Compile Data Set for Download or QSAR
maximum 50k data
Found 19 Enz. Inhib. hit(s) with all data for entry = 50008153
TargetSubstance-K receptor(Homo sapiens (Human))
Zeneca Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50403654(CHEMBL2115073)
Affinity DataKi:  0.840nMAssay Description:Displacement of [3H]- NKA from human NK-2 receptor expressed in MEL cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-K receptor(Homo sapiens (Human))
Zeneca Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50071118(CHEMBL2111522 | CHEMBL443264 | N-[2-(3,4-Dichloro-...)
Affinity DataKi:  1.30nMAssay Description:Displacement of [3H]- NKA from human NK-2 receptor expressed in MEL cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-K receptor(Homo sapiens (Human))
Zeneca Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50071112(CHEMBL56835 | N-[4-(4-Acetylamino-4-phenyl-piperid...)
Affinity DataKi:  1.75nMAssay Description:Displacement of [3H]- NKA from human NK-2 receptor expressed in MEL cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-K receptor(Homo sapiens (Human))
Zeneca Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50071112(CHEMBL56835 | N-[4-(4-Acetylamino-4-phenyl-piperid...)
Affinity DataKi:  1.80nMAssay Description:Displacement of [3H]- NKA from human NK-2 receptor expressed in MEL cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-K receptor(Homo sapiens (Human))
Zeneca Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50216091(CHEMBL2111522)
Affinity DataKi:  2.10nMAssay Description:Displacement of [3H]- NKA from human NK-2 receptor expressed in MEL cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-K receptor(Homo sapiens (Human))
Zeneca Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50071118(CHEMBL2111522 | CHEMBL443264 | N-[2-(3,4-Dichloro-...)
Affinity DataKi:  2.70nMAssay Description:Displacement of [3H]- NKA from human NK-2 receptor expressed in MEL cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-K receptor(Homo sapiens (Human))
Zeneca Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50071125(CHEMBL56481 | N-{2-(3,4-Dichloro-phenyl)-4-[4-(1-e...)
Affinity DataKi:  3.5nMAssay Description:Displacement of [3H]- NKA from human NK-2 receptor expressed in MEL cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-K receptor(Homo sapiens (Human))
Zeneca Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50071120(CHEMBL56788 | N-{2-(3,4-Dichloro-phenyl)-4-[4-(1-h...)
Affinity DataKi:  3.70nMAssay Description:Displacement of [3H]- NKA from human NK-2 receptor expressed in MEL cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-K receptor(Homo sapiens (Human))
Zeneca Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50071119(CHEMBL56143 | N-{2-(3,4-Dichloro-phenyl)-4-[4-(1-h...)
Affinity DataKi:  4.70nMAssay Description:Displacement of [3H]- NKA from human NK-2 receptor expressed in MEL cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-K receptor(Homo sapiens (Human))
Zeneca Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50071115(CHEMBL58638 | N-[2-(3,4-Dichloro-phenyl)-4-(4-{1-[...)
Affinity DataKi:  6.5nMAssay Description:Displacement of [3H]- NKA from human NK-2 receptor expressed in MEL cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-K receptor(Homo sapiens (Human))
Zeneca Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50071121(CHEMBL301437 | N-{2-(3,4-Dichloro-phenyl)-4-[4-(1-...)
Affinity DataKi:  7.70nMAssay Description:Displacement of [3H]- NKA from human NK-2 receptor expressed in MEL cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-K receptor(Homo sapiens (Human))
Zeneca Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50071122(CHEMBL417940 | N-[2-(3,4-Dichloro-phenyl)-4-(4-pro...)
Affinity DataKi:  9.20nMAssay Description:Displacement of [3H]- NKA from human NK-2 receptor expressed in MEL cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-K receptor(Homo sapiens (Human))
Zeneca Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50071126(CHEMBL59542 | N-[2-(3,4-Dichloro-phenyl)-4-(4-prop...)
Affinity DataKi:  9.90nMAssay Description:Displacement of [3H]- NKA from human NK-2 receptor expressed in MEL cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-K receptor(Homo sapiens (Human))
Zeneca Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50071124(CHEMBL56739 | N-{2-(3,4-Dichloro-phenyl)-4-[4-(1-h...)
Affinity DataKi:  13nMAssay Description:Displacement of [3H]- NKA from human NK-2 receptor expressed in MEL cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-K receptor(Homo sapiens (Human))
Zeneca Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50071123(CHEMBL56274 | N-{2-(3,4-Dichloro-phenyl)-4-[4-(1-h...)
Affinity DataKi:  34nMAssay Description:Displacement of [3H]- NKA from human NK-2 receptor expressed in MEL cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-K receptor(Homo sapiens (Human))
Zeneca Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50071113(Acetic acid 2-{1-[4-(benzoyl-methyl-amino)-3-(3,4-...)
Affinity DataKi:  40nMAssay Description:Displacement of [3H]- NKA from human NK-2 receptor expressed in MEL cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-K receptor(Homo sapiens (Human))
Zeneca Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50071117(CHEMBL292415 | N-{2-(3,4-Dichloro-phenyl)-4-[4-(2-...)
Affinity DataKi:  47nMAssay Description:Displacement of [3H]- NKA from human NK-2 receptor expressed in MEL cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-K receptor(Homo sapiens (Human))
Zeneca Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50071116(CHEMBL58331 | N-[4-[4-(2-Acetylamino-ethyl)-piperi...)
Affinity DataKi:  66nMAssay Description:Displacement of [3H]- NKA from human NK-2 receptor expressed in MEL cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-K receptor(Homo sapiens (Human))
Zeneca Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50071114(CHEMBL57224 | N-[2-(3,4-Dichloro-phenyl)-4-(4-hydr...)
Affinity DataKi:  142nMAssay Description:Displacement of [3H]- NKA from human NK-2 receptor expressed in MEL cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed