Compile Data Set for Download or QSAR
maximum 50k data
Found 14 Enz. Inhib. hit(s) with all data for entry = 50008028
TargetHistamine H3 receptor(Rattus norvegicus (rat))
Gliatech

Curated by ChEMBL
LigandPNGBDBM22541(Clobenpropit | N''-[(4-chlorophenyl)methyl]{[3-(1H...)
Affinity DataKi:  0.180nMAssay Description:Inhibition of [3H]- N-alpha-methylhistamine from histamine H3 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Rattus norvegicus (rat))
Gliatech

Curated by ChEMBL
LigandPNGBDBM50070217(3-(3-Bromo-4-methoxy-phenyl)-2-[(E)-hydroxyimino]-...)
Affinity DataKi:  0.5nMAssay Description:Inhibition of [3H]- N-alpha-methylhistamine from histamine H3 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Rattus norvegicus (rat))
Gliatech

Curated by ChEMBL
LigandPNGBDBM50070214(4-(7,7-Dimethyl-oct-3-ynyl)-1H-imidazole | CHEMBL2...)
Affinity DataKi:  0.800nMAssay Description:Inhibition of [3H]- N-alpha-methylhistamine from histamine H3 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Rattus norvegicus (rat))
Gliatech

Curated by ChEMBL
LigandPNGBDBM50070220(4-(6-Cyclopentyl-hex-3-ynyl)-1H-imidazole | CHEMBL...)
Affinity DataKi:  0.950nMAssay Description:Inhibition of [3H]- N-alpha-methylhistamine from histamine H3 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Rattus norvegicus (rat))
Gliatech

Curated by ChEMBL
LigandPNGBDBM7967(1-methyl-5-(beta-aminoethyl)-imidazole | 2-(1-meth...)
Affinity DataKi:  1nMAssay Description:Inhibition of [3H]- N-alpha-methylhistamine from histamine H3 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Rattus norvegicus (rat))
Gliatech

Curated by ChEMBL
LigandPNGBDBM22914(CHEMBL260374 | N-cyclohexyl-4-(1H-imidazol-5-yl)pi...)
Affinity DataKi:  1.5nMAssay Description:Antagonistic activity of the compound was evaluated against histamine H3 receptor using [3H]- N-alpha-methylhistamine as radioligand in experiment 2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Rattus norvegicus (rat))
Gliatech

Curated by ChEMBL
LigandPNGBDBM50070211(4-(6-Cyclohexyl-hex-3-ynyl)-1H-imidazole | CHEMBL1...)
Affinity DataKi:  2.90nMAssay Description:Inhibition of [3H]- N-alpha-methylhistamine from histamine H3 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Rattus norvegicus (rat))
Gliatech

Curated by ChEMBL
LigandPNGBDBM50070216(4-(8-Phenyl-oct-3-ynyl)-1H-imidazole | CHEMBL14811)
Affinity DataKi:  3.5nMAssay Description:Inhibition of [3H]- N-alpha-methylhistamine from histamine H3 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Rattus norvegicus (rat))
Gliatech

Curated by ChEMBL
LigandPNGBDBM50070212(4-(7-Methyl-oct-3-ynyl)-1H-imidazole | CHEMBL14497)
Affinity DataKi:  3.70nMAssay Description:Inhibition of [3H]- N-alpha-methylhistamine from histamine H3 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Rattus norvegicus (rat))
Gliatech

Curated by ChEMBL
LigandPNGBDBM22914(CHEMBL260374 | N-cyclohexyl-4-(1H-imidazol-5-yl)pi...)
Affinity DataKi:  4.30nMAssay Description:Antagonistic activity of the compound was evaluated against histamine H3 receptor using [3H]- N-alpha-methylhistamine as radioligand in experiment 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Rattus norvegicus (rat))
Gliatech

Curated by ChEMBL
LigandPNGBDBM50070213(3-(4-Chloro-benzyl)-5-[2-(1H-imidazol-4-yl)-ethyl]...)
Affinity DataKi:  7nMAssay Description:Inhibition of [3H]- N-alpha-methylhistamine from histamine H3 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Rattus norvegicus (rat))
Gliatech

Curated by ChEMBL
LigandPNGBDBM50070215(4-Hept-3-ynyl-1H-imidazole | CHEMBL276804)
Affinity DataKi:  27nMAssay Description:Inhibition of [3H]- N-alpha-methylhistamine from histamine H3 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Rattus norvegicus (rat))
Gliatech

Curated by ChEMBL
LigandPNGBDBM86490(CAS_0 | CHEMBL14812 | GT 2016 | NSC_0)
Affinity DataKi:  40nMAssay Description:Inhibition of [3H]- N-alpha-methylhistamine from histamine H3 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Rattus norvegicus (rat))
Gliatech

Curated by ChEMBL
LigandPNGBDBM50070219(4-Hex-3-ynyl-1H-imidazole | CHEMBL14721)
Affinity DataKi:  79nMAssay Description:Inhibition of [3H]- N-alpha-methylhistamine from histamine H3 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed