogenateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Rat)
Solvay Duphar Research Laboratories

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50001862BDBM50001862(CHEMBL9666 | 2-METHOXYPHENYLPIPERAZINE | 4-(2-Meth...)
Affinity DataKi:  170nMAssay Description:Displacement of radioligand [3H]2-(di-N-propylamino)-8-hydroxytetralin from 5-hydroxytryptamine 1A receptor in rat frontal cortex homogenateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50231233BDBM50231233(CHEMBL92960)
Affinity DataIC50: 200nMAssay Description:Tested for displacement of radioligand [3H]-Naloxone from opiate receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Rat)
Solvay Duphar Research Laboratories

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50001915BDBM50001915(mCPP | 1-(3-chlorophenyl)piperazine | CHEMBL478 | ...)
Affinity DataKi:  200nMAssay Description:Displacement of radioligand [3H]2-(di-N-propylamino)-8-hydroxytetralin from 5-hydroxytryptamine 1A receptor in rat frontal cortex homogenate (experim...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Rat)
Solvay Duphar Research Laboratories

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50005139BDBM50005139(CHEMBL413527 | 1-(3-Chloro-phenyl)-4-ethyl-piperaz...)
Affinity DataKi:  220nMAssay Description:Displacement of radioligand [3H]2-(di-N-propylamino)-8-hydroxytetralin from 5-hydroxytryptamine 1A receptor in rat frontal cortex homogenateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50231240BDBM50231240(CHEMBL92779)
Affinity DataIC50: 400nMAssay Description:Tested for displacement of radioligand [3H]-Naloxone from opiate receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50026752BDBM50026752(4-Ethoxycarbonyl-1-methyl-4-phenyl-piperidinium | ...)
Affinity DataIC50: 500nMAssay Description:Tested for displacement of radioligand [3H]-Naloxone from opiate receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50231231BDBM50231231(CHEMBL92124)
Affinity DataIC50: 900nMAssay Description:Tested for displacement of radioligand [3H]-Naloxone from opiate receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50231236BDBM50231236(CHEMBL89961)
Affinity DataIC50: 4.00E+3nMAssay Description:Tested for displacement of radioligand [3H]-Naloxone from opiate receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50231241BDBM50231241(CHEMBL285244)
Affinity DataIC50: 5.00E+3nMAssay Description:Tested for displacement of radioligand [3H]-Naloxone from opiate receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50231237BDBM50231237(CHEBI:6125 | Cetobemidone | Cliradon | Cymidon | K...)
Affinity DataIC50: 7.00E+3nMAssay Description:Tested for displacement of radioligand [3H]-Naloxone from opiate receptor; value ranges from 7-10 uMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50231228BDBM50231228(CHEMBL96626)
Affinity DataIC50: 8.00E+3nMAssay Description:Tested for displacement of radioligand [3H]-Naloxone from opiate receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
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