Compile Data Set for Download or QSAR
maximum 50k data
Found 28 Enz. Inhib. hit(s) with all data for entry = 50003467
LigandPNGBDBM50471350(CHEMBL102763)
Affinity DataKi:  8.80nMAssay Description:Displacement of [3H]rauwolscine from Alpha-2 adrenergic receptor of rat brain membranesMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
LigandPNGBDBM50036913((+-)-4-(alpha,2,3-trimethylbenzyl)imidazole | 4-[1...)
Affinity DataKi:  25nMAssay Description:Displacement of [3H]rauwolscine from Alpha-2 adrenergic receptor of rat brain membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50471342(CHEMBL322907)
Affinity DataKi:  31nMAssay Description:Displacement of [3H]rauwolscine from Alpha-2 adrenergic receptor of rat brain membranesMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
LigandPNGBDBM50471340(CHEMBL317912)
Affinity DataKi:  63nMAssay Description:Displacement of [3H]rauwolscine from Alpha-2 adrenergic receptor of rat brain membranesMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAlpha-1A/Alpha-1B/Alpha-1D adrenergic receptor(Rattus norvegicus (rat))
University Of Tennessee

Curated by ChEMBL
LigandPNGBDBM50471350(CHEMBL102763)
Affinity DataKi:  73nMAssay Description:Displacement of [3H]-prazosin from Alpha-1 adrenergic receptor of rat brain membranesMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
LigandPNGBDBM50471338(CHEMBL105347)
Affinity DataKi:  95nMAssay Description:Displacement of [3H]rauwolscine from Alpha-2 adrenergic receptor of rat brain membranesMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
LigandPNGBDBM50471346(CHEMBL330185)
Affinity DataKi:  98nMAssay Description:Displacement of [3H]rauwolscine from Alpha-2 adrenergic receptor of rat brain membranesMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
LigandPNGBDBM50471343(CHEMBL319221)
Affinity DataKi:  103nMAssay Description:Displacement of [3H]rauwolscine from Alpha-2 adrenergic receptor of rat brain membranesMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAlpha-1A/Alpha-1B/Alpha-1D adrenergic receptor(Rattus norvegicus (rat))
University Of Tennessee

Curated by ChEMBL
LigandPNGBDBM50471340(CHEMBL317912)
Affinity DataKi:  126nMAssay Description:Displacement of [3H]-prazosin from Alpha-1 adrenergic receptor of rat brain membranesMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAlpha-1A/Alpha-1B/Alpha-1D adrenergic receptor(Rattus norvegicus (rat))
University Of Tennessee

Curated by ChEMBL
LigandPNGBDBM50471343(CHEMBL319221)
Affinity DataKi:  131nMAssay Description:Displacement of [3H]-prazosin from Alpha-1 adrenergic receptor of rat brain membranesMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
LigandPNGBDBM50471347(CHEMBL319984)
Affinity DataKi:  169nMAssay Description:Displacement of [3H]rauwolscine from Alpha-2 adrenergic receptor of rat brain membranesMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAlpha-1A/Alpha-1B/Alpha-1D adrenergic receptor(Rattus norvegicus (rat))
University Of Tennessee

Curated by ChEMBL
LigandPNGBDBM50471338(CHEMBL105347)
Affinity DataKi:  191nMAssay Description:Displacement of [3H]-prazosin from Alpha-1 adrenergic receptor of rat brain membranesMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAlpha-1A/Alpha-1B/Alpha-1D adrenergic receptor(Rattus norvegicus (rat))
University Of Tennessee

Curated by ChEMBL
LigandPNGBDBM50471347(CHEMBL319984)
Affinity DataKi:  198nMAssay Description:Displacement of [3H]-prazosin from Alpha-1 adrenergic receptor of rat brain membranesMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
LigandPNGBDBM50471348(CHEMBL103448)
Affinity DataKi:  201nMAssay Description:Displacement of [3H]rauwolscine from Alpha-2 adrenergic receptor of rat brain membranesMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
LigandPNGBDBM50471344(CHEMBL422247)
Affinity DataKi:  232nMAssay Description:Displacement of [3H]rauwolscine from Alpha-2 adrenergic receptor of rat brain membranesMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAlpha-1A/Alpha-1B/Alpha-1D adrenergic receptor(Rattus norvegicus (rat))
University Of Tennessee

Curated by ChEMBL
LigandPNGBDBM50471346(CHEMBL330185)
Affinity DataKi:  243nMAssay Description:Displacement of [3H]-prazosin from Alpha-1 adrenergic receptor of rat brain membranesMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
LigandPNGBDBM50471339(CHEMBL103500)
Affinity DataKi:  580nMAssay Description:Displacement of [3H]rauwolscine from Alpha-2 adrenergic receptor of rat brain membranesMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAlpha-1A/Alpha-1B/Alpha-1D adrenergic receptor(Rattus norvegicus (rat))
University Of Tennessee

Curated by ChEMBL
LigandPNGBDBM50471342(CHEMBL322907)
Affinity DataKi:  992nMAssay Description:Displacement of [3H]-prazosin from Alpha-1 adrenergic receptor of rat brain membranesMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAlpha-1A/Alpha-1B/Alpha-1D adrenergic receptor(Rattus norvegicus (rat))
University Of Tennessee

Curated by ChEMBL
LigandPNGBDBM50036913((+-)-4-(alpha,2,3-trimethylbenzyl)imidazole | 4-[1...)
Affinity DataKi:  1.11E+3nMAssay Description:Displacement of [3H]-prazosin from Alpha-1 adrenergic receptor of rat brain membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50471349(CHEMBL321964)
Affinity DataKi:  1.42E+3nMAssay Description:Displacement of [3H]rauwolscine from Alpha-2 adrenergic receptor of rat brain membranesMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
LigandPNGBDBM50471345(CHEMBL102538)
Affinity DataKi:  1.57E+3nMAssay Description:Displacement of [3H]rauwolscine from Alpha-2 adrenergic receptor of rat brain membranesMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAlpha-1A/Alpha-1B/Alpha-1D adrenergic receptor(Rattus norvegicus (rat))
University Of Tennessee

Curated by ChEMBL
LigandPNGBDBM50471339(CHEMBL103500)
Affinity DataKi:  1.63E+3nMAssay Description:Displacement of [3H]-prazosin from Alpha-1 adrenergic receptor of rat brain membranesMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAlpha-1A/Alpha-1B/Alpha-1D adrenergic receptor(Rattus norvegicus (rat))
University Of Tennessee

Curated by ChEMBL
LigandPNGBDBM50471348(CHEMBL103448)
Affinity DataKi:  1.77E+3nMAssay Description:Displacement of [3H]-prazosin from Alpha-1 adrenergic receptor of rat brain membranesMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
LigandPNGBDBM50471341(CHEMBL103438)
Affinity DataKi:  2.67E+3nMAssay Description:Displacement of [3H]rauwolscine from Alpha-2 adrenergic receptor of rat brain membranesMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAlpha-1A/Alpha-1B/Alpha-1D adrenergic receptor(Rattus norvegicus (rat))
University Of Tennessee

Curated by ChEMBL
LigandPNGBDBM50471344(CHEMBL422247)
Affinity DataKi:  2.96E+3nMAssay Description:Displacement of [3H]-prazosin from Alpha-1 adrenergic receptor of rat brain membranesMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAlpha-1A/Alpha-1B/Alpha-1D adrenergic receptor(Rattus norvegicus (rat))
University Of Tennessee

Curated by ChEMBL
LigandPNGBDBM50471349(CHEMBL321964)
Affinity DataKi:  2.97E+3nMAssay Description:Displacement of [3H]-prazosin from Alpha-1 adrenergic receptor of rat brain membranesMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAlpha-1A/Alpha-1B/Alpha-1D adrenergic receptor(Rattus norvegicus (rat))
University Of Tennessee

Curated by ChEMBL
LigandPNGBDBM50471341(CHEMBL103438)
Affinity DataKi:  8.25E+3nMAssay Description:Displacement of [3H]-prazosin from Alpha-1 adrenergic receptor of rat brain membranesMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAlpha-1A/Alpha-1B/Alpha-1D adrenergic receptor(Rattus norvegicus (rat))
University Of Tennessee

Curated by ChEMBL
LigandPNGBDBM50471345(CHEMBL102538)
Affinity DataKi:  1.42E+4nMAssay Description:Displacement of [3H]-prazosin from Alpha-1 adrenergic receptor of rat brain membranesMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed