Compile Data Set for Download or QSAR
maximum 50k data
Report error Found 50 Enz. Inhib. hit(s) with all data for entry = 50006502
TargetEndothelin-1 receptor(Rat)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50049983(2-[(R)-1-{(S)-2-[(Azepane-1-carbonyl)-amino]-4-met...)
Affinity DataIC50:  570nMAssay Description:Inhibition of Endothelin-1 binding to Endothelin A receptor binding sites in MMQ cell membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetEndothelin-1 receptor(Rat)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50049996(2-[(R)-1-{(S)-2-[(Azepane-1-carbonyl)-amino]-4-met...)
Affinity DataIC50:  730nMAssay Description:Inhibition of Endothelin-1 binding to Endothelin A receptor binding sites in MMQ cell membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetEndothelin-1 receptor(Rat)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50049981(2-[(R)-1-{(S)-2-[(Azepane-1-carbonyl)-amino]-4-met...)
Affinity DataIC50:  1.43E+3nMAssay Description:Inhibition of Endothelin-1 binding to Endothelin A receptor binding sites in MMQ cell membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetEndothelin-1 receptor(Rat)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50049998(2-[(R)-1-{(S)-2-[(Azepane-1-carbonyl)-amino]-4-met...)
Affinity DataIC50:  1.50E+3nMAssay Description:Inhibition of Endothelin-1 binding to Endothelin A receptor binding sites in MMQ cell membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetEndothelin-1 receptor(Rat)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50049994(2-[(R)-1-{(S)-2-[(Azepane-1-carbonyl)-amino]-4-met...)
Affinity DataIC50:  1.90E+3nMAssay Description:Inhibition of Endothelin-1 binding to Endothelin A receptor binding sites in MMQ cell membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetEndothelin-1 receptor(Rat)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50049978(2-[(R)-1-{(S)-2-[(Azepane-1-carbonyl)-amino]-4-met...)
Affinity DataIC50:  2.50E+3nMAssay Description:Inhibition of Endothelin-1 binding to Endothelin A receptor binding sites in MMQ cell membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetEndothelin-1 receptor(Rat)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50049974(2-[(R)-1-{(S)-2-[(Azepane-1-carbonyl)-amino]-4-met...)
Affinity DataIC50:  3.70E+3nMAssay Description:Inhibition of Endothelin-1 binding to Endothelin A receptor binding sites in MMQ cell membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetEndothelin-1 receptor(Rat)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50049975(2-[(R)-1-{(S)-2-[(Azepane-1-carbonyl)-amino]-4-met...)
Affinity DataIC50:  5.20E+3nMAssay Description:Inhibition of Endothelin-1 binding to Endothelin A receptor binding sites in MMQ cell membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetEndothelin-1 receptor(Rat)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50049992(2-[(R)-1-{(S)-2-[(Azepane-1-carbonyl)-amino]-4-met...)
Affinity DataIC50:  7.30E+3nMAssay Description:Inhibition of Endothelin-1 binding to Endothelin A receptor binding sites in MMQ cell membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetEndothelin-1 receptor(Rat)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50049997(2-[(R)-1-{(S)-2-[(Azepane-1-carbonyl)-amino]-4-met...)
Affinity DataIC50:  7.70E+3nMAssay Description:Inhibition of Endothelin-1 binding to Endothelin A receptor binding sites in MMQ cell membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetEndothelin-1 receptor(Rat)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50049995(2-[(R)-1-{(S)-2-[(Azepane-1-carbonyl)-amino]-4-met...)
Affinity DataIC50:  7.80E+3nMAssay Description:Inhibition of Endothelin-1 binding to Endothelin A receptor binding sites in MMQ cell membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetEndothelin-1 receptor(Rat)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50049991(2-[(R)-1-{(S)-2-[(Azepane-1-carbonyl)-amino]-4-met...)
Affinity DataIC50:  8.00E+3nMAssay Description:Inhibition of Endothelin-1 binding to Endothelin A receptor binding sites in MMQ cell membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetEndothelin-1 receptor(Rat)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50049987(2-[(R)-1-{(S)-2-[(Azepane-1-carbonyl)-amino]-4-met...)
Affinity DataIC50:  1.10E+4nMAssay Description:Inhibition of Endothelin-1 binding to Endothelin A receptor binding sites in MMQ cell membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetEndothelin-1 receptor(Rat)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50049989(2-[(R)-1-{(S)-2-[(Azepane-1-carbonyl)-amino]-4-met...)
Affinity DataIC50:  1.60E+4nMAssay Description:Inhibition of Endothelin-1 binding to Endothelin A receptor binding sites in MMQ cell membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetEndothelin-1 receptor(Rat)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50049979(2-[(R)-1-{(S)-2-[(Azepane-1-carbonyl)-amino]-4-met...)
Affinity DataIC50:  2.40E+4nMAssay Description:Inhibition of Endothelin-1 binding to Endothelin A receptor binding sites in MMQ cell membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetEndothelin-1 receptor(Rat)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50049993(2-[(R)-1-{(S)-2-[(Azepane-1-carbonyl)-amino]-4-met...)
Affinity DataIC50:  3.60E+4nMAssay Description:Inhibition of Endothelin-1 binding to Endothelin A receptor binding sites in MMQ cell membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetEndothelin-1 receptor(Rat)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50049988(2-[(R)-1-{(S)-2-[(Azepane-1-carbonyl)-amino]-4-met...)
Affinity DataIC50:  3.90E+4nMAssay Description:Inhibition of Endothelin-1 binding to Endothelin A receptor binding sites in MMQ cell membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetEndothelin-1 receptor(Rat)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50049976(2-[(R)-1-{(S)-2-[(Azepane-1-carbonyl)-amino]-4-met...)
Affinity DataIC50:  4.10E+4nMAssay Description:Inhibition of Endothelin-1 binding to Endothelin A receptor binding sites in MMQ cell membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetEndothelin-1 receptor(Rat)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50049977(2-[(R)-1-{(S)-2-[(Azepane-1-carbonyl)-amino]-4-met...)
Affinity DataIC50:  4.10E+4nMAssay Description:Inhibition of Endothelin-1 binding to Endothelin A receptor binding sites in MMQ cell membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetEndothelin-1 receptor(Rat)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50049985(2-[(R)-1-{(S)-2-[(Azepane-1-carbonyl)-amino]-4-met...)
Affinity DataIC50:  5.10E+4nMAssay Description:Inhibition of Endothelin-1 binding to Endothelin A receptor binding sites in MMQ cell membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetEndothelin-1 receptor(Rat)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50049980(2-[(R)-1-{(S)-2-[(Azepane-1-carbonyl)-amino]-4-met...)
Affinity DataIC50:  5.10E+4nMAssay Description:Inhibition of Endothelin-1 binding to Endothelin A receptor binding sites in MMQ cell membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetEndothelin receptor type B(Pig)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50049978(2-[(R)-1-{(S)-2-[(Azepane-1-carbonyl)-amino]-4-met...)
Affinity DataIC50: >6.00E+4nMAssay Description:Inhibition of Endothelin-3(ET-3) binding to Endothelin B receptor binding sites in porcine cerebellar membranes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetEndothelin receptor type B(Pig)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50049974(2-[(R)-1-{(S)-2-[(Azepane-1-carbonyl)-amino]-4-met...)
Affinity DataIC50:  6.50E+4nMAssay Description:Inhibition of Endothelin-3(ET-3) binding to Endothelin B receptor binding sites in porcine cerebellar membranes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetEndothelin-1 receptor(Rat)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50049982((R)-2-{[2-{(S)-1-[(Azepane-1-carbonyl)-amino]-3-me...)
Affinity DataIC50:  6.80E+4nMAssay Description:Inhibition of Endothelin-1 binding to Endothelin A receptor binding sites in MMQ cell membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetEndothelin receptor type B(Pig)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50049991(2-[(R)-1-{(S)-2-[(Azepane-1-carbonyl)-amino]-4-met...)
Affinity DataIC50:  6.90E+4nMAssay Description:Inhibition of Endothelin-3(ET-3) binding to Endothelin B receptor binding sites in porcine cerebellar membranes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetEndothelin receptor type B(Pig)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50049994(2-[(R)-1-{(S)-2-[(Azepane-1-carbonyl)-amino]-4-met...)
Affinity DataIC50: >8.00E+4nMAssay Description:Inhibition of Endothelin-3(ET-3) binding to Endothelin B receptor binding sites in porcine cerebellar membranes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetEndothelin receptor type B(Pig)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50049992(2-[(R)-1-{(S)-2-[(Azepane-1-carbonyl)-amino]-4-met...)
Affinity DataIC50: >8.50E+4nMAssay Description:Inhibition of Endothelin-3(ET-3) binding to Endothelin B receptor binding sites in porcine cerebellar membranes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetEndothelin-1 receptor(Rat)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50049986((R)-2-{[2-{(S)-1-[(Azepane-1-carbonyl)-amino]-3-me...)
Affinity DataIC50: >9.00E+4nMAssay Description:Inhibition of Endothelin-1 binding to Endothelin A receptor binding sites in MMQ cell membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetEndothelin receptor type B(Pig)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50049988(2-[(R)-1-{(S)-2-[(Azepane-1-carbonyl)-amino]-4-met...)
Affinity DataIC50: >9.00E+4nMAssay Description:Inhibition of Endothelin-3(ET-3) binding to Endothelin B receptor binding sites in porcine cerebellar membranes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetEndothelin receptor type B(Pig)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50049989(2-[(R)-1-{(S)-2-[(Azepane-1-carbonyl)-amino]-4-met...)
Affinity DataIC50:  9.00E+4nMAssay Description:Inhibition of Endothelin-3(ET-3) binding to Endothelin B receptor binding sites in porcine cerebellar membranes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetEndothelin-1 receptor(Rat)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50049990((R)-2-{[2-{(S)-1-[(Azepane-1-carbonyl)-amino]-3-me...)
Affinity DataIC50: >9.00E+4nMAssay Description:Inhibition of Endothelin-1 binding to Endothelin A receptor binding sites in MMQ cell membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetEndothelin receptor type B(Pig)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50049983(2-[(R)-1-{(S)-2-[(Azepane-1-carbonyl)-amino]-4-met...)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of Endothelin-3(ET-3) binding to Endothelin B receptor binding sites in porcine cerebellar membranes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetEndothelin receptor type B(Pig)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50049990((R)-2-{[2-{(S)-1-[(Azepane-1-carbonyl)-amino]-3-me...)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of Endothelin-3(ET-3) binding to Endothelin B receptor binding sites in porcine cerebellar membranes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetEndothelin receptor type B(Pig)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50049984((R)-2-{[2-{(S)-1-[(Azepane-1-carbonyl)-amino]-3-me...)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of Endothelin-3(ET-3) binding to Endothelin B receptor binding sites in porcine cerebellar membranes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetEndothelin receptor type B(Pig)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50049993(2-[(R)-1-{(S)-2-[(Azepane-1-carbonyl)-amino]-4-met...)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of Endothelin-3(ET-3) binding to Endothelin B receptor binding sites in porcine cerebellar membranes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetEndothelin receptor type B(Pig)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50049987(2-[(R)-1-{(S)-2-[(Azepane-1-carbonyl)-amino]-4-met...)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of Endothelin-3(ET-3) binding to Endothelin B receptor binding sites in porcine cerebellar membranes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetEndothelin-1 receptor(Rat)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50049984((R)-2-{[2-{(S)-1-[(Azepane-1-carbonyl)-amino]-3-me...)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of Endothelin-1 binding to Endothelin A receptor binding sites in MMQ cell membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetEndothelin receptor type B(Pig)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50049986((R)-2-{[2-{(S)-1-[(Azepane-1-carbonyl)-amino]-3-me...)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of Endothelin-3(ET-3) binding to Endothelin B receptor binding sites in porcine cerebellar membranes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetEndothelin receptor type B(Pig)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50049982((R)-2-{[2-{(S)-1-[(Azepane-1-carbonyl)-amino]-3-me...)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of Endothelin-3(ET-3) binding to Endothelin B receptor binding sites in porcine cerebellar membranes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetEndothelin receptor type B(Pig)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50049981(2-[(R)-1-{(S)-2-[(Azepane-1-carbonyl)-amino]-4-met...)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of Endothelin-3(ET-3) binding to Endothelin B receptor binding sites in porcine cerebellar membranes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetEndothelin receptor type B(Pig)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50049979(2-[(R)-1-{(S)-2-[(Azepane-1-carbonyl)-amino]-4-met...)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of Endothelin-3(ET-3) binding to Endothelin B receptor binding sites in porcine cerebellar membranes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetEndothelin receptor type B(Pig)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50049980(2-[(R)-1-{(S)-2-[(Azepane-1-carbonyl)-amino]-4-met...)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of Endothelin-3(ET-3) binding to Endothelin B receptor binding sites in porcine cerebellar membranes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetEndothelin receptor type B(Pig)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50049975(2-[(R)-1-{(S)-2-[(Azepane-1-carbonyl)-amino]-4-met...)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of Endothelin-3(ET-3) binding to Endothelin B receptor binding sites in porcine cerebellar membranes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetEndothelin receptor type B(Pig)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50049977(2-[(R)-1-{(S)-2-[(Azepane-1-carbonyl)-amino]-4-met...)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of Endothelin-3(ET-3) binding to Endothelin B receptor binding sites in porcine cerebellar membranes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetEndothelin receptor type B(Pig)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50049976(2-[(R)-1-{(S)-2-[(Azepane-1-carbonyl)-amino]-4-met...)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of Endothelin-3(ET-3) binding to Endothelin B receptor binding sites in porcine cerebellar membranes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetEndothelin receptor type B(Pig)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50049985(2-[(R)-1-{(S)-2-[(Azepane-1-carbonyl)-amino]-4-met...)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of Endothelin-3(ET-3) binding to Endothelin B receptor binding sites in porcine cerebellar membranes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetEndothelin receptor type B(Pig)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50049996(2-[(R)-1-{(S)-2-[(Azepane-1-carbonyl)-amino]-4-met...)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of Endothelin-3(ET-3) binding to Endothelin B receptor binding sites in porcine cerebellar membranes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetEndothelin receptor type B(Pig)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50049998(2-[(R)-1-{(S)-2-[(Azepane-1-carbonyl)-amino]-4-met...)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of Endothelin-3(ET-3) binding to Endothelin B receptor binding sites in porcine cerebellar membranes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetEndothelin receptor type B(Pig)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50049997(2-[(R)-1-{(S)-2-[(Azepane-1-carbonyl)-amino]-4-met...)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of Endothelin-3(ET-3) binding to Endothelin B receptor binding sites in porcine cerebellar membranes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetEndothelin receptor type B(Pig)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50049995(2-[(R)-1-{(S)-2-[(Azepane-1-carbonyl)-amino]-4-met...)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of Endothelin-3(ET-3) binding to Endothelin B receptor binding sites in porcine cerebellar membranes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed