Compile Data Set for Download or QSAR
Report error Found 13 Enz. Inhib. hit(s) with all data for entry = 50041250
TargetB2 bradykinin receptor(Rat)
Cortech

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50408045BDBM50408045(CHEMBL2372278)
Affinity DataKd:  0.490nMAssay Description:In vitro Bradykinin receptor B2 antagonist activity by using rat uterus functional assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/20/2013
Entry Details Article
PubMed
TargetB2 bradykinin receptor(Rat)
Cortech

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50408053BDBM50408053(CHEMBL3038094)
Affinity DataKd:  3.16nMAssay Description:In vitro Bradykinin receptor B2 antagonist activity by using rat uterus functional assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/20/2013
Entry Details Article
PubMed
TargetB2 bradykinin receptor(Rat)
Cortech

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50408047BDBM50408047(CHEMBL3038096)
Affinity DataKd:  18.6nMAssay Description:In vitro Bradykinin receptor B2 antagonist activity by using rat uterus functional assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/20/2013
Entry Details Article
PubMed
TargetB2 bradykinin receptor(Rat)
Cortech

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50408055BDBM50408055(CHEMBL3038102)
Affinity DataKd:  50.1nMAssay Description:In vitro Bradykinin receptor B2 antagonist activity by using rat uterus functional assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/20/2013
Entry Details Article
PubMed
TargetB2 bradykinin receptor(Rat)
Cortech

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50408044BDBM50408044(CHEMBL3038104)
Affinity DataKd:  174nMAssay Description:In vitro Bradykinin receptor B2 antagonist activity by using rat uterus functional assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/20/2013
Entry Details Article
PubMed
TargetB1 bradykinin receptor(Human)
Cortech

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50408044BDBM50408044(CHEMBL3038104)
Affinity DataIC50: 1.62E+3nMAssay Description:In vitro Bradykinin receptor B1 antagonist activity in functional tissue within rabbit aortaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/20/2013
Entry Details Article
PubMed
TargetB1 bradykinin receptor(Human)
Cortech

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50408047BDBM50408047(CHEMBL3038096)
Affinity DataIC50: 3.02E+3nMAssay Description:In vitro Bradykinin receptor B1 antagonist activity in functional tissue within rabbit aortaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/20/2013
Entry Details Article
PubMed
TargetB1 bradykinin receptor(Human)
Cortech

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50408058BDBM50408058(CHEMBL2028982)
Affinity DataIC50: 1.00E+4nMAssay Description:In vitro Bradykinin receptor B1 antagonist activity in functional tissue within rabbit aortaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/20/2013
Entry Details Article
PubMed
TargetB1 bradykinin receptor(Human)
Cortech

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50408055BDBM50408055(CHEMBL3038102)
Affinity DataIC50: 1.00E+4nMAssay Description:In vitro Bradykinin receptor B1 antagonist activity in functional tissue within rabbit aortaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/20/2013
Entry Details Article
PubMed
TargetB1 bradykinin receptor(Human)
Cortech

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50408053BDBM50408053(CHEMBL3038094)
Affinity DataIC50: 1.00E+4nMAssay Description:In vitro Bradykinin receptor B1 antagonist activity in functional tissue within rabbit aortaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/20/2013
Entry Details Article
PubMed
TargetB1 bradykinin receptor(Human)
Cortech

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50408049BDBM50408049(CHEMBL3038098)
Affinity DataIC50: 1.00E+4nMAssay Description:In vitro Bradykinin receptor B1 antagonist activity in functional tissue within rabbit aortaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/20/2013
Entry Details Article
PubMed
TargetB1 bradykinin receptor(Human)
Cortech

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50408048BDBM50408048(CHEMBL3038099)
Affinity DataIC50: 1.00E+4nMAssay Description:In vitro Bradykinin receptor B1 antagonist activity in functional tissue within rabbit aortaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/20/2013
Entry Details Article
PubMed
TargetB1 bradykinin receptor(Human)
Cortech

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50408052BDBM50408052(CHEMBL3038097)
Affinity DataIC50: 1.00E+4nMAssay Description:In vitro Bradykinin receptor B1 antagonist activity in functional tissue within rabbit aortaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/20/2013
Entry Details Article
PubMed