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Found 48 Enz. Inhib. hit(s) with all data for entry = 50003452
TargetMelatonin receptor type 1C(Gallus gallus)
Universit£

Curated by ChEMBL
LigandPNGBDBM50230657(CHEMBL290493)
Affinity DataKi:  0.0295nMAssay Description:Binding affinity against chicken brain melatonin receptors using 2-[125I]iodomelatonin as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelatonin receptor type 1C(Gallus gallus)
Universit£

Curated by ChEMBL
LigandPNGBDBM29611(2-Iodomelatonin | CHEMBL289233 | Melatonin,2-Iodo)
Affinity DataKi:  0.0324nMAssay Description:Binding affinity against chicken brain melatonin receptors using 2-[125I]iodomelatonin as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelatonin receptor type 1C(Gallus gallus)
Universit£

Curated by ChEMBL
LigandPNGBDBM50035202(CHEMBL291857 | N-[2-(2,7-Dimethoxy-naphthalen-1-yl...)
Affinity DataKi:  0.0724nMAssay Description:Binding affinity against chicken brain melatonin receptors using 2-[125I]iodomelatonin as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelatonin receptor type 1C(Gallus gallus)
Universit£

Curated by ChEMBL
LigandPNGBDBM50470007(CHEMBL322269)
Affinity DataKi:  0.120nMAssay Description:Binding affinity against chicken brain melatonin receptors using 2-[125I]iodomelatonin as radioligandMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMelatonin receptor type 1C(Gallus gallus)
Universit£

Curated by ChEMBL
LigandPNGBDBM50470000(CHEMBL111599)
Affinity DataKi:  0.141nMAssay Description:Binding affinity against chicken brain melatonin receptors using 2-[125I]iodomelatonin as radioligandMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMelatonin receptor type 1C(Gallus gallus)
Universit£

Curated by ChEMBL
LigandPNGBDBM50408556(CHEMBL37771)
Affinity DataKi:  0.182nMAssay Description:Binding affinity against chicken brain melatonin receptors using 2-[125I]iodomelatonin as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelatonin receptor type 1C(Gallus gallus)
Universit£

Curated by ChEMBL
LigandPNGBDBM50470187(CHEMBL428882)
Affinity DataKi:  0.240nMAssay Description:Binding affinity against chicken brain melatonin receptors using 2-[125I]iodomelatonin as radioligandMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMelatonin receptor type 1C(Gallus gallus)
Universit£

Curated by ChEMBL
LigandPNGBDBM50470180(CHEMBL61626)
Affinity DataKi:  0.389nMAssay Description:Binding affinity against chicken brain melatonin receptors using 2-[125I]iodomelatonin as radioligandMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMelatonin receptor type 1C(Gallus gallus)
Universit£

Curated by ChEMBL
LigandPNGBDBM50035179(Agomelatine | CHEMBL10878 | N-[2-(7-Methoxy-naphth...)
Affinity DataKi:  0.537nMAssay Description:Binding affinity against chicken brain melatonin receptors using 2-[125I]iodomelatonin as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelatonin receptor type 1C(Gallus gallus)
Universit£

Curated by ChEMBL
LigandPNGBDBM50470174(CHEMBL62992)
Affinity DataKi:  0.550nMAssay Description:Binding affinity against chicken brain melatonin receptors using 2-[125I]iodomelatonin as radioligandMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMelatonin receptor type 1C(Gallus gallus)
Universit£

Curated by ChEMBL
LigandPNGBDBM50470172(CHEMBL294517)
Affinity DataKi:  0.676nMAssay Description:Binding affinity against chicken brain melatonin receptors using 2-[125I]iodomelatonin as radioligandMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMelatonin receptor type 1C(Gallus gallus)
Universit£

Curated by ChEMBL
LigandPNGBDBM9019(CHEMBL45 | Melatonin | N-[2-(5-methoxy-1H-indol-3-...)
Affinity DataKi:  0.676nMAssay Description:Binding affinity against chicken brain melatonin receptors using 2-[125I]iodomelatonin as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelatonin receptor type 1C(Gallus gallus)
Universit£

Curated by ChEMBL
LigandPNGBDBM50471087(CHEMBL124462)
Affinity DataKi:  1.10nMAssay Description:Binding affinity against chicken brain melatonin receptors using 2-[125I]iodomelatonin as radioligandMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMelatonin receptor type 1C(Gallus gallus)
Universit£

Curated by ChEMBL
LigandPNGBDBM50470183(CHEMBL305383)
Affinity DataKi:  1.10nMAssay Description:Binding affinity against chicken brain melatonin receptors using 2-[125I]iodomelatonin as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelatonin receptor type 1C(Gallus gallus)
Universit£

Curated by ChEMBL
LigandPNGBDBM50470193(CHEMBL64142)
Affinity DataKi:  1.40nMAssay Description:Binding affinity against chicken brain melatonin receptors using 2-[125I]iodomelatonin as radioligandMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMelatonin receptor type 1C(Gallus gallus)
Universit£

Curated by ChEMBL
LigandPNGBDBM50408625(CHEMBL138549)
Affinity DataKi:  1.70nMAssay Description:Binding affinity against chicken brain melatonin receptors using 2-[125I]iodomelatonin as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelatonin receptor type 1C(Gallus gallus)
Universit£

Curated by ChEMBL
LigandPNGBDBM50037249(CHEMBL109086 | Cyclopropanecarboxylic acid [2-(6-f...)
Affinity DataKi:  2.5nMAssay Description:Binding affinity against chicken brain melatonin receptors using 2-[125I]iodomelatonin as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelatonin receptor type 1C(Gallus gallus)
Universit£

Curated by ChEMBL
LigandPNGBDBM50230659(CHEMBL37549)
Affinity DataKi:  2.5nMAssay Description:Binding affinity against chicken brain melatonin receptors using 2-[125I]iodomelatonin as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelatonin receptor type 1C(Gallus gallus)
Universit£

Curated by ChEMBL
LigandPNGBDBM50470175(CHEMBL64471)
Affinity DataKi:  2.70nMAssay Description:Binding affinity against chicken brain melatonin receptors using 2-[125I]iodomelatonin as radioligandMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMelatonin receptor type 1C(Gallus gallus)
Universit£

Curated by ChEMBL
LigandPNGBDBM50471088(CHEMBL126143)
Affinity DataKi:  3.5nMAssay Description:Binding affinity against chicken brain melatonin receptors using 2-[125I]iodomelatonin as radioligandMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMelatonin receptor type 1C(Gallus gallus)
Universit£

Curated by ChEMBL
LigandPNGBDBM50471084(CHEMBL428342)
Affinity DataKi:  5.90nMAssay Description:Binding affinity against chicken brain melatonin receptors using 2-[125I]iodomelatonin as radioligandMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMelatonin receptor type 1C(Gallus gallus)
Universit£

Curated by ChEMBL
LigandPNGBDBM50470869(CHEMBL12477)
Affinity DataKi:  6nMAssay Description:Binding affinity against chicken brain melatonin receptors using 2-[125I]iodomelatonin as radioligandMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMelatonin receptor type 1C(Gallus gallus)
Universit£

Curated by ChEMBL
LigandPNGBDBM50408596(CHEMBL137949)
Affinity DataKi:  6.80nMAssay Description:Binding affinity against chicken brain melatonin receptors using 2-[125I]iodomelatonin as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelatonin receptor type 1C(Gallus gallus)
Universit£

Curated by ChEMBL
LigandPNGBDBM50470009(CHEMBL109842)
Affinity DataKi:  9.30nMAssay Description:Binding affinity against chicken brain melatonin receptors using 2-[125I]iodomelatonin as radioligandMore data for this Ligand-Target Pair
Ligand InfoKEGGPC cidPC sid
In DepthDetails ArticlePubMed
TargetMelatonin receptor type 1C(Gallus gallus)
Universit£

Curated by ChEMBL
LigandPNGBDBM50471083(CHEMBL349435)
Affinity DataKi:  12nMAssay Description:Binding affinity against chicken brain melatonin receptors using 2-[125I]iodomelatonin as radioligandMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMelatonin receptor type 1C(Gallus gallus)
Universit£

Curated by ChEMBL
LigandPNGBDBM50408578(CHEMBL417151)
Affinity DataKi:  19nMAssay Description:Binding affinity against chicken brain melatonin receptors using 2-[125I]iodomelatonin as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelatonin receptor type 1C(Gallus gallus)
Universit£

Curated by ChEMBL
LigandPNGBDBM50408659(CHEMBL342162)
Affinity DataKi:  22nMAssay Description:Binding affinity against chicken brain melatonin receptors using 2-[125I]iodomelatonin as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelatonin receptor type 1C(Gallus gallus)
Universit£

Curated by ChEMBL
LigandPNGBDBM50469991(CHEMBL109784)
Affinity DataKi:  30nMAssay Description:Binding affinity against chicken brain melatonin receptors using 2-[125I]iodomelatonin as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelatonin receptor type 1C(Gallus gallus)
Universit£

Curated by ChEMBL
LigandPNGBDBM50470868(CHEMBL12795)
Affinity DataKi:  35nMAssay Description:Binding affinity against chicken brain melatonin receptors using 2-[125I]iodomelatonin as radioligandMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMelatonin receptor type 1C(Gallus gallus)
Universit£

Curated by ChEMBL
LigandPNGBDBM50470182(CHEMBL62306)
Affinity DataKi:  42nMAssay Description:Binding affinity against chicken brain melatonin receptors using 2-[125I]iodomelatonin as radioligandMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMelatonin receptor type 1C(Gallus gallus)
Universit£

Curated by ChEMBL
LigandPNGBDBM50230663(CHEMBL34349)
Affinity DataKi:  45nMAssay Description:Binding affinity against chicken brain melatonin receptors using 2-[125I]iodomelatonin as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelatonin receptor type 1C(Gallus gallus)
Universit£

Curated by ChEMBL
LigandPNGBDBM50471094(CHEMBL162456)
Affinity DataKi:  56nMAssay Description:Binding affinity against chicken brain melatonin receptors using 2-[125I]iodomelatonin as radioligandMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMelatonin receptor type 1C(Gallus gallus)
Universit£

Curated by ChEMBL
LigandPNGBDBM50471092(CHEMBL162914)
Affinity DataKi:  65nMAssay Description:Binding affinity against chicken brain melatonin receptors using 2-[125I]iodomelatonin as radioligandMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMelatonin receptor type 1C(Gallus gallus)
Universit£

Curated by ChEMBL
LigandPNGBDBM50470194(CHEMBL63006)
Affinity DataKi:  71nMAssay Description:Binding affinity against chicken brain melatonin receptors using 2-[125I]iodomelatonin as radioligandMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMelatonin receptor type 1C(Gallus gallus)
Universit£

Curated by ChEMBL
LigandPNGBDBM50471085(CHEMBL162154)
Affinity DataKi:  115nMAssay Description:Binding affinity against chicken brain melatonin receptors using 2-[125I]iodomelatonin as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelatonin receptor type 1C(Gallus gallus)
Universit£

Curated by ChEMBL
LigandPNGBDBM50471090(CHEMBL124076)
Affinity DataKi:  158nMAssay Description:Binding affinity against chicken brain melatonin receptors using 2-[125I]iodomelatonin as radioligandMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMelatonin receptor type 1C(Gallus gallus)
Universit£

Curated by ChEMBL
LigandPNGBDBM50470173(CHEMBL304685)
Affinity DataKi:  195nMAssay Description:Binding affinity against chicken brain melatonin receptors using 2-[125I]iodomelatonin as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelatonin receptor type 1C(Gallus gallus)
Universit£

Curated by ChEMBL
LigandPNGBDBM50035176(8-M-ADOT | CHEMBL53015 | N-(8-Methoxy-1,2,3,4-tetr...)
Affinity DataKi:  204nMAssay Description:Binding affinity against chicken brain melatonin receptors using 2-[125I]iodomelatonin as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelatonin receptor type 1C(Gallus gallus)
Universit£

Curated by ChEMBL
LigandPNGBDBM50231305(CHEMBL52801)
Affinity DataKi:  214nMAssay Description:Binding affinity against chicken brain melatonin receptors using 2-[125I]iodomelatonin as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelatonin receptor type 1C(Gallus gallus)
Universit£

Curated by ChEMBL
LigandPNGBDBM50470870(CHEMBL104997)
Affinity DataKi:  214nMAssay Description:Binding affinity against chicken brain melatonin receptors using 2-[125I]iodomelatonin as radioligandMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMelatonin receptor type 1C(Gallus gallus)
Universit£

Curated by ChEMBL
LigandPNGBDBM50470176(CHEMBL291378)
Affinity DataKi:  219nMAssay Description:Binding affinity against chicken brain melatonin receptors using 2-[125I]iodomelatonin as radioligandMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMelatonin receptor type 1C(Gallus gallus)
Universit£

Curated by ChEMBL
LigandPNGBDBM50471089(CHEMBL165186)
Affinity DataKi:  229nMAssay Description:Binding affinity against chicken brain melatonin receptors using 2-[125I]iodomelatonin as radioligandMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMelatonin receptor type 1C(Gallus gallus)
Universit£

Curated by ChEMBL
LigandPNGBDBM50471091(CHEMBL350753)
Affinity DataKi:  240nMAssay Description:Binding affinity against chicken brain melatonin receptors using 2-[125I]iodomelatonin as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelatonin receptor type 1C(Gallus gallus)
Universit£

Curated by ChEMBL
LigandPNGBDBM50231306(CHEMBL53722)
Affinity DataKi:  251nMAssay Description:Binding affinity against chicken brain melatonin receptors using 2-[125I]iodomelatonin as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelatonin receptor type 1C(Gallus gallus)
Universit£

Curated by ChEMBL
LigandPNGBDBM50471093(CHEMBL125081)
Affinity DataKi:  288nMAssay Description:Binding affinity against chicken brain melatonin receptors using 2-[125I]iodomelatonin as radioligandMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMelatonin receptor type 1C(Gallus gallus)
Universit£

Curated by ChEMBL
LigandPNGBDBM50470188(CHEMBL62495)
Affinity DataKi:  324nMAssay Description:Binding affinity against chicken brain melatonin receptors using 2-[125I]iodomelatonin as radioligandMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMelatonin receptor type 1C(Gallus gallus)
Universit£

Curated by ChEMBL
LigandPNGBDBM50282758(CHEMBL33171 | N-Acetyltryptamine | N-[2-(1H-Indol-...)
Affinity DataKi:  490nMAssay Description:Binding affinity against chicken brain melatonin receptors using 2-[125I]iodomelatonin as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelatonin receptor type 1C(Gallus gallus)
Universit£

Curated by ChEMBL
LigandPNGBDBM50471086(CHEMBL165685)
Affinity DataKi:  1.91E+3nMAssay Description:Binding affinity against chicken brain melatonin receptors using 2-[125I]iodomelatonin as radioligandMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed