Compile Data Set for Download or QSAR
Report error Found 17 Enz. Inhib. hit(s) with all data for entry = 289
TargetDimer of Gag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Ciba-Geigy

LigandChemical structure of BindingDB Monomer ID 201BDBM201((2S)-N-[(2S,3S)-4-[(2S)-N'-(cyclohexylmethyl)-2-ac...)
Affinity DataIC50: 8.5nMpH: 6.0 T: 2°CAssay Description:A peptide cleavage assay was performed using the icosapeptide H-Arg-Arg-Ser-Asn-Gln-Val-Ser-Gln-Asn-Tyr-Pro-Ile-Val-Gln-Asn-Ile-Gln-Gly-Arg-Arg-OH, a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/9/2002
Entry Details Article
PubMed
TargetDimer of Gag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Ciba-Geigy

LigandChemical structure of BindingDB Monomer ID 213BDBM213(methyl N-[(1S)-1-{N'-[(2S,3S)-2-hydroxy-4-phenyl-3...)
Affinity DataIC50: 23nMpH: 6.0 T: 2°CAssay Description:A peptide cleavage assay was performed using the icosapeptide H-Arg-Arg-Ser-Asn-Gln-Val-Ser-Gln-Asn-Tyr-Pro-Ile-Val-Gln-Asn-Ile-Gln-Gly-Arg-Arg-OH, a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/9/2002
Entry Details Article
PubMed
TargetDimer of Gag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Ciba-Geigy

LigandChemical structure of BindingDB Monomer ID 206BDBM206(1-Cyclohexyl-2-N-[[(methoxycarbonyl)-L-valinyl]ami...)
Affinity DataIC50: 27nMpH: 6.0 T: 2°CAssay Description:A peptide cleavage assay was performed using the icosapeptide H-Arg-Arg-Ser-Asn-Gln-Val-Ser-Gln-Asn-Tyr-Pro-Ile-Val-Gln-Asn-Ile-Gln-Gly-Arg-Arg-OH, a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/9/2002
Entry Details Article
PubMed
TargetDimer of Gag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Ciba-Geigy

LigandChemical structure of BindingDB Monomer ID 214BDBM214(1-(4-Methoxyphenyl)-2-[[N-(methoxycarbonyl)-L-vali...)
Affinity DataIC50: 31nMpH: 6.0 T: 2°CAssay Description:A peptide cleavage assay was performed using the icosapeptide H-Arg-Arg-Ser-Asn-Gln-Val-Ser-Gln-Asn-Tyr-Pro-Ile-Val-Gln-Asn-Ile-Gln-Gly-Arg-Arg-OH, a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/9/2002
Entry Details Article
PubMed
TargetDimer of Gag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Ciba-Geigy

LigandChemical structure of BindingDB Monomer ID 216BDBM216(benzyl N-[(1S)-1-{N'-[(2S,3S)-2-hydroxy-4-phenyl-3...)
Affinity DataIC50: 37nMpH: 6.0 T: 2°CAssay Description:A peptide cleavage assay was performed using the icosapeptide H-Arg-Arg-Ser-Asn-Gln-Val-Ser-Gln-Asn-Tyr-Pro-Ile-Val-Gln-Asn-Ile-Gln-Gly-Arg-Arg-OH, a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/9/2002
Entry Details Article
PubMed
TargetDimer of Gag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Ciba-Geigy

LigandChemical structure of BindingDB Monomer ID 215BDBM215(benzyl N-[(1S)-1-[N'-(cyclohexylmethyl)-N'-[(2S,3S...)
Affinity DataIC50: 41nMpH: 6.0 T: 2°CAssay Description:A peptide cleavage assay was performed using the icosapeptide H-Arg-Arg-Ser-Asn-Gln-Val-Ser-Gln-Asn-Tyr-Pro-Ile-Val-Gln-Asn-Ile-Gln-Gly-Arg-Arg-OH, a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/9/2002
Entry Details Article
PubMed
TargetDimer of Gag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Ciba-Geigy

LigandChemical structure of BindingDB Monomer ID 217BDBM217(benzyl N-[(1S)-1-{N'-[(2S,3S)-2-hydroxy-4-phenyl-3...)
Affinity DataIC50: 49nMpH: 6.0 T: 2°CAssay Description:A peptide cleavage assay was performed using the icosapeptide H-Arg-Arg-Ser-Asn-Gln-Val-Ser-Gln-Asn-Tyr-Pro-Ile-Val-Gln-Asn-Ile-Gln-Gly-Arg-Arg-OH, a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/9/2002
Entry Details Article
PubMed
TargetDimer of Gag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Ciba-Geigy

LigandChemical structure of BindingDB Monomer ID 207BDBM207(methyl N-[(1S)-1-{[(2S,3S)-4-[(2S)-N'-(cyclohexylm...)
Affinity DataIC50: 56nMpH: 6.0 T: 2°CAssay Description:A peptide cleavage assay was performed using the icosapeptide H-Arg-Arg-Ser-Asn-Gln-Val-Ser-Gln-Asn-Tyr-Pro-Ile-Val-Gln-Asn-Ile-Gln-Gly-Arg-Arg-OH, a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/9/2002
Entry Details Article
PubMed
TargetDimer of Gag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Ciba-Geigy

LigandChemical structure of BindingDB Monomer ID 211BDBM211(2-methoxyethyl N-[(1S)-1-{[(2S,3S)-4-[(2S)-N'-(cyc...)
Affinity DataIC50: 62nMpH: 6.0 T: 2°CAssay Description:A peptide cleavage assay was performed using the icosapeptide H-Arg-Arg-Ser-Asn-Gln-Val-Ser-Gln-Asn-Tyr-Pro-Ile-Val-Gln-Asn-Ile-Gln-Gly-Arg-Arg-OH, a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/9/2002
Entry Details Article
PubMed
TargetDimer of Gag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Ciba-Geigy

LigandChemical structure of BindingDB Monomer ID 205BDBM205(2-(2-methoxyethoxy)ethyl N-[(1S)-1-{[(2S,3S)-4-[(2...)
Affinity DataIC50: 67nMpH: 6.0 T: 2°CAssay Description:A peptide cleavage assay was performed using the icosapeptide H-Arg-Arg-Ser-Asn-Gln-Val-Ser-Gln-Asn-Tyr-Pro-Ile-Val-Gln-Asn-Ile-Gln-Gly-Arg-Arg-OH, a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/9/2002
Entry Details Article
PubMed
TargetDimer of Gag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Ciba-Geigy

LigandChemical structure of BindingDB Monomer ID 208BDBM208(methyl N-[(1S)-1-{[(2S,3S)-4-[(2S)-N'-(cyclohexylm...)
Affinity DataIC50: 67nMpH: 6.0 T: 2°CAssay Description:A peptide cleavage assay was performed using the icosapeptide H-Arg-Arg-Ser-Asn-Gln-Val-Ser-Gln-Asn-Tyr-Pro-Ile-Val-Gln-Asn-Ile-Gln-Gly-Arg-Arg-OH, a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/9/2002
Entry Details Article
PubMed
TargetDimer of Gag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Ciba-Geigy

LigandChemical structure of BindingDB Monomer ID 209BDBM209(ethyl N-[(1S)-1-{[(2S,3S)-4-[(2S)-N'-(cyclohexylme...)
Affinity DataIC50: 76nMpH: 6.0 T: 2°CAssay Description:A peptide cleavage assay was performed using the icosapeptide H-Arg-Arg-Ser-Asn-Gln-Val-Ser-Gln-Asn-Tyr-Pro-Ile-Val-Gln-Asn-Ile-Gln-Gly-Arg-Arg-OH, a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/9/2002
Entry Details Article
PubMed
TargetDimer of Gag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Ciba-Geigy

LigandChemical structure of BindingDB Monomer ID 218BDBM218(ethyl N-[(1S)-1-[N'-(cyclohexylmethyl)-N'-[(2S,3S)...)
Affinity DataIC50: 126nMpH: 6.0 T: 2°CAssay Description:A peptide cleavage assay was performed using the icosapeptide H-Arg-Arg-Ser-Asn-Gln-Val-Ser-Gln-Asn-Tyr-Pro-Ile-Val-Gln-Asn-Ile-Gln-Gly-Arg-Arg-OH, a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/9/2002
Entry Details Article
PubMed
TargetDimer of Gag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Ciba-Geigy

LigandChemical structure of BindingDB Monomer ID 212BDBM212(2-methoxyethyl N-[(1S)-1-{[(2S,3S)-4-[(2S)-N'-(cyc...)
Affinity DataIC50: 134nMpH: 6.0 T: 2°CAssay Description:A peptide cleavage assay was performed using the icosapeptide H-Arg-Arg-Ser-Asn-Gln-Val-Ser-Gln-Asn-Tyr-Pro-Ile-Val-Gln-Asn-Ile-Gln-Gly-Arg-Arg-OH, a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/9/2002
Entry Details Article
PubMed
TargetDimer of Gag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Ciba-Geigy

LigandChemical structure of BindingDB Monomer ID 210BDBM210(ethyl N-[(1S)-1-{[(2S,3S)-4-[(2S)-N'-(cyclohexylme...)
Affinity DataIC50: 150nMpH: 6.0 T: 2°CAssay Description:A peptide cleavage assay was performed using the icosapeptide H-Arg-Arg-Ser-Asn-Gln-Val-Ser-Gln-Asn-Tyr-Pro-Ile-Val-Gln-Asn-Ile-Gln-Gly-Arg-Arg-OH, a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/9/2002
Entry Details Article
PubMed
TargetDimer of Gag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Ciba-Geigy

LigandChemical structure of BindingDB Monomer ID 204BDBM204(2-methoxyethyl N-[(1S)-1-{[(2S,3S)-4-[(2S)-N'-(cyc...)
Affinity DataIC50: 164nMpH: 6.0 T: 2°CAssay Description:A peptide cleavage assay was performed using the icosapeptide H-Arg-Arg-Ser-Asn-Gln-Val-Ser-Gln-Asn-Tyr-Pro-Ile-Val-Gln-Asn-Ile-Gln-Gly-Arg-Arg-OH, a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/9/2002
Entry Details Article
PubMed
TargetDimer of Gag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Ciba-Geigy

LigandChemical structure of BindingDB Monomer ID 202BDBM202(CHEMBL324572 | ethyl N-[(1S)-1-{[(2S,3S)-4-[(2S)-N...)
Affinity DataIC50: 177nMpH: 6.0 T: 2°CAssay Description:A peptide cleavage assay was performed using the icosapeptide H-Arg-Arg-Ser-Asn-Gln-Val-Ser-Gln-Asn-Tyr-Pro-Ile-Val-Gln-Asn-Ile-Gln-Gly-Arg-Arg-OH, a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/9/2002
Entry Details Article
PubMed