Compile Data Set for Download or QSAR
Report error Found 54 Enz. Inhib. hit(s) with all data for entry = 50003470
TargetcAMP-specific 3',5'-cyclic phosphodiesterase 4A/4B/4C/4D(Human)
Hokuriku University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50471409BDBM50471409(CHEMBL326464)
Affinity DataIC50: 1.40E+3nMAssay Description:Inhibitory activity against Phosphodiesterase 4 from heart.More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2020
Entry Details Article
PubMed
TargetcAMP-specific 3',5'-cyclic phosphodiesterase 4A/4B/4C/4D(Human)
Hokuriku University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50471416BDBM50471416(CHEMBL333599)
Affinity DataIC50: 1.60E+3nMAssay Description:Inhibitory activity against Phosphodiesterase 4 from heart.More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2020
Entry Details Article
PubMed
TargetcAMP-specific 3',5'-cyclic phosphodiesterase 4A/4B/4C/4D(Human)
Hokuriku University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50471421BDBM50471421(CHEMBL109574)
Affinity DataIC50: 1.90E+3nMAssay Description:Inhibitory activity against Phosphodiesterase 4 from heart.More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2020
Entry Details Article
PubMed
TargetcAMP-specific 3',5'-cyclic phosphodiesterase 4A/4B/4C/4D(Human)
Hokuriku University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50471412BDBM50471412(CHEMBL110304 | XT-44)
Affinity DataIC50: 2.20E+3nMAssay Description:Inhibitory activity against Phosphodiesterase 4 from heart.More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2020
Entry Details Article
PubMed
TargetcAMP-specific 3',5'-cyclic phosphodiesterase 4A/4B/4C/4D(Human)
Hokuriku University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50471418BDBM50471418(CHEMBL326285)
Affinity DataIC50: 3.10E+3nMAssay Description:Inhibitory activity against Phosphodiesterase 4 from heart.More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2020
Entry Details Article
PubMed
TargetcAMP-specific 3',5'-cyclic phosphodiesterase 4A/4B/4C/4D(Human)
Hokuriku University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50471411BDBM50471411(CHEMBL109550)
Affinity DataIC50: 4.70E+3nMAssay Description:Inhibitory activity against Phosphodiesterase 4 from heart.More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2020
Entry Details Article
PubMed
TargetcAMP-specific 3',5'-cyclic phosphodiesterase 4A/4B/4C/4D(Human)
Hokuriku University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50010981BDBM50010981(4-(3-Butoxy-4-methoxy-benzyl)-imidazolidin-2-one |...)
Affinity DataIC50: 4.80E+3nMAssay Description:Inhibitory activity against Phosphodiesterase 4 from heart.More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2020
Entry Details Article
PubMed
TargetcAMP-specific 3',5'-cyclic phosphodiesterase 4A/4B/4C/4D(Human)
Hokuriku University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50471413BDBM50471413(CHEMBL111486)
Affinity DataIC50: 5.10E+3nMAssay Description:Inhibitory activity against Phosphodiesterase 4 from heart.More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2020
Entry Details Article
PubMed
TargetcAMP-specific 3',5'-cyclic phosphodiesterase 4A/4B/4C/4D(Human)
Hokuriku University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50471408BDBM50471408(CHEMBL109427)
Affinity DataIC50: 1.30E+4nMAssay Description:Inhibitory activity against Phosphodiesterase 4 from heart.More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2020
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50471421BDBM50471421(CHEMBL109574)
Affinity DataIC50: 1.40E+4nMAssay Description:Inhibitory activity against PDE1 from cerebral cortexMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2020
Entry Details Article
PubMed
TargetcGMP-inhibited 3',5'-cyclic phosphodiesterase 3A/3B(Human)
Hokuriku University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 34651BDBM34651(MLS000069829 | cid_3698 | SMR000058850 | CHEMBL128...)
Affinity DataIC50: 1.60E+4nMAssay Description:Inhibitory activity against Phosphodiesterase 3 from heart.More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2020
Entry Details Article
PubMed
TargetcAMP-specific 3',5'-cyclic phosphodiesterase 4A/4B/4C/4D(Human)
Hokuriku University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50471410BDBM50471410(CHEMBL322358)
Affinity DataIC50: 1.80E+4nMAssay Description:Inhibitory activity against Phosphodiesterase 4 from heart.More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2020
Entry Details Article
PubMed
TargetcAMP-specific 3',5'-cyclic phosphodiesterase 4A/4B/4C/4D(Human)
Hokuriku University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50471422BDBM50471422(CHEMBL320350)
Affinity DataIC50: 3.90E+4nMAssay Description:Inhibitory activity against Phosphodiesterase 4 from heart.More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2020
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50471409BDBM50471409(CHEMBL326464)
Affinity DataIC50: 4.00E+4nMAssay Description:Inhibitory activity against PDE1 from cerebral cortexMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2020
Entry Details Article
PubMed
TargetcAMP-specific 3',5'-cyclic phosphodiesterase 4A/4B/4C/4D(Human)
Hokuriku University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50471414BDBM50471414(CHEMBL109639)
Affinity DataIC50: 4.90E+4nMAssay Description:Inhibitory activity against Phosphodiesterase 4 from heart.More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2020
Entry Details Article
PubMed
TargetcAMP-specific 3',5'-cyclic phosphodiesterase 4A/4B/4C/4D(Human)
Hokuriku University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 82053BDBM82053(8-(2-Furyl)theophylline | US9138393, Theophylline ...)
Affinity DataIC50: 8.10E+4nMAssay Description:Inhibitory activity against Phosphodiesterase 4 from heart.More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2020
Entry Details Article
PubMed
TargetcGMP-inhibited 3',5'-cyclic phosphodiesterase 3A/3B(Human)
Hokuriku University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50471419BDBM50471419(CHEMBL111071)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibitory activity against Phosphodiesterase 3 from heart.More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2020
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50471413BDBM50471413(CHEMBL111486)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibitory activity against PDE1 from cerebral cortexMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2020
Entry Details Article
PubMed
TargetcGMP-inhibited 3',5'-cyclic phosphodiesterase 3A/3B(Human)
Hokuriku University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50471417BDBM50471417(CHEMBL111466)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibitory activity against Phosphodiesterase 3 from heart.More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2020
Entry Details Article
PubMed
TargetcGMP-inhibited 3',5'-cyclic phosphodiesterase 3A/3B(Human)
Hokuriku University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50471414BDBM50471414(CHEMBL109639)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibitory activity against Phosphodiesterase 3 from heart.More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2020
Entry Details Article
PubMed
TargetcGMP-inhibited 3',5'-cyclic phosphodiesterase 3A/3B(Human)
Hokuriku University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50471415BDBM50471415(CHEMBL111990)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibitory activity against Phosphodiesterase 3 from heart.More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2020
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50471416BDBM50471416(CHEMBL333599)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibitory activity against PDE1 from cerebral cortexMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2020
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50471410BDBM50471410(CHEMBL322358)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibitory activity against PDE1 from cerebral cortexMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2020
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50471411BDBM50471411(CHEMBL109550)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibitory activity against PDE1 from cerebral cortexMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2020
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50471418BDBM50471418(CHEMBL326285)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibitory activity against PDE1 from cerebral cortexMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2020
Entry Details Article
PubMed
TargetcAMP-specific 3',5'-cyclic phosphodiesterase 4A/4B/4C/4D(Human)
Hokuriku University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50471417BDBM50471417(CHEMBL111466)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibitory activity against Phosphodiesterase 4 from heart.More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2020
Entry Details Article
PubMed
TargetcGMP-inhibited 3',5'-cyclic phosphodiesterase 3A/3B(Human)
Hokuriku University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50471409BDBM50471409(CHEMBL326464)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibitory activity against Phosphodiesterase 3 from heart.More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2020
Entry Details Article
PubMed
TargetcGMP-inhibited 3',5'-cyclic phosphodiesterase 3A/3B(Human)
Hokuriku University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50471418BDBM50471418(CHEMBL326285)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibitory activity against Phosphodiesterase 3 from heart.More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2020
Entry Details Article
PubMed
TargetcAMP-specific 3',5'-cyclic phosphodiesterase 4A/4B/4C/4D(Human)
Hokuriku University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50471419BDBM50471419(CHEMBL111071)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibitory activity against Phosphodiesterase 4 from heart.More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2020
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50471419BDBM50471419(CHEMBL111071)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibitory activity against PDE1 from cerebral cortexMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2020
Entry Details Article
PubMed
TargetcGMP-inhibited 3',5'-cyclic phosphodiesterase 3A/3B(Human)
Hokuriku University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50471416BDBM50471416(CHEMBL333599)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibitory activity against Phosphodiesterase 3 from heart.More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2020
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50471417BDBM50471417(CHEMBL111466)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibitory activity against PDE1 from cerebral cortexMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2020
Entry Details Article
PubMed
TargetcGMP-inhibited 3',5'-cyclic phosphodiesterase 3A/3B(Human)
Hokuriku University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50471411BDBM50471411(CHEMBL109550)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibitory activity against Phosphodiesterase 3 from heart.More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2020
Entry Details Article
PubMed
TargetcGMP-inhibited 3',5'-cyclic phosphodiesterase 3A/3B(Human)
Hokuriku University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50471410BDBM50471410(CHEMBL322358)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibitory activity against Phosphodiesterase 3 from heart.More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2020
Entry Details Article
PubMed
TargetcGMP-inhibited 3',5'-cyclic phosphodiesterase 3A/3B(Human)
Hokuriku University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50471420BDBM50471420(CHEMBL108884)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibitory activity against Phosphodiesterase 3 from heart.More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2020
Entry Details Article
PubMed
TargetcAMP-specific 3',5'-cyclic phosphodiesterase 4A/4B/4C/4D(Human)
Hokuriku University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50471415BDBM50471415(CHEMBL111990)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibitory activity against Phosphodiesterase 4 from heart.More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2020
Entry Details Article
PubMed
TargetcGMP-inhibited 3',5'-cyclic phosphodiesterase 3A/3B(Human)
Hokuriku University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50471413BDBM50471413(CHEMBL111486)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibitory activity against Phosphodiesterase 3 from heart.More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2020
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50471415BDBM50471415(CHEMBL111990)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibitory activity against PDE1 from cerebral cortexMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2020
Entry Details Article
PubMed
TargetcAMP-specific 3',5'-cyclic phosphodiesterase 4A/4B/4C/4D(Human)
Hokuriku University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50471420BDBM50471420(CHEMBL108884)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibitory activity against Phosphodiesterase 4 from heart.More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2020
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50471408BDBM50471408(CHEMBL109427)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibitory activity against PDE1 from cerebral cortexMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2020
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50471414BDBM50471414(CHEMBL109639)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibitory activity against PDE1 from cerebral cortexMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2020
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50471420BDBM50471420(CHEMBL108884)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibitory activity against PDE1 from cerebral cortexMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2020
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50471422BDBM50471422(CHEMBL320350)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibitory activity against PDE1 from cerebral cortexMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2020
Entry Details Article
PubMed
TargetcGMP-inhibited 3',5'-cyclic phosphodiesterase 3A/3B(Human)
Hokuriku University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50471408BDBM50471408(CHEMBL109427)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibitory activity against Phosphodiesterase 3 from heart.More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2020
Entry Details Article
PubMed
TargetcGMP-inhibited 3',5'-cyclic phosphodiesterase 3A/3B(Human)
Hokuriku University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50471422BDBM50471422(CHEMBL320350)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibitory activity against Phosphodiesterase 3 from heart.More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2020
Entry Details Article
PubMed
TargetcGMP-inhibited 3',5'-cyclic phosphodiesterase 3A/3B(Human)
Hokuriku University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50471421BDBM50471421(CHEMBL109574)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibitory activity against Phosphodiesterase 3 from heart.More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2020
Entry Details Article
PubMed
TargetcAMP-specific 3',5'-cyclic phosphodiesterase 4A/4B/4C/4D(Human)
Hokuriku University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 34651BDBM34651(MLS000069829 | cid_3698 | SMR000058850 | CHEMBL128...)
Affinity DataIC50: 1.01E+5nMAssay Description:Inhibitory activity against Phosphodiesterase 4 from heart.More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2020
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50471412BDBM50471412(CHEMBL110304 | XT-44)
Affinity DataIC50: 1.49E+5nMAssay Description:Inhibitory activity against PDE1 from cerebral cortexMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2020
Entry Details Article
PubMed
TargetcGMP-inhibited 3',5'-cyclic phosphodiesterase 3A/3B(Human)
Hokuriku University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 82053BDBM82053(8-(2-Furyl)theophylline | US9138393, Theophylline ...)
Affinity DataIC50: 2.40E+5nMAssay Description:Inhibitory activity against Phosphodiesterase 3 from heart.More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2020
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 34651BDBM34651(MLS000069829 | cid_3698 | SMR000058850 | CHEMBL128...)
Affinity DataIC50: 3.00E+5nMAssay Description:Inhibitory activity against PDE1 from cerebral cortexMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2020
Entry Details Article
PubMed
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