Compile Data Set for Download or QSAR
Report error Found 18 Enz. Inhib. hit(s) with all data for entry = 50007231
TargetProthrombin(Human)
Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50060001({(R)-1-Cyclohexyl-2-[(S)-2-((S)-1-formyl-4-guanidi...)
Affinity DataIC50: 12nMAssay Description:In vitro inhibitory activity against human ProthrombinMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProthrombin(Human)
Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50029506(tert-butyloxy carbonyl-D-ethylphenylglycine-Pro-Ar...)
Affinity DataIC50: 16nMAssay Description:In vitro inhibitory activity against human ProthrombinMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProthrombin(Human)
Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50060000((S)-1-((R)-2-Methylamino-2-phenyl-acetyl)-pyrrolid...)
Affinity DataIC50: 18nMAssay Description:In vitro inhibitory activity against human ProthrombinMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProthrombin(Human)
Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50060009((S)-1-((R)-2-Amino-2-phenyl-acetyl)-pyrrolidine-2-...)
Affinity DataIC50: 18nMAssay Description:In vitro inhibitory activity against human ProthrombinMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProthrombin(Human)
Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50060007({(R)-2-[(S)-2-((S)-1-Formyl-4-guanidino-butylcarba...)
Affinity DataIC50: 18nMAssay Description:In vitro inhibitory activity against human ProthrombinMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProthrombin(Human)
Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50060005((S)-1-((S)-1,2,3,4-Tetrahydro-isoquinoline-1-carbo...)
Affinity DataIC50: 19nMAssay Description:In vitro inhibitory activity against human ProthrombinMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProthrombin(Human)
Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50060008({(R)-2-[(S)-2-((S)-1-Formyl-4-guanidino-butylcarba...)
Affinity DataIC50: 23nMAssay Description:In vitro inhibitory activity against human ProthrombinMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProthrombin(Human)
Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50029500((S)-1-((S)-1,2,3,4-Tetrahydro-isoquinoline-3-carbo...)
Affinity DataIC50: 25nMAssay Description:In vitro inhibitory activity against human ProthrombinMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProthrombin(Human)
Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50060011([(R)-2-[(S)-2-((S)-1-Formyl-4-guanidino-butylcarba...)
Affinity DataIC50: 27nMAssay Description:In vitro inhibitory activity against human ProthrombinMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProthrombin(Human)
Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50060002({(R)-1-(4-Fluoro-phenyl)-2-[(S)-2-((S)-1-formyl-4-...)
Affinity DataIC50: 30nMAssay Description:In vitro inhibitory activity against human ProthrombinMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProthrombin(Human)
Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50029511({(R)-1-Benzyl-2-[(S)-2-((S)-1-formyl-4-guanidino-b...)
Affinity DataIC50: 45nMAssay Description:In vitro inhibitory activity against human ProthrombinMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProthrombin(Human)
Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50060003({2-[(S)-2-((S)-1-Formyl-4-guanidino-butylcarbamoyl...)
Affinity DataIC50: 85nMAssay Description:In vitro inhibitory activity against human ProthrombinMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProthrombin(Human)
Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50060003({2-[(S)-2-((S)-1-Formyl-4-guanidino-butylcarbamoyl...)
Affinity DataIC50: 85nMAssay Description:In vitro inhibitory activity against human ProthrombinMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProthrombin(Human)
Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50060006([(R)-2-[(S)-2-((S)-1-Formyl-4-guanidino-butylcarba...)
Affinity DataIC50: 89nMAssay Description:In vitro inhibitory activity against human ProthrombinMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProthrombin(Human)
Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50060013((S)-1-((R)-2-Phenyl-propionyl)-pyrrolidine-2-carbo...)
Affinity DataIC50: 94nMAssay Description:In vitro inhibitory activity against human ProthrombinMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProthrombin(Human)
Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50060010((S)-1-((R)-2-Phenyl-butyryl)-pyrrolidine-2-carboxy...)
Affinity DataIC50: 130nMAssay Description:In vitro inhibitory activity against human ProthrombinMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProthrombin(Human)
Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50060004((S)-1-((R)-2-Methoxy-2-phenyl-acetyl)-pyrrolidine-...)
Affinity DataIC50: 250nMAssay Description:In vitro inhibitory activity against human ProthrombinMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProthrombin(Human)
Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50060012((S)-1-((S)-2-Phenyl-propionyl)-pyrrolidine-2-carbo...)
Affinity DataIC50: 5.10E+3nMAssay Description:In vitro inhibitory activity against human ProthrombinMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed