Report error Found 57 Enz. Inhib. hit(s) with all data for entry = 50006949
Affinity DataKi: 0.150nMAssay Description:Binding affinity was evaluated by determining in vitro displacement of [3H]8-OH-DPAT from the central 5-hydroxytryptamine 1A receptor recognition sit...More data for this Ligand-Target Pair
Affinity DataKi: 0.300nMAssay Description:Binding affinity was evaluated by determining in vitro displacement of [3H]8-OH-DPAT from the central 5-hydroxytryptamine 1A receptor recognition sit...More data for this Ligand-Target Pair
Affinity DataKi: 0.320nMAssay Description:Binding affinity was evaluated by determining in vitro displacement of [3H]8-OH-DPAT from the central 5-hydroxytryptamine 1A receptor recognition sit...More data for this Ligand-Target Pair
Affinity DataEC50: 0.780nMAssay Description:In vitro potency at human 5-hydroxytryptamine 1A receptor in inhibiting forskolin-stimulated accumulation of intracellular cAMPMore data for this Ligand-Target Pair
Affinity DataEC50: 0.780nMAssay Description:In vitro potency at human 5-hydroxytryptamine 1A receptor in inhibiting forskolin-stimulated accumulation of intracellular cAMPMore data for this Ligand-Target Pair
Affinity DataKi: 0.800nMAssay Description:Binding affinity was evaluated by determining in vitro displacement of [3H]8-OH-DPAT from the central 5-hydroxytryptamine 1A receptor recognition sit...More data for this Ligand-Target Pair
Affinity DataKi: 1nMAssay Description:Binding affinity was evaluated by determining in vitro displacement of [3H]8-OH-DPAT from the central 5-hydroxytryptamine 1A receptor recognition sit...More data for this Ligand-Target Pair
Affinity DataKi: 1nMAssay Description:Binding affinity was evaluated by determining in vitro displacement of [3H]8-OH-DPAT from the central 5-hydroxytryptamine 1A receptor recognition sit...More data for this Ligand-Target Pair
Affinity DataKi: 1nMAssay Description:Binding affinity was evaluated by determining in vitro displacement of [3H]8-OH-DPAT from the central 5-hydroxytryptamine 1A receptor recognition sit...More data for this Ligand-Target Pair
Affinity DataKi: 1.10nMAssay Description:Binding affinity was evaluated by determining in vitro displacement of [3H]8-OH-DPAT from the central 5-hydroxytryptamine 1A receptor recognition sit...More data for this Ligand-Target Pair
Affinity DataKi: 1.30nMAssay Description:Binding affinity was evaluated by determining in vitro displacement of [3H]8-OH-DPAT from the central 5-hydroxytryptamine 1A receptor recognition sit...More data for this Ligand-Target Pair
Affinity DataKi: 1.60nMAssay Description:Binding affinity was evaluated by determining in vitro displacement of [3H]8-OH-DPAT from the central 5-hydroxytryptamine 1A receptor recognition sit...More data for this Ligand-Target Pair
Affinity DataKi: 1.70nMAssay Description:Binding affinity was evaluated by determining in vitro displacement of [3H]8-OH-DPAT from the central 5-hydroxytryptamine 1A receptor recognition sit...More data for this Ligand-Target Pair
Affinity DataKi: 1.80nMAssay Description:Binding affinity was evaluated by determining in vitro displacement of [3H]8-OH-DPAT from the central 5-hydroxytryptamine 1A receptor recognition sit...More data for this Ligand-Target Pair
Affinity DataKi: 2.5nMAssay Description:Binding affinity was evaluated by determining in vitro displacement of [3H]8-OH-DPAT from the central 5-hydroxytryptamine 1A receptor recognition sit...More data for this Ligand-Target Pair
Affinity DataKi: 3.10nMAssay Description:In vitro displacement of [3H]spiperone from Dopamine receptor D2 binding site in rat striatum.More data for this Ligand-Target Pair
Affinity DataKi: 3.30nMAssay Description:In vitro displacement of [3H]spiperone from Dopamine receptor D2 binding site in rat striatum.More data for this Ligand-Target Pair
Affinity DataKi: 3.30nMAssay Description:In vitro displacement of [3H]spiperone from Dopamine receptor D2 binding site in rat striatum.More data for this Ligand-Target Pair
Affinity DataKi: 3.40nMAssay Description:In vitro displacement of [3H]spiperone from Dopamine receptor D2 binding site in rat striatum.More data for this Ligand-Target Pair
Affinity DataKi: 3.40nMAssay Description:Binding affinity was evaluated by determining in vitro displacement of [3H]8-OH-DPAT from the central 5-hydroxytryptamine 1A receptor recognition sit...More data for this Ligand-Target Pair
Affinity DataKi: 4.10nMAssay Description:In vitro displacement of [3H]spiperone from Dopamine receptor D2 binding site in rat striatum.More data for this Ligand-Target Pair
Affinity DataKi: 4.5nMAssay Description:Binding affinity was evaluated by determining in vitro displacement of [3H]8-OH-DPAT from the central 5-hydroxytryptamine 1A receptor recognition sit...More data for this Ligand-Target Pair
Affinity DataKi: 4.90nMAssay Description:Binding affinity was evaluated by determining in vitro displacement of [3H]8-OH-DPAT from the central 5-hydroxytryptamine 1A receptor recognition sit...More data for this Ligand-Target Pair
Affinity DataKi: 5nMAssay Description:In vitro displacement of [3H]spiperone from Dopamine receptor D2 binding site in rat striatum.More data for this Ligand-Target Pair
Affinity DataKi: 5.30nMAssay Description:In vitro displacement of [3H]spiperone from Dopamine receptor D2 binding site in rat striatum.More data for this Ligand-Target Pair
Affinity DataKi: 6.40nMAssay Description:In vitro displacement of [3H]spiperone from Dopamine receptor D2 binding site in rat striatum.More data for this Ligand-Target Pair
Affinity DataKi: 10nMAssay Description:In vitro displacement of [3H]spiperone from Dopamine receptor D2 binding site in rat striatum.More data for this Ligand-Target Pair
Affinity DataKi: 13nMAssay Description:In vitro displacement of [3H]spiperone from Dopamine receptor D2 binding site in rat striatum.More data for this Ligand-Target Pair
Affinity DataKi: 13nMAssay Description:Binding affinity was evaluated by determining in vitro displacement of [3H]8-OH-DPAT from the central 5-hydroxytryptamine 1A receptor recognition sit...More data for this Ligand-Target Pair
Affinity DataKi: 14nMAssay Description:In vitro displacement of [3H]spiperone from Dopamine receptor D2 binding site in rat striatum.More data for this Ligand-Target Pair
Affinity DataKi: 15nMAssay Description:Binding affinity was evaluated by determining in vitro displacement of [3H]8-OH-DPAT from the central 5-hydroxytryptamine 1A receptor recognition sit...More data for this Ligand-Target Pair
Affinity DataKi: 16nMAssay Description:Binding affinity was evaluated by determining in vitro displacement of [3H]8-OH-DPAT from the central 5-hydroxytryptamine 1A receptor recognition sit...More data for this Ligand-Target Pair
Affinity DataKi: 17nMAssay Description:In vitro displacement of [3H]spiperone from Dopamine receptor D2 binding site in rat striatum.More data for this Ligand-Target Pair
Affinity DataKi: 18nMAssay Description:Binding affinity was evaluated by determining in vitro displacement of [3H]8-OH-DPAT from the central 5-hydroxytryptamine 1A receptor recognition sit...More data for this Ligand-Target Pair
Affinity DataKi: 18nMAssay Description:Binding affinity was evaluated by determining in vitro displacement of [3H]8-OH-DPAT from the central 5-hydroxytryptamine 1A receptor recognition sit...More data for this Ligand-Target Pair
Affinity DataKi: 22nMAssay Description:Binding affinity was evaluated by determining in vitro displacement of [3H]8-OH-DPAT from the central 5-hydroxytryptamine 1A receptor recognition sit...More data for this Ligand-Target Pair
Affinity DataKi: 23nMAssay Description:In vitro displacement of [3H]spiperone from Dopamine receptor D2 binding site in rat striatum.More data for this Ligand-Target Pair
Affinity DataKi: 40nMAssay Description:Binding affinity was evaluated by determining in vitro displacement of [3H]8-OH-DPAT from the central 5-hydroxytryptamine 1A receptor recognition sit...More data for this Ligand-Target Pair
Affinity DataKi: 59nMAssay Description:Binding affinity was evaluated by determining in vitro displacement of [3H]8-OH-DPAT from the central 5-hydroxytryptamine 1A receptor recognition sit...More data for this Ligand-Target Pair
Affinity DataKi: 64nMAssay Description:In vitro displacement of [3H]spiperone from Dopamine receptor D2 binding site in rat striatum.More data for this Ligand-Target Pair
Affinity DataKi: 73nMAssay Description:In vitro displacement of [3H]spiperone from Dopamine receptor D2 binding site in rat striatum.More data for this Ligand-Target Pair
Affinity DataKi: 92nMAssay Description:In vitro displacement of [3H]spiperone from Dopamine receptor D2 binding site in rat striatum.More data for this Ligand-Target Pair
Affinity DataKi: 130nMAssay Description:In vitro displacement of [3H]spiperone from Dopamine receptor D2 binding site in rat striatum.More data for this Ligand-Target Pair
Affinity DataKi: 140nMAssay Description:In vitro displacement of [3H]spiperone from Dopamine receptor D2 binding site in rat striatum.More data for this Ligand-Target Pair
Affinity DataKi: 140nMAssay Description:Binding affinity was evaluated by determining in vitro displacement of [3H]8-OH-DPAT from the central 5-hydroxytryptamine 1A receptor recognition sit...More data for this Ligand-Target Pair
Affinity DataKi: 170nMAssay Description:Binding affinity was evaluated by determining in vitro displacement of [3H]8-OH-DPAT from the central 5-hydroxytryptamine 1A receptor recognition sit...More data for this Ligand-Target Pair
Affinity DataKi: 230nMAssay Description:In vitro displacement of [3H]spiperone from Dopamine receptor D2 binding site in rat striatum.More data for this Ligand-Target Pair
Affinity DataKi: 250nMAssay Description:In vitro displacement of [3H]spiperone from Dopamine receptor D2 binding site in rat striatum.More data for this Ligand-Target Pair
Affinity DataKi: 500nMAssay Description:Binding affinity was evaluated by determining in vitro displacement of [3H]8-OH-DPAT from the central 5-hydroxytryptamine 1A receptor recognition sit...More data for this Ligand-Target Pair
Affinity DataKi: 570nMAssay Description:In vitro displacement of [3H]spiperone from Dopamine receptor D2 binding site in rat striatum.More data for this Ligand-Target Pair


























