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Found 54 Enz. Inhib. hit(s) with all data for entry = 50003470
TargetcAMP-specific 3',5'-cyclic phosphodiesterase 4A/4B/4C/4D(Homo sapiens (Human))
Hokuriku University

Curated by ChEMBL
LigandPNGBDBM50471409(CHEMBL326464)
Affinity DataIC50:  1.40E+3nMAssay Description:Inhibitory activity against Phosphodiesterase 4 from heart.More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetcAMP-specific 3',5'-cyclic phosphodiesterase 4A/4B/4C/4D(Homo sapiens (Human))
Hokuriku University

Curated by ChEMBL
LigandPNGBDBM50471416(CHEMBL333599)
Affinity DataIC50:  1.60E+3nMAssay Description:Inhibitory activity against Phosphodiesterase 4 from heart.More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetcAMP-specific 3',5'-cyclic phosphodiesterase 4A/4B/4C/4D(Homo sapiens (Human))
Hokuriku University

Curated by ChEMBL
LigandPNGBDBM50471421(CHEMBL109574)
Affinity DataIC50:  1.90E+3nMAssay Description:Inhibitory activity against Phosphodiesterase 4 from heart.More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetcAMP-specific 3',5'-cyclic phosphodiesterase 4A/4B/4C/4D(Homo sapiens (Human))
Hokuriku University

Curated by ChEMBL
LigandPNGBDBM50471412(CHEMBL110304 | XT-44)
Affinity DataIC50:  2.20E+3nMAssay Description:Inhibitory activity against Phosphodiesterase 4 from heart.More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetcAMP-specific 3',5'-cyclic phosphodiesterase 4A/4B/4C/4D(Homo sapiens (Human))
Hokuriku University

Curated by ChEMBL
LigandPNGBDBM50471418(CHEMBL326285)
Affinity DataIC50:  3.10E+3nMAssay Description:Inhibitory activity against Phosphodiesterase 4 from heart.More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetcAMP-specific 3',5'-cyclic phosphodiesterase 4A/4B/4C/4D(Homo sapiens (Human))
Hokuriku University

Curated by ChEMBL
LigandPNGBDBM50471411(CHEMBL109550)
Affinity DataIC50:  4.70E+3nMAssay Description:Inhibitory activity against Phosphodiesterase 4 from heart.More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetcAMP-specific 3',5'-cyclic phosphodiesterase 4A/4B/4C/4D(Homo sapiens (Human))
Hokuriku University

Curated by ChEMBL
LigandPNGBDBM50010981((Ro 20-1724)4-(3-Butoxy-4-methoxy-benzyl)-imidazol...)
Affinity DataIC50:  4.80E+3nMAssay Description:Inhibitory activity against Phosphodiesterase 4 from heart.More data for this Ligand-Target Pair
TargetcAMP-specific 3',5'-cyclic phosphodiesterase 4A/4B/4C/4D(Homo sapiens (Human))
Hokuriku University

Curated by ChEMBL
LigandPNGBDBM50471413(CHEMBL111486)
Affinity DataIC50:  5.10E+3nMAssay Description:Inhibitory activity against Phosphodiesterase 4 from heart.More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetcAMP-specific 3',5'-cyclic phosphodiesterase 4A/4B/4C/4D(Homo sapiens (Human))
Hokuriku University

Curated by ChEMBL
LigandPNGBDBM50471408(CHEMBL109427)
Affinity DataIC50:  1.30E+4nMAssay Description:Inhibitory activity against Phosphodiesterase 4 from heart.More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
LigandPNGBDBM50471421(CHEMBL109574)
Affinity DataIC50:  1.40E+4nMAssay Description:Inhibitory activity against PDE1 from cerebral cortexMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetcGMP-inhibited 3',5'-cyclic phosphodiesterase 3A/3B(Homo sapiens (Human))
Hokuriku University

Curated by ChEMBL
LigandPNGBDBM34651(Amrinon | Amrinone | CHEMBL12856 | Cordemcura | IN...)
Affinity DataIC50:  1.60E+4nMAssay Description:Inhibitory activity against Phosphodiesterase 3 from heart.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcAMP-specific 3',5'-cyclic phosphodiesterase 4A/4B/4C/4D(Homo sapiens (Human))
Hokuriku University

Curated by ChEMBL
LigandPNGBDBM50471410(CHEMBL322358)
Affinity DataIC50:  1.80E+4nMAssay Description:Inhibitory activity against Phosphodiesterase 4 from heart.More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetcAMP-specific 3',5'-cyclic phosphodiesterase 4A/4B/4C/4D(Homo sapiens (Human))
Hokuriku University

Curated by ChEMBL
LigandPNGBDBM50471422(CHEMBL320350)
Affinity DataIC50:  3.90E+4nMAssay Description:Inhibitory activity against Phosphodiesterase 4 from heart.More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
LigandPNGBDBM50471409(CHEMBL326464)
Affinity DataIC50:  4.00E+4nMAssay Description:Inhibitory activity against PDE1 from cerebral cortexMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetcAMP-specific 3',5'-cyclic phosphodiesterase 4A/4B/4C/4D(Homo sapiens (Human))
Hokuriku University

Curated by ChEMBL
LigandPNGBDBM50471414(CHEMBL109639)
Affinity DataIC50:  4.90E+4nMAssay Description:Inhibitory activity against Phosphodiesterase 4 from heart.More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetcAMP-specific 3',5'-cyclic phosphodiesterase 4A/4B/4C/4D(Homo sapiens (Human))
Hokuriku University

Curated by ChEMBL
LigandPNGBDBM82053(8-(2-Furyl)theophylline | US9138393, Theophylline ...)
Affinity DataIC50:  8.10E+4nMAssay Description:Inhibitory activity against Phosphodiesterase 4 from heart.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50471422(CHEMBL320350)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibitory activity against PDE1 from cerebral cortexMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetcGMP-inhibited 3',5'-cyclic phosphodiesterase 3A/3B(Homo sapiens (Human))
Hokuriku University

Curated by ChEMBL
LigandPNGBDBM50471408(CHEMBL109427)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibitory activity against Phosphodiesterase 3 from heart.More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetcGMP-inhibited 3',5'-cyclic phosphodiesterase 3A/3B(Homo sapiens (Human))
Hokuriku University

Curated by ChEMBL
LigandPNGBDBM50471422(CHEMBL320350)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibitory activity against Phosphodiesterase 3 from heart.More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetcGMP-inhibited 3',5'-cyclic phosphodiesterase 3A/3B(Homo sapiens (Human))
Hokuriku University

Curated by ChEMBL
LigandPNGBDBM50471421(CHEMBL109574)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibitory activity against Phosphodiesterase 3 from heart.More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
LigandPNGBDBM50471420(CHEMBL108884)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibitory activity against PDE1 from cerebral cortexMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetcAMP-specific 3',5'-cyclic phosphodiesterase 4A/4B/4C/4D(Homo sapiens (Human))
Hokuriku University

Curated by ChEMBL
LigandPNGBDBM50471415(CHEMBL111990)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibitory activity against Phosphodiesterase 4 from heart.More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetcGMP-inhibited 3',5'-cyclic phosphodiesterase 3A/3B(Homo sapiens (Human))
Hokuriku University

Curated by ChEMBL
LigandPNGBDBM50471411(CHEMBL109550)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibitory activity against Phosphodiesterase 3 from heart.More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
LigandPNGBDBM50471415(CHEMBL111990)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibitory activity against PDE1 from cerebral cortexMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
LigandPNGBDBM50471414(CHEMBL109639)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibitory activity against PDE1 from cerebral cortexMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
LigandPNGBDBM50471408(CHEMBL109427)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibitory activity against PDE1 from cerebral cortexMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetcAMP-specific 3',5'-cyclic phosphodiesterase 4A/4B/4C/4D(Homo sapiens (Human))
Hokuriku University

Curated by ChEMBL
LigandPNGBDBM50471420(CHEMBL108884)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibitory activity against Phosphodiesterase 4 from heart.More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetcGMP-inhibited 3',5'-cyclic phosphodiesterase 3A/3B(Homo sapiens (Human))
Hokuriku University

Curated by ChEMBL
LigandPNGBDBM50471409(CHEMBL326464)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibitory activity against Phosphodiesterase 3 from heart.More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetcAMP-specific 3',5'-cyclic phosphodiesterase 4A/4B/4C/4D(Homo sapiens (Human))
Hokuriku University

Curated by ChEMBL
LigandPNGBDBM50471417(CHEMBL111466)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibitory activity against Phosphodiesterase 4 from heart.More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
LigandPNGBDBM50471418(CHEMBL326285)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibitory activity against PDE1 from cerebral cortexMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
LigandPNGBDBM50471419(CHEMBL111071)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibitory activity against PDE1 from cerebral cortexMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetcAMP-specific 3',5'-cyclic phosphodiesterase 4A/4B/4C/4D(Homo sapiens (Human))
Hokuriku University

Curated by ChEMBL
LigandPNGBDBM50471419(CHEMBL111071)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibitory activity against Phosphodiesterase 4 from heart.More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetcGMP-inhibited 3',5'-cyclic phosphodiesterase 3A/3B(Homo sapiens (Human))
Hokuriku University

Curated by ChEMBL
LigandPNGBDBM50471418(CHEMBL326285)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibitory activity against Phosphodiesterase 3 from heart.More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
LigandPNGBDBM50471417(CHEMBL111466)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibitory activity against PDE1 from cerebral cortexMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetcGMP-inhibited 3',5'-cyclic phosphodiesterase 3A/3B(Homo sapiens (Human))
Hokuriku University

Curated by ChEMBL
LigandPNGBDBM50471416(CHEMBL333599)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibitory activity against Phosphodiesterase 3 from heart.More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetcGMP-inhibited 3',5'-cyclic phosphodiesterase 3A/3B(Homo sapiens (Human))
Hokuriku University

Curated by ChEMBL
LigandPNGBDBM50471420(CHEMBL108884)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibitory activity against Phosphodiesterase 3 from heart.More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetcGMP-inhibited 3',5'-cyclic phosphodiesterase 3A/3B(Homo sapiens (Human))
Hokuriku University

Curated by ChEMBL
LigandPNGBDBM50471410(CHEMBL322358)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibitory activity against Phosphodiesterase 3 from heart.More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetcGMP-inhibited 3',5'-cyclic phosphodiesterase 3A/3B(Homo sapiens (Human))
Hokuriku University

Curated by ChEMBL
LigandPNGBDBM50471413(CHEMBL111486)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibitory activity against Phosphodiesterase 3 from heart.More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
LigandPNGBDBM50471413(CHEMBL111486)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibitory activity against PDE1 from cerebral cortexMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetcGMP-inhibited 3',5'-cyclic phosphodiesterase 3A/3B(Homo sapiens (Human))
Hokuriku University

Curated by ChEMBL
LigandPNGBDBM50471419(CHEMBL111071)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibitory activity against Phosphodiesterase 3 from heart.More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetcGMP-inhibited 3',5'-cyclic phosphodiesterase 3A/3B(Homo sapiens (Human))
Hokuriku University

Curated by ChEMBL
LigandPNGBDBM50471417(CHEMBL111466)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibitory activity against Phosphodiesterase 3 from heart.More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
LigandPNGBDBM50471416(CHEMBL333599)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibitory activity against PDE1 from cerebral cortexMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetcGMP-inhibited 3',5'-cyclic phosphodiesterase 3A/3B(Homo sapiens (Human))
Hokuriku University

Curated by ChEMBL
LigandPNGBDBM50471415(CHEMBL111990)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibitory activity against Phosphodiesterase 3 from heart.More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetcGMP-inhibited 3',5'-cyclic phosphodiesterase 3A/3B(Homo sapiens (Human))
Hokuriku University

Curated by ChEMBL
LigandPNGBDBM50471414(CHEMBL109639)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibitory activity against Phosphodiesterase 3 from heart.More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
LigandPNGBDBM50471411(CHEMBL109550)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibitory activity against PDE1 from cerebral cortexMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
LigandPNGBDBM50471410(CHEMBL322358)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibitory activity against PDE1 from cerebral cortexMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetcAMP-specific 3',5'-cyclic phosphodiesterase 4A/4B/4C/4D(Homo sapiens (Human))
Hokuriku University

Curated by ChEMBL
LigandPNGBDBM34651(Amrinon | Amrinone | CHEMBL12856 | Cordemcura | IN...)
Affinity DataIC50:  1.01E+5nMAssay Description:Inhibitory activity against Phosphodiesterase 4 from heart.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50471412(CHEMBL110304 | XT-44)
Affinity DataIC50:  1.49E+5nMAssay Description:Inhibitory activity against PDE1 from cerebral cortexMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetcGMP-inhibited 3',5'-cyclic phosphodiesterase 3A/3B(Homo sapiens (Human))
Hokuriku University

Curated by ChEMBL
LigandPNGBDBM82053(8-(2-Furyl)theophylline | US9138393, Theophylline ...)
Affinity DataIC50:  2.40E+5nMAssay Description:Inhibitory activity against Phosphodiesterase 3 from heart.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50010981((Ro 20-1724)4-(3-Butoxy-4-methoxy-benzyl)-imidazol...)
Affinity DataIC50: >3.00E+5nMAssay Description:Inhibitory activity against PDE1 from cerebral cortexMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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