Compile Data Set for Download or QSAR
Report error Found 5 Enz. Inhib. hit(s) with all data for entry = 50007277
TargetGlutamate receptor ionotropic, NMDA 1(Rat)
Cocensys

Curated by ChEMBL
LigandPNGBDBM50048173(C,C,C-Trifluoro-N-(7-nitro-2-oxo-1,2-dihydro-quino...)
Affinity DataIC50: 620nMAssay Description:Inhibition of binding of [3H]DCKA to N-methyl-D-aspartate glutamate receptor 1 in rat brain membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGlutamate receptor ionotropic, NMDA 1(Rat)
Cocensys

Curated by ChEMBL
LigandPNGBDBM50060699(7-Nitro-5-oxy-1,4-dihydro-pyrido[2,3-b]pyrazine-2,...)
Affinity DataIC50: 690nMAssay Description:Binding affinity in rat brain cortical membranes by the displacement of [3H]- DCKA at N-methyl-D-aspartate glutamate receptor 1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGlutamate receptor ionotropic, NMDA 1(Rat)
Cocensys

Curated by ChEMBL
LigandPNGBDBM50060694(7-Bromo-5-oxy-1,4-dihydro-pyrido[2,3-b]pyrazine-2,...)
Affinity DataIC50: 1.00E+3nMAssay Description:Binding affinity in rat brain cortical membranes by the displacement of [3H]- DCKA at N-methyl-D-aspartate glutamate receptor 1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGlutamate receptor ionotropic, NMDA 1(Rat)
Cocensys

Curated by ChEMBL
LigandPNGBDBM50060700(5-Oxy-7-trifluoromethyl-1,4-dihydro-pyrido[2,3-b]p...)
Affinity DataIC50: 1.05E+3nMAssay Description:Binding affinity in rat brain cortical membranes by the displacement of [3H]- DCKA at N-methyl-D-aspartate glutamate receptor 1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGlutamate receptor ionotropic, NMDA 1(Rat)
Cocensys

Curated by ChEMBL
LigandPNGBDBM50060695(7-Methyl-5-oxy-1,4-dihydro-pyrido[2,3-b]pyrazine-2...)
Affinity DataIC50: 5.90E+3nMAssay Description:Binding affinity in rat brain cortical membranes by the displacement of [3H]- DCKA at N-methyl-D-aspartate glutamate receptor 1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed