Compile Data Set for Download or QSAR
Report error Found 11 Enz. Inhib. hit(s) with all data for entry = 50036434
TargetTransient receptor potential cation channel subfamily V member 1(Rat)
Institute For Medical Research

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50366620BDBM50366620(RESINIFERATOXIN)
Affinity DataKi:  0.120nMAssay Description:Binding affinity against Vanilloid receptor in dorsal Root Ganglion (DRG) membranes using [3H]RTX binding assay.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/1/2012
Entry Details Article
PubMed
TargetTransient receptor potential cation channel subfamily V member 1(Rat)
Institute For Medical Research

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50366620BDBM50366620(RESINIFERATOXIN)
Affinity DataKi:  0.120nMAssay Description:Binding affinity against Vanilloid receptor in dorsal Root Ganglion (DRG) membranes using [3H]RTX binding assay.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/1/2012
Entry Details Article
PubMed
TargetTransient receptor potential cation channel subfamily V member 1(Rat)
Institute For Medical Research

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50052327BDBM50052327(6-hydroxy-15-isopropenyl-4,13,17-trimethyl-5-oxo-(...)
Affinity DataKi:  0.170nMAssay Description:Binding affinity against Vanilloid receptor in dorsal Root Ganglion (DRG) membranes using [3H]RTX binding assay.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/1/2012
Entry Details Article
PubMed
TargetTransient receptor potential cation channel subfamily V member 1(Rat)
Institute For Medical Research

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50052320BDBM50052320(13-benzyl-6-hydroxy-15-isopropenyl-4,17-dimethyl-5...)
Affinity DataKi:  1nMAssay Description:Binding affinity against Vanilloid receptor in dorsal Root Ganglion (DRG) membranes using [3H]RTX binding assay.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/1/2012
Entry Details Article
PubMed
TargetTransient receptor potential cation channel subfamily V member 1(Rat)
Institute For Medical Research

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50052323BDBM50052323((4-Hydroxy-3-methoxy-phenyl)-acetic acid 4a,7b-dih...)
Affinity DataKi:  3.20nMAssay Description:Binding affinity against Vanilloid receptor in dorsal Root Ganglion (DRG) membranes using [3H]RTX binding assay.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/1/2012
Entry Details Article
PubMed
TargetTransient receptor potential cation channel subfamily V member 1(Rat)
Institute For Medical Research

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50052333BDBM50052333(13-benzyl-6-hydroxy-15-isopropenyl-4,17-dimethyl-5...)
Affinity DataKi:  4.30nMAssay Description:Binding affinity against Vanilloid receptor in dorsal Root Ganglion (DRG) membranes using [3H]RTX binding assay.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/1/2012
Entry Details Article
PubMed
TargetTransient receptor potential cation channel subfamily V member 1(Rat)
Institute For Medical Research

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50052328BDBM50052328(13-benzyl-6-hydroxy-15-isopropenyl-4,17-dimethyl-5...)
Affinity DataKi:  8.30nMAssay Description:Binding affinity against Vanilloid receptor in dorsal Root Ganglion (DRG) membranes using [3H]RTX binding assay.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/1/2012
Entry Details Article
PubMed
TargetTransient receptor potential cation channel subfamily V member 1(Rat)
Institute For Medical Research

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50052330BDBM50052330(13-benzyl-5,6-dihydroxy-15-isopropenyl-4,17-dimeth...)
Affinity DataKi:  11nMAssay Description:Binding affinity against Vanilloid receptor in dorsal Root Ganglion (DRG) membranes using [3H]RTX binding assay.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/1/2012
Entry Details Article
PubMed
TargetTransient receptor potential cation channel subfamily V member 1(Rat)
Institute For Medical Research

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50052321BDBM50052321(Phenyl-acetic acid (1aR,1bS,4aR,7aS,8R,9aS)-7b-hyd...)
Affinity DataKi:  600nMAssay Description:Binding affinity against Vanilloid receptor in dorsal Root Ganglion (DRG) membranes using [3H]RTX binding assay.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/1/2012
Entry Details Article
PubMed
TargetTransient receptor potential cation channel subfamily V member 1(Rat)
Institute For Medical Research

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 20461BDBM20461(Zostrix | (E)-N-[(4-hydroxy-3-methoxyphenyl)methyl...)
Affinity DataKi:  2.00E+3nMAssay Description:Binding affinity against Vanilloid receptor in dorsal Root Ganglion (DRG) membranes using [3H]RTX binding assay.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/1/2012
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetTransient receptor potential cation channel subfamily V member 1(Rat)
Institute For Medical Research

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50052324BDBM50052324(13-benzyl-6-hydroxy-8-hydroxymethyl-15-isopropenyl...)
Affinity DataKi: >1.00E+4nMAssay Description:Binding affinity against Vanilloid receptor in dorsal Root Ganglion (DRG) membranes using [3H]RTX binding assay.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/1/2012
Entry Details Article
PubMed