Compile Data Set for Download or QSAR
maximum 50k data
Found 17 Enz. Inhib. hit(s) with all data for entry = 50036484
TargetPlatelet-activating factor receptor(Cavia porcellus)
Sankyo

Curated by ChEMBL
LigandPNGBDBM50366241(CHEMBL297624 | L-652731)
Affinity DataIC50:  24nMAssay Description:Inhibiting Platelet activating factor receptor by radioreceptor binding assay using rabbit platelets and [3H]-PAFMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlatelet-activating factor receptor(Cavia porcellus)
Sankyo

Curated by ChEMBL
LigandPNGBDBM50055488(CHEMBL148491 | Carbonic acid methyl ester (E)-(1R,...)
Affinity DataIC50:  26nMAssay Description:Inhibiting Platelet activating factor receptor by radioreceptor binding assay using rabbit platelets and [3H]-PAFMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlatelet-activating factor receptor(Cavia porcellus)
Sankyo

Curated by ChEMBL
LigandPNGBDBM50055491((E)-(1R,2R,3R,5R,12S,13R,16S)-16-(Isoxazol-3-yloxy...)
Affinity DataIC50:  31nMAssay Description:Inhibiting Platelet activating factor receptor by radioreceptor binding assay using rabbit platelets and [3H]-PAFMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlatelet-activating factor receptor(Cavia porcellus)
Sankyo

Curated by ChEMBL
LigandPNGBDBM50055482((E)-(1R,3S,5R,12S,13R,16S)-16-(Isoxazol-3-yloxymet...)
Affinity DataIC50:  50nMAssay Description:Inhibiting Platelet activating factor receptor by radioreceptor binding assay using rabbit platelets and [3H]-PAFMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlatelet-activating factor receptor(Cavia porcellus)
Sankyo

Curated by ChEMBL
LigandPNGBDBM50055479(Acetic acid (E)-(1R,2R,3R,5R,12S,13R,16S)-2-hydrox...)
Affinity DataIC50:  80nMAssay Description:Inhibiting Platelet activating factor receptor by radioreceptor binding assay using rabbit platelets and [3H]-PAFMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlatelet-activating factor receptor(Cavia porcellus)
Sankyo

Curated by ChEMBL
LigandPNGBDBM50055489((E)-(1R,3S,5R,12S,13R,16S)-5,9,12,13-Tetramethyl-2...)
Affinity DataIC50:  120nMAssay Description:Inhibiting Platelet activating factor receptor by radioreceptor binding assay using rabbit platelets and [3H]-PAFMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlatelet-activating factor receptor(Cavia porcellus)
Sankyo

Curated by ChEMBL
LigandPNGBDBM50055493(CHEMBL148549 | Carbonic acid (E)-(1R,2R,3R,5R,12S,...)
Affinity DataIC50:  130nMAssay Description:Inhibiting Platelet activating factor receptor by radioreceptor binding assay using rabbit platelets and [3H]-PAFMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlatelet-activating factor receptor(Cavia porcellus)
Sankyo

Curated by ChEMBL
LigandPNGBDBM50055495(CHEMBL151075 | Dimethyl-carbamic acid (E)-(1R,2R,3...)
Affinity DataIC50:  180nMAssay Description:Inhibiting Platelet activating factor receptor by radioreceptor binding assay using rabbit platelets and [3H]-PAFMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlatelet-activating factor receptor(Cavia porcellus)
Sankyo

Curated by ChEMBL
LigandPNGBDBM50055483(CHEMBL151310 | Dimethyl-carbamic acid (E)-(1R,3S,5...)
Affinity DataIC50:  180nMAssay Description:Inhibiting Platelet activating factor receptor by radioreceptor binding assay using rabbit platelets and [3H]-PAFMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlatelet-activating factor receptor(Cavia porcellus)
Sankyo

Curated by ChEMBL
LigandPNGBDBM50055492(CHEMBL147337 | Propionic acid (E)-(1R,2R,3R,5R,12S...)
Affinity DataIC50:  340nMAssay Description:Inhibiting Platelet activating factor receptor by radioreceptor binding assay using rabbit platelets and [3H]-PAFMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlatelet-activating factor receptor(Cavia porcellus)
Sankyo

Curated by ChEMBL
LigandPNGBDBM50055487(Acetic acid (E)-(1R,3S,5R,12S,13R,16S)-5,9,12,13-t...)
Affinity DataIC50:  410nMAssay Description:Inhibiting Platelet activating factor receptor by radioreceptor binding assay using rabbit platelets and [3H]-PAFMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlatelet-activating factor receptor(Cavia porcellus)
Sankyo

Curated by ChEMBL
LigandPNGBDBM50055484(CHEMBL421954 | Carbonic acid phenyl ester (E)-(1R,...)
Affinity DataIC50:  550nMAssay Description:Inhibiting Platelet activating factor receptor by radioreceptor binding assay using rabbit platelets and [3H]-PAFMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlatelet-activating factor receptor(Cavia porcellus)
Sankyo

Curated by ChEMBL
LigandPNGBDBM50055494(CHEMBL147079 | Propionic acid (E)-(1R,3S,5R,12S,13...)
Affinity DataIC50:  1.00E+3nMAssay Description:Inhibiting Platelet activating factor receptor by radioreceptor binding assay using rabbit platelets and [3H]-PAFMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlatelet-activating factor receptor(Cavia porcellus)
Sankyo

Curated by ChEMBL
LigandPNGBDBM50055480((E)-(1R,3S,5R,12S,13R,16S)-16-Hydroxymethyl-5,9,12...)
Affinity DataIC50:  1.30E+3nMAssay Description:Inhibiting Platelet activating factor receptor by radioreceptor binding assay using rabbit platelets and [3H]-PAFMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlatelet-activating factor receptor(Cavia porcellus)
Sankyo

Curated by ChEMBL
LigandPNGBDBM50055485(16-(Isoxazol-3-yloxymethyl)-5,9,12,13-tetramethyl-...)
Affinity DataIC50:  1.70E+4nMAssay Description:Inhibiting Platelet activating factor receptor by radioreceptor binding assay using rabbit platelets and [3H]-PAFMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlatelet-activating factor receptor(Cavia porcellus)
Sankyo

Curated by ChEMBL
LigandPNGBDBM50055481(16-(Isoxazol-3-yloxymethyl)-5,9,12,13-tetramethyl-...)
Affinity DataIC50:  3.00E+4nMAssay Description:Inhibiting Platelet activating factor receptor by radioreceptor binding assay using rabbit platelets and [3H]-PAFMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlatelet-activating factor receptor(Cavia porcellus)
Sankyo

Curated by ChEMBL
LigandPNGBDBM50055486((1R,3S,5R,8S,9S,12S,13R,16S)-8,9-Dihydroxy-16-hydr...)
Affinity DataIC50: >2.80E+5nMAssay Description:Inhibiting Platelet activating factor receptor by radioreceptor binding assay using rabbit platelets and [3H]-PAFMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed