Compile Data Set for Download or QSAR
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Report error Found 39 Enz. Inhib. hit(s) with all data for entry = 50006301
TargetThromboxane A2 receptor(Human)
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50456020(CHEMBL2368531)
Affinity DataKd:  22nMAssay Description:Inhibitory binding activity against TXA2 receptor in human platelet membrane, using [3H]-SQ 29548 as the radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetThromboxane A2 receptor(Human)
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50047303((3-{3-[4-(4-Cyclohexyl-butylcarbamoyl)-oxazol-2-yl...)
Affinity DataKd:  1.20nMAssay Description:Inhibitory binding activity against TXA2 receptor in human platelet membrane, using [3H]-SQ 29548 as the radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetThromboxane A2 receptor(Human)
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50047266(3-(2-{3-[4-(4-Cyclohexyl-butylcarbamoyl)-oxazol-2-...)
Affinity DataKd:  0.100nMAssay Description:Inhibitory binding activity against TXA2 receptor in human platelet membrane, using [3H]-SQ 29548 as the radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetThromboxane A2 receptor(Human)
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50047267(2-{3-[2-(3-Hydroxy-propyl)-benzyl]-7-oxa-bicyclo[2...)
Affinity DataKd:  112nMAssay Description:Inhibitory binding activity against TXA2 receptor in human platelet membrane, using [3H]-SQ 29548 as the radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetThromboxane A2 receptor(Human)
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50047268(3-(2-{3-[4-(4-Cyclohexylcarbamoyl-butylcarbamoyl)-...)
Affinity DataKd:  22nMAssay Description:Inhibitory binding activity against TXA2 receptor in human platelet membrane, using [3H]-SQ 29548 as the radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetThromboxane A2 receptor(Human)
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50047270(3-[2-(3-{4-[4-(4-Methoxy-phenyl)-butylcarbamoyl]-o...)
Affinity DataKd:  0.300nMAssay Description:Inhibitory binding activity against TXA2 receptor in human platelet membrane, using [3H]-SQ 29548 as the radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetThromboxane A2 receptor(Human)
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50047269(3-(2-{3-[4-(5,5,5-Trifluoro-pentylcarbamoyl)-oxazo...)
Affinity DataKd:  4.80nMAssay Description:Inhibitory binding activity against TXA2 receptor in human platelet membrane, using [3H]-SQ 29548 as the radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetThromboxane A2 receptor(Human)
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50047271(3-{2-[3-(4-tert-Butylcarbamoyl-oxazol-2-yl)-7-oxa-...)
Affinity DataKd:  19nMAssay Description:Inhibitory binding activity against TXA2 receptor in human platelet membrane, using [3H]-SQ 29548 as the radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetThromboxane A2 receptor(Human)
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50047272(3-(2-{3-[4-(4-Cyclohexyl-butylcarbamoyl)-oxazol-2-...)
Affinity DataKd:  36nMAssay Description:Inhibitory binding activity against TXA2 receptor in human platelet membrane, using [3H]-SQ 29548 as the radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetThromboxane A2 receptor(Human)
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50047273(2-{3-[2-(2-Carboxy-ethyl)-benzyl]-7-oxa-bicyclo[2....)
Affinity DataKd:  1nMAssay Description:Inhibitory binding activity against TXA2 receptor in human platelet membrane, using [3H]-SQ 29548 as the radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetThromboxane A2 receptor(Human)
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50047275(3-{2-[3-(4-Methylcarbamoyl-oxazol-2-yl)-7-oxa-bicy...)
Affinity DataKd:  45nMAssay Description:Inhibitory binding activity against TXA2 receptor in human platelet membrane, using [3H]-SQ 29548 as the radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetThromboxane A2 receptor(Human)
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50047274(3-{2-[3-(4-Pentylcarbamoyl-oxazol-2-yl)-7-oxa-bicy...)
Affinity DataKd:  4nMAssay Description:Inhibitory binding activity against TXA2 receptor in human platelet membrane, using [3H]-SQ 29548 as the radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetThromboxane A2 receptor(Human)
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50047276(3-(2-{3-[4-(Methyl-pentyl-carbamoyl)-oxazol-2-yl]-...)
Affinity DataKd:  11nMAssay Description:Inhibitory binding activity against TXA2 receptor in human platelet membrane, using [3H]-SQ 29548 as the radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetThromboxane A2 receptor(Human)
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50047277((2-{3-[4-(4-Cyclohexyl-butylcarbamoyl)-oxazol-2-yl...)
Affinity DataKd:  3.20nMAssay Description:Inhibitory binding activity against TXA2 receptor in human platelet membrane, using [3H]-SQ 29548 as the radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetThromboxane A2 receptor(Human)
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50047278(3-[2-(3-{4-[4-(4-Chloro-phenyl)-butylcarbamoyl]-ox...)
Affinity DataKd:  0.200nMAssay Description:Inhibitory binding activity against TXA2 receptor in human platelet membrane, using [3H]-SQ 29548 as the radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetThromboxane A2 receptor(Human)
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50047279(3-{2-[3-(4-Propylcarbamoyl-oxazol-2-yl)-7-oxa-bicy...)
Affinity DataKd:  10nMAssay Description:Inhibitory binding activity against TXA2 receptor in human platelet membrane, using [3H]-SQ 29548 as the radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetThromboxane A2 receptor(Human)
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50047281(2-{3-[2-(3-Methanesulfonylamino-3-oxo-propyl)-benz...)
Affinity DataKd:  1.60nMAssay Description:Inhibitory binding activity against TXA2 receptor in human platelet membrane, using [3H]-SQ 29548 as the radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetThromboxane A2 receptor(Human)
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50047280(3-[2-(3-{4-[4-(4-Hydroxy-phenyl)-butylcarbamoyl]-o...)
Affinity DataKd:  0.5nMAssay Description:Inhibitory binding activity against TXA2 receptor in human platelet membrane, using [3H]-SQ 29548 as the radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetThromboxane A2 receptor(Human)
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50047282(3-[2-(3-{4-[2-(4-Chloro-phenyl)-ethylcarbamoyl]-ox...)
Affinity DataKd:  1.30nMAssay Description:Inhibitory binding activity against TXA2 receptor in human platelet membrane, using [3H]-SQ 29548 as the radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetThromboxane A2 receptor(Human)
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50047286((2-{3-[4-(4-Cyclohexyl-butylcarbamoyl)-oxazol-2-yl...)
Affinity DataKd:  19nMAssay Description:Inhibitory binding activity against TXA2 receptor in human platelet membrane, using [3H]-SQ 29548 as the radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetThromboxane A2 receptor(Human)
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50047283(3-{2-[3-(4-Phenethylcarbamoyl-oxazol-2-yl)-7-oxa-b...)
Affinity DataKd:  0.700nMAssay Description:Inhibitory binding activity against TXA2 receptor in human platelet membrane, using [3H]-SQ 29548 as the radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetThromboxane A2 receptor(Human)
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50047285(3-[2-(3-{4-[4-(4-Fluoro-phenyl)-butylcarbamoyl]-ox...)
Affinity DataKd:  3.90nMAssay Description:Inhibitory binding activity against TXA2 receptor in human platelet membrane, using [3H]-SQ 29548 as the radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetThromboxane A2 receptor(Human)
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50047284(3-{2-[3-(4-Heptylcarbamoyl-oxazol-2-yl)-7-oxa-bicy...)
Affinity DataKd:  0.200nMAssay Description:Inhibitory binding activity against TXA2 receptor in human platelet membrane, using [3H]-SQ 29548 as the radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetThromboxane A2 receptor(Human)
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50047289(3-(2-{3-[4-(5,5-Dimethyl-hexylcarbamoyl)-oxazol-2-...)
Affinity DataKd:  0.600nMAssay Description:Inhibitory binding activity against TXA2 receptor in human platelet membrane, using [3H]-SQ 29548 as the radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetThromboxane A2 receptor(Human)
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50047288(3-(2-{3-[4-(2-Cyclohexyl-ethylcarbamoyl)-oxazol-2-...)
Affinity DataKd:  0.700nMAssay Description:Inhibitory binding activity against TXA2 receptor in human platelet membrane, using [3H]-SQ 29548 as the radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetThromboxane A2 receptor(Human)
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50047296(3-(2-{3-[4-(3,3-Dimethyl-butylcarbamoyl)-oxazol-2-...)
Affinity DataKd:  2.90nMAssay Description:Inhibitory binding activity against TXA2 receptor in human platelet membrane, using [3H]-SQ 29548 as the radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetThromboxane A2 receptor(Human)
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50047295(3-{2-[3-(4-Isopropylcarbamoyl-oxazol-2-yl)-7-oxa-b...)
Affinity DataKd:  26nMAssay Description:Inhibitory binding activity against TXA2 receptor in human platelet membrane, using [3H]-SQ 29548 as the radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetThromboxane A2 receptor(Human)
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50047291(3-(2-{3-[4-(6-Cyclohexyl-hexanoyl)-oxazol-2-yl]-7-...)
Affinity DataKd:  0.0500nMAssay Description:Inhibitory binding activity against TXA2 receptor in human platelet membrane, using [3H]-SQ 29548 as the radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetThromboxane A2 receptor(Human)
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50047290(3-{2-[3-(4-Decylcarbamoyl-oxazol-2-yl)-7-oxa-bicyc...)
Affinity DataKd:  5.80nMAssay Description:Inhibitory binding activity against TXA2 receptor in human platelet membrane, using [3H]-SQ 29548 as the radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetThromboxane A2 receptor(Human)
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50047292(3-[2-(3-{4-[4-(4-Methylsulfanyl-phenyl)-butylcarba...)
Affinity DataKd:  2.90nMAssay Description:Inhibitory binding activity against TXA2 receptor in human platelet membrane, using [3H]-SQ 29548 as the radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetThromboxane A2 receptor(Human)
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50047293(3-(2-{3-[4-(4-Cyclohexyl-butylcarbamoyl)-oxazol-2-...)
Affinity DataKd:  18nMAssay Description:Inhibitory binding activity against TXA2 receptor in human platelet membrane, using [3H]-SQ 29548 as the radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetThromboxane A2 receptor(Human)
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50047298(3-(2-{3-[4-(1,1-Dimethyl-propylcarbamoyl)-oxazol-2...)
Affinity DataKd:  0.800nMAssay Description:Inhibitory binding activity against TXA2 receptor in human platelet membrane, using [3H]-SQ 29548 as the radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetThromboxane A2 receptor(Human)
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50047294(4-(2-{3-[4-(4-Cyclohexyl-butylcarbamoyl)-oxazol-2-...)
Affinity DataKd:  0.850nMAssay Description:Inhibitory binding activity against TXA2 receptor in human platelet membrane, using [3H]-SQ 29548 as the radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetThromboxane A2 receptor(Human)
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50047297(3-{2-[3-(4-Cyclohexylcarbamoyl-oxazol-2-yl)-7-oxa-...)
Affinity DataKd:  4.5nMAssay Description:Inhibitory binding activity against TXA2 receptor in human platelet membrane, using [3H]-SQ 29548 as the radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetThromboxane A2 receptor(Human)
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50047299(3-{2-[3-(4-Hept-6-ynylcarbamoyl-oxazol-2-yl)-7-oxa...)
Affinity DataKd:  4.70nMAssay Description:Inhibitory binding activity against TXA2 receptor in human platelet membrane, using [3H]-SQ 29548 as the radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetThromboxane A2 receptor(Human)
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50047300(3-(2-{3-[4-(4-Phenyl-butylcarbamoyl)-oxazol-2-yl]-...)
Affinity DataKd:  0.300nMAssay Description:Inhibitory binding activity against TXA2 receptor in human platelet membrane, using [3H]-SQ 29548 as the radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetThromboxane A2 receptor(Human)
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50047302(3-(2-{3-[4-(4-Cyclohexyl-butylthiocarbamoyl)-oxazo...)
Affinity DataKd:  11nMAssay Description:Inhibitory binding activity against TXA2 receptor in human platelet membrane, using [3H]-SQ 29548 as the radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetThromboxane A2 receptor(Human)
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50047301(CHEMBL280786 | [3-(2-{3-[4-(4-Cyclohexyl-butylcarb...)
Affinity DataKd:  16nMAssay Description:Inhibitory binding activity against TXA2 receptor in human platelet membrane, using [3H]-SQ 29548 as the radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetThromboxane A2 receptor(Human)
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50047265(3-(2-{3-[4-(5-Hydroxy-pentylcarbamoyl)-oxazol-2-yl...)
Affinity DataKd:  20nMAssay Description:Inhibitory binding activity against TXA2 receptor in human platelet membrane, using [3H]-SQ 29548 as the radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed