Compile Data Set for Download or QSAR
maximum 50k data
Found 18 Enz. Inhib. hit(s) with all data for entry = 5183
TargetMelatonin receptor type 1A(Homo sapiens (Human))
Universita Degli Studi Di Milano

Curated by PDSP Ki Database
LigandPNGBDBM85372(CAS_121-75-5 | MLT | Malathion)
Affinity DataKi:  0.290nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelatonin receptor type 1A(Homo sapiens (Human))
Universita Degli Studi Di Milano

Curated by PDSP Ki Database
LigandPNGBDBM85361(N-[(1H-Indol-2-yl)alkyl]acylamino Derivatives 5h)
Affinity DataKi:  63.1nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelatonin receptor type 1A(Homo sapiens (Human))
Universita Degli Studi Di Milano

Curated by PDSP Ki Database
LigandPNGBDBM85371(N-[(1H-Indol-2-yl)alkyl]acylamino Derivatives 5f)
Affinity DataKi:  87.1nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelatonin receptor type 1A(Homo sapiens (Human))
Universita Degli Studi Di Milano

Curated by PDSP Ki Database
LigandPNGBDBM85360(N-[(1H-Indol-2-yl)alkyl]acylamino Derivatives 5g)
Affinity DataKi:  135nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelatonin receptor type 1A(Homo sapiens (Human))
Universita Degli Studi Di Milano

Curated by PDSP Ki Database
LigandPNGBDBM50034101(CHEMBL14701 | Compound 6 | Cyclobutanecarboxylic a...)
Affinity DataKi:  200nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelatonin receptor type 1A(Homo sapiens (Human))
Universita Degli Studi Di Milano

Curated by PDSP Ki Database
LigandPNGBDBM85368(N-[(1H-Indol-2-yl)alkyl]acylamino Derivatives 9)
Affinity DataKi:  407nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelatonin receptor type 1A(Homo sapiens (Human))
Universita Degli Studi Di Milano

Curated by PDSP Ki Database
LigandPNGBDBM82271(CAS_260803 | NAS | NSC_260803)
Affinity DataKi:  490nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelatonin receptor type 1A(Homo sapiens (Human))
Universita Degli Studi Di Milano

Curated by PDSP Ki Database
LigandPNGBDBM85359
Affinity DataKi:  631nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMelatonin receptor type 1A(Homo sapiens (Human))
Universita Degli Studi Di Milano

Curated by PDSP Ki Database
LigandPNGBDBM85373(N-[(1H-Indol-2-yl)alkyl]acylamino Derivatives 5a)
Affinity DataKi:  631nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelatonin receptor type 1A(Homo sapiens (Human))
Universita Degli Studi Di Milano

Curated by PDSP Ki Database
LigandPNGBDBM85362(N-[(1H-Indol-2-yl)alkyl]acylamino Derivatives 5j)
Affinity DataKi:  832nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMelatonin receptor type 1A(Homo sapiens (Human))
Universita Degli Studi Di Milano

Curated by PDSP Ki Database
LigandPNGBDBM85363(N-[(1H-Indol-2-yl)alkyl]acylamino Derivatives 8)
Affinity DataKi:  1.23E+3nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelatonin receptor type 1A(Homo sapiens (Human))
Universita Degli Studi Di Milano

Curated by PDSP Ki Database
LigandPNGBDBM85365(N-[(1H-Indol-2-yl)alkyl]acylamino Derivatives 5i)
Affinity DataKi:  1.82E+3nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelatonin receptor type 1A(Homo sapiens (Human))
Universita Degli Studi Di Milano

Curated by PDSP Ki Database
LigandPNGBDBM85364(N-[(1H-Indol-2-yl)alkyl]acylamino Derivatives 5d)
Affinity DataKi:  2.45E+3nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelatonin receptor type 1A(Homo sapiens (Human))
Universita Degli Studi Di Milano

Curated by PDSP Ki Database
LigandPNGBDBM85366(N-[(1H-Indol-2-yl)alkyl]acylamino Derivatives 13)
Affinity DataKi:  2.95E+3nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMelatonin receptor type 1A(Homo sapiens (Human))
Universita Degli Studi Di Milano

Curated by PDSP Ki Database
LigandPNGBDBM85358(N-[(1H-Indol-2-yl)alkyl]acylamino Derivatives 5c)
Affinity DataKi:  3.80E+3nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelatonin receptor type 1A(Homo sapiens (Human))
Universita Degli Studi Di Milano

Curated by PDSP Ki Database
LigandPNGBDBM85370(N-[(1H-Indol-2-yl)alkyl]acylamino Derivatives 5k)
Affinity DataKi:  3.98E+3nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMelatonin receptor type 1A(Homo sapiens (Human))
Universita Degli Studi Di Milano

Curated by PDSP Ki Database
LigandPNGBDBM85367(N-[(1H-Indol-2-yl)alkyl]acylamino Derivatives 5b)
Affinity DataKi:  8.51E+3nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelatonin receptor type 1A(Homo sapiens (Human))
Universita Degli Studi Di Milano

Curated by PDSP Ki Database
LigandPNGBDBM85369(N-[(1H-Indol-2-yl)alkyl]acylamino Derivatives 5e)
Affinity DataKi: >1.00E+4nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed