Compile Data Set for Download or QSAR
maximum 50k data
Found 23 Enz. Inhib. hit(s) with all data for entry = 50036612
Target5-hydroxytryptamine receptor 1B(Rattus norvegicus (Rat))
Astra Arcus

Curated by ChEMBL
LigandPNGBDBM50369356(CHEMBL1744087)
Affinity DataKi:  47nMAssay Description:Binding affinity against 5-hydroxytryptamine 1B receptor in membranes of Rat cerebral cortexMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1B(Rattus norvegicus (Rat))
Astra Arcus

Curated by ChEMBL
LigandPNGBDBM50369357(CHEMBL1201939)
Affinity DataKi:  60nMAssay Description:Binding affinity against 5-hydroxytryptamine 1B receptor in membranes of Rat cerebral cortexMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1B(Rattus norvegicus (Rat))
Astra Arcus

Curated by ChEMBL
LigandPNGBDBM50064466(CHEMBL58961 | Morpholin-4-yl-[8-(morpholin-2-ylmet...)
Affinity DataKi:  240nMAssay Description:Binding affinity against 5-hydroxytryptamine 1B receptor in membranes of Rat cerebral cortexMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1B(Rattus norvegicus (Rat))
Astra Arcus

Curated by ChEMBL
LigandPNGBDBM50064462(8-(Morpholin-2-ylmethoxy)-2H-chromene-3-carbonitri...)
Affinity DataKi:  250nMAssay Description:Binding affinity against 5-hydroxytryptamine 1B receptor in membranes of Rat cerebral cortexMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1B(Rattus norvegicus (Rat))
Astra Arcus

Curated by ChEMBL
LigandPNGBDBM50369355(CHEMBL1202783)
Affinity DataKi:  275nMAssay Description:Binding affinity against 5-hydroxytryptamine 1B receptor in membranes of Rat cerebral cortexMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1B(Rattus norvegicus (Rat))
Astra Arcus

Curated by ChEMBL
LigandPNGBDBM50064464(5-(Morpholin-2-ylmethoxy)-3,4-dihydro-naphthalene-...)
Affinity DataKi:  445nMAssay Description:Binding affinity against 5-hydroxytryptamine 1B receptor in membranes of Rat cerebral cortexMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M3(RAT)
Astra Arcus

Curated by ChEMBL
LigandPNGBDBM50369356(CHEMBL1744087)
Affinity DataKi: >1.00E+3nMAssay Description:Binding affinity against Muscarinic acetylcholine receptor using [3H]QNB as the radioligand.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1B(Rattus norvegicus (Rat))
Astra Arcus

Curated by ChEMBL
LigandPNGBDBM50064467(8-(Piperidin-3-ylmethoxy)-2H-chromene-3-carbonitri...)
Affinity DataKi:  1.40E+3nMAssay Description:Binding affinity against 5-hydroxytryptamine 1B receptor in membranes of Rat cerebral cortexMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 6(RAT)
Astra Arcus

Curated by ChEMBL
LigandPNGBDBM50369356(CHEMBL1744087)
Affinity DataKi: >3.00E+3nMAssay Description:Binding affinity against 5-hydroxytryptamine 6 receptor from CHO cell membranes using [3H]5-HT as the radioligand.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1B(Rattus norvegicus (Rat))
Astra Arcus

Curated by ChEMBL
LigandPNGBDBM50064465(8-(4-Methyl-morpholin-2-ylmethoxy)-2H-chromene-3-c...)
Affinity DataKi:  3.60E+3nMAssay Description:Binding affinity against 5-hydroxytryptamine 1B receptor in membranes of Rat cerebral cortexMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
Astra Arcus

Curated by ChEMBL
LigandPNGBDBM50369356(CHEMBL1744087)
Affinity DataKi: >1.00E+4nMAssay Description:Binding affinity against 5-hydroxytryptamine 1A receptor from rat hippocampus using [3H]8-OH-DPAT as the radioligand.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
Astra Arcus

Curated by ChEMBL
LigandPNGBDBM50369355(CHEMBL1202783)
Affinity DataKi: >1.00E+4nMAssay Description:Binding affinity against 5-hydroxytryptamine 1A receptor from rat hippocampus using [3H]8-OH-DPAT as the radioligand.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
Astra Arcus

Curated by ChEMBL
LigandPNGBDBM50369355(CHEMBL1202783)
Affinity DataKi: >1.00E+4nMAssay Description:Binding affinity against Dopamine receptor D2 from cell LtkhD2A membranes using [3H]raclopride as the radioligand.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2C(Rattus norvegicus (Rat))
Astra Arcus

Curated by ChEMBL
LigandPNGBDBM50369355(CHEMBL1202783)
Affinity DataKi: >1.00E+4nMAssay Description:Binding affinity against 5-hydroxytryptamine 2C receptor from rat cortex using [3H]mesulergine as the radioligand.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSigma non-opioid intracellular receptor 1(RAT)
Astra Arcus

Curated by ChEMBL
LigandPNGBDBM50369355(CHEMBL1202783)
Affinity DataKi: >1.00E+4nMAssay Description:Binding affinity against sigma receptor from rat whole brains using [3H]DTG as the radioligand.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 7(Rattus norvegicus (rat))
Astra Arcus

Curated by ChEMBL
LigandPNGBDBM50369356(CHEMBL1744087)
Affinity DataKi: >1.00E+4nMAssay Description:Binding affinity against 5-hydroxytryptamine 7 receptor using from CHO cell membranes [3H]5-HT as the radioligand.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSigma non-opioid intracellular receptor 1(RAT)
Astra Arcus

Curated by ChEMBL
LigandPNGBDBM50369356(CHEMBL1744087)
Affinity DataKi: >1.00E+4nMAssay Description:Binding affinity against sigma receptor from rat whole brains using [3H]DTG as the radioligand.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
Astra Arcus

Curated by ChEMBL
LigandPNGBDBM50369356(CHEMBL1744087)
Affinity DataKi: >1.00E+4nMAssay Description:Binding affinity against Dopamine receptor D2 from cell LtkhD2A membranes using [3H]raclopride as the radioligand.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2A(Rattus norvegicus (rat))
Astra Arcus

Curated by ChEMBL
LigandPNGBDBM50369355(CHEMBL1202783)
Affinity DataKi: >1.00E+4nMAssay Description:Binding affinity against 5-hydroxytryptamine 2A receptor from rat cortex using [3H]ketanserin as the radioligand.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(1A) dopamine receptor(RAT)
Astra Arcus

Curated by ChEMBL
LigandPNGBDBM50369356(CHEMBL1744087)
Affinity DataKi: >1.00E+4nMAssay Description:Binding affinity against Dopamine receptor D1 in rat striatum using [3H]-SCH- 23390 as the radioligand.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2A(Rattus norvegicus (rat))
Astra Arcus

Curated by ChEMBL
LigandPNGBDBM50369356(CHEMBL1744087)
Affinity DataKi: >1.00E+4nMAssay Description:Binding affinity against 5-hydroxytryptamine 2A receptor from rat cortex using [3H]ketanserin as the radioligand.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(1A) dopamine receptor(RAT)
Astra Arcus

Curated by ChEMBL
LigandPNGBDBM50369355(CHEMBL1202783)
Affinity DataKi: >1.00E+4nMAssay Description:Binding affinity against Dopamine receptor D1 in rat striatum using [3H]-SCH- 23390 as the radioligand.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2C(Rattus norvegicus (Rat))
Astra Arcus

Curated by ChEMBL
LigandPNGBDBM50369356(CHEMBL1744087)
Affinity DataKi: >1.00E+4nMAssay Description:Binding affinity against 5-hydroxytryptamine 2C receptor from rat cortex using [3H]mesulergine as the radioligand.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed