Compile Data Set for Download or QSAR
Report error Found 17 Enz. Inhib. hit(s) with all data for entry = 50036484
TargetPlatelet-activating factor receptor(Guinea pig)
Sankyo

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50366241BDBM50366241(L-652731 | CHEMBL297624)
Affinity DataIC50: 24nMAssay Description:Inhibiting Platelet activating factor receptor by radioreceptor binding assay using rabbit platelets and [3H]-PAFMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/3/2012
Entry Details Article
PubMed
TargetPlatelet-activating factor receptor(Guinea pig)
Sankyo

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50055488BDBM50055488(Carbonic acid methyl ester (E)-(1R,3S,5R,12S,13R,1...)
Affinity DataIC50: 26nMAssay Description:Inhibiting Platelet activating factor receptor by radioreceptor binding assay using rabbit platelets and [3H]-PAFMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/3/2012
Entry Details Article
PubMed
TargetPlatelet-activating factor receptor(Guinea pig)
Sankyo

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50055491BDBM50055491((E)-(1R,2R,3R,5R,12S,13R,16S)-16-(Isoxazol-3-yloxy...)
Affinity DataIC50: 31nMAssay Description:Inhibiting Platelet activating factor receptor by radioreceptor binding assay using rabbit platelets and [3H]-PAFMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/3/2012
Entry Details Article
PubMed
TargetPlatelet-activating factor receptor(Guinea pig)
Sankyo

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50055482BDBM50055482((E)-(1R,3S,5R,12S,13R,16S)-16-(Isoxazol-3-yloxymet...)
Affinity DataIC50: 50nMAssay Description:Inhibiting Platelet activating factor receptor by radioreceptor binding assay using rabbit platelets and [3H]-PAFMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/3/2012
Entry Details Article
PubMed
TargetPlatelet-activating factor receptor(Guinea pig)
Sankyo

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50055479BDBM50055479(Acetic acid (E)-(1R,2R,3R,5R,12S,13R,16S)-2-hydrox...)
Affinity DataIC50: 80nMAssay Description:Inhibiting Platelet activating factor receptor by radioreceptor binding assay using rabbit platelets and [3H]-PAFMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/3/2012
Entry Details Article
PubMed
TargetPlatelet-activating factor receptor(Guinea pig)
Sankyo

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50055489BDBM50055489((E)-(1R,3S,5R,12S,13R,16S)-5,9,12,13-Tetramethyl-2...)
Affinity DataIC50: 120nMAssay Description:Inhibiting Platelet activating factor receptor by radioreceptor binding assay using rabbit platelets and [3H]-PAFMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/3/2012
Entry Details Article
PubMed
TargetPlatelet-activating factor receptor(Guinea pig)
Sankyo

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50055493BDBM50055493(Carbonic acid (E)-(1R,2R,3R,5R,12S,13R,16S)-2-hydr...)
Affinity DataIC50: 130nMAssay Description:Inhibiting Platelet activating factor receptor by radioreceptor binding assay using rabbit platelets and [3H]-PAFMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/3/2012
Entry Details Article
PubMed
TargetPlatelet-activating factor receptor(Guinea pig)
Sankyo

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50055495BDBM50055495(Dimethyl-carbamic acid (E)-(1R,2R,3R,5R,12S,13R,16...)
Affinity DataIC50: 180nMAssay Description:Inhibiting Platelet activating factor receptor by radioreceptor binding assay using rabbit platelets and [3H]-PAFMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/3/2012
Entry Details Article
PubMed
TargetPlatelet-activating factor receptor(Guinea pig)
Sankyo

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50055483BDBM50055483(Dimethyl-carbamic acid (E)-(1R,3S,5R,12S,13R,16S)-...)
Affinity DataIC50: 180nMAssay Description:Inhibiting Platelet activating factor receptor by radioreceptor binding assay using rabbit platelets and [3H]-PAFMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/3/2012
Entry Details Article
PubMed
TargetPlatelet-activating factor receptor(Guinea pig)
Sankyo

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50055492BDBM50055492(Propionic acid (E)-(1R,2R,3R,5R,12S,13R,16S)-2-hyd...)
Affinity DataIC50: 340nMAssay Description:Inhibiting Platelet activating factor receptor by radioreceptor binding assay using rabbit platelets and [3H]-PAFMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/3/2012
Entry Details Article
PubMed
TargetPlatelet-activating factor receptor(Guinea pig)
Sankyo

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50055487BDBM50055487(Acetic acid (E)-(1R,3S,5R,12S,13R,16S)-5,9,12,13-t...)
Affinity DataIC50: 410nMAssay Description:Inhibiting Platelet activating factor receptor by radioreceptor binding assay using rabbit platelets and [3H]-PAFMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/3/2012
Entry Details Article
PubMed
TargetPlatelet-activating factor receptor(Guinea pig)
Sankyo

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50055484BDBM50055484(Carbonic acid phenyl ester (E)-(1R,3S,5R,12S,13R,1...)
Affinity DataIC50: 550nMAssay Description:Inhibiting Platelet activating factor receptor by radioreceptor binding assay using rabbit platelets and [3H]-PAFMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/3/2012
Entry Details Article
PubMed
TargetPlatelet-activating factor receptor(Guinea pig)
Sankyo

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50055494BDBM50055494(Propionic acid (E)-(1R,3S,5R,12S,13R,16S)-5,9,12,1...)
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibiting Platelet activating factor receptor by radioreceptor binding assay using rabbit platelets and [3H]-PAFMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/3/2012
Entry Details Article
PubMed
TargetPlatelet-activating factor receptor(Guinea pig)
Sankyo

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50055480BDBM50055480((E)-(1R,3S,5R,12S,13R,16S)-16-Hydroxymethyl-5,9,12...)
Affinity DataIC50: 1.30E+3nMAssay Description:Inhibiting Platelet activating factor receptor by radioreceptor binding assay using rabbit platelets and [3H]-PAFMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/3/2012
Entry Details Article
PubMed
TargetPlatelet-activating factor receptor(Guinea pig)
Sankyo

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50055485BDBM50055485(16-(Isoxazol-3-yloxymethyl)-5,9,12,13-tetramethyl-...)
Affinity DataIC50: 1.70E+4nMAssay Description:Inhibiting Platelet activating factor receptor by radioreceptor binding assay using rabbit platelets and [3H]-PAFMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/3/2012
Entry Details Article
PubMed
TargetPlatelet-activating factor receptor(Guinea pig)
Sankyo

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50055481BDBM50055481(16-(Isoxazol-3-yloxymethyl)-5,9,12,13-tetramethyl-...)
Affinity DataIC50: 3.00E+4nMAssay Description:Inhibiting Platelet activating factor receptor by radioreceptor binding assay using rabbit platelets and [3H]-PAFMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/3/2012
Entry Details Article
PubMed
TargetPlatelet-activating factor receptor(Guinea pig)
Sankyo

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50055486BDBM50055486((1R,3S,5R,8S,9S,12S,13R,16S)-8,9-Dihydroxy-16-hydr...)
Affinity DataIC50: 2.80E+5nMAssay Description:Inhibiting Platelet activating factor receptor by radioreceptor binding assay using rabbit platelets and [3H]-PAFMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/3/2012
Entry Details Article
PubMed