Compile Data Set for Download or QSAR
Report error Found 140 Enz. Inhib. hit(s) with all data for entry = 3480
TargetProtein arginine N-methyltransferase 5(Human)
Ctxt

US Patent
LigandPNGBDBM401715(US10005792, Compound 77 | US10005792, Compound 135)
Affinity DataIC50: 15nMAssay Description:Compounds of the invention may be tested for in vitro activity in the following assay: A histone H4 derived peptide is used as substrate (amino acid ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/18/2020
Entry Details
US Patent

TargetProtein arginine N-methyltransferase 5(Human)
Ctxt

US Patent
LigandPNGBDBM401715(US10005792, Compound 77 | US10005792, Compound 135)
Affinity DataIC50: 29nMAssay Description:Compounds of the invention may be tested for in vitro activity in the following assay: A histone H4 derived peptide is used as substrate (amino acid ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/18/2020
Entry Details
US Patent

TargetProtein arginine N-methyltransferase 5(Human)
Ctxt

US Patent
LigandPNGBDBM401764(US10005792, Compound 123)
Affinity DataIC50: 40nMAssay Description:Compounds of the invention may be tested for in vitro activity in the following assay: A histone H4 derived peptide is used as substrate (amino acid ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/18/2020
Entry Details
US Patent

TargetProtein arginine N-methyltransferase 5(Human)
Ctxt

US Patent
LigandPNGBDBM401765(US10005792, Compound 124)
Affinity DataIC50: 48nMAssay Description:Compounds of the invention may be tested for in vitro activity in the following assay: A histone H4 derived peptide is used as substrate (amino acid ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/18/2020
Entry Details
US Patent

TargetProtein arginine N-methyltransferase 5(Human)
Ctxt

US Patent
LigandPNGBDBM401741(US10005792, Compound 103 | US10005792, Compound 13...)
Affinity DataIC50: 50nMAssay Description:Compounds of the invention may be tested for in vitro activity in the following assay: A histone H4 derived peptide is used as substrate (amino acid ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/18/2020
Entry Details
US Patent

TargetProtein arginine N-methyltransferase 5(Human)
Ctxt

US Patent
LigandPNGBDBM401672(US10005792, Compound 35)
Affinity DataIC50: 50nMAssay Description:Compounds of the invention may be tested for in vitro activity in the following assay: A histone H4 derived peptide is used as substrate (amino acid ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/18/2020
Entry Details
US Patent

TargetProtein arginine N-methyltransferase 5(Human)
Ctxt

US Patent
LigandPNGBDBM401677(US10005792, Compound 40)
Affinity DataIC50: 57nMAssay Description:Compounds of the invention may be tested for in vitro activity in the following assay: A histone H4 derived peptide is used as substrate (amino acid ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/18/2020
Entry Details
US Patent

TargetProtein arginine N-methyltransferase 5(Human)
Ctxt

US Patent
LigandPNGBDBM401713(US10005792, Compound 75)
Affinity DataIC50: 64nMAssay Description:Compounds of the invention may be tested for in vitro activity in the following assay: A histone H4 derived peptide is used as substrate (amino acid ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/18/2020
Entry Details
US Patent

TargetProtein arginine N-methyltransferase 5(Human)
Ctxt

US Patent
LigandPNGBDBM401755(US10005792, Compound 114)
Affinity DataIC50: 66nMAssay Description:Compounds of the invention may be tested for in vitro activity in the following assay: A histone H4 derived peptide is used as substrate (amino acid ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/18/2020
Entry Details
US Patent

TargetProtein arginine N-methyltransferase 5(Human)
Ctxt

US Patent
LigandPNGBDBM401673(US10005792, Compound 37)
Affinity DataIC50: 95nMAssay Description:Compounds of the invention may be tested for in vitro activity in the following assay: A histone H4 derived peptide is used as substrate (amino acid ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/18/2020
Entry Details
US Patent

TargetProtein arginine N-methyltransferase 5(Human)
Ctxt

US Patent
LigandPNGBDBM401693(US10005792, Compound 56)
Affinity DataIC50: 98nMAssay Description:Compounds of the invention may be tested for in vitro activity in the following assay: A histone H4 derived peptide is used as substrate (amino acid ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/18/2020
Entry Details
US Patent

TargetProtein arginine N-methyltransferase 5(Human)
Ctxt

US Patent
LigandPNGBDBM401741(US10005792, Compound 103 | US10005792, Compound 13...)
Affinity DataIC50: 120nMAssay Description:Compounds of the invention may be tested for in vitro activity in the following assay: A histone H4 derived peptide is used as substrate (amino acid ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/18/2020
Entry Details
US Patent

TargetProtein arginine N-methyltransferase 5(Human)
Ctxt

US Patent
LigandPNGBDBM401676(US10005792, Compound 39)
Affinity DataIC50: 120nMAssay Description:Compounds of the invention may be tested for in vitro activity in the following assay: A histone H4 derived peptide is used as substrate (amino acid ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/18/2020
Entry Details
US Patent

TargetProtein arginine N-methyltransferase 5(Human)
Ctxt

US Patent
LigandPNGBDBM401762(US10005792, Compound 121)
Affinity DataIC50: 130nMAssay Description:Compounds of the invention may be tested for in vitro activity in the following assay: A histone H4 derived peptide is used as substrate (amino acid ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/18/2020
Entry Details
US Patent

TargetProtein arginine N-methyltransferase 5(Human)
Ctxt

US Patent
LigandPNGBDBM401774(US10005792, Compound 133)
Affinity DataIC50: 131nMAssay Description:Compounds of the invention may be tested for in vitro activity in the following assay: A histone H4 derived peptide is used as substrate (amino acid ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/18/2020
Entry Details
US Patent

TargetProtein arginine N-methyltransferase 5(Human)
Ctxt

US Patent
LigandPNGBDBM401768(US10005792, Compound 127)
Affinity DataIC50: 137nMAssay Description:Compounds of the invention may be tested for in vitro activity in the following assay: A histone H4 derived peptide is used as substrate (amino acid ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/18/2020
Entry Details
US Patent

TargetProtein arginine N-methyltransferase 5(Human)
Ctxt

US Patent
LigandPNGBDBM401679(US10005792, Compound 42)
Affinity DataIC50: 137nMAssay Description:Compounds of the invention may be tested for in vitro activity in the following assay: A histone H4 derived peptide is used as substrate (amino acid ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/18/2020
Entry Details
US Patent

TargetProtein arginine N-methyltransferase 5(Human)
Ctxt

US Patent
LigandPNGBDBM401672(US10005792, Compound 35)
Affinity DataIC50: 155nMAssay Description:Compounds of the invention may be tested for in vitro activity in the following assay: A histone H4 derived peptide is used as substrate (amino acid ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/18/2020
Entry Details
US Patent

TargetProtein arginine N-methyltransferase 5(Human)
Ctxt

US Patent
LigandPNGBDBM401678(US10005792, Compound 41)
Affinity DataIC50: 157nMAssay Description:Compounds of the invention may be tested for in vitro activity in the following assay: A histone H4 derived peptide is used as substrate (amino acid ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/18/2020
Entry Details
US Patent

TargetProtein arginine N-methyltransferase 5(Human)
Ctxt

US Patent
LigandPNGBDBM401708(US10005792, Compound 70)
Affinity DataIC50: 157nMAssay Description:Compounds of the invention may be tested for in vitro activity in the following assay: A histone H4 derived peptide is used as substrate (amino acid ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/18/2020
Entry Details
US Patent

TargetProtein arginine N-methyltransferase 5(Human)
Ctxt

US Patent
LigandPNGBDBM401673(US10005792, Compound 37)
Affinity DataIC50: 163nMAssay Description:Compounds of the invention may be tested for in vitro activity in the following assay: A histone H4 derived peptide is used as substrate (amino acid ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/18/2020
Entry Details
US Patent

TargetProtein arginine N-methyltransferase 5(Human)
Ctxt

US Patent
LigandPNGBDBM401690(US10005792, Compound 53)
Affinity DataIC50: 164nMAssay Description:Compounds of the invention may be tested for in vitro activity in the following assay: A histone H4 derived peptide is used as substrate (amino acid ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/18/2020
Entry Details
US Patent

TargetProtein arginine N-methyltransferase 5(Human)
Ctxt

US Patent
LigandPNGBDBM401763(US10005792, Compound 122)
Affinity DataIC50: 166nMAssay Description:Compounds of the invention may be tested for in vitro activity in the following assay: A histone H4 derived peptide is used as substrate (amino acid ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/18/2020
Entry Details
US Patent

TargetProtein arginine N-methyltransferase 5(Human)
Ctxt

US Patent
LigandPNGBDBM401751(US10005792, Compound 110)
Affinity DataIC50: 166nMAssay Description:Compounds of the invention may be tested for in vitro activity in the following assay: A histone H4 derived peptide is used as substrate (amino acid ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/18/2020
Entry Details
US Patent

TargetProtein arginine N-methyltransferase 5(Human)
Ctxt

US Patent
LigandPNGBDBM401658(US10005792, Compound 22)
Affinity DataIC50: 171nMAssay Description:Compounds of the invention may be tested for in vitro activity in the following assay: A histone H4 derived peptide is used as substrate (amino acid ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/18/2020
Entry Details
US Patent

TargetProtein arginine N-methyltransferase 5(Human)
Ctxt

US Patent
LigandPNGBDBM401698(US10005792, Compound 61)
Affinity DataIC50: 180nMAssay Description:Compounds of the invention may be tested for in vitro activity in the following assay: A histone H4 derived peptide is used as substrate (amino acid ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/18/2020
Entry Details
US Patent

TargetProtein arginine N-methyltransferase 5(Human)
Ctxt

US Patent
LigandPNGBDBM401743(US10005792, Compound 105)
Affinity DataIC50: 196nMAssay Description:Compounds of the invention may be tested for in vitro activity in the following assay: A histone H4 derived peptide is used as substrate (amino acid ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/18/2020
Entry Details
US Patent

TargetProtein arginine N-methyltransferase 5(Human)
Ctxt

US Patent
LigandPNGBDBM401714(US10005792, Compound 76)
Affinity DataIC50: 209nMAssay Description:Compounds of the invention may be tested for in vitro activity in the following assay: A histone H4 derived peptide is used as substrate (amino acid ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/18/2020
Entry Details
US Patent

TargetProtein arginine N-methyltransferase 5(Human)
Ctxt

US Patent
LigandPNGBDBM401675(US10005792, Compound 38)
Affinity DataIC50: 210nMAssay Description:Compounds of the invention may be tested for in vitro activity in the following assay: A histone H4 derived peptide is used as substrate (amino acid ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/18/2020
Entry Details
US Patent

TargetProtein arginine N-methyltransferase 5(Human)
Ctxt

US Patent
LigandPNGBDBM401652(US10005792, Compound 15)
Affinity DataIC50: 218nMAssay Description:Compounds of the invention may be tested for in vitro activity in the following assay: A histone H4 derived peptide is used as substrate (amino acid ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/18/2020
Entry Details
US Patent

TargetProtein arginine N-methyltransferase 5(Human)
Ctxt

US Patent
LigandPNGBDBM401767(US10005792, Compound 126)
Affinity DataIC50: 226nMAssay Description:Compounds of the invention may be tested for in vitro activity in the following assay: A histone H4 derived peptide is used as substrate (amino acid ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/18/2020
Entry Details
US Patent

TargetProtein arginine N-methyltransferase 5(Human)
Ctxt

US Patent
LigandPNGBDBM401727(US10005792, Compound 88)
Affinity DataIC50: 229nMAssay Description:Compounds of the invention may be tested for in vitro activity in the following assay: A histone H4 derived peptide is used as substrate (amino acid ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/18/2020
Entry Details
US Patent

TargetProtein arginine N-methyltransferase 5(Human)
Ctxt

US Patent
LigandPNGBDBM401709(US10005792, Compound 71)
Affinity DataIC50: 237nMAssay Description:Compounds of the invention may be tested for in vitro activity in the following assay: A histone H4 derived peptide is used as substrate (amino acid ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/18/2020
Entry Details
US Patent

TargetProtein arginine N-methyltransferase 5(Human)
Ctxt

US Patent
LigandPNGBDBM401655(US10005792, Compound 18)
Affinity DataIC50: 238nMAssay Description:Compounds of the invention may be tested for in vitro activity in the following assay: A histone H4 derived peptide is used as substrate (amino acid ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/18/2020
Entry Details
US Patent

TargetProtein arginine N-methyltransferase 5(Human)
Ctxt

US Patent
LigandPNGBDBM401775(US10005792, Compound 134)
Affinity DataIC50: 238nMAssay Description:Compounds of the invention may be tested for in vitro activity in the following assay: A histone H4 derived peptide is used as substrate (amino acid ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/18/2020
Entry Details
US Patent

TargetProtein arginine N-methyltransferase 5(Human)
Ctxt

US Patent
LigandPNGBDBM401718(US10005792, Compound 80)
Affinity DataIC50: 253nMAssay Description:Compounds of the invention may be tested for in vitro activity in the following assay: A histone H4 derived peptide is used as substrate (amino acid ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/18/2020
Entry Details
US Patent

TargetProtein arginine N-methyltransferase 5(Human)
Ctxt

US Patent
LigandPNGBDBM401645(US10005792, Compound 8)
Affinity DataIC50: 263nMAssay Description:Compounds of the invention may be tested for in vitro activity in the following assay: A histone H4 derived peptide is used as substrate (amino acid ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/18/2020
Entry Details
US Patent

TargetProtein arginine N-methyltransferase 5(Human)
Ctxt

US Patent
LigandPNGBDBM401757(US10005792, Compound 116)
Affinity DataIC50: 276nMAssay Description:Compounds of the invention may be tested for in vitro activity in the following assay: A histone H4 derived peptide is used as substrate (amino acid ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/18/2020
Entry Details
US Patent

TargetProtein arginine N-methyltransferase 5(Human)
Ctxt

US Patent
LigandPNGBDBM401737(US10005792, Compound 98)
Affinity DataIC50: 281nMAssay Description:Compounds of the invention may be tested for in vitro activity in the following assay: A histone H4 derived peptide is used as substrate (amino acid ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/18/2020
Entry Details
US Patent

TargetProtein arginine N-methyltransferase 5(Human)
Ctxt

US Patent
LigandPNGBDBM401653(US10005792, Compound 16)
Affinity DataIC50: 301nMAssay Description:Compounds of the invention may be tested for in vitro activity in the following assay: A histone H4 derived peptide is used as substrate (amino acid ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/18/2020
Entry Details
US Patent

TargetProtein arginine N-methyltransferase 5(Human)
Ctxt

US Patent
LigandPNGBDBM401756(US10005792, Compound 115)
Affinity DataIC50: 305nMAssay Description:Compounds of the invention may be tested for in vitro activity in the following assay: A histone H4 derived peptide is used as substrate (amino acid ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/18/2020
Entry Details
US Patent

TargetProtein arginine N-methyltransferase 5(Human)
Ctxt

US Patent
LigandPNGBDBM401618(US10005792, Compound 3)
Affinity DataIC50: 309nMAssay Description:Compounds of the invention may be tested for in vitro activity in the following assay: A histone H4 derived peptide is used as substrate (amino acid ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/18/2020
Entry Details
US Patent

TargetProtein arginine N-methyltransferase 5(Human)
Ctxt

US Patent
LigandPNGBDBM401675(US10005792, Compound 38)
Affinity DataIC50: 310nMAssay Description:Compounds of the invention may be tested for in vitro activity in the following assay: A histone H4 derived peptide is used as substrate (amino acid ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/18/2020
Entry Details
US Patent

TargetProtein arginine N-methyltransferase 5(Human)
Ctxt

US Patent
LigandPNGBDBM401617(US10005792, Compound 2)
Affinity DataIC50: 310nMAssay Description:Compounds of the invention may be tested for in vitro activity in the following assay: A histone H4 derived peptide is used as substrate (amino acid ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/18/2020
Entry Details
US Patent

TargetProtein arginine N-methyltransferase 5(Human)
Ctxt

US Patent
LigandPNGBDBM401710(US10005792, Compound 72)
Affinity DataIC50: 341nMAssay Description:Compounds of the invention may be tested for in vitro activity in the following assay: A histone H4 derived peptide is used as substrate (amino acid ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/18/2020
Entry Details
US Patent

TargetProtein arginine N-methyltransferase 5(Human)
Ctxt

US Patent
LigandPNGBDBM401681(US10005792, Compound 44)
Affinity DataIC50: 373nMAssay Description:Compounds of the invention may be tested for in vitro activity in the following assay: A histone H4 derived peptide is used as substrate (amino acid ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/18/2020
Entry Details
US Patent

TargetProtein arginine N-methyltransferase 5(Human)
Ctxt

US Patent
LigandPNGBDBM401660(US10005792, Compound 24)
Affinity DataIC50: 425nMAssay Description:Compounds of the invention may be tested for in vitro activity in the following assay: A histone H4 derived peptide is used as substrate (amino acid ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/18/2020
Entry Details
US Patent

TargetProtein arginine N-methyltransferase 5(Human)
Ctxt

US Patent
LigandPNGBDBM401664(US10005792, Compound 27)
Affinity DataIC50: 434nMAssay Description:Compounds of the invention may be tested for in vitro activity in the following assay: A histone H4 derived peptide is used as substrate (amino acid ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/18/2020
Entry Details
US Patent

TargetProtein arginine N-methyltransferase 5(Human)
Ctxt

US Patent
LigandPNGBDBM401651(US10005792, Compound 14)
Affinity DataIC50: 445nMAssay Description:Compounds of the invention may be tested for in vitro activity in the following assay: A histone H4 derived peptide is used as substrate (amino acid ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/18/2020
Entry Details
US Patent

TargetProtein arginine N-methyltransferase 5(Human)
Ctxt

US Patent
LigandPNGBDBM401692(US10005792, Compound 55)
Affinity DataIC50: 450nMAssay Description:Compounds of the invention may be tested for in vitro activity in the following assay: A histone H4 derived peptide is used as substrate (amino acid ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/18/2020
Entry Details
US Patent

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