Compile Data Set for Download or QSAR
Report error Found 19 Enz. Inhib. hit(s) with all data for entry = 50006194
TargetTyrosine-protein kinase Lck(Human)
Purdue University

Curated by ChEMBL
LigandPNGBDBM50045933(5-[2-(3,5-dihydroxyphenyl)-(E)-1-ethenyl]-1,3-benz...)
Affinity DataIC50: 1.60E+4nMAssay Description:Tested in vitro for the inhibition of protein-tyrosine kinase p56lck using angiotensin I (1.2 mM) and [gamma-32P]-ATP (50 pM)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetTyrosine-protein kinase Lck(Human)
Purdue University

Curated by ChEMBL
LigandPNGBDBM50045922(5-[2-(3-Hydroxy-phenyl)-vinyl]-benzene-1,3-diol | ...)
Affinity DataIC50: 1.70E+4nMAssay Description:Tested in vitro for the inhibition of protein-tyrosine kinase p56lck using angiotensin I (1.2 mM) and [gamma-32P]-ATP (50 pM)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetTyrosine-protein kinase Lck(Human)
Purdue University

Curated by ChEMBL
LigandPNGBDBM50045921(4-[2-(4-Hydroxy-phenyl)-vinyl]-benzene-1,2-diol | ...)
Affinity DataIC50: 1.90E+4nMAssay Description:Tested in vitro for the inhibition of protein-tyrosine kinase p56lck using angiotensin I (1.2 mM) and [gamma-32P]-ATP (50 pM)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetTyrosine-protein kinase Lck(Human)
Purdue University

Curated by ChEMBL
LigandPNGBDBM50045935(1-(3-benzyloxyphenyl)-2-(4-benzyloxyphenyl)-(E)-1-...)
Affinity DataIC50: 3.60E+4nMAssay Description:Tested in vitro for the inhibition of protein-tyrosine kinase p56lck using angiotensin I (1.2 mM) and [gamma-32P]-ATP (50 pM)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetTyrosine-protein kinase Lck(Human)
Purdue University

Curated by ChEMBL
LigandPNGBDBM50045937(4-[2-(3-Hydroxy-phenyl)-vinyl]-benzene-1,2-diol | ...)
Affinity DataIC50: 5.80E+4nMAssay Description:Tested in vitro for the inhibition of protein-tyrosine kinase p56lck using angiotensin I (1.2 mM) and [gamma-32P]-ATP (50 pM)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetTyrosine-protein kinase Lck(Human)
Purdue University

Curated by ChEMBL
LigandPNGBDBM50045936(CHEMBL69863 | 4-(3,5-dihydroxystyryl)benzene-1,2-d...)
Affinity DataIC50: 6.60E+4nMAssay Description:Tested in vitro for the inhibition of protein-tyrosine kinase p56lck using angiotensin I (1.2 mM) and [gamma-32P]-ATP (50 pM)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetTyrosine-protein kinase Lck(Human)
Purdue University

Curated by ChEMBL
LigandPNGBDBM50045929(4-[2-(3,4-dihydroxyphenyl)-(E)-1-ethenyl]-1,2-benz...)
Affinity DataIC50: 7.40E+4nMAssay Description:Tested in vitro for the inhibition of protein-tyrosine kinase p56lck using angiotensin I (1.2 mM) and [gamma-32P]-ATP (50 pM)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetTyrosine-protein kinase Lck(Human)
Purdue University

Curated by ChEMBL
LigandPNGBDBM23926(5-[(E)-2-(4-hydroxyphenyl)ethenyl]benzene-1,3-diol...)
Affinity DataIC50: 1.12E+5nMAssay Description:Tested in vitro for the inhibition of protein-tyrosine kinase p56lck using angiotensin I (1.2 mM) and [gamma-32P]-ATP (50 pM)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetTyrosine-protein kinase Lck(Human)
Purdue University

Curated by ChEMBL
LigandPNGBDBM50045924((E)-5-(2-phenylethenyl)-1,3-benzenediol | pinosylv...)
Affinity DataIC50: 1.93E+5nMAssay Description:Tested in vitro for the inhibition of protein-tyrosine kinase p56lck using angiotensin I (1.2 mM) and [gamma-32P]-ATP (50 pM)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetTyrosine-protein kinase Lck(Human)
Purdue University

Curated by ChEMBL
LigandPNGBDBM50045934(4-Styryl-benzene-1,2-diol | 3,4-dihydroxy-trans-st...)
Affinity DataIC50: 2.03E+5nMAssay Description:Tested in vitro for the inhibition of protein-tyrosine kinase p56lck using angiotensin I (1.2 mM) and [gamma-32P]-ATP (50 pM)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetTyrosine-protein kinase Lck(Human)
Purdue University

Curated by ChEMBL
LigandPNGBDBM50045926(3-[2-(3-hydroxyphenyl)-(E)-1-ethenyl]phenol | CHEM...)
Affinity DataIC50: 2.34E+5nMAssay Description:Tested in vitro for the inhibition of protein-tyrosine kinase p56lck using angiotensin I (1.2 mM) and [gamma-32P]-ATP (50 pM)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetTyrosine-protein kinase Lck(Human)
Purdue University

Curated by ChEMBL
LigandPNGBDBM50045923(5-(3,5-dihydroxyphenethyl)-1,3-benzenediol | CHEMB...)
Affinity DataIC50: 4.87E+5nMAssay Description:Tested in vitro for the inhibition of protein-tyrosine kinase p56lck using angiotensin I (1.2 mM) and [gamma-32P]-ATP (50 pM)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetTyrosine-protein kinase Lck(Human)
Purdue University

Curated by ChEMBL
LigandPNGBDBM50045930(4-[2-(3,5-dihydroxyphenyl)ethyl]benzene-1,2-diol |...)
Affinity DataIC50: 1.56E+6nMAssay Description:Tested in vitro for the inhibition of protein-tyrosine kinase p56lck using angiotensin I (1.2 mM) and [gamma-32P]-ATP (50 pM)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetTyrosine-protein kinase Lck(Human)
Purdue University

Curated by ChEMBL
LigandPNGBDBM50045920(1,3-Bis-benzyloxy-5-[2-(4-benzyloxy-phenyl)-vinyl]...)
Affinity DataIC50: 2.03E+6nMAssay Description:Tested in vitro for the inhibition of protein-tyrosine kinase p56lck using angiotensin I (1.2 mM) and [gamma-32P]-ATP (50 pM)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetTyrosine-protein kinase Lck(Human)
Purdue University

Curated by ChEMBL
LigandPNGBDBM50045932(1,3-Bis-benzyloxy-5-styryl-benzene | 1,3-Bis-benzy...)
Affinity DataIC50: 2.03E+6nMAssay Description:Tested in vitro for the inhibition of protein-tyrosine kinase p56lck using angiotensin I (1.2 mM) and [gamma-32P]-ATP (50 pM)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetTyrosine-protein kinase Lck(Human)
Purdue University

Curated by ChEMBL
LigandPNGBDBM50045927(1,2-Bis-benzyloxy-4-[2-(3-benzyloxy-phenyl)-vinyl]...)
Affinity DataIC50: 2.03E+6nMAssay Description:Tested in vitro for the inhibition of protein-tyrosine kinase p56lck using angiotensin I (1.2 mM) and [gamma-32P]-ATP (50 pM)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetTyrosine-protein kinase Lck(Human)
Purdue University

Curated by ChEMBL
LigandPNGBDBM50045928(1,3-Bis-benzyloxy-5-[2-(3-benzyloxy-phenyl)-vinyl]...)
Affinity DataIC50: 2.03E+6nMAssay Description:Tested in vitro for the inhibition of protein-tyrosine kinase p56lck using angiotensin I (1.2 mM) and [gamma-32P]-ATP (50 pM)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetTyrosine-protein kinase Lck(Human)
Purdue University

Curated by ChEMBL
LigandPNGBDBM50045931(1,2-Bis-benzyloxy-4-styryl-benzene | CHEMBL101337)
Affinity DataIC50: 2.03E+6nMAssay Description:Tested in vitro for the inhibition of protein-tyrosine kinase p56lck using angiotensin I (1.2 mM) and [gamma-32P]-ATP (50 pM)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetTyrosine-protein kinase Lck(Human)
Purdue University

Curated by ChEMBL
LigandPNGBDBM50045925(1,2-Bis-benzyloxy-4-[2-(4-benzyloxy-phenyl)-vinyl]...)
Affinity DataIC50: 2.03E+6nMAssay Description:Tested in vitro for the inhibition of protein-tyrosine kinase p56lck using angiotensin I (1.2 mM) and [gamma-32P]-ATP (50 pM)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed