Compile Data Set for Download or QSAR
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Found 30 Enz. Inhib. hit(s) with all data for entry = 50007845
Target5-hydroxytryptamine receptor 2C(Homo sapiens (Human))
Purdue University

Curated by ChEMBL
LigandPNGBDBM50068516(2-(5-Methoxy-1H-indol-3-yl)-propylamine | CHEMBL14...)
Affinity DataKi:  1nMAssay Description:Binding affinity against the cloned human 5-hydroxytryptamine 2C receptor using [125I]-DOI as the radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2C(Homo sapiens (Human))
Purdue University

Curated by ChEMBL
LigandPNGBDBM50068514(2-(5-Fluoro-1H-indol-3-yl)-cyclopropylamine | CHEM...)
Affinity DataKi:  1.90nMAssay Description:Binding affinity against the cloned human 5-hydroxytryptamine 2C receptor using [125I]-DOI as the radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
Purdue University

Curated by ChEMBL
LigandPNGBDBM21393(7-(dipropylamino)-5,6,7,8-tetrahydronaphthalen-1-o...)
Affinity DataKi:  2.10nMAssay Description:Binding affinity against the 5-hydroxytryptamine 1A receptor labelled with [3H]-8-OH-DPAT in rat hippocampal homogenatesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2A(Homo sapiens (Human))
Purdue University

Curated by ChEMBL
LigandPNGBDBM50068516(2-(5-Methoxy-1H-indol-3-yl)-propylamine | CHEMBL14...)
Affinity DataKi:  2.20nMAssay Description:Binding affinity against the cloned human 5-hydroxytryptamine 2A receptor using [125I]-DOI as the radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2B(Homo sapiens (Human))
Purdue University

Curated by ChEMBL
LigandPNGBDBM50068514(2-(5-Fluoro-1H-indol-3-yl)-cyclopropylamine | CHEM...)
Affinity DataKi:  5.70nMAssay Description:Binding affinity against the cloned human 5-hydroxytryptamine 2B receptor using [3H]-5-HT as the radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2B(Homo sapiens (Human))
Purdue University

Curated by ChEMBL
LigandPNGBDBM50068516(2-(5-Methoxy-1H-indol-3-yl)-propylamine | CHEMBL14...)
Affinity DataKi:  8.30nMAssay Description:Binding affinity against the cloned human 5-hydroxytryptamine 2B receptor using [3H]-5-HT as the radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2C(Homo sapiens (Human))
Purdue University

Curated by ChEMBL
LigandPNGBDBM50068509(2-(1H-Indol-3-yl)-propylamine | CHEMBL148463)
Affinity DataKi:  9.30nMAssay Description:Binding affinity against the cloned human 5-hydroxytryptamine 2C receptor using [125I]-DOI as the radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2A(Homo sapiens (Human))
Purdue University

Curated by ChEMBL
LigandPNGBDBM50068514(2-(5-Fluoro-1H-indol-3-yl)-cyclopropylamine | CHEM...)
Affinity DataKi:  10.2nMAssay Description:Binding affinity against the cloned human 5-hydroxytryptamine 2A receptor using [125I]-DOI as the radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2C(Homo sapiens (Human))
Purdue University

Curated by ChEMBL
LigandPNGBDBM50068515(2-(4-Methoxy-1H-indol-3-yl)-cyclopropylamine | CHE...)
Affinity DataKi:  11.8nMAssay Description:Binding affinity against the cloned human 5-hydroxytryptamine 2C receptor using [125I]-DOI as the radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2C(Homo sapiens (Human))
Purdue University

Curated by ChEMBL
LigandPNGBDBM50068510(2-(5-Methoxy-1H-indol-3-yl)-cyclopropylamine | CHE...)
Affinity DataKi:  17.8nMAssay Description:Binding affinity against the cloned human 5-hydroxytryptamine 2C receptor using [125I]-DOI as the radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2C(Homo sapiens (Human))
Purdue University

Curated by ChEMBL
LigandPNGBDBM50068512((1S,2R)-2-(1H-Indol-3-yl)-cyclopropylamine | CHEMB...)
Affinity DataKi:  21.3nMAssay Description:Binding affinity against the cloned human 5-hydroxytryptamine 2C receptor using [125I]-DOI as the radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2C(Homo sapiens (Human))
Purdue University

Curated by ChEMBL
LigandPNGBDBM50068511(2-(1H-Indol-3-yl)-cyclopropylamine | CHEMBL358810)
Affinity DataKi:  29.9nMAssay Description:Binding affinity against the cloned human 5-hydroxytryptamine 2C receptor using [125I]-DOI as the radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2A(Homo sapiens (Human))
Purdue University

Curated by ChEMBL
LigandPNGBDBM50068510(2-(5-Methoxy-1H-indol-3-yl)-cyclopropylamine | CHE...)
Affinity DataKi:  30.9nMAssay Description:Binding affinity against the cloned human 5-hydroxytryptamine 2A receptor using [125I]-DOI as the radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2B(Homo sapiens (Human))
Purdue University

Curated by ChEMBL
LigandPNGBDBM50068510(2-(5-Methoxy-1H-indol-3-yl)-cyclopropylamine | CHE...)
Affinity DataKi:  38.1nMAssay Description:Binding affinity against the cloned human 5-hydroxytryptamine 2B receptor using [3H]-5-HT as the radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
Purdue University

Curated by ChEMBL
LigandPNGBDBM50068510(2-(5-Methoxy-1H-indol-3-yl)-cyclopropylamine | CHE...)
Affinity DataKi:  40.1nMAssay Description:Binding affinity against the 5-hydroxytryptamine 1A receptor labelled with [3H]-8-OH-DPAT in rat hippocampal homogenatesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2A(Homo sapiens (Human))
Purdue University

Curated by ChEMBL
LigandPNGBDBM50068509(2-(1H-Indol-3-yl)-propylamine | CHEMBL148463)
Affinity DataKi:  41nMAssay Description:Binding affinity against the cloned human 5-hydroxytryptamine 2A receptor using [125I]-DOI as the radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2C(Homo sapiens (Human))
Purdue University

Curated by ChEMBL
LigandPNGBDBM50068513((1R,2S)-2-(1H-Indol-3-yl)-cyclopropylamine | CHEMB...)
Affinity DataKi:  44.1nMAssay Description:Binding affinity against the cloned human 5-hydroxytryptamine 2C receptor using [125I]-DOI as the radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2A(Homo sapiens (Human))
Purdue University

Curated by ChEMBL
LigandPNGBDBM50068515(2-(4-Methoxy-1H-indol-3-yl)-cyclopropylamine | CHE...)
Affinity DataKi:  45.9nMAssay Description:Binding affinity against the cloned human 5-hydroxytryptamine 2A receptor using [125I]-DOI as the radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2B(Homo sapiens (Human))
Purdue University

Curated by ChEMBL
LigandPNGBDBM50068511(2-(1H-Indol-3-yl)-cyclopropylamine | CHEMBL358810)
Affinity DataKi:  58.3nMAssay Description:Binding affinity against the cloned human 5-hydroxytryptamine 2B receptor using [3H]-5-HT as the radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2B(Homo sapiens (Human))
Purdue University

Curated by ChEMBL
LigandPNGBDBM50068513((1R,2S)-2-(1H-Indol-3-yl)-cyclopropylamine | CHEMB...)
Affinity DataKi:  58.5nMAssay Description:Binding affinity against the cloned human 5-hydroxytryptamine 2B receptor using [3H]-5-HT as the radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2B(Homo sapiens (Human))
Purdue University

Curated by ChEMBL
LigandPNGBDBM50068515(2-(4-Methoxy-1H-indol-3-yl)-cyclopropylamine | CHE...)
Affinity DataKi:  64.9nMAssay Description:Binding affinity against the cloned human 5-hydroxytryptamine 2B receptor using [3H]-5-HT as the radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2B(Homo sapiens (Human))
Purdue University

Curated by ChEMBL
LigandPNGBDBM50068509(2-(1H-Indol-3-yl)-propylamine | CHEMBL148463)
Affinity DataKi:  87nMAssay Description:Binding affinity against the cloned human 5-hydroxytryptamine 2B receptor using [3H]-5-HT as the radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2B(Homo sapiens (Human))
Purdue University

Curated by ChEMBL
LigandPNGBDBM50068512((1S,2R)-2-(1H-Indol-3-yl)-cyclopropylamine | CHEMB...)
Affinity DataKi:  93.5nMAssay Description:Binding affinity against the cloned human 5-hydroxytryptamine 2B receptor using [3H]-5-HT as the radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2A(Homo sapiens (Human))
Purdue University

Curated by ChEMBL
LigandPNGBDBM50068513((1R,2S)-2-(1H-Indol-3-yl)-cyclopropylamine | CHEMB...)
Affinity DataKi:  98.2nMAssay Description:Binding affinity against the cloned human 5-hydroxytryptamine 2A receptor using [125I]-DOI as the radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2A(Homo sapiens (Human))
Purdue University

Curated by ChEMBL
LigandPNGBDBM50068512((1S,2R)-2-(1H-Indol-3-yl)-cyclopropylamine | CHEMB...)
Affinity DataKi:  132nMAssay Description:Binding affinity against the cloned human 5-hydroxytryptamine 2A receptor using [125I]-DOI as the radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2A(Homo sapiens (Human))
Purdue University

Curated by ChEMBL
LigandPNGBDBM50068511(2-(1H-Indol-3-yl)-cyclopropylamine | CHEMBL358810)
Affinity DataKi:  164nMAssay Description:Binding affinity against the cloned human 5-hydroxytryptamine 2A receptor using [125I]-DOI as the radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
Purdue University

Curated by ChEMBL
LigandPNGBDBM50068514(2-(5-Fluoro-1H-indol-3-yl)-cyclopropylamine | CHEM...)
Affinity DataKi:  258nMAssay Description:Binding affinity against the 5-hydroxytryptamine 1A receptor labelled with [3H]-8-OH-DPAT in rat hippocampal homogenatesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
Purdue University

Curated by ChEMBL
LigandPNGBDBM50068513((1R,2S)-2-(1H-Indol-3-yl)-cyclopropylamine | CHEMB...)
Affinity DataKi:  258nMAssay Description:Binding affinity against the 5-hydroxytryptamine 1A receptor labelled with [3H]-8-OH-DPAT in rat hippocampal homogenatesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
Purdue University

Curated by ChEMBL
LigandPNGBDBM50068512((1S,2R)-2-(1H-Indol-3-yl)-cyclopropylamine | CHEMB...)
Affinity DataKi:  810nMAssay Description:Binding affinity against the 5-hydroxytryptamine 1A receptor labelled with [3H]-8-OH-DPAT in rat hippocampal homogenatesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
Purdue University

Curated by ChEMBL
LigandPNGBDBM50068515(2-(4-Methoxy-1H-indol-3-yl)-cyclopropylamine | CHE...)
Affinity DataKi:  1.53E+3nMAssay Description:Binding affinity against the 5-hydroxytryptamine 1A receptor labelled with [3H]-8-OH-DPAT in rat hippocampal homogenatesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed