Compile Data Set for Download or QSAR
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Found 37 Enz. Inhib. hit(s) with all data for entry = 50036620
TargetSomatostatin receptor type 2(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50064772(Ala-Gly-cyclo[Cys-Lys-Asn-Phe-Phe-Trp-Lys-Thr-Phe-...)
Affinity DataKi:  0.0400nMAssay Description:Binding affinity towards human sst2 receptor expressed in CHO-K1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 1(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50064772(Ala-Gly-cyclo[Cys-Lys-Asn-Phe-Phe-Trp-Lys-Thr-Phe-...)
Affinity DataKi:  0.380nMAssay Description:Binding affinity towards human sst1 receptor expressed in CHO-K1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 2(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50454938(CHEMBL2052017 | L-363377)
Affinity DataKi:  0.5nMAssay Description:Binding affinity towards human sst2 receptor expressed in CHO-K1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 3(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50064772(Ala-Gly-cyclo[Cys-Lys-Asn-Phe-Phe-Trp-Lys-Thr-Phe-...)
Affinity DataKi:  0.660nMAssay Description:Binding affinity towards human sst3 receptor expressed in CHO-K1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 1(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50064773(1'N-[1-[3-aminomethyl-(1S,3R)-cyclohexylmethylcarb...)
Affinity DataKi:  1.60nMAssay Description:Binding affinity towards human sst1 receptor expressed in CHO-K1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 4(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50064772(Ala-Gly-cyclo[Cys-Lys-Asn-Phe-Phe-Trp-Lys-Thr-Phe-...)
Affinity DataKi:  1.80nMAssay Description:Binding affinity towards human sst4 receptor expressed in CHO-K1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 5(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50064772(Ala-Gly-cyclo[Cys-Lys-Asn-Phe-Phe-Trp-Lys-Thr-Phe-...)
Affinity DataKi:  2.30nMAssay Description:Binding affinity towards human sst5 receptor expressed in CHO-K1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 2(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50064774(1'N-[1-(3-aminomethylcyclohexylmethylcarbamoyl)-2-...)
Affinity DataKi:  4nMAssay Description:Binding affinity towards human sst2 receptor expressed in CHO-K1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 2(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50064776(1'N-[1-[3-aminomethyl-(1R,3S)-cyclohexylmethylcarb...)
Affinity DataKi:  20nMAssay Description:Binding affinity towards human sst2 receptor expressed in CHO-K1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 2(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50454937(CHEMBL2112223)
Affinity DataKi:  46nMAssay Description:Binding affinity towards human sst2 receptor expressed in CHO-K1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 2(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50454936(CHEMBL2112222)
Affinity DataKi:  53nMAssay Description:Binding affinity towards human sst2 receptor expressed in CHO-K1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 2(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50064775(1'N-[1-(6-aminohexylcarbamoyl)-2-(1H-3-indolyl)-(1...)
Affinity DataKi:  225nMAssay Description:Binding affinity towards human sst2 receptor expressed in CHO-K1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 2(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50064782(1'N-[1-(4-aminobutylcarbamoyl)-2-(1H-3-indolyl)-(1...)
Affinity DataKi:  300nMAssay Description:Binding affinity towards human sst2 receptor expressed in CHO-K1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 1(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50064774(1'N-[1-(3-aminomethylcyclohexylmethylcarbamoyl)-2-...)
Affinity DataKi:  537nMAssay Description:Binding affinity towards human sst1 receptor expressed in CHO-K1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 2(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50064770(1'N-[1-(4-aminobutylcarbamoyl)-2-(1H-3-indolyl)eth...)
Affinity DataKi:  615nMAssay Description:Binding affinity towards human sst2 receptor expressed in CHO-K1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 2(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50064780(1'N-[1-(3-aminopropylcarbamoyl)-2-(1H-3-indolyl)-(...)
Affinity DataKi:  815nMAssay Description:Binding affinity towards human sst2 receptor expressed in CHO-K1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 2(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50064777(6-amino-2-[2-(1H-3-indolyl)-1-spiro[1H-indene-1,4'...)
Affinity DataKi:  1.11E+3nMAssay Description:Binding affinity towards human sst2 receptor expressed in CHO-K1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 2(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50064773(1'N-[1-[3-aminomethyl-(1S,3R)-cyclohexylmethylcarb...)
Affinity DataKi:  1.74E+3nMAssay Description:Binding affinity towards human sst2 receptor expressed in CHO-K1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 4(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50064773(1'N-[1-[3-aminomethyl-(1S,3R)-cyclohexylmethylcarb...)
Affinity DataKi:  2.00E+3nMAssay Description:Binding affinity towards human sst4 receptor expressed in CHO-K1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 4(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50064776(1'N-[1-[3-aminomethyl-(1R,3S)-cyclohexylmethylcarb...)
Affinity DataKi:  2.18E+3nMAssay Description:Binding affinity towards human sst4 receptor expressed in CHO-K1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 1(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50064776(1'N-[1-[3-aminomethyl-(1R,3S)-cyclohexylmethylcarb...)
Affinity DataKi:  2.43E+3nMAssay Description:Binding affinity towards human sst1 receptor expressed in CHO-K1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 4(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50064774(1'N-[1-(3-aminomethylcyclohexylmethylcarbamoyl)-2-...)
Affinity DataKi:  2.48E+3nMAssay Description:Binding affinity towards human sst4 receptor expressed in CHO-K1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 3(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50454937(CHEMBL2112223)
Affinity DataKi:  2.57E+3nMAssay Description:Binding affinity towards human sst3 receptor expressed in CHO-K1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 3(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50064773(1'N-[1-[3-aminomethyl-(1S,3R)-cyclohexylmethylcarb...)
Affinity DataKi:  2.95E+3nMAssay Description:Binding affinity towards human sst3 receptor expressed in CHO-K1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 5(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50064776(1'N-[1-[3-aminomethyl-(1R,3S)-cyclohexylmethylcarb...)
Affinity DataKi:  3.32E+3nMAssay Description:Binding affinity towards human sst5 receptor expressed in CHO-K1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 3(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50064774(1'N-[1-(3-aminomethylcyclohexylmethylcarbamoyl)-2-...)
Affinity DataKi:  3.61E+3nMAssay Description:Binding affinity towards human sst3 receptor expressed in CHO-K1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 3(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50064776(1'N-[1-[3-aminomethyl-(1R,3S)-cyclohexylmethylcarb...)
Affinity DataKi:  3.69E+3nMAssay Description:Binding affinity towards human sst3 receptor expressed in CHO-K1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 1(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50064770(1'N-[1-(4-aminobutylcarbamoyl)-2-(1H-3-indolyl)eth...)
Affinity DataKi:  4.26E+3nMAssay Description:Binding affinity towards human sst1 receptor expressed in CHO-K1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 5(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50064773(1'N-[1-[3-aminomethyl-(1S,3R)-cyclohexylmethylcarb...)
Affinity DataKi:  4.47E+3nMAssay Description:Binding affinity towards human sst5 receptor expressed in CHO-K1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 5(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50064774(1'N-[1-(3-aminomethylcyclohexylmethylcarbamoyl)-2-...)
Affinity DataKi:  5.02E+3nMAssay Description:Binding affinity towards human sst5 receptor expressed in CHO-K1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 1(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50454937(CHEMBL2112223)
Affinity DataKi:  5.38E+3nMAssay Description:Binding affinity towards human sst1 receptor expressed in CHO-K1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 3(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50064770(1'N-[1-(4-aminobutylcarbamoyl)-2-(1H-3-indolyl)eth...)
Affinity DataKi:  5.69E+3nMAssay Description:Binding affinity towards human sst3 receptor expressed in CHO-K1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 4(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50454937(CHEMBL2112223)
Affinity DataKi:  6.84E+3nMAssay Description:Binding affinity towards human sst4 receptor expressed in CHO-K1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 2(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50064781(1'N-[1-(4-aminobutylcarbamoyl)-2-(1H-3-indolyl)-(1...)
Affinity DataKi:  1.00E+4nMAssay Description:Binding affinity towards human sst2 receptor expressed in CHO-K1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 5(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50064770(1'N-[1-(4-aminobutylcarbamoyl)-2-(1H-3-indolyl)eth...)
Affinity DataKi: >1.00E+4nMAssay Description:Binding affinity towards human sst5 receptor expressed in CHO-K1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 5(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50454937(CHEMBL2112223)
Affinity DataKi: >1.00E+4nMAssay Description:Binding affinity towards human sst5 receptor expressed in CHO-K1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 4(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50064770(1'N-[1-(4-aminobutylcarbamoyl)-2-(1H-3-indolyl)eth...)
Affinity DataKi: >1.00E+4nMAssay Description:Binding affinity towards human sst4 receptor expressed in CHO-K1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed